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Neuroscience

Neuroscience

Neuroscience inhibitors are compounds designed to modulate the activity of specific proteins, enzymes, or receptors within the nervous system. These inhibitors are crucial for studying the molecular mechanisms underlying neural function, synaptic transmission, and neurodegenerative diseases. By targeting neurotransmitter receptors, ion channels, and signaling pathways, neuroscience inhibitors aid in the exploration of brain function and the development of therapeutic strategies for neurological disorders such as Alzheimer's, Parkinson's, and epilepsy. At CymitQuimica, we offer a comprehensive range of high-quality neuroscience inhibitors to support your research in neurobiology, neuropharmacology, and cognitive sciences.

Subcategories of "Neuroscience"

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Found 5389 products of "Neuroscience"

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  • Naronapride

    CAS:
    <p>Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.</p>
    Formula:C27H41ClN4O5
    Color and Shape:Solid
    Molecular weight:537.09
  • 5-HT7 agonist 2

    CAS:
    <p>Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.</p>
    Formula:C23H29N3O
    Color and Shape:Solid
    Molecular weight:363.5
  • p-MPPF dihydrochloride

    CAS:
    <p>p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.</p>
    Formula:C25H29Cl2FN4O2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:507.43
  • GlyT1 Inhibitor 1

    CAS:
    <p>GlyT1 Inhibitor 1 is a selective and potent GlyT1 inhibitor, inhibiting rGlyT1, used in research on neurological disorders.</p>
    Formula:C22H21N5O2
    Color and Shape:Solid
    Molecular weight:387.43
  • Memoquin

    CAS:
    <p>Memoquin is a multi-target-directed ligand for the therapy of Alzheimer's disease.</p>
    Formula:C38H56N4O4
    Color and Shape:Solid
    Molecular weight:632.88
  • Ro 67-4853

    CAS:
    <p>Ro 67-4853 is a positive allosteric modulator of mGluR1, selectively enhancing the response to the agonist (S)-3,5-dihydroxy-phenylglycine (DHPG).</p>
    Formula:C19H19NO4
    Purity:98.57%
    Color and Shape:Solid
    Molecular weight:325.36
  • GAT107

    CAS:
    <p>GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.</p>
    Formula:C18H17BrN2O2S
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:405.31
  • SCH 57790

    CAS:
    SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.
    Formula:C25H31N3O2S
    Purity:99.12% - 99.69%
    Color and Shape:Solid
    Molecular weight:437.6
  • VU6001376

    CAS:
    <p>VU6001376 is an effective and selective positive allosteric modulator of the metabotropic glutamate receptor 4 (EC50: 50.1 nM).</p>
    Formula:C18H14F2N6OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:400.41
  • 2-Iodomelatonin

    CAS:
    <p>2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, &gt;5x selective over MT2, used to map melatonin sites in brain/tissues.</p>
    Formula:C13H15IN2O2
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:358.17
  • EMD 56551

    CAS:
    <p>EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.</p>
    Formula:C24H31N3O2
    Purity:95.64% - 99.39%
    Color and Shape:Solid
    Molecular weight:393.522
  • AP521

    CAS:
    <p>AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).</p>
    Formula:C20H19ClN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.89
  • Dizocilpine

    CAS:
    <p>MK-801 (Dizocilpine (MK-801)) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.</p>
    Formula:C16H15N
    Purity:99.85% - 99.97%
    Color and Shape:Solid
    Molecular weight:221.3
  • Tarafenacin D-tartrate

    CAS:
    Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.
    Formula:C25H26F4N2O8
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:558.48
  • Pridefine

    CAS:
    <p>Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.</p>
    Formula:C19H21N
    Purity:99.15% - 99.66%
    Color and Shape:Solid
    Molecular weight:263.38
  • Donitriptan

    CAS:
    <p>Donitriptan 是一种 5-HT 受体激动剂,对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。</p>
    Formula:C23H25N5O2
    Purity:98.76%
    Color and Shape:Solid
    Molecular weight:403.48
  • F13714 fumarate

    CAS:
    <p>F13714 fumarate is a 5-HT1A receptor-biased agonist.</p>
    Formula:C25H29ClF2N4O5
    Purity:98.86%
    Color and Shape:Solid
    Molecular weight:538.97
  • ASP2535

    CAS:
    <p>ASP2535 is a potent, selective, orally bioavailable, brain permeable and centrally-active glycine transporter-1 (GlyT1) inhibitor.ASP2535 can improve cognitive</p>
    Formula:C22H18N6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:382.42
  • Glemanserin

    CAS:
    <p>Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.</p>
    Formula:C20H25NO
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:295.42
  • Aβ42-IN-2

    CAS:
    <p>Aβ42-IN-2 is a γ-secretase modulator. Aβ42-IN-2 has an IC 50 of 6.5 nM for Αβ 42. Aβ42-IN-2 can be used for the Alzheimer's disease research[1].</p>
    Formula:C24H26N6O2
    Purity:98.09% - 99.87%
    Color and Shape:Solid
    Molecular weight:430.5
  • JNJ-55308942

    CAS:
    <p>JNJ-55308942: selective, brain-penetrant P2X7 antagonist; IC50s: 10nM (human), 15nM (rat); Kis: 7.1nM (h), 2.9nM (r).</p>
    Formula:C17H12F5N7O
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:425.32
  • SCH 50911

    CAS:
    <p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>
    Formula:C8H15NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:173.21
  • MAO-B-IN-22

