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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66669 products of "Inhibitors"

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  • PF-06463922 acetate

    CAS:
    PF-06463922 acetate: ALK/ROS1 inhibitor, brain- penetrable, active vs crizotinib-resistant mutants, in NSCLC trials.
    Formula:C23H23FN6O4
    Color and Shape:Solid
    Molecular weight:466.46
  • Silvestrol

    CAS:
    Silvestrol is a eukaryotic translation initiation factor 4A inhibitor. Silvestrol causes autophagy and caspase-mediated apoptosis.
    Formula:C34H38O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:654.66
  • FAK-IN-6


    FAK-IN-6: Potent FAK inhibitor (IC50=1.415 nM), anti-cancer, for pancreatic studies.
    Formula:C25H31ClN5O6PS
    Color and Shape:Solid
    Molecular weight:596.04
  • RSV-IN-5

    CAS:
    RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM & 8.1 nM. Potent anti-RSV.
    Formula:C28H37N7O2
    Color and Shape:Solid
    Molecular weight:503.64
  • Antitrypanosomal agent 5


    Antitrypanosal agent 5 is a selective anti-trypanosomal agent that acts on T. brucei (IC50: 1 nM) and HEK293 cells (IC50: 483.3 μM).
    Formula:C30H30N6O4S
    Color and Shape:Solid
    Molecular weight:570.66
  • 5-HT6R/MAO-B modulator 1


    5-HT6R/MAO-B modulator 1 blocks 5-HT6R and permanently inhibits MAO-B, protects glial cells, and reverses memory loss.
    Formula:C33H38N4O3S
    Color and Shape:Solid
    Molecular weight:570.74
  • PPARγ agonist 1


    PPARγ agonist 1 is a potent agonist of PPARγ that efficiently activates hPPARγ without causing full agonism, thereby avoiding adverse effects.
    Formula:C34H39NO3
    Color and Shape:Solid
    Molecular weight:509.68
  • MtTMPK-IN-9


    MtTMPK-IN-9 moderately inhibits MtbTMPK (IC50: 48 μM), has submicromolar Mycobacterium activity, and is non-toxic, aiding tuberculosis research.
    Formula:C25H26N6O7
    Color and Shape:Solid
    Molecular weight:522.51
  • Brostallicin HCl

    CAS:
    Brostallicin, a synthetic MGB, inhibits DNA replication in cancer cells, inducing cell death, effective against MMR-defective tumors.
    Formula:C30H36BrClN12O5
    Color and Shape:Solid
    Molecular weight:760.04
  • c-Myc inhibitor 4


    Potent oral c-Myc inhibitor 4 reduces the proto-oncogene linked to tumor development.
    Formula:C26H33FN6O3
    Color and Shape:Solid
    Molecular weight:496.58
  • PARP1-IN-5


    PARP1-IN-5 is a potent, selective, orally active, low-toxicity PARP-1 inhibitor with an IC50 value of 14.7 nM. PARP1-IN-5 can be used in cancer research.
    Formula:C25H24N2O5S
    Color and Shape:Solid
    Molecular weight:464.53
  • Isobetanin

    CAS:
    <p>Isobetanin is a betacyanin that has been shown to enhance vitexin-2-O-xyloside mediated inhibition of proliferation of T24 bladder cancer cells.</p>
    Formula:C24H26N2O13
    Color and Shape:Solid
    Molecular weight:550.47
  • SHP2 IN-1

    CAS:
    SHP2 IN-1 is an allergic SHP2 (PTPN11) inhibitor(IC50 : 3 nM).
    Formula:C18H22Cl2N6OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.38
  • NPR-C activator 1

    CAS:
    NPR-C activator 1 is an activator of the natriuretic peptide receptor C (NPR-C), which can be used to study cardiovascular diseases.
    Formula:C18H24N6O3
    Purity:98.74%
    Color and Shape:Solid
    Molecular weight:372.42
  • C.I. Pigment Red 60

    CAS:
    C.I. Pigment Red 60 is a bright, scarlet, semi-transparent red pigment.
    Formula:C17H9N2Na3O9S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:518.35
  • RORγt/DHODH-IN-3


    RORγt/DHODH-IN-3 (compound (S)-14d) is a potent, orally active dual inhibitor of RORγt (IC50: 0.098 μM) and DHODH (IC50: 0.432 μM).RORγt/DHODH-IN-1 has
    Formula:C24H26ClF6N3O3S
    Color and Shape:Solid
    Molecular weight:585.99
  • Anticancer agent 65

