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G-protein Coupled Receptors and 7-TM Receptors

G-protein Coupled Receptors and 7-TM Receptors

G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.

Found 5708 products of "G-protein Coupled Receptors and 7-TM Receptors"

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  • Moxisylyte hydrochloride
    Targetmol
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    Moxisylyte hydrochloride

    CAS:
    Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
    Formula:C16H26ClNO3
    Purity:99.94% - ≥95%
    Color and Shape:Solid
    Molecular weight:315.84

    Ref: TM-T0394

  • Zolmitriptan
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    Zolmitriptan

    CAS:
    <p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>
    Formula:C16H21N3O2
    Purity:99.69% - 99.91%
    Color and Shape:White Or Kind Of White Powder
    Molecular weight:287.36

    Ref: TM-T1092

  • Mifentidine
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    Mifentidine

    CAS:
    <p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>
    Formula:C13H16N4
    Purity:98.34% - 99.73%
    Color and Shape:Solid
    Molecular weight:228.29

    Ref: TM-T68100

  • YNT-185
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    YNT-185

    CAS:
    YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,
    Formula:C33H37N5O5S
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:615.74

    Ref: TM-T39229

  • Terlipressin Acetate
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    Terlipressin Acetate

    CAS:
    Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).
    Formula:C56H82N16O19S2
    Purity:98.50% - 99.69%
    Color and Shape:Solid
    Molecular weight:1347.5

    Ref: TM-T13920L

  • PF-06882961
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    PF-06882961

    CAS:
    PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Formula:C31H30FN5O4
    Purity:97.19% - 99.56%
    Color and Shape:Solid
    Molecular weight:555.6

    Ref: TM-T12431

  • AH 6809
    Targetmol
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    AH 6809

    CAS:
    <p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>
    Formula:C17H14O5
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:298.29

    Ref: TM-T14148

  • Noradrenaline bitartrate
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    Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Formula:C12H19NO10
    Purity:99.53% - >99.99%
    Color and Shape:Solid
    Molecular weight:337.28

    Ref: TM-T0871

  • Desipramine hydrochloride
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    Desipramine hydrochloride

    CAS:
    Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.
    Formula:C18H23ClN2
    Purity:99.58% - 99.94%
    Color and Shape:White To Off-White Powder
    Molecular weight:302.842

    Ref: TM-T0991

  • Evocalcet
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    Evocalcet

    CAS:
    Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).
    Formula:C24H26N2O2
    Purity:98.88% - 99.68%
    Color and Shape:Solid
    Molecular weight:374.48

    Ref: TM-T15261

  • Ticlopidine hydrochloride
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    Ticlopidine hydrochloride

    CAS:
    <p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>
    Formula:C14H15Cl2NS
    Purity:99.85% - >99.99%
    Color and Shape:White Powder
    Molecular weight:300.25

    Ref: TM-T0362

  • Senktide acetate
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    Senktide acetate

    <p>Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of ELM and can be used to study Alzheimer's disease.</p>
    Formula:C42H59N7O13S
    Purity:98.26%
    Color and Shape:Solid
    Molecular weight:902.02

    Ref: TM-T7633L

  • Venlafaxine hydrochloride
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    Venlafaxine hydrochloride

    CAS:
    <p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>
    Formula:C17H28ClNO2
    Purity:97.32% - 99.86%
    Color and Shape:White Crystalline Powder
    Molecular weight:313.86

    Ref: TM-T0472

  • Methyldopa
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    Methyldopa

    CAS:
    Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or
    Formula:C10H13NO4
    Purity:98.95% - 99.86%
    Color and Shape:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Molecular weight:211.21

    Ref: TM-T0505

  • Frovatriptan succinate hydrate
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    Frovatriptan succinate hydrate

    CAS:
    <p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>
    Formula:C18H25N3O6
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:379.41

    Ref: TM-T11326

  • Bambuterol hydrochloride
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    Bambuterol hydrochloride

    CAS:
    Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.
    Formula:C18H30ClN3O5
    Purity:99.53% - 99.61%
    Color and Shape:White Solid
    Molecular weight:403.91

    Ref: TM-T1446

  • Nylidrin hydrochloride
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    Nylidrin hydrochloride