    CAS:
    <p>MAO-B-IN-22 (compound 6h) represents a powerful MAO-B inhibitor, boasting an IC50 value of 0.014 μM, and exhibits high antioxidant activity alongside effective</p>
    Formula:C20H18FNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:323.36
  • E2730

    CAS:
    <p>E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.</p>
    Formula:C9H8F4N2O2S
    Purity:98.22% - 98.54%
    Color and Shape:Solid
    Molecular weight:284.23
  • PD-102807

    CAS:
    <p>PD-102807 is a selective and competitive M4 muscarinic receptor antagonist for Parkinson's disease research, inhibit airway smooth muscle (ASM) contraction.</p>
    Formula:C23H24N2O4
    Purity:98.90%
    Color and Shape:Solid
    Molecular weight:392.45
  • Amitifadine hydrochloride

    CAS:
    <p>Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).</p>
    Formula:C11H12Cl3N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:264.58
  • Nexopamil racemate

    CAS:
    <p>Nexopamil racemate((Rac)-Nexopamil) is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.</p>
    Formula:C24H40N2O3
    Purity:98.61%
    Color and Shape:Solid
    Molecular weight:404.59
  • Alniditan

    CAS:
    <p>Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.</p>
    Formula:C17H26N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.41
  • PNU-96391

    CAS:
    <p>PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.</p>
    Formula:C15H23NO2S
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:281.41
  • PNU-142633

    CAS:
    <p>PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; &gt;18,000 nM for 5-HT1B.</p>
    Formula:C24H30N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:422.52
  • Glutaminyl Cyclase Inhibitor 5


    <p>Glutaminyl Cyclase Inhibitor 5 is a potent, selective inhibitor of human glutaminyl cyclase (hQC), demonstrating an inhibition concentration half-max (IC 50) of</p>
    Formula:C22H30N6O
    Color and Shape:Solid
    Molecular weight:394.51
  • AS19

    CAS:
    <p>AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).</p>
    Formula:C18H25N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:283.41
  • YM-58790

    CAS:
    <p>YM-58790 is a potent mAChR blocker with Ki values of 28 nM (M1), 260 nM (M2), 15 nM (M3), and reduces bladder contractions in rats.</p>
    Formula:C27H31N3O2
    Purity:98.59%
    Color and Shape:Soild
    Molecular weight:429.55
  • Asoxime dichloride

    CAS:
    <p>Asoxime dichloride (HI-6) blocks AChRs, including α7 nAChR, and boosts vaccination in the nervous system.</p>
    Formula:C14H16Cl2N4O3
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:359.21
  • Glutaminyl Cyclase Inhibitor 2

    CAS:
    <p>Glutaminyl Cyclase Inhibitor 2 is a glutaminyl cyclase inhibitor (IC50: 1.23 μM).</p>
    Formula:C19H20FN3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:309.38
  • mAChr-in-1

    CAS:
    <p>mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).</p>
    Formula:C23H25IN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:488.36
  • S(-)-8-Hydroxy-DPAT hydrobromide

    CAS:
    <p>S(-)-8-Hydroxy-DPAT hydrobromide is an agonist of 5-HT1A serotonin receptor.</p>
    Formula:C16H26BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.29
  • GW-876167

    CAS:
    <p>GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.</p>
    Formula:C16H21N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.37
  • JN403

    CAS:
    <p>JN403 is a selective agonist of nicotinic acetylcholine receptor alpha7.</p>
    Formula:C16H21FN2O2
    Color and Shape:Solid
    Molecular weight:292.35
  • (S)-3-Carboxy-4-hydroxyphenylglycine

    CAS:
    <p>group I metabotropic glutamate receptor antagonist and group II mGlu agonist</p>
    Formula:C9H9NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:211.17
  • AL-37350A

    CAS:
    <p>AL-37350A is a 5-HT2 receptor-selective agonist with ocular hypotensive activity.</p>
    Formula:C14H18N2O
    Color and Shape:Solid
    Molecular weight:230.31
  • DBO-83

    CAS:
    <p>DBO-83, an agonist of nicotinic acetylcholine receptors (nAChRs), has anti-amnesic and antinociceptive activities.</p>
    Formula:C10H15Cl3N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.61
  • Aganodine

    CAS:
    <p>Aganodine, a guanidine, activates imidazoline receptors to inhibit norepinephrine release.</p>
    Formula:C9H10Cl2N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:245.11
  • Pridinol

    CAS:
    Pridinol is an antispasmodic and muscle relaxant.
    Formula:C20H25NO
    Purity:98%
    Color and Shape:Crystals Solid
    Molecular weight:295.42
  • NPS ALX Compound 4a dihydrochloride

    CAS:
    <p>NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>
    Formula:C25H27Cl2N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:504.47
  • RS 45041-190 hydrochloride

    CAS:
    <p>Highly selective I2 imidazoline receptor ligand</p>
    Formula:C11H13Cl2N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:258.15
  • Hyoscyamine hydrobromide

    CAS:
    <p>Hyoscyamine hydrobromide is an agent of anticholinergic.</p>
    Formula:C17H24BrNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.28
  • Epibatidine 2HCl

    CAS:
    <p>Epibatidine 2HCl is a potent nicotinic agonist.</p>
    Formula:C11H15Cl3N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:281.61
  • CPP-115

    CAS:
    <p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>
    Formula:C7H9F2NO2
    Color and Shape:Solid
    Molecular weight:177.15
  • Btm 1042