    CAS:
    Anticancer agent 65: Effective on A549 cells, IC50 1.07 μM, halts S phase, triggers apoptosis, elevates p53/p21, causes ROS and MMP collapse.
    Formula:C36H63NO5
    Color and Shape:Solid
    Molecular weight:589.89
  • CDK/HDAC-IN-1


    CDK/HDAC-IN-1 inhibits CDK2/4/6 & HDAC6 with IC50s: 60.9, 276, 27.2, and 128.6 nM respectively.
    Formula:C20H18N4O4
    Color and Shape:Solid
    Molecular weight:378.38
  • MRS2279 diammonium

    CAS:
    MRS2279 diammonium, a P2Y1 antagonist with K i 2.5 nM, IC 50 51.6 nM, blocks ADP-induced platelet aggregation, pK b 8.05.
    Formula:C13H24ClN7O8P2
    Color and Shape:Solid
    Molecular weight:503.77
  • Mt KARI-IN-1


    <p>Mt KARI-IN-1 inhibits Mtb KARI with a 3.06 μM Ki, targeting tuberculosis.</p>
    Formula:C14H11N5O4S2
    Color and Shape:Solid
    Molecular weight:377.4
  • Lobaric acid

    CAS:
    Lobaric acid, from Stereocaulon lichen, has antioxidant and anticancer properties, inhibits PTP1B and 12(S)-LOX, and reduces TMV lesions in plants.
    Formula:C25H28O8
    Color and Shape:Solid
    Molecular weight:456.48
  • Pyruvate Carboxylase-IN-2

    CAS:
    Pyruvate Carboxylase-IN-2, erianin analog, inhibits PC with IC50s of 0.065/0.097 μM in lysate/cell assays, targets HCC.
    Formula:C21H22O8
    Color and Shape:Solid
    Molecular weight:402.39
  • Zorubicin

    CAS:
    <p>Zorubicin, a Daunorubicin derivative, targets topoisomerase II, inhibits DNA polymerase, and researches acute leukemia, sarcomas.</p>
    Formula:C34H35N3O10
    Color and Shape:Solid
    Molecular weight:645.66
  • Udifitimod

    CAS:
    Udifitimod (BMS-986166) is a potent, selective, and orally active modulator of the S1P1R receptor, showing potential for research in autoimmune diseases.
    Formula:C25H33NO2
    Color and Shape:Solid
    Molecular weight:379.54
  • NCI-006

    CAS:
    NCI-006, an LDH inhibitor, slows tumor growth and enhances pyruvate's role in mitochondrial metabolism.
    Formula:C31H24F2N4O4S3
    Color and Shape:Solid
    Molecular weight:650.74
  • Heparastatin

    CAS:
    Heparastatin is an inhibitor of heparanase.
    Formula:C8H11F3N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:272.18
  • TT15

    CAS:
    TT15 is an agonist of the GLP-1R.
    Formula:C51H44Cl2N4O6
    Color and Shape:Solid
    Molecular weight:879.82
  • OUN58101

    CAS:
    OUN58101, also MDK-8101/BI-D, is an RSV L-protein inhibitor with no formal name, first reported in patent WO 2005042530.
    Formula:C32H36N6O6
    Color and Shape:Solid
    Molecular weight:600.66
  • NTU281

    CAS:
    NTU281 inhibits transglutaminase-2, lowers creatinine in diabetic rats, reduces proteinuria, and fights glomerulosclerosis.
    Formula:C25H31N2O6S
    Color and Shape:Solid
    Molecular weight:487.59
  • HIV-1 inhibitor-13


    HIV-1 inhibitor-13: oral NNRTI, IC50=0.14μM for HIV-1 RT, effective on resistant strains (EC50=2.85-18nM).
    Formula:C30H32N6O3
    Color and Shape:Solid
    Molecular weight:524.61
  • Homodestcardin

    CAS:
    <p>Homodestcardin: cyclic depsipeptide from T. roseum with immunosuppressant properties; inhibits mouse T cell proliferation.</p>
    Formula:C32H55N5O7
    Color and Shape:Solid
    Molecular weight:621.81
  • USP7-IN-6

    CAS:
    USP7-IN-6 is a potent inhibitor of ubiquitin-specific protease 7 (USP7, IC50: 6.8 nM).
    Formula:C41H43N7O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:729.89
  • Emd 52297