    CAS:
    Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.
    Formula:C19H26ClNO2
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:335.87

    Ref: TM-T0173

  • Chlorprothixene hydrochloride
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    Chlorprothixene hydrochloride

    CAS:
    Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.
    Formula:C18H18ClNS·HCl
    Purity:99.76%
    Color and Shape:White Powder
    Molecular weight:352.32

    Ref: TM-T0074L

  • Roxatidine Acetate hydrochloride
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    Roxatidine Acetate hydrochloride

    CAS:
    Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.
    Formula:C19H29ClN2O4
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:384.9

    Ref: TM-T0157

  • JP1302 dihydrochloride
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    JP1302 dihydrochloride

    CAS:
    JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.
    Formula:C24H26Cl2N4
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:441.4

    Ref: TM-T11726

  • Moxonidine
    Targetmol
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    Moxonidine

    CAS:
    Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.
    Formula:C9H12ClN5O
    Purity:99.81% - 99.94%
    Color and Shape:Crystal
    Molecular weight:241.68

    Ref: TM-T1028

  • Levodropropizine
    Targetmol
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    Levodropropizine

    CAS:
    Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.
    Formula:C13H20N2O2
    Purity:99.87% - 99.93%
    Color and Shape:White Or Off White Crystalline Powder
    Molecular weight:236.31

    Ref: TM-T0217

  • CD80-IN-3
    Targetmol
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    CD80-IN-3

    CAS:
    <p>CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).</p>
    Formula:C17H10FN3O3
    Purity:98.08%
    Color and Shape:Solid
    Molecular weight:323.28

    Ref: TM-T10722

  • Heptaminol hydrochloride
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    Heptaminol hydrochloride

    CAS:
    <p>Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.</p>
    Formula:C8H20ClNO
    Purity:98.61%
    Color and Shape:White Crystalline Powder
    Molecular weight:181.71

    Ref: TM-T0045

  • Rimonabant
    Targetmol
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    Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Formula:C22H21Cl3N4O
    Purity:98% - 99.91%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:463.79

    Ref: TM-T1519L

  • LCKLSL hydrochloride
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    LCKLSL hydrochloride

    <p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>
    Formula:C30H58ClN7O8S
    Purity:98.02% - 99.31%
    Color and Shape:Solid
    Molecular weight:712.34

    Ref: TM-T78015

  • Blonanserin
    Targetmol
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    Blonanserin

    CAS:
    Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.
    Formula:C23H30FN3
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:367.5

    Ref: TM-T1180

  • Fluvoxamine maleate
    Targetmol
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    Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Formula:C19H25F3N2O6
    Purity:99.92% - 99.94%
    Color and Shape:White Crystalline Powder
    Molecular weight:434.41

    Ref: TM-T1077

  • Dimenhydrinate
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    Dimenhydrinate

    CAS:
    Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.
    Formula:C24H28ClN5O3
    Purity:99.57% - 99.77%
    Color and Shape:Crystals Physical Description Crystalline White Powder (Ntp 1992)
    Molecular weight:469.96

    Ref: TM-T0298

  • Urocortin (rat) acetate
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    Urocortin (rat) acetate

    Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.
    Purity:97.76%
    Color and Shape:Soild

    Ref: TM-TP1020L

  • Aripiprazole
    Targetmol
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    Aripiprazole

    CAS:
    Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.
    Formula:C23H27Cl2N3O2
    Purity:99.43% - 99.62%
    Color and Shape:Colourless Flake Crystalline Solid
    Molecular weight:448.39

    Ref: TM-T1566

  • Metaproterenol hemisulfate
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    Metaproterenol hemisulfate

    CAS:
    Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
    Formula:C11H17NO3·5H2O4S
    Purity:98.53% - 99.74%
    Color and Shape:Solid
    Molecular weight:260.3

    Ref: TM-T0277

  • Trimipramine maleate
    Targetmol
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    Trimipramine maleate

    CAS:
    Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.
    Formula:C24H30N2O4
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:410.51

    Ref: TM-T1045

  • Pericyazine
    Targetmol
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    Pericyazine

    CAS:
    <p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>
    Formula:C21H23N3OS
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:365.49