    CAS:
    <p>Btm 1042 is an antispasmodic drug. It has been found to depress twitch responses in the ileum of guinea pigs.</p>
    Formula:C21H26ClN3OS
    Color and Shape:Solid
    Molecular weight:403.97
  • SDZ 205-557 hydrochloride

    CAS:
    <p>5-HT3/5-HT4 receptor antagonist</p>
    Formula:C14H22Cl2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:337.24
  • ML 10375

    CAS:
    <p>ML 10375 is an antagonist of 5-HT4 receptor.</p>
    Formula:C17H25ClN2O3
    Color and Shape:Solid
    Molecular weight:340.85
  • U 90042

    CAS:
    <p>GABAA receptor ligand</p>
    Formula:C17H13ClN6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.78
  • KW-6055

    CAS:
    <p>KW-6055 has anti-amnesic activity, is a benzylpyridine derivative.</p>
    Formula:C16H17N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.32
  • AZ4800

    CAS:
    <p>AZD4800 is a gamma secretase modulators.</p>
    Formula:C24H29N5O3
    Color and Shape:Solid
    Molecular weight:435.52
  • Astrophloxine

    CAS:
    <p>Astrophloxine is a fluorescent imaging probe that targets antiparallel dimers.Astrophloxine can be used to detect aggregated Aβ in brain tissue and</p>
    Formula:C27H33IN2
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:512.47
  • Mirisetron

    CAS:
    <p>Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.</p>
    Formula:C24H31N3O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:393.52
  • Nitroflurbiprofen

    CAS:
    <p>Nitroflurbiprofen (Nitroxybutyl flurbiprofen) is a NO-releasing COX inhibitor and modulates the increased intrahepatic vascular tone in portal hypertensive</p>
    Formula:C19H20FNO5
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:361.36
  • S 14506 hydrochloride

    CAS:
    <p>S 14506 hydrochloride is a 5-HT1A receptor full agonist.</p>
    Formula:C24H27ClFN3O2
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:443.94
  • SC58451

    CAS:
    <p>SC58451 is a novel potent, orally active and selective COX-2 inhibitor.SC58451 showed anti-inflammatory activity in a rat model of arthritis.</p>
    Formula:C20H19FO2S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:342.43
  • (+)-Nipecotic acid

    CAS:
    <p>(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.</p>
    Formula:C6H11NO2
    Purity:99.38%
    Color and Shape:Solid
    Molecular weight:129.16
  • CP94253 hydrochloride

    CAS:
    <p>CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).</p>
    Formula:C15H20ClN3O
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:293.79
  • SSAO inhibitor-3

    CAS:
    <p>SSAO inhibitor-3 targets human AOC1/SSAO in atherosclerosis, diabetes, obesity, CKD, and more, with IC50s of 0.1-10 μM/&lt;10 nM.</p>
    Formula:C15H23FN4O3
    Color and Shape:Solid
    Molecular weight:326.37
  • BChE-IN-9

    CAS:
    <p>BChE-IN-9 (Azepano-11-deoxo-glycyrrhetol) is a hybrid BChE inhibitor (Ki: 0.21 μM).</p>
    Formula:C30H51NO
    Color and Shape:Solid
    Molecular weight:441.73
  • RLH 033

    CAS:
    <p>RLH 033 is a selective ligand for the sigma 1 recognition site.</p>
    Formula:C25H31ClN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:458.98
  • SGC-AAK1-1N

    CAS:
    <p>SGC-AAK1-1N is a potent and selective inhibitor of AAK1 (AP2 associated kinase 1) with an IC 50 of 1.8 μM [1].</p>
    Formula:C20H22N4O3S
    Color and Shape:Solid
    Molecular weight:398.48
  • 2-PAT

    CAS:
    <p>2-PAT: reversible MAO-A inhib., IC50=0.721 µM; MAO-B inactivator, IC50=14.6 µM; potential in Parkinson's/depression study.</p>
    Formula:C13H15N
    Color and Shape:Solid
    Molecular weight:185.26
  • VU6001966

    CAS:
    <p>VU6001966: potent, selective mGlu2 inhibitor (IC50=78 nM), negative modulator, with good CNS penetration.</p>
    Formula:C17H15FN4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:326.33
  • Aβ Fibrillization modulator 1

    CAS:
    <p>Aβ Fibrillization Modulator 1 stabilizes amyloid-beta (Aβ) monomers, preventing their aggregation into fibrils.</p>
    Formula:C17H12N4O3SSe
    Color and Shape:Solid
    Molecular weight:431.33
  • BMS-911172

    CAS:
    <p>BMS-911172 is an adaptor associated kinase 1 (AAK1 kinase) inhibitor with an IC 50 of 35 nM.</p>
    Formula:C16H19F2N3O3
    Color and Shape:Solid
    Molecular weight:339.34
  • Prucalopride hydrochloride

    CAS:
    <p>Prucalopride hydrochloride is a selective agonist of the 5-HT4.</p>
    Formula:C18H27Cl2N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:404.33
  • TC-2153

    CAS:
    <p>TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.</p>
    Formula:C7H5ClF3NS5
    Color and Shape:Solid
    Molecular weight:355.89
  • Pimprinine

    CAS:
    <p>Pimprinine: an alkaloid, inhibits MAO, and has anticonvulsant properties.</p>
    Formula:C12H10N2O
    Color and Shape:Solid
    Molecular weight:198.22
  • AChE-IN-9