    CAS:
    Emd 52297 is an inhibitor of renin.
    Formula:C39H59N11O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:793.96
  • (S)-MALT1-IN-5

    CAS:
    (S)-MALT1-IN-5: Potent MALT1 protease inhibitor, may help in abnormal T/B-cell signalling and MALT1-linked diseases.
    Formula:C17H17ClF2N6O3
    Color and Shape:Solid
    Molecular weight:426.80
  • CS-003 HCl

    CAS:
    CS-003 HCl is a TNRA - triple neurokinin receptor antagonist.
    Formula:C34H39Cl3N2O6S
    Color and Shape:Solid
    Molecular weight:710.1
  • VEGFR-2-IN-18


    VEGFR-2-IN-18 is a potent VEGFR-2 inhibitor with a 60 nM IC50, promoting cell apoptosis and anticancer effects.
    Formula:C20H13ClN4O2
    Color and Shape:Solid
    Molecular weight:376.8
  • KMN-80

    CAS:
    KMN-80 is a potent, selective EP4 agonist with IC50 3 nM, spurring osteoblast differentiation, and showing in vivo bone repair efficacy.
    Formula:C21H33NO4
    Color and Shape:Solid
    Molecular weight:363.49
  • Antiproliferative agent-4


    Antiproliferative agent-4 suppresses cancer cell growth with low toxicity, inhibits tumors in mice, and induces apoptosis in EC109 cells.
    Formula:C29H35ClO8
    Color and Shape:Solid
    Molecular weight:547.04
  • L-697639

    CAS:
    L-697639 inhibits of HIV-1 reverse transcriptase and HIV-1 replication.
    Formula:C18H21N3O2
    Color and Shape:Solid
    Molecular weight:311.38
  • eIF4A3-IN-4


    eIF4A3-IN-4 is a novel inhibitor of eIF4A (IC50: 8.6 μM).
    Formula:C24H20N2O5
    Color and Shape:Solid
    Molecular weight:416.43
  • SGE-516

    CAS:
    SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.
    Formula:C23H35N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:385.54
  • Isoleucyl tRNA synthetase-IN-2

    CAS:
    Isoleucyl tRNA synthetase-IN-2 is a selective and potent inhibitor (Ki: 114 nM) that targets isoleucyl tRNA synthetase (IleRS).
    Formula:C22H33N5O8S
    Color and Shape:Solid
    Molecular weight:527.59
  • 14α-Demethylase/DNA Gyrase-IN-1


    14α-Demethylase/DNA Gyrase-IN-1 (Compound 7c) is a potent inhibitor of 14α-Demethylase/DNA Gyrase with antibacterial activity.
    Formula:C26H22N4O4
    Color and Shape:Solid
    Molecular weight:454.48
  • Mopivabil


    Mopivabil is the angiotensin II receptor antagonist[1].
    Formula:C14H20O3
    Color and Shape:Solid
    Molecular weight:236.31
  • Carbonic anhydrase inhibitor 5


    Potent hCA inhibitor: targets hCA II, IX & XII with IC50s of 42.9, 47.6, & 6.7 nM respectively.
    Formula:C24H20ClN3O3S
    Color and Shape:Solid
    Molecular weight:465.95
  • Desacetylravidomycin

    CAS:
    Desacetylravidomycin is a new inhibitor of IL-4 signal transduction, produced by Streptomyces sp. WK-6326.
    Formula:C29H31NO8
    Color and Shape:Solid
    Molecular weight:521.56
  • Ambelline

    CAS:
    Ambelline has antitumor activity.
    Formula:C18H21NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.36
  • ddCTP trisodium


    ddCTP trisodium, an HIV reverse transcriptase target, aids AIDS research and DNA sequencing as a ddNTP.
    Formula:C9H13N3Na3O12P3
    Color and Shape:Solid
    Molecular weight:517.1
  • KC-11404

    CAS:
    KC-11404 is an LTB4 inhibitor for the treatment of b-cell leukemias and lymphomas, potently inhibiting histamine, platelet activating factor and 5-lipoxygenase.
    Formula:C28H38N4O
    Color and Shape:Solid
    Molecular weight:446.63
  • PF-9404C

    CAS:
    PF-9404C: S-S diastereoisomer, beta-blocker with vasodilation, boosts cyclic GMP in rat aorta cells from 3 to 53 pmol/mg protein.
    Formula:C16H25N3O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:403.38
  • LP-284