    Ref: TM-T16472

  • Adrenalone hydrochloride
    Targetmol
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    Adrenalone hydrochloride

    CAS:
    Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.
    Formula:C9H11NO3·HCl
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:217.65

    Ref: TM-T0948

  • Cefaclor monohydrate
    Targetmol
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    Cefaclor monohydrate

    CAS:
    <p>Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.</p>
    Formula:C15H16ClN3O5S
    Purity:97.36% - 99.9%
    Color and Shape:White Crystaling Powder
    Molecular weight:385.82

    Ref: TM-T1495

  • Indacaterol maleate
    Targetmol
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    Indacaterol maleate

    CAS:
    <p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>
    Formula:C28H32N2O7
    Purity:99.03% - 99.67%
    Color and Shape:Solid
    Molecular weight:508.56

    Ref: TM-T1239

  • Agomelatine
    Targetmol
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    Agomelatine

    CAS:
    Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.
    Formula:C15H17NO2
    Purity:99.92%
    Color and Shape:White Solid
    Molecular weight:243.3

    Ref: TM-T1445

  • Ziprasidone
    Targetmol
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    Ziprasidone

    CAS:
    <p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>
    Formula:C21H21ClN4OS
    Purity:99.55%
    Color and Shape:Tan Solid
    Molecular weight:412.94

    Ref: TM-T0031L2

  • Fexofenadine hydrochloride
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    Fexofenadine hydrochloride

    CAS:
    Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with
    Formula:C32H40ClNO4
    Purity:>99.99%
    Color and Shape:White Crystalline Powder
    Molecular weight:538.12

    Ref: TM-T1470L

  • CYM 50769
    Targetmol
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    CYM 50769

    CAS:
    <p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>
    Formula:C24H17ClN2O3
    Purity:98% - 99.08%
    Color and Shape:Solid
    Molecular weight:416.86

    Ref: TM-T22702

  • Levocetirizine
    Targetmol
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    Levocetirizine

    CAS:
    Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.
    Formula:C21H25ClN2O3
    Purity:98% - 99.94%
    Color and Shape:White Powder
    Molecular weight:388.89

    Ref: TM-T1469

  • Talastine
    Targetmol
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    Talastine

    CAS:
    Talastine is an antihistamine compound that can induce an allergic rash.
    Formula:C19H21N3O
    Purity:99.44% - 99.84%
    Color and Shape:Solid
    Molecular weight:307.39

    Ref: TM-T68150

  • Filorexant
    Targetmol
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    Filorexant

    CAS:
    Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).
    Formula:C24H25FN4O2
    Purity:98.88%
    Color and Shape:Solid
    Molecular weight:420.48

    Ref: TM-T16096

  • Clonidine hydrochloride
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    Clonidine hydrochloride

    CAS:
    Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.
    Formula:C9H10Cl3N3
    Purity:99.16% - 99.86%
    Color and Shape:Solid
    Molecular weight:266.55

    Ref: TM-T1247

  • Olinciguat
    Targetmol
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    Olinciguat

    CAS:
    Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.
    Formula:C21H16F5N7O3
    Purity:99.33% - 99.71%
    Color and Shape:Solid
    Molecular weight:509.39

    Ref: TM-T16383

  • ML-180
    Targetmol
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    ML-180

    CAS:
    <p>ML-180 (SR1848) is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 μM) .</p>
    Formula:C20H25ClN4O2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:388.89

    Ref: TM-T12075

  • Ondansetron hydrochloride dihydrate
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    Ondansetron hydrochloride dihydrate

    CAS:
    <p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>
    Formula:C18H19N3O·HCl·2H2O
    Purity:99.92%
    Color and Shape:White Crystal Powder
    Molecular weight:365.86

    Ref: TM-T1478

  • Tetrahydrozoline
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    Tetrahydrozoline

    CAS:
    <p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>
    Formula:C13H16N2
    Purity:97.85% - 99.77%
    Color and Shape:Solid
    Molecular weight:200.28

    Ref: TM-T0397

  • CymitQuimica logo
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    Latozinemab

    Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.
    Purity:> 95%
    Color and Shape:Liquid
    Molecular weight:146.28 kDa

    Ref: TM-T77053