Cannabinoid Receptor
Cannabinoid receptors are GPCRs that mediate the effects of endogenous cannabinoids (endocannabinoids) and phytocannabinoids, such as those found in cannabis. The two main types of cannabinoid receptors, CB1 and CB2, are involved in regulating a wide range of physiological processes, including pain perception, appetite, mood, and immune function. Cannabinoid receptor modulators have therapeutic potential in treating conditions such as chronic pain, epilepsy, and multiple sclerosis. At CymitQuimica, we offer a wide range of high-quality cannabinoid receptor modulators to support your research in neuropharmacology, pain management, and immunology.
Found 196 products of "Cannabinoid Receptor"
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Linoleoyl Ethanolamide
CAS:<p>Linoleoyl Ethanolamide is an endocannabinoid agent.</p>Formula:C20H37NO2Purity:99.97%Color and Shape:SolidMolecular weight:323.51Otenabant
CAS:<p>Otenabant (CP-945598) has been investigated for the treatment of Obesity.</p>Formula:C25H25Cl2N7OPurity:99.43%Color and Shape:SolidMolecular weight:510.42CB1 antagonist 4
CAS:<p>TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.</p>Formula:C30H25Cl2F3N4OSPurity:98.97%Color and Shape:SolidMolecular weight:617.51LY2828360
CAS:<p>LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.</p>Formula:C22H27ClN6OPurity:98.45% - 99.51%Color and Shape:SolidMolecular weight:426.94A-836339
CAS:<p>A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.</p>Formula:C16H26N2O2SPurity:99.94%Color and Shape:SolidMolecular weight:310.45Tetrahydromagnolol
CAS:<p>Tetrahydromagnolol can activate cannabinoid (CB) receptors.</p>Formula:C18H22O2Purity:99.86% - >99.99%Color and Shape:SolidMolecular weight:270.37CB1-IN-1
CAS:<p>CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.</p>Formula:C33H31Cl2F3N6O3S2Purity:99.08% - 99.76%Color and Shape:SolidMolecular weight:751.67ML-193
CAS:<p>ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.</p>Formula:C28H25N5O4SPurity:97.74%Color and Shape:SolidMolecular weight:527.59Otenabant hydrochloride
CAS:<p>Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).</p>Formula:C25H26Cl3N7OPurity:99.79% - ≥95%Color and Shape:SolidMolecular weight:546.88Cannabigerol
CAS:<p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>Formula:C21H32O2Purity:99.59% - 99.92%Color and Shape:SolidMolecular weight:316.48AM251
CAS:<p>AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).</p>Formula:C22H21Cl2IN4OPurity:97.43% - 98.79%Color and Shape:A Crystalline SolidMolecular weight:555.24Hemopressin (human, mouse) acetate
<p>Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.</p>Formula:C52H83N13O14Purity:99.86%Color and Shape:SolidMolecular weight:1114.29ARN272
CAS:<p>ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).</p>Formula:C27H20N4O2Purity:98.23%Color and Shape:SolidMolecular weight:432.47Voacamine
CAS:<p>Voacamine: an indole alkaloid, CB1 antagonist, inhibits P-gp, may affect rhythm.</p>Formula:C43H52N4O5Purity:98.54% - 99.82%Color and Shape:SolidMolecular weight:704.9AM1241
CAS:<p>AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.</p>Formula:C22H22IN3O3Purity:98.937% - 99.1%Color and Shape:SolidMolecular weight:503.33yangonin
CAS:<p>Yangonin (Y100550) is a novel CB1 receptor ligand with affinity for human recombinant CB1 receptors.</p>Formula:C15H14O4Purity:98.82% - 99.55%Color and Shape:Pale Yellow PowderMolecular weight:258.27Olivetol
CAS:<p>Olivetol, found in lichens, is an organic antioxidant and THC synthesis precursor.</p>Formula:C11H16O2Purity:99.98%Color and Shape:(Melting Point 102-106°F) (Ntp 1992)Molecular weight:180.24ML-191
CAS:<p>ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.</p>Formula:C24H25N3O3Purity:99.58%Color and Shape:SolidMolecular weight:403.47Hemopressin (rat) acetate(568588-77-2 free base)
<p>Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.</p>Formula:C5H81N13O14Purity:99.37%Color and Shape:SolidMolecular weight:1148.31Org 27569
CAS:<p>Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity and</p>Formula:C24H28ClN3OPurity:>99.99% - ≥95%Color and Shape:SolidMolecular weight:409.95JD-5037
CAS:<p>JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.</p>Formula:C27H27Cl2N5O3SPurity:99.54% - 99.84%Color and Shape:SolidMolecular weight:572.51PSB-SB-487
CAS:<p>PSB-SB-487 is antagonist of GPR55.</p>Formula:C26H32O4Purity:98.53%Color and Shape:SolidMolecular weight:408.53BML-190
CAS:<p>BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。</p>Formula:C23H23ClN2O4Purity:97.70%Color and Shape:SolidMolecular weight:426.89CID 16020046