    CAS:
    LP-284 is a DNA alkylating agent effective against solid tumors and hematologic cancers like MCL.
    Formula:C16H20N2O4
    Color and Shape:Solid
    Molecular weight:304.34
  • AM-3189

    CAS:
    AM-3189: potent, selective GPR40 agonist with low CNS penetration, good pharmacokinetics, and efficacy mirroring AMG 837.
    Formula:C27H25ClN2O3
    Color and Shape:Solid
    Molecular weight:460.95
  • Latrunculin M

    CAS:
    Latrunculin M, a novel marine toxin, disrupts microfilament organization in cultured cells.
    Formula:C21H33NO5S
    Color and Shape:Solid
    Molecular weight:411.55
  • GNE-203

    CAS:
    GNE-203 is a Met inhibitor.
    Formula:C30H29Cl2F3N8O3
    Color and Shape:Solid
    Molecular weight:677.50
  • Detajmium

    CAS:
    Detajmium is an anti-arrhythmia compound. It is an Na(+)-channel-blocking drug with an extremely long recovery from use-dependent sodium channel block.
    Formula:C27H42N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:456.64
  • Luffolide

    CAS:
    Luffolide, a Luffariella sponge metabolite, shares manoalide's anti-inflammatory traits and fully inhibits PLA2's cleavage of phosphatidylcholine.
    Formula:C27H40O6
    Color and Shape:Solid
    Molecular weight:460.60
  • Anticancer agent 53

    CAS:
    Anticancer agent 53 exhibits potent in vitro cytotoxicity, triggers apoptosis, halts S/G2/M cycle, and has antitumor effects without toxicity.
    Formula:C31H25FN4O6S
    Color and Shape:Solid
    Molecular weight:600.62
  • KMH-233

    CAS:
    KMH-233 effectively blocks LAT1, inhibiting L-leucine uptake and cell growth, boosting betastatin and cisplatin efficacy at 25 μM.
    Formula:C32H25N7O5
    Color and Shape:Solid
    Molecular weight:587.58
  • DL-Buthionine-(S,R)-sulfoximine hydrochloride


    DL-Buthionine-(S,R)-sulfoximine hydrochloride (Buthionine sulfoximine hydrochloride) is a potent and specific glutamylcysteine synthetase biosynthesis inhibitor
    Formula:C8H19ClN2O3S
    Color and Shape:Solid
    Molecular weight:258.77
  • Glutaminyl cyclases-IN-1


    Glutaminyl cyclase inhibitor IsoQC-IN-1: IC50=12 nM for QC, 73 nM for isoQC; blocks CD47/SIRPα; boosts THP-1, U937 macrophage phagocytosis.
    Formula:C25H30N6O2S
    Color and Shape:Solid
    Molecular weight:478.61
  • CM-352

    CAS:
    CM-352 is a metalloproteinase inhibitor that reduces brain damage and improves functional recovery in rat models of cerebral hemorrhage.
    Formula:C24H29N3O6S
    Purity:97.24%
    Color and Shape:Solid
    Molecular weight:487.57
  • GS-9822

    CAS:
    GS-9822 is a new LEDGIN inhibitor targeting LEDGF/p75 to alter HIV integration, showing a block-and-lock effect in cells.
    Formula:C36H39ClN4O4S
    Color and Shape:Solid
    Molecular weight:659.24
  • (+)-Sparteine sulfate pentahydrate


    (+)-sparteine (sulfate pentahydrate) is a ganglion blocker that competitively blocks nicotinic acetylcholine receptors in neurons.
    Formula:C15H38N2O9S
    Color and Shape:Solid
    Molecular weight:422.54
  • α-Glucosidase-IN-13


    α-Glucosidase-IN-13 is an inhibitor of α-glucosidase (IC50: 5.69 μM).
    Formula:C25H28N4O3S2
    Color and Shape:Solid
    Molecular weight:496.64
  • DNA-PK-IN-8

    CAS:
    DNA-PK-IN-8: Potent, selective oral DNA-PK inhibitor, IC50 = 0.8 nM, boosts anti-cancer effects with Doxorubicin.
    Formula:C19H22N8O2
    Color and Shape:Solid
    Molecular weight:394.43
  • AKR1C3-IN-8