    <p>AChE-IN-9: Tacrine-β-glucose glycoconjugate; IC50 0.4μM; reduced hepatotoxicity; Alzheimer's research.</p>
    Formula:C30H35N5O9
    Color and Shape:Solid
    Molecular weight:609.63
  • ACDPP hydrochloride

    CAS:
    <p>mGlu5 receptor antagonist</p>
    Formula:C12H13ClN6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:292.72
  • NNC052090

    CAS:
    <p>NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).</p>
    Formula:C27H30N2O2
    Color and Shape:Solid
    Molecular weight:414.54
  • AChE/BChE-IN-5

    CAS:
    <p>AChE/BChE-IN-5 (BMC-16) crosses BBB; IC50: hAChE 266 nM, hBChE 10.6 nM. Dual AChE/BChE inhibitor.</p>
    Formula:C17H26N2O3
    Color and Shape:Solid
    Molecular weight:306.4
  • DREADD agonist 21 dihydrochloride

    CAS:
    <p>DREADD agonist 21 dihydrochloride is a potent human muscarinic acetylcholine M3 receptors ( hM3Dq ) agonist with EC 50 of 1.7 nM [1].</p>
    Formula:C17H20Cl2N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.27
  • Alvameline maleate

    CAS:
    <p>Alvameline maleate is used as a Partial M1 Agonist and M2/M3 Antagonist.</p>
    Formula:C13H19N5O4
    Color and Shape:Solid
    Molecular weight:309.32
  • BACE1-IN-12

    CAS:
    <p>BACE1-IN-12: potent BACE1 and BuChE inhibitor, IC50s - 8.9 μM and 3.2 μM, blood-brain barrier permeable, anti-Alzheimer's potential.</p>
    Formula:C29H28Cl2N6O
    Color and Shape:Solid
    Molecular weight:547.48
  • ST1936

    CAS:
    <p>ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.</p>
    Formula:C13H17ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:236.74
  • Befloxatone

    CAS:
    <p>Befloxatone is a potent, selective and reversible inhibitor of monoamine oxidase A.</p>
    Formula:C15H18F3NO5
    Color and Shape:Solid
    Molecular weight:349.3
  • SD-6

    CAS:
    <p>SD-6, oral hAChE/hBChE inhibitor (IC50: 0.907/1.579 µM), crosses BBB, non-toxic, for Alzheimer's research.</p>
    Formula:C20H22N4OS
    Color and Shape:Solid
    Molecular weight:366.48
  • AChE/BChE/MAO-B-IN-4


    <p>AChE/BChE/MAO-B-IN-4 inhibits MAO-B (IC50: 0.0393 µM), AChE (IC50: 0.0458 µM), BChE (IC50: 0.075 µM), and fights AD with antioxidant action.</p>
    Formula:C26H33N3O4
    Color and Shape:Solid
    Molecular weight:451.56
  • Ambenonium dichloride

    CAS:
    <p>AChE inhibitor</p>
    Formula:C28H42Cl3N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:573.02
  • RS 23597-190 hydrochloride

    CAS:
    <p>RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.</p>
    Formula:C16H24Cl2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.28
  • AChE/BChE-IN-4

    CAS:
    <p>AChE/BChE-IN-4 (BMC-3) crosses the BBB; IC50: hAChE 792 nM, hBChE 2.2 nM. Dual AChE/BChE inhibitor.</p>
    Formula:C17H26N2O3
    Color and Shape:Solid
    Molecular weight:306.4
  • MRK-623

    CAS:
    <p>MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.</p>
    Formula:C20H17FN4O
    Color and Shape:Solid
    Molecular weight:348.37
  • Eplivanserin hemifumarate

    CAS:
    <p>Eplivanserin is an inverse agonist of 5-HT2A.</p>
    Formula:C23H25FN2O6
    Color and Shape:Solid
    Molecular weight:444.45
  • RJR-2403 oxalate

    CAS:
    <p>RJR-2403 oxalate is a highly selective agonist of α4β2 subtype nicotinic receptor.</p>
    Formula:C14H18N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:278.308
  • Belaperidone

    CAS:
    <p>Belaperidone, an antipsychotic, resembles clozapine, binds D(4) and 5-HT(2A) receptors, minimally extends Q-T without causing arrhythmias.</p>
    Formula:C22H22FN3O2
    Color and Shape:Solid
    Molecular weight:379.43
  • RS 56812 hydrochloride

    CAS:
    <p>5-HT3 partial agonist</p>
    Formula:C18H22ClN3O2
    Purity:98.62%
    Color and Shape:Solid
    Molecular weight:347.84
  • A-794282

    CAS:
    <p>A-794282 is a selective antagonist of mGluR1.</p>
    Formula:C19H18N4OS
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:350.44
  • Lenumlostat

    CAS:
    <p>Lenumlostat is a lysyl oxidase-like protein 2 (LOXL2) inhibitor with inhibitory effects on hLOXL2, hLOXL3 and LOXL2 for the study of fibrotic diseases.</p>
    Formula:C18H17F4N3O3
    Purity:99.11%
    Color and Shape:Solid
    Molecular weight:399.34
  • Mibampator

    CAS:
    <p>Mibampator (LY451395) is an effective and selective AMPA receptor potentiator.</p>
    Formula:C21H30N2O4S2
    Purity:99.34%
    Color and Shape:Solid
    Molecular weight:438.6
  • Ru-32514

    CAS:
    Ru-32514 is a benzodiazepine receptor agonist.
    Formula:C18H17N3O2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:307.35
  • LY266097 hydrochloride