CAS:<p>CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.</p>Formula:C25H19N3O4Purity:99.03%Color and Shape:SolidMolecular weight:425.44GW 405833
CAS:<p>GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selective</p>Formula:C23H24Cl2N2O3Purity:99.82% - 99.93%Color and Shape:SolidMolecular weight:447.35GW842166X
CAS:<p>GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.</p>Formula:C18H17Cl2F3N4O2Purity:99.47%Color and Shape:SolidMolecular weight:449.25RTICBM-189
CAS:<p>RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.</p>Formula:C15H14Cl2N2OPurity:99.96%Color and Shape:SolidMolecular weight:309.19Bay 59-3074
CAS:<p>Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).</p>Formula:C18H13F6NO4SPurity:97.68% - 99.69%Color and Shape:SolidMolecular weight:453.36(±)-Ibipinabant
CAS:<p>(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.</p>Formula:C23H20Cl2N4O2SPurity:99.28% - 99.83%Color and Shape:SolidMolecular weight:487.4N-Oleoyl glycine
CAS:<p>N-Oleoyl glycine, a lipoamino acid, was able to promote 3T3-L1 adipogenesis through the activation of CB1 receptor and the enhancement of insulin-mediated Akt</p>Formula:C20H37NO3Purity:97.43%Color and Shape:SolidMolecular weight:339.51RVD-Hpα acetate(1193362-76-3 free base)
<p>RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.</p>Formula:C67H109N19O19Purity:99.87%Color and Shape:SolidMolecular weight:1484.71CB1/2 agonist 3
CAS:<p>CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.</p>Formula:C25H41NO2Purity:98.78%Color and Shape:SolidMolecular weight:387.6S-Methoprene
CAS:<p>S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.</p>Formula:C19H34O3Purity:97.05% - 98.55%Color and Shape:SolidMolecular weight:310.47Dehydroabiethylamine
CAS:<p>Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.</p>Formula:C20H31NPurity:98.79%Color and Shape:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidMolecular weight:285.47AM404
CAS:<p>AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.</p>Formula:C26H37NO2Color and Shape:SolidMolecular weight:395.58LEI-101
CAS:<p>LEI-101: potent CB2 agonist, pEC50=8, bioavailable, >100x selective over CB1, potential for inflammatory diseases.</p>Formula:C23H25FN4O4SPurity:98%Color and Shape:SolidMolecular weight:472.53UCM 707
CAS:<p>endocannabinoid transport inhibitor</p>Formula:C25H37NO2Purity:98%Color and Shape:SolidMolecular weight:383.57CB1-IN-2
CAS:<p>CB1-IN-2 (4g) inhibits CB1 receptor with 0.644 μM IC50; crosses blood-brain barrier, may cause CNS side effects like Rimonabant.</p>Formula:C17H19Cl2N5OColor and Shape:SolidMolecular weight:380.27VSN-16
CAS:<p>VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.</p>Formula:C18H26N2O3Color and Shape:SolidMolecular weight:318.41CB1R Allosteric modulator 4
CAS:<p>Modulates CB1R positively; inhibits cAMP production; strong β-arrestin-2 recruitment.</p>Formula:C20H17N3O2SColor and Shape:SolidMolecular weight:363.43UCM710
CAS:<p>UCM710 is a dual inhibitor of α/β hydrolase domain 6 (ABHD6) and fatty acid amide hydrolase (FAAH).</p>Formula:C19H34O3Purity:98%Color and Shape:SolidMolecular weight:310.47CB1/2 agonist 4
CAS:<p>CB1/2 agonist 4 is a potent CB1 full agonist (EC50: 15.09 nM) and CB2 partial agonist (EC50: 1.16 nM), with anti-pain and TRPV1 activation properties.</p>Formula:C27H45NO3Color and Shape:SolidMolecular weight:431.65Palmitoyl serinol
CAS:<p>Anticancer agent 110 is an anticancer compound with cytotoxic, antitumor and antileukemic activities.</p>Formula:C19H39NO3Color and Shape:SolidMolecular weight:329.52(R)-SLV 319
CAS:<p>(R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.</p>Formula:C23H20Cl2N4O2SColor and Shape:SolidMolecular weight:487.4LH 21
CAS:<p>LH-21, a strong CB1 receptor antagonist, curbs eating and lessens weight gain in obese rats.</p>Formula:C20H20Cl3N3Color and Shape:SolidMolecular weight:408.75NIDA 41020
CAS:<p>NIDA 41020 is a CB1 receptor antagonist.</p>Formula:C23H24Cl2N4O2Purity:98%Color and Shape:SolidMolecular weight:459.37AM-6538
CAS:<p>AM6538: long-acting, high-affinity CB antagonist similar to rimonabant, useful for studying cannabinoid agonists.</p>Formula:C26H25Cl2N5O4Color and Shape:SolidMolecular weight:542.41CID1792197
CAS:<p>CID1792197 is a selective agonist of GPR55.</p>Formula:C24H23N3O4S2Purity:98%Color and Shape:SolidMolecular weight:481.59PM226
CAS:<p>CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.</p>Formula:C22H31NO3Color and Shape:SolidMolecular weight:357.49GPR55 agonist 3
CAS:<p>Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.</p>Formula:C19H16F4N4Color and Shape:SolidMolecular weight:376.35
