5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
Found 1025 products of "5-HT Receptor"
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Tiprenolol
CAS:Tiprenolol is a beta adrenergic receptor antagonist.[1]Formula:C13H21NO2SPurity:99.43%Color and Shape:SolidMolecular weight:255.38Ref: TM-T50081
1mg52.00€1mL*10mM (DMSO)89.00€5mg98.00€10mg146.00€25mg235.00€50mg319.00€100mg447.00€200mg587.00€Geissoschizine methyl ether
CAS:Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.Formula:C22H26N2O3Purity:99.24% - 99.68%Color and Shape:SolidMolecular weight:366.45Ref: TM-TN1032
1mg130.00€2mg187.00€5mg319.00€1mL*10mM (DMSO)326.00€10mg485.00€25mg770.00€50mg1,035.00€100mg1,395.00€Tandospirone hydrochloride
CAS:Tandospirone (SM-3997) HCl: potent 5-HT1A partial agonist; Ki: 27 nM; anxiolytic, antidepressant, for CNS disorder research.Formula:C21H30ClN5O2Color and Shape:SolidMolecular weight:419.95Vortioxetine
CAS:Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Formula:C18H22N2SPurity:99.34% - 99.34%Color and Shape:SolidMolecular weight:298.45Ref: TM-T2395
1mL*10mM (DMSO)46.00€10mg48.00€25mg65.00€50mg90.00€100mg117.00€200mg203.00€500mg333.00€1g477.00€γ-Mangostin
CAS:Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.Formula:C23H24O6Purity:98.55% - 99.08%Color and Shape:SolidMolecular weight:396.43Xanthotoxol
CAS:Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.Formula:C11H6O4Purity:98.44% - 99.97%Color and Shape:SolidMolecular weight:202.16Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Formula:C21H25ClN2O4SPurity:99.04%Color and Shape:SolidMolecular weight:436.95Ansofaxine hydrochloride
CAS:Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formula:C24H32ClNO3Purity:99.57% - 99.77%Color and Shape:SolidMolecular weight:417.97Aripiprazole monohydrate
CAS:Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.Formula:C23H29Cl2N3O3Color and Shape:SolidMolecular weight:466.4MDL 100009
CAS:MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.Formula:C22H28FNO3Purity:98.96%Color and Shape:SolidMolecular weight:373.46Ref: TM-T22359
1mg99.00€5mg187.00€1mL*10mM (DMSO)222.00€10mg280.00€25mg434.00€50mg585.00€100mg775.00€200mg1,054.00€SB399885
CAS:SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.Formula:C18H21Cl2N3O4SPurity:98.94%Color and Shape:SolidMolecular weight:446.35Ref: TM-T19669
1mg67.00€5mg123.00€1mL*10mM (DMSO)150.00€10mg177.00€25mg291.00€50mg393.00€100mg553.00€200mg743.00€Relenopride hydrochloride
CAS:Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.Formula:C24H31Cl2FN4O4Color and Shape:SolidMolecular weight:529.43Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formula:C23H30N4O2SPurity:99.23%Color and Shape:White PowderMolecular weight:426.57LY334370
CAS:LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nMFormula:C21H22FN3OPurity:99.32%Color and Shape:SolidMolecular weight:351.42Clozapine HCl
CAS:Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.Formula:C18H20Cl2N4Color and Shape:SolidMolecular weight:363.29Niaprazine
CAS:Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.Formula:C20H25FN4OPurity:99.56%Color and Shape:SolidMolecular weight:356.44Sevoflurane
CAS:Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.Formula:C4H3F7OPurity:98%Color and Shape:Less Oil Colorless OilMolecular weight:200.05Ref: TM-T22425
2mg39.00€5mg54.00€1mL*10mM (DMSO)56.00€10mg75.00€25mg110.00€50mg158.00€100mg226.00€200mg339.00€Piboserod
CAS:Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formula:C22H31N3O2Purity:97.21% - 99.49%Color and Shape:SolidMolecular weight:369.5Ref: TM-T2278
1mg38.00€2mg50.00€5mg84.00€10mg118.00€1mL*10mM (DMSO)120.00€25mg220.00€50mg403.00€100mg582.00€500mg1,198.00€Frovatriptan Succinate
CAS:Frovatriptan Succinate is a synthetic triptan with 5-HT1B/1D receptors agonist activity. It is indicated for the acute treatment of migraine.Formula:C18H25N3O6Color and Shape:SolidMolecular weight:379.41AVN-492
CAS:AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).Formula:C17H21N5O2SPurity:99.81%Color and Shape:SolidMolecular weight:359.45Ref: TM-T5179
1mg37.00€2mg50.00€5mg77.00€1mL*10mM (DMSO)85.00€10mg114.00€25mg225.00€50mg335.00€100mg484.00€Methiothepin mesylate
CAS:Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.Formula:C21H28N2O3S3Purity:98% - 99.92%Color and Shape:SolidMolecular weight:452.65Alprenolol benzoate
CAS:Alprenolol benzoate is the benzoate salt of Alprenolol -- a beta blocker.Formula:C22H29NO4Color and Shape:SolidMolecular weight:371.48lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formula:C31H36FN3O4SPurity:95.83% - 99.95%Color and Shape:SolidMolecular weight:565.7Eltoprazine hydrochloride
CAS:Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formula:C12H17ClN2O2Purity:99.35%Color and Shape:SolidMolecular weight:256.73Naluzotan
CAS:Naluzotan（PRX 00023） is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+Formula:C23H38N4O3SPurity:>99.99%Color and Shape:SolidMolecular weight:450.64Dolasetron
CAS:Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.Formula:C19H20N2O3Purity:99.84% - 99.86%Color and Shape:White PowderMolecular weight:324.37AC-90179 HCl
CAS:AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Formula:C23H31ClN2O2Purity:99.71%Color and Shape:SolidMolecular weight:402.96Escitalopram Oxalate
CAS:Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Formula:C22H23FN2O5Purity:97.39% - 99.73%Color and Shape:White SolidMolecular weight:414.43Ref: TM-T6493
10mg37.00€1mL*10mM (DMSO)42.00€25mg52.00€50mg63.00€100mg86.00€200mg118.00€500mg187.00€1g268.00€Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formula:C27H25F2N3OSPurity:99.77% - 99.89%Color and Shape:SolidMolecular weight:477.57Opiranserin hydrochloride
CAS:Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormula:C21H35ClN2O5Purity:99.33%Color and Shape:SolidMolecular weight:430.97Ref: TM-T9833
1mg90.00€5mg215.00€1mL*10mM (DMSO)236.00€10mg340.00€25mg618.00€50mg879.00€100mg1,224.00€500mg2,457.00€Eltoprazine dihydrochloride
CAS:Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.Formula:C12H18Cl2N2O2Purity:99.64%Color and Shape:SolidMolecular weight:293.19Indophagolin
CAS:Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Formula:C19H15BrClF3N2O3SPurity:99.76%Color and Shape:SolidMolecular weight:523.75Adoprazine hydrochloride
CAS:Adoprazine hydrochloride is a dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.Formula:C24H25ClFN3O2Color and Shape:SolidMolecular weight:441.93Nefazodone hydrochloride
CAS:Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Formula:C25H33Cl2N5O2Purity:99% - 99.86%Color and Shape:White SolidMolecular weight:506.47Ref: TM-T3275
5mg47.00€10mg70.00€1mL*10mM (DMSO)77.00€25mg120.00€50mg216.00€100mg325.00€200mg472.00€500mg775.00€NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = 10.19).Formula:C20H23Cl2F2N3O2Purity:99.59%Color and Shape:SolidMolecular weight:446.32Idalopirdine Hydrochloride
CAS:Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.Formula:C20H20ClF5N2OPurity:99.77%Color and Shape:SolidMolecular weight:434.83Almotriptan Malate
CAS:Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.Formula:C17H25N3O2S·C4H6O5Purity:99.95%Color and Shape:Pale Yellow SolidMolecular weight:469.55Anpirtoline free base
CAS:Anpirtoline: potent 5-HT1B agonist; lowers serotonin synthesis; reduces aggression; 5-HT3 antagonist; crosses blood-brain barrier.Formula:C10H13ClN2SColor and Shape:SolidMolecular weight:228.74Naratriptan
CAS:Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.Formula:C17H25N3O2SPurity:99.08%Color and Shape:SolidMolecular weight:335.47Ref: TM-T8666
1mg39.00€2mg50.00€5mg73.00€1mL*10mM (DMSO)88.00€10mg92.00€25mg166.00€50mg240.00€100mg360.00€SB 204741
CAS:SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.Formula:C14H14N4OSPurity:99.83%Color and Shape:SolidMolecular weight:286.35Ref: TM-T23312
1mg38.00€2mg50.00€5mg84.00€1mL*10mM (DMSO)84.00€10mg119.00€25mg234.00€50mg439.00€100mg600.00€200mg837.00€Serotonin hydrochloride
CAS:Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (Formula:C10H13ClN2OPurity:98.05% - 99.93%Color and Shape:White To Cream PowderMolecular weight:212.676Cerlapirdine hydrochloride
CAS:Cerlapirdine/SAM-531, potent 5-HT6 antagonist, targets Alzheimer's and schizophrenia cognitive issues; phase II trials, promising efficacy, safe profile.Formula:C22H24ClN3O3SColor and Shape:SolidMolecular weight:445.96Cilansetron Hydrochloride
CAS:Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.Formula:C20H24ClN3O2Color and Shape:SolidMolecular weight:373.88Naratriptan hydrochloride
CAS:Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.Formula:C17H25N3O2S·HClPurity:99.17% - 99.93%Color and Shape:Beige SolidMolecular weight:371.93Rizatriptan sulfate
CAS:Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine.Formula:C15H21N5O4SColor and Shape:SolidMolecular weight:367.42Ralmitaront
CAS:Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).Formula:C17H22N4O2Purity:99.71% - 99.79%Color and Shape:SolidMolecular weight:314.38Ref: TM-T9183
1mg105.00€5mg260.00€1mL*10mM (DMSO)286.00€10mg401.00€25mg668.00€50mg897.00€100mg1,243.00€200mg1,693.00€Mosapride Citrate
CAS:Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.Formula:C21H25ClFN3O3·C6H8O7Purity:99.70%Color and Shape:White PowderMolecular weight:614.02Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderateFormula:C21H32Cl2N4OPurity:99.68% - 99.87%Color and Shape:SolidMolecular weight:427.41Ref: TM-T4577
1mg49.00€5mg92.00€1mL*10mM (DMSO)103.00€10mg145.00€25mg281.00€50mg394.00€100mg550.00€200mg780.00€Pipamperone HCl
CAS:Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.Formula:C21H31ClFN3O2Color and Shape:SolidMolecular weight:411.95Intepirdine
CAS:Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.Formula:C19H19N3O2SPurity:98% - 98.63%Color and Shape:SolidMolecular weight:353.44