    CAS:
    <p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>
    Formula:C21H24Cl2N2O2
    Purity:98.58%
    Color and Shape:Solid
    Molecular weight:407.33
  • Eltenac

    CAS:
    <p>Eltenac, a cyclooxygenase (COX) inhibitor, is used potentially for the treatment of pain.</p>
    Formula:C12H9Cl2NO2S
    Purity:98.53%
    Color and Shape:Solid
    Molecular weight:302.18
  • LSN2463359

    CAS:
    <p>LSN2463359 is a positive allosteric modulators of the mGlu5 receptor.</p>
    Formula:C16H15N3O
    Purity:99.26%
    Color and Shape:Solid
    Molecular weight:265.31
  • ADR-851 free base

    CAS:
    ADR-851 free base is an antagonist of the HT3 receptor.
    Formula:C14H18ClN3O2
    Purity:97.88% - 98.39%
    Color and Shape:Solid
    Molecular weight:295.77
  • Gavestinel sodium

    CAS:
    <p>Gavestinel (GV 150526): potent, selective oral NMDA antagonist; binds glycine site, pKi 8.5; studied for acute ischemic stroke.</p>
    Formula:C18H11Cl2N2NaO3
    Purity:99.04%
    Color and Shape:Solid
    Molecular weight:397.19
  • Landipirdine

    CAS:
    <p>Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.</p>
    Formula:C18H19FN2O3S
    Purity:97.61% - 99.37%
    Color and Shape:Solid
    Molecular weight:362.42
  • Dipraglurant

    CAS:
    <p>Dipraglurant: a blood-brain permeable mGluR5 NAM, orally active, selective, IC50 = 21 nM, treats PD-LID.</p>
    Formula:C16H12FN3
    Purity:98.7%
    Color and Shape:Solid
    Molecular weight:265.29
  • LRRK2-IN-7

    CAS:
    <p>LRRK2-IN-7: potent, selective CNS-active LRRK2 inhibitor, IC50 0.9 nM, &gt;1000x selectivity vs kinases/channels/CYPs.</p>
    Formula:C24H26N6O
    Purity:99.26%
    Color and Shape:Solid
    Molecular weight:414.5
  • RS 67333 hydrochloride

    CAS:
    <p>RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.</p>
    Formula:C19H30Cl2N2O2
    Purity:98.78%
    Color and Shape:Solid
    Molecular weight:389.36
  • W-9 hydrochloride

    CAS:
    <p>W-9 hydrochloride is a calmodulin antagonist.</p>
    Formula:C16H22Cl2N2O2S
    Purity:98.9%
    Color and Shape:Solid
    Molecular weight:377.33
  • Riluzole hydrochloride

    CAS:
    <p>Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).</p>
    Formula:C8H6ClF3N2OS
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:270.66
  • MK-3328

    CAS:
    <p>MK-3328, a potential Alzheimer's drug, binds β-Amyloid with strong affinity (IC50:10.5 nM) and may serve as a PET ligand to gauge plaque load.</p>
    Formula:C14H9FN4O
    Purity:99.70% - >99.99%
    Color and Shape:Solid
    Molecular weight:268.25
  • LY-2300559

    CAS:
    <p>LY-2300559 is an agonist of metabotropic glutamate receptor 2 (mGluR2) and can be used in studies about the treatment of migraine.</p>
    Formula:C26H26O6
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:434.48
  • (E/Z)-SIB-1893

    CAS:
    <p>(E/Z)-SIB-1893 (SIB 1893) is the racemate of (E)-SIB-1893 and (Z)-SIB-1893.</p>
    Formula:C14H13N
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:195.26
  • Liafensine

    CAS:
    Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.
    Formula:C24H22N4
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:366.46
  • JNJ-54175446

    CAS:
    <p>JNJ-54175446 (JNJ-5446) is a P2X7 receptor antagonist that attenuates the release of IL-1β/IL-18 from microglia and is used in the study of depression.</p>
    Formula:C18H13ClF4N6O
    Purity:97.98% - 99.79%
    Color and Shape:Solid
    Molecular weight:440.78
  • SPD-473 citrate

    CAS:
    <p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>
    Formula:C23H31Cl2NO8S
    Purity:99.37%
    Color and Shape:Solid
    Molecular weight:552.47
  • Nexopamil

    CAS:
    <p>Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.</p>
    Formula:C24H40N2O3
    Purity:97.87% - >99.99%
    Color and Shape:Solid
    Molecular weight:404.59
  • Cyamemazine

    CAS:
    Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.
    Formula:C19H21N3S
    Purity:97.01%
    Color and Shape:Solid
    Molecular weight:323.46
  • DSP-0565

    CAS:
    <p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>
    Formula:C14H12FNO
    Purity:99.51% - 99.56%
    Color and Shape:Solid
    Molecular weight:229.25
  • Buntanetap

    CAS:
    Buntanetap ((+)-Phenserine) is an inhibitor of TINAPs used in the study of neurological disorders, endocrine and metabolic disorders, and cardiovascular disease
    Formula:C20H23N3O2
    Purity:98.2%
    Color and Shape:Solid
    Molecular weight:337.42
  • Aceclidine

    CAS:
    <p>Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies about treating glaucoma by reducing intraocular</p>
    Formula:C9H15NO2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:169.22
  • Sarizotan HCl

    CAS:
    <p>Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.</p>
    Formula:C22H22ClFN2O
    Purity:96%
    Color and Shape:Solid
    Molecular weight:384.87
  • ML 10302 hydrochloride

    CAS:
    ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.
    Formula:C15H22Cl2N2O3
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:349.25
  • DSS30

    CAS:
    <p>DSS30 is a P25/CDK5 inhibitor that reduces β-amyloid secretion to help prevent Alzheimer's.</p>
    Formula:C16H14ClNO3S2
    Purity:99.19% - 99.4%
    Color and Shape:Solid
    Molecular weight:367.87
  • Suriclone

    CAS:
    <p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>
    Formula:C20H20ClN5O3S2
    Purity:99.21% - 99.73%
    Color and Shape:Solid
    Molecular weight:477.99
  • GR 46611

    CAS:
    GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.
    Formula:C23H27N3O2
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:377.48
  • Sudoxicam

    CAS:
    <p>Sudoxicam (4-Hydroxy-2-methyl-N-2-thiazolyl-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide) is a reversible antagonist of COX with anti-inflammatory, anti-edema</p>
    Formula:C13H11N3O4S2
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:337.37
  • Lirequinil

    CAS:
    <p>Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.</p>
    Formula:C26H25ClN2O3
    Purity:98.54%
    Color and Shape:Solid
    Molecular weight:448.94
  • DMCM hydrochloride

    CAS:
    <p>DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.</p>
    Formula:C17H19ClN2O4
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:350.8
  • Otenzepad

    CAS:
    Otenzepad (AF-DX 116) is a selective antagonist of M2 mAChR with IC50s of 386 nM and 640 nM for rat heart and rabbit peripheral lung.
    Formula:C24H31N5O2
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:421.54
  • CP-810123

    CAS:
    <p>CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or neurological disorders such as schizophrenia.</p>
    Formula:C14H18N4O
    Purity:98.63% - 99.60%
    Color and Shape:Solid
    Molecular weight:258.32
  • Adoprazine

    CAS:
    <p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>
    Formula:C24H24FN3O2
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:405.46
  • Lecozotan HCl

    CAS:
    <p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>
    Formula:C28H30ClN5O3
    Purity:99.04%
    Color and Shape:Solid
    Molecular weight:520.02
  • 5-HT2 antagonist 1

    CAS:
    <p>5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.</p>
    Formula:C22H29FN4O2
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:400.49
  • PHA 543613

    CAS:
    <p>PHA 543613 is a specific agonist of α7 nAChR (Ki = 8.8 nM) and can be used in studies about the cognitive deficits of Alzheimer's disease and schizophrenia.</p>
    Formula:C15H17N3O2
    Purity:99.43% - 99.96%
    Color and Shape:Solid
    Molecular weight:271.31
  • Ecopipam

    CAS:
    <p>Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.</p>
    Formula:C19H20ClNO
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:313.82
  • Aβ-IN-1

    CAS:
    <p>Aβ-IN-1 is a novel, potent and orally active γ-secretase modulator (GSM).</p>
    Formula:C35H49N
    Purity:99.1%
    Color and Shape:Soild
    Molecular weight:483.77
  • CP 96021

    CAS:
    <p>"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."</p>
    Formula:C29H21FN4OS
    Purity:97.81% - 99.62%
    Color and Shape:Soild
    Molecular weight:492.57
  • AZD6538

    CAS:
    <p>AZD6538 is an mGluR5 negative allosteric modulator used in the study of CNS-related diseases such as Alzheimer's disease.</p>
    Formula:C15H6FN5O
    Purity:98.68%
    Color and Shape:Solid
    Molecular weight:291.24
  • PPI-1019

    CAS:
    <p>PPI-1019 is an APP (β-amyloid A4) inhibitor for the treatment of neurological disorders and the study of Alzheimer's disease (AD).</p>
    Formula:C36H54N6O5
    Purity:95.16% - 98.16%
    Color and Shape:Solid
    Molecular weight:650.85
  • MNI 137

    CAS:
    <p>MNI 137 is a negative allosteric modulator of mGlu2. MNI 137 inhibits glutamate-induced calcium mobilization with IC50s of 8.3 and 12.6 nM for human and rat.</p>
    Formula:C15H9BrN4O
    Purity:97.49%
    Color and Shape:Solid
    Molecular weight:341.16
  • Fengabine

    CAS:
    <p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>
    Formula:C17H17Cl2NO
    Purity:99%
    Color and Shape:Solid
    Molecular weight:322.23
  • Ensaculin

    CAS:
    <p>Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.</p>
    Formula:C26H32N2O5
    Purity:99.17% - 99.67%
    Color and Shape:Solid
    Molecular weight:452.54
  • cis-Urocanic acid

    CAS:
    <p>cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).</p>
    Formula:C6H6N2O2
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:138.12
  • Ricasetron

    CAS:
    <p>Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.</p>
    Formula:C19H27N3O
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:313.44
  • Tedatioxetine

    CAS:
    <p>Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.</p>
    Formula:C18H21NS
    Purity:99.76% - >99.99%
    Color and Shape:Solid
    Molecular weight:283.43
  • Xanomeline

    CAS:
    <p>Xanomeline: orally active, M1/M4 selective activator for neurological disorders; promising in trials, crosses blood-brain barrier, liver metabolized.</p>
    Formula:C14H23N3OS
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:281.42
  • AQW051

    CAS:
    <p>AQW051 (VQW-765) is an oral α7-nAChR activator for cognitive impairments, used in anxiety disorder studies.</p>
    Formula:C19H22N2O
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:294.39
  • Itasetron