    AKR1C3-IN-8 (Compound 5) is an effective and selective AKR1C3 inhibitor (IC50=0.069 μM). AKR1C3-IN-8 has antitumor activity.
    Formula:C23H20N4O3
    Color and Shape:Solid
    Molecular weight:400.43
  • TK-129


    TK-129: Oral KDM5B inhibitor, IC50=44 nM, low-toxicity, cardioprotective, aids in heart disease research.
    Formula:C15H23N5O2
    Color and Shape:Solid
    Molecular weight:305.38
  • GSK3527497 HCl

    CAS:
    GSK3527497: potent TRPV4 inhibitor, IC50=12 nM, targets heart/respiratory issues, for oral/IV use, low-dose effective.
    Formula:C17H17Cl2FN4O4S
    Color and Shape:Solid
    Molecular weight:463.3054
  • Etamicastat

    CAS:
    Etamicastat can be used in the research of cardiovascular diseases.
    Formula:C14H15F2N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:311.35
  • Musettamycin

    CAS:
    Musettamycin triggers erythroid differentiation in blood cells, acts like anthracycline antibiotics, but only inhibits gram-positive bacteria.
    Formula:C36H45NO14
    Color and Shape:Solid
    Molecular weight:715.74
  • BRD-9526

    CAS:
    BRD-9526 is a potent and selective inhibitor of Sonic Hedgehog (Shh).
    Formula:C26H31Cl2N3O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:584.51
  • FtsZ-IN-4


    FtsZ-IN-4 is an oral FtsZ inhibitor with strong antibacterial effects and good drug traits, low toxicity (CC50 >20μg/mL).
    Formula:C21H16ClF2NO2
    Color and Shape:Solid
    Molecular weight:387.81
  • (R)-FL118

    CAS:
    FL118 inhibits human survivinion expression and activates tumor suppressor p53 as a MOA in p53 wild-type cancer cells.
    Formula:C21H16N2O6
    Color and Shape:Solid
    Molecular weight:392.36
  • Cilobamine (free base)

    CAS:
    Cilobamine: a stimulant antidepressant, inhibits norepinephrine-dopamine reuptake, based on dichloroisoprenaline structure.
    Formula:C17H23Cl2NO
    Color and Shape:Solid
    Molecular weight:328.28
  • HBV-IN-18


    HBV-IN-18 (Compound 3) is an HBV capsid assembly modulator (CpAM) (EC50: 2790 nM).
    Formula:C17H15F6N5O2
    Color and Shape:Solid
    Molecular weight:435.32
  • SARS-CoV-2 nsp14-IN-1


    SARS-CoV-2 nsp14-IN-1 inhibits Nsp14 Mtase with an IC50 of 0.061 μM, affecting multiple substrates.
    Formula:C20H20N6O5S
    Color and Shape:Solid
    Molecular weight:456.48
  • Nepaprazole sodium

    CAS:
    Nepaprazole Na (TY-11345), a proton pump inhibitor, may treat gastric ulcers; it reduces H+/K(+)-ATPase activity, with IC50 of 5.8-9.9 microM.
    Formula:C18H18N3NaO2S
    Color and Shape:Solid
    Molecular weight:363.41
  • Karenitecin

    CAS:
    <p>Karenitecin (Cositecan) is an inhibitor of topoisomerase I. It has potent anti-cancer activity.</p>
    Formula:C25H28N2O4Si
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.59
  • L 365209

    CAS:
    L 365209 is an oxytocin antagonist.
    Formula:C40H50N8O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:738.88
  • Hexedine

    CAS:
    Hexedine is a biochemical.
    Formula:C22H45N3
    Color and Shape:Solid
    Molecular weight:351.61
  • CCT369260

    CAS:
    CCT369260 (compound 1), an orally active inhibitor targeting B-cell lymphoma 6 (BCL6), demonstrates anti-tumor efficacy with an IC50 value of 520 nM [1].
    Formula:C24H31ClF2N6O2
    Color and Shape:Solid
    Molecular weight:508.99
  • B-3852

    CAS:
    B-3852 is a Bradykinin inhibitor.
    Formula:C55H74F3N15O11
    Color and Shape:Solid
    Molecular weight:1178.27
  • Org-6906

    CAS:
    DCB-3503, a tylophorine analog, may treat cancer and suppress immunity by blocking protein synthesis and modulating HSC70's ATPase activity.
    Formula:C13H16ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:221.73
  • BAY-3153

