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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66618 products of "Inhibitors"

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  • (RS)-AMPA monohydrate

    CAS:
    <p>(RS)-AMPA monohydrate, potent glutamate analogue, selectively activates L-glutamic acid without affecting kainic acid or NMDA receptors.</p>
    Formula:C7H12N2O5
    Color and Shape:Solid
    Molecular weight:204.182
  • S1P1 agonist 4

    CAS:
    <p>S1P1 agonist 4 exhibits enhanced potency with an EC 50 value of less than 0.05 mg/kg and a predicted human half-life (t1/2) of approximately 5 days, indicating</p>
    Formula:C24H31NO3
    Color and Shape:Solid
    Molecular weight:381.51
  • Anticancer agent 45


    <p>Anticancer agent 46, potent and selective, induces apoptosis, is cytotoxic to cancer cells, with low toxicity to human lymphocytes.</p>
    Formula:C22H14ClN3O6S2
    Color and Shape:Solid
    Molecular weight:515.95
  • OICR-9429-N-C2-NH2

    CAS:
    <p>OICR-9429-N-C2-NH2, a ligand for WDR5, intermediate 2, serves as a crucial compound in the synthesis of PROTACs.</p>
    Formula:C31H38F3N7O2
    Color and Shape:Solid
    Molecular weight:597.687
  • A 76889

    CAS:
    A 76889 is an inhibitor of HIV-1 protease.
    Formula:C44H58N8O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:794.98
  • Org-31710

    CAS:
    <p>Org-31710 is a progesterone receptor antagonist potentially for contraception.</p>
    Formula:C30H39NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:445.64
  • LLS30

    CAS:
    <p>LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.</p>
    Formula:C34H33Cl4N5O3
    Color and Shape:Solid
    Molecular weight:701.47
  • ATR-IN-11


    <p>ATR-IN-11, a potent ATR kinase inhibitor, shows promise as a lead for DNA damage response-targeted cancer drugs.</p>
    Formula:C25H30N6O2
    Color and Shape:Solid
    Molecular weight:446.54
  • Cemdomespib

    CAS:
    <p>Cemdomespib (KU-596) is a potent Hsp90 modulator with neuroprotective effects and can improve diabetic neuropathy.</p>
    Formula:C24H30FNO6
    Color and Shape:Solid
    Molecular weight:447.5
  • AMG-315

    CAS:
    <p>AMG-315: Chiral AEA analogue, potent CB1 agonist (Ki 7.8 nM, EC50 0.6 nM), stable against hydrolyzing/oxidative enzymes.</p>
    Formula:C24H41NO2
    Color and Shape:Solid
    Molecular weight:375.59
  • Aβ-IN-2


    <p>Aβ-IN-2 is a peptide inhibitor of Aβ1-42.</p>
    Formula:C37H51NO
    Color and Shape:Solid
    Molecular weight:525.81
  • (E)-10-Hydroxynortriptyline maleate

    CAS:
    <p>(E)-10-Hydroxy Nortriptyline maleate, a derivative of antidepressant Nortriptyline, eases depression symptoms.</p>
    Formula:C23H25NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:395.455
  • (-)-Adenophorine

    CAS:
    <p>(-)-Adenophorine is a moderate alpha-l-fucosidase inhibitor.</p>
    Formula:C8H17NO4
    Color and Shape:Solid
    Molecular weight:191.22
  • MK-7128

    CAS:
    <p>MK-7128 is a CB1 receptor inverse agonist.</p>
    Formula:C29H25ClF2N4O2
    Color and Shape:Solid
    Molecular weight:534.98
  • RS 61756-007

    CAS:
    <p>RS 61756-007 is a selective thromboxane receptor (TP) agonist.</p>
    Formula:C23H28O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:384.47
  • EB-0156


    <p>EB-0156: potent ER α-glucosidase inhibitor, IC50 of 0.0479/ &lt;0.001 μM, N-substituted valerian, broad-spectrum antiviral potential.</p>
    Formula:C21H32N6O7
    Color and Shape:Solid
    Molecular weight:480.51
  • MRTX-EX185


    <p>MRTX-EX185 inhibits GDP-KRAS/G12D; IC50=90 nM on G12D. It also binds GDP-HRAS.</p>
    Formula:C33H33FN6O2
    Color and Shape:Solid
    Molecular weight:564.65
  • Fosmanogepix

    CAS:
    Fosmanogepix (APX001) is a broad-spectrum oral antifungal that targets Gwt1 enzyme, transforming into active APX001A in the body.
    Formula:C22H21N4O6P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.40
  • AChE-IN-22


    <p>AChE-IN-22 (10q) selectively inhibits AChE (IC50: 0.88 μM), less on BuChE (IC50: 10 μM), targets CAS and PAS, useful in Alzheimer's research.</p>
    Formula:C21H20N4O5S
    Color and Shape:Solid
    Molecular weight:440.47
  • TRK-IN-19


    <p>TRK-IN-19 (I-10) inhibits TRKA (1.1 nM IC50) &amp; TRKAG595R (5.3 nM), promising for cancer research.</p>
    Formula:C22H26FN5O2
    Color and Shape:Solid
    Molecular weight:411.47
  • NusB-IN-1


    <p>NusB-IN-1 (22r) is an oral bacterial rRNA inhibitor, effective against MRSA and VRSA.</p>
    Formula:C21H16N2O3
    Color and Shape:Solid
    Molecular weight:344.36
  • HMG499

    CAS:
    <p>HMG499 inhibits HMG-CoA reductase (IC50: 0.41μM), reduces statin-induced HMGCR, lowers cholesterol, and lessens atherosclerosis.</p>
    Formula:C33H54O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.78
  • MtMetAP1-IN-1


    <p>MtMetAP1-IN-1 is an inhibitor of methionine aminopeptidase 1 ( MetAP1 ). MtMetAP1-IN-1 shows antimycobacterial activity.</p>
    Formula:C15H10BrN5O2S
    Color and Shape:Solid
    Molecular weight:404.24
  • PF-06815345 hydrochloride

    CAS:
    <p>PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.</p>
    Formula:C27H30Cl2FN9O4
    Color and Shape:Solid
    Molecular weight:634.49
  • Anticancer agent 30


    <p>Anticancer agent 30 (6f-Z), a 3-arylidene-2-oxindole, selectively inhibits CDK2, showing potent anticancer potential.</p>
    Formula:C22H15ClFNO
    Color and Shape:Solid
    Molecular weight:363.81
  • HBV-IN-20


    <p>HBV-IN-20 is a potent, orally active HBV inhibitor (EC50: 0.46 μM). HBV-IN-20 is a classical type II CpAM (core protein assembly regulator).</p>
    Color and Shape:Solid
  • Epothilone E

    CAS:
    <p>Epothilone E, a derivative of epothilone, functions by inhibiting microtubule protein activity, thereby halting cell division and exhibiting anti-tumor</p>
    Formula:C26H39NO7S
    Color and Shape:Solid
    Molecular weight:509.66
  • KP 10614

    CAS:
    <p>KP 10614 is a new prostacyclin analog that inhibits platelet-polymorphonuclear