    CAS:
    <p>Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.</p>
    Formula:C16H20N4O2
    Purity:98.58% - 99.33%
    Color and Shape:Solid
    Molecular weight:300.36
  • ELB-139

    CAS:
    <p>ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.</p>
    Formula:C14H16ClN3O
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:277.75
  • BL-1020 Mesylate

    CAS:
    <p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>
    Formula:C28H45ClN4O11S4
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:777.39
  • Progabide

    CAS:
    <p>Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.</p>
    Formula:C17H16ClFN2O2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:334.77
  • Muscimol HBr

    CAS:
    Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.
    Formula:C4H7BrN2O2
    Purity:98.13%
    Color and Shape:Off-White Powder
    Molecular weight:195.01
  • Viloxazine

    CAS:
    <p>Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activity</p>
    Formula:C13H19NO3
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:237.29
  • (Z)-Thiothixene

    CAS:
    <p>(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.</p>
    Formula:C23H29N3O2S2
    Purity:99.21%
    Color and Shape:Yellow To Yellow With A Tan Cast Powder
    Molecular weight:443.63
  • Divaplon

    CAS:
    <p>Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.</p>
    Formula:C17H17N3O2
    Purity:97.44% - 98.25%
    Color and Shape:Solid
    Molecular weight:295.34
  • 2-BFI hydrochloride

    CAS:
    2-BFI hydrochloride: High-affinity I2 agonist; used in researching stroke and immune disease protection.
    Formula:C11H11ClN2O
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:222.67
  • Repinotan

    CAS:
    <p>Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.</p>
    Formula:C21H24N2O4S
    Purity:99%
    Color and Shape:Solid
    Molecular weight:400.49
  • NB001

    CAS:
    <p>NB001 (HTS 09836) is an inhibitor of adenyl cyclase 1 exhibiting effects on neural and non-neural pain.</p>
    Formula:C12H20N6O
    Purity:99.69%
    Color and Shape:Off-White To Pale Pink Solid
    Molecular weight:264.33
  • Faxeladol

    CAS:
    <p>Faxeladol: adrenergic, serotonin inhibitor &amp; opioid agonist for neurological studies.</p>
    Formula:C15H23NO
    Purity:98.09% - 98.77%
    Color and Shape:Solid
    Molecular weight:233.35
  • Alpidem

    CAS:
    <p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>
    Formula:C21H23Cl2N3O
    Purity:99.56% - 99.97%
    Color and Shape:White To Off-White Solid
    Molecular weight:404.33
  • Teniloxazine

    CAS:
    Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.
    Formula:C16H19NO2S
    Purity:99.29%
    Color and Shape:Solid
    Molecular weight:289.39
  • Fananserin

    CAS:
    <p>Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).</p>
    Formula:C23H24FN3O2S
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:425.52
  • AZD 9272

    CAS:
    <p>AZD 9272 is a brain-permeable mGluR5 antagonist for the study of gastroesophageal reflux.</p>
    Formula:C14H6F2N4O
    Purity:98.29%
    Color and Shape:Solid
    Molecular weight:284.22
  • Cirsimaritin

    CAS:
    <p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>
    Formula:C17H14O6
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:314.29
  • CBiPES hydrochloride

    CAS:
    CBiPES hydrochloride (CBiPES HCl) is an orthosteric modulator of the mGlu2 receptor and is used to study neurological disorders like epilepsy.
    Formula:C21H20ClN3O2S
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:413.92
  • Panadiplon

    CAS:
    <p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>
    Formula:C18H17N5O2
    Purity:98.30% - 98.94%
    Color and Shape:Solid
    Molecular weight:335.36
  • VU 0285683

    CAS:
    VU 0285683 is a specific negative allosteric modulator of mGluR5 with a high affinity for the MPEP binding site. VU 0285683 shows anxiolytic-like activity.
    Formula:C14H7FN4O
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:266.23
  • ATC 0175 hydrochloride

    CAS:
    <p>ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.</p>
    Formula:C23H26ClF2N5O
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:461.93
  • Tribendimidine

    CAS:
    <p>Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.</p>
    Formula:C28H32N6
    Purity:≥98%
    Color and Shape:Solid
    Molecular weight:452.59
  • Piromelatine

    CAS:
    <p>Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity with</p>
    Formula:C17H16N2O4
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:312.32
  • Cianopramine

    CAS:
    <p>Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.</p>
    Formula:C20H23N3
    Purity:99.92% - 99.92%
    Color and Shape:Solid
    Molecular weight:305.42
  • Oxotremorine M iodide

    CAS:
    <p>Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.</p>
    Formula:C11H19IN2O
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:322.19
  • L-838417

    CAS:
    <p>L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disorders</p>
    Formula:C19H19F2N7O
    Purity:98.12% - 99.70%
    Color and Shape:Solid
    Molecular weight:399.4
  • Cilansetron

    CAS:
    Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.
    Formula:C20H21N3O
    Purity:99.82% - 99.98%
    Color and Shape:Solid
    Molecular weight:319.4
  • Ticalopride

    CAS:
    <p>Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.</p>
    Formula:C14H20ClN3O3
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:313.78
  • Roxindole

    CAS:
    Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.
    Formula:C23H26N2O
    Purity:98.03% - 98.93%
    Color and Shape:Solid
    Molecular weight:346.47
  • Masupirdine free base

    CAS:
    <p>Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.</p>
    Formula:C21H24BrN3O3S
    Purity:98.36% - 99.65%
    Color and Shape:Solid
    Molecular weight:478.4
  • Aplindore Fumarate