    CAS:
    BAY-3153 is a selective CCR1 ( C-C motif chemokine receptor 1 ) antagonist (human IC 50 =3 nM ; rat IC 50 =11 nM ; mice IC 50 =81 nM) .
    Formula:C25H29Cl2N3O4
    Color and Shape:Solid
    Molecular weight:506.42
  • IRAK4-IN-15

    CAS:
    IRAK4-IN-15: selective IRAK4 inhibitor, IC50 0.002 μM, good PK, low clearance, synergizes with Acalabrutinib in MyD88/CD79 mutant ABC-DLBCL.
    Formula:C25H29FN10
    Color and Shape:Solid
    Molecular weight:488.56
  • PTP1B-IN-17


    PTP1B-IN-17, a benzimidazole derivative, inhibits PTP1B (Ki: 30.2 μM) and may help study type 2 diabetes.
    Formula:C26H19N3O4S
    Color and Shape:Solid
    Molecular weight:469.51
  • QPX7728 methoxy acetoxy methy ester

    CAS:
    QPX7728 methoxy acetoxy methy ester is an inhibitor of boronic acid β-lactamase.
    Formula:C14H14BFO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.07
  • Anti-TSWV agent 1


    Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV).
    Formula:C22H27ClN4OS3
    Color and Shape:Solid
    Molecular weight:495.12
  • Pan-Trk-IN-3


    Pan-Trk-IN-3: potent Trk inhibitor (IC50: 2-26 nM), effective against drug-resistant mutants, induces apoptosis, anti-tumor effects.
    Formula:C29H31ClN8O3
    Color and Shape:Solid
    Molecular weight:575.06
  • CXCR7 antagonist-1 hydrochloride

    CAS:
    CXCR7 antagonist-1 hydrochloride blocks SDF-1 and I-TAC from CXCR7; may prevent cancer and inflammation.
    Formula:C21H20ClFN6O
    Color and Shape:Solid
    Molecular weight:426.87
  • Topoisomerase II inhibitor 6


    Topoisomerase II inhibitor 6, a potent tryptanthrin derivative, blocks G2 phase in CCRF-CEM cells, induces DNA breaks, and may be used for cancer research.
    Formula:C19H18N4O2
    Color and Shape:Solid
    Molecular weight:334.37
  • α-Glucosidase-IN-12


    α-Glucosidase-IN-12 is a potent inhibitor of α-glucosidase (IC50: 10.20 μM).
    Formula:C25H30N4O4S2
    Color and Shape:Solid
    Molecular weight:514.66
  • YM-355179

    CAS:
    YM-355179 is a novel, selective antagonist of CC chemokine receptor 3 with oral activity.
    Formula:C33H34FN4O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:617.64
  • TP-6076

    CAS:
    TP-6076 is a fluorocycline antibiotic, inhibiting bacterial protein synthesis, exhibiting great antimicrobial activity against carbapenem-resistant A.
    Formula:C28H32F3N3O7
    Color and Shape:Solid
    Molecular weight:579.56
  • 264W94

    CAS:
    264W94 robustly inhibits IBAT, induces CYP7A1, and significantly reduces cholesterol.
    Formula:C23H31NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:417.56
  • Fasitibant

    CAS:
    <p>Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.</p>
    Formula:C36H49Cl2N6O6S
    Color and Shape:Solid
    Molecular weight:764.78
  • MEN-10354

    CAS:
    MEN-10354 is a less potent and less selective NK-2 tachykinin receptor antagonist compared to the linear analog, R 396.
    Formula:C37H46N8O9
    Color and Shape:Solid
    Molecular weight:746.81
  • 3-IN-PP1

    CAS:
    3-IN-PP1: PKD inhibitor (IC50: 94-108 nM for PKD1/2/3), broad anticancer agent for research.
    Formula:C17H18N6
    Color and Shape:Solid
    Molecular weight:306.36
  • GLS-1-IN-1


    GLS-1-IN-1 (compound 1d) is a GLS-1 inhibitor that inhibits Hep G2, MCF 7 and MCF 10A cells.
    Formula:C26H25FN4OS
    Color and Shape:Solid
    Molecular weight:460.57
  • KPH2f

    CAS:
    KPH2f: dual URAT1/GLUT9 inhibitor, orally active, IC50: 0.24μM (URAT1), 9.37μM (GLUT9), minimal OAT1/ABCG2 impact.
    Formula:C24H16N3NaO2S
    Color and Shape:Solid
    Molecular weight:433.46