Cannabinoid Receptor
Cannabinoid receptors are GPCRs that mediate the effects of endogenous cannabinoids (endocannabinoids) and phytocannabinoids, such as those found in cannabis. The two main types of cannabinoid receptors, CB1 and CB2, are involved in regulating a wide range of physiological processes, including pain perception, appetite, mood, and immune function. Cannabinoid receptor modulators have therapeutic potential in treating conditions such as chronic pain, epilepsy, and multiple sclerosis. At CymitQuimica, we offer a wide range of high-quality cannabinoid receptor modulators to support your research in neuropharmacology, pain management, and immunology.
Found 217 products of "Cannabinoid Receptor"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Δ9-THCH
CAS:Δ9-THCH, a phytocannabinoid analytical reference standard, is present in a Cannabis variety cultivated for medicinal use. In the United States, it is classified as a Schedule I compound. This product is designated for research and forensic applications.Formula:C22H32O2Color and Shape:SolidMolecular weight:328.49CB1-IN-3
CB1-IN-3 (Compound 6i) is a potent inhibitor of the cannabinoid receptor type 1 (CB1). It holds potential for research in obesity, inflammation, and neurological disorders.Color and Shape:Odour SolidCannabidivarinic acid
CAS:Cannabidivarinic acid (CBDVA), the carboxylic acid precursor to cannabidivarin (CBDV), is a non-psychoactive cannabinoid found in Cannabis and known for its anti-inflammatory properties.Formula:C20H26O4Color and Shape:SolidMolecular weight:330.42Taranabant racemate
CAS:Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.Formula:C27H25ClF3N3O2Purity:98%Color and Shape:SolidMolecular weight:515.95Virodhamine
CAS:Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.Formula:C22H37NO2Purity:98%Color and Shape:SoildMolecular weight:347.53WIN 55,212-2 Mesylate
CAS:WIN 55,212-2 Mesylate ((R)-(+)-WIN 55212) is a potent aminoalkylindole cannabinoid (CB) receptor agonist with Kis of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively. Cannabinoid analogue WIN 55,212-2 Mesylate exhibited a novel anticancer effect against human tumors.Formula:C28H30N2O6SPurity:98% - 99.71%Color and Shape:White To Off-White SolidMolecular weight:522.61AM251
CAS:AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).Formula:C22H21Cl2IN4OPurity:97.43% - 98.79%Color and Shape:A Crystalline SolidMolecular weight:555.24Hemopressin (human, mouse) acetate
Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.Formula:C52H83N13O14Purity:99.86%Color and Shape:SolidMolecular weight:1114.29Cannabigerol
CAS:Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFormula:C21H32O2Purity:99.59% - 99.92%Color and Shape:SolidMolecular weight:316.48Ref: TM-TN1465
1mg138.00€2mg203.00€5mg298.00€10mg449.00€25mg765.00€50mg1,054.00€100mg1,423.00€1mL*10mM (DMSO)306.00€PSB-SB-487
CAS:PSB-SB-487 is antagonist of GPR55.Formula:C26H32O4Purity:98.53%Color and Shape:SolidMolecular weight:408.53Ref: TM-T8975
1mg35.00€5mg80.00€10mg119.00€25mg231.00€50mg344.00€100mg480.00€200mg660.00€1mL*10mM (DMSO)87.00€ML-191
CAS:ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.Formula:C24H25N3O3Purity:99.58%Color and Shape:SolidMolecular weight:403.47ML-184
CAS:ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.Formula:C25H34N4O3SPurity:99.45%Color and Shape:SolidMolecular weight:470.63JD-5037
CAS:JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.Formula:C27H27Cl2N5O3SPurity:99.54% - 99.84%Color and Shape:SolidMolecular weight:572.51Ref: TM-T4453
1mg42.00€2mg55.00€5mg90.00€10mg133.00€25mg234.00€50mg350.00€100mg522.00€1mL*10mM (DMSO)101.00€ML-193
CAS:ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.Formula:C28H25N5O4SPurity:97.74%Color and Shape:SolidMolecular weight:527.59Otenabant hydrochloride
CAS:Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).Formula:C25H26Cl3N7OPurity:99.79% - ≥95%Color and Shape:SolidMolecular weight:546.88Olivetol
CAS:Olivetol, found in lichens, is an organic antioxidant and THC synthesis precursor.Formula:C11H16O2Purity:99.98%Color and Shape:(Melting Point 102-106°F) (Ntp 1992)Molecular weight:180.24CB1 antagonist 4
CAS:TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.Formula:C30H25Cl2F3N4OSPurity:98.97%Color and Shape:SolidMolecular weight:617.51Ref: TM-T8511
2mg46.00€5mg92.00€10mg152.00€25mg259.00€50mg405.00€100mg597.00€200mg848.00€1mL*10mM (DMSO)155.00€Bay 59-3074
CAS:Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).