    CAS:
    Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.
    Formula:C22H22N2O7
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:426.42
  • Litoxetine

    CAS:
    <p>Litoxetine: a selective 5-HT inhibitor &amp; 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.</p>
    Formula:C16H19NO
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:241.33
  • TAK-137

    CAS:
    <p>TAK-137 is an AMPA receptor enhancer with antidepressant effects. TAK-137 has the ability to improve cognition and could be used to study schizophrenia.</p>
    Formula:C19H16N2O3S
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:352.41
  • McN-A 343

    CAS:
    <p>McN-A 343: Selective M1 muscarinic agonist; reduces inflammation in colitis models.</p>
    Formula:C14H18Cl2N2O2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:317.21
  • E6801

    CAS:
    <p>E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.</p>
    Formula:C17H18ClN5O2S2
    Purity:96.32% - 99.53%
    Color and Shape:Solid
    Molecular weight:423.94
  • Rilapine

    CAS:
    <p>Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.</p>
    Formula:C22H20ClN3
    Purity:97.76% - 99.20%
    Color and Shape:Solid
    Molecular weight:361.87
  • amyloid P-IN-1

    CAS:
    <p>amyloid P-IN-1 can be used in studies about diseases with depletion of serum amyloid P components such as Alzheimer's disease, amyloidosis, osteoarthritis, and</p>
    Formula:C30H44N2O14
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:656.68
  • ASM-024

    CAS:
    <p>ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment with anti-inflammatory effects.</p>
    Formula:C15H25N2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:233.37
  • Desformylflustrabromine hydrochloride

    CAS:
    <p>Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 neurons, with pEC50 of 6.</p>
    Formula:C17H12INO5
    Purity:98.12%
    Color and Shape:Solid
    Molecular weight:437.19
  • Anpirtoline hydrochloride

    CAS:
    <p>Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.</p>
    Formula:C10H14Cl2N2S
    Purity:>99.99% - >99.99%
    Color and Shape:Solid
    Molecular weight:265.20
  • Saripidem

    CAS:
    <p>Saripidem (SL-85.0274) is a compound with anxiolytic activity.</p>
    Formula:C19H20ClN3O
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:341.83
  • SCH-900271

    CAS:
    <p>SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.</p>
    Formula:C14H16N2O4
    Purity:98.82% - 99.93%
    Color and Shape:Solid
    Molecular weight:276.29
  • Xanomeline oxalate

    CAS:
    <p>Xanomeline oxalate (LY246708), a potent SMRA, boosts phosphoinositide hydrolysis; key for Alzheimer's research.</p>
    Formula:C16H25N3O5S
    Purity:99.1%
    Color and Shape:Solid
    Molecular weight:371.45
  • LM-1685

    CAS:
    <p>LM-1685是一种有效且具有选择性的人单核细胞和全血中COX-2抑制剂,IC50分别为0.65 µM 和IC50 = 4.3 μM,是治疗炎症的潜在化合物。</p>
    Formula:C18H16ClNO4S
    Purity:98.16%
    Color and Shape:Solid
    Molecular weight:377.84
  • Selurampanel

    CAS:
    <p>Selurampanel (BGG492), an oral AMPA antagonist for epilepsy, migraine, and tinnitus studies.</p>
    Formula:C16H19N5O4S
    Purity:99.60% - 99.78%
    Color and Shape:Solid
    Molecular weight:377.42
  • SB 699551 dihydrochloride

    CAS:
    <p>SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.</p>
    Formula:C34H47Cl2N3O
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:584.66
  • CGP 37849

    CAS:
    <p>CGP 37849: oral NMDA antagonist (Ki=35 nM), anticonvulsant, with antidepressant/anxiolytic effects.</p>
    Formula:C6H12NO5P
    Purity:99.87%
    Color and Shape:White Solid
    Molecular weight:209.14
  • Agomelatine hydrochloride

    CAS:
    <p>Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).</p>
    Formula:C15H18ClNO2
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:279.76
  • PAT-1251

    CAS:
    <p>PAT-1251 is an inhibitor of LOXL2 with IC50s of 10, 0.12, and 0.16 μM for the mouse, rat, and dog and can be used in studies about fibrotic diseases.</p>
    Formula:C18H17F4N3O3
    Purity:97.27% - 98.46%
    Color and Shape:Solid
    Molecular weight:399.34
  • Tiospirone

    CAS:
    <p>Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.</p>
    Formula:C24H32N4O2S
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:440.6
  • MAO-B-IN-9

    CAS:
    <p>MAO-B-IN-9 is a monoamine oxidase B MAO-B inhibitor (IC50: 0.18 μM) that crosses the blood-brain barrier with potency, selectivity and time-dependence.</p>
    Formula:C18H24N2O2
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:300.4
  • 5-HT6/7 antagonist 1

    CAS:
    <p>5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.</p>
    Formula:C22H20FN3O3
    Purity:98.78% - 99.26%
    Color and Shape:Solid
    Molecular weight:393.41
  • Quinupramine

    CAS:
    Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.
    Formula:C21H24N2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:304.43
  • PF-03635659

    CAS:
    <p>PF-03635659: potent M3 antagonist, Ki=0.2 nM, long half-life, potential COPD treatment.</p>
    Formula:C28H32N2O3
    Purity:98.39% - 99.83%
    Color and Shape:Solid
    Molecular weight:444.57
  • SB228357

    CAS:
    <p>SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.</p>
    Formula:C22H17F4N3O2
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:431.38