Formula:C18H13F6NO4SPurity:97.68% - 99.69%Color and Shape:SolidMolecular weight:453.36AM1241
CAS:AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.Formula:C22H22IN3O3Purity:98.937% - 99.1%Color and Shape:SolidMolecular weight:503.33Ref: TM-T6755
2mg35.00€5mg49.00€10mg84.00€25mg168.00€50mg275.00€100mg495.00€500mg1,071.00€1mL*10mM (DMSO)87.00€Org 27569
CAS:Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity andFormula:C24H28ClN3OPurity:>99.99% - ≥95%Color and Shape:SolidMolecular weight:409.95A-836339
CAS:A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.Formula:C16H26N2O2SPurity:99.94%Color and Shape:SolidMolecular weight:310.45Ref: TM-T7375
2mg34.00€5mg67.00€10mg109.00€25mg177.00€50mg260.00€100mg369.00€200mg500.00€1mL*10mM (DMSO)63.00€RTICBM-189
CAS:RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.Formula:C15H14Cl2N2OPurity:99.96%Color and Shape:SolidMolecular weight:309.19Ref: TM-T9466
2mg34.00€5mg52.00€10mg84.00€25mg161.00€50mg250.00€100mg369.00€200mg522.00€1mL*10mM (DMSO)67.00€GW842166X
CAS:GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.Formula:C18H17Cl2F3N4O2Purity:99.47%Color and Shape:SolidMolecular weight:449.25β-Caryophyllene
CAS:β-Caryophyllene ((-)-(E)-Caryophyllene) acts as an CB2 receptor agonist.Formula:C15H24Purity:95.43% - 99.11%Color and Shape:Turpentine (Ntp 1992)Molecular weight:204.35RVD-Hpα acetate(1193362-76-3 free base)
RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.Formula:C67H109N19O19Purity:99.87%Color and Shape:SolidMolecular weight:1484.71Hemopressin (rat) acetate(568588-77-2 free base)
Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.Formula:C5H81N13O14Purity:99.37%Color and Shape:SolidMolecular weight:1148.31N-Oleoyl glycine
CAS:N-Oleoyl glycine, a lipoamino acid, was able to promote 3T3-L1 adipogenesis through the activation of CB1 receptor and the enhancement of insulin-mediated AktFormula:C20H37NO3Purity:97.43%Color and Shape:SolidMolecular weight:339.51ARN272
CAS:ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).Formula:C27H20N4O2Purity:98.23%Color and Shape:SolidMolecular weight:432.47Voacamine
CAS:Voacamine: an indole alkaloid, CB1 antagonist, inhibits P-gp, may affect rhythm.
Formula:C43H52N4O5Purity:98.54% - 99.82%Color and Shape:SolidMolecular weight:704.9yangonin
CAS:Yangonin (Y100550) is a novel CB1 receptor ligand with affinity for human recombinant CB1 receptors.Formula:C15H14O4Purity:98.82% - 99.55%Color and Shape:Pale Yellow PowderMolecular weight:258.27Ref: TM-T3S0738
1mg70.00€5mg135.00€10mg207.00€25mg349.00€50mg515.00€100mg735.00€1mL*10mM (DMSO)177.00€(±)-Ibipinabant
CAS:(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Formula:C23H20Cl2N4O2SPurity:99.28% - 99.83%Color and Shape:SolidMolecular weight:487.4GW 405833
CAS:GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFormula:C23H24Cl2N2O3Purity:99.82% - 99.93%Color and Shape:SolidMolecular weight:447.35Linoleoyl Ethanolamide
CAS:Linoleoyl Ethanolamide is an endocannabinoid agent.Formula:C20H37NO2Purity:99.97%Color and Shape:SolidMolecular weight:323.51Ref: TM-T8425
1mg35.00€5mg67.00€10mg90.00€25mg164.00€50mg239.00€100mg348.00€200mg522.00€1mL*10mM (DMSO)85.00€AM281
CAS:AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.Formula:C21H19Cl2IN4O2Purity:98.6% - >99.99%Color and Shape:White To Off-White SolidMolecular weight:557.21Ref: TM-T2264
1mg80.00€5mg169.00€10mg259.00€25mg523.00€50mg750.00€100mg1,035.00€500mg2,062.00€1mL*10mM (DMSO)233.00€AM-2232
CAS:AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.Formula:C24H20N2OPurity:99.37%Color and Shape:SolidMolecular weight:352.43LY2828360
CAS:LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.Formula:C22H27ClN6OPurity:98.45% - 99.51%Color and Shape:SolidMolecular weight:426.94CID 16020046
CAS:CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.Formula:C25H19N3O4Purity:99.03%Color and Shape:SolidMolecular weight:425.44Otenabant
CAS:Otenabant (CP-945598) has been investigated for the treatment of Obesity.Formula:C25H25Cl2N7OPurity:99.43%Color and Shape:SolidMolecular weight:510.42CB1-IN-1
CAS:CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.Formula:C33H31Cl2F3N6O3S2Purity:99.08% - 99.76%Color and Shape:SolidMolecular weight:751.67Ref: TM-T5996
1mg82.00€2mg110.00€5mg180.00€10mg258.00€25mg423.00€50mg588.00€100mg793.00€500mg1,594.00€1mL*10mM (DMSO)215.00€Tetrahydromagnolol
CAS:Tetrahydromagnolol can activate cannabinoid (CB) receptors.Formula:C18H22O2Purity:99.86% - >99.99%Color and Shape:SolidMolecular weight:270.37Ref: TM-TN2268
2mgTo inquire5mg52.00€10mg81.00€25mgTo inquire50mg170.00€100mg243.00€1mL*10mM (DMSO)63.00€BML-190
CAS:BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。Formula:C23H23ClN2O4Purity:97.70%Color and Shape:SolidMolecular weight:426.89CB1/2 agonist 3
CAS:CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.Formula:C25H41NO2Purity:98.78%Color and Shape:SolidMolecular weight:387.6S-Methoprene
CAS:S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.
Formula:C19H34O3Purity:97.05% - 98.55%Color and Shape:SolidMolecular weight:310.47Dehydroabiethylamine
CAS:Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.Formula:C20H31NPurity:98.79%Color and Shape:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidMolecular weight:285.47PSB-KK1445
CAS:PSB-KK1445 is a potent and selective agonist of GPR18, exhibiting EC50 values of 45.4 nM for humans and 124 nM for mice. The selectivity of PSB-KK1445 for GPR18 over the CB receptor subtypes GPR55 and GPR183 exceeds 200-fold.Formula:C24H23FN6O2Molecular weight:446.48GPR55 agonist 3
CAS:Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.Formula:C19H16F4N4Color and Shape:SolidMolecular weight:376.35PM226
CAS:CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.Formula:C22H31NO3Color and Shape:SolidMolecular weight:357.49CID1792197
CAS:CID1792197 is a selective agonist of GPR55.Formula:C24H23N3O4S2Purity:98%Color and Shape:SolidMolecular weight:481.59VSN-16
CAS:VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.Formula:C18H26N2O3Color and Shape:SolidMolecular weight:318.41GAT229
CAS:GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.Formula:C22H18N2O2Color and Shape:SolidMolecular weight:342.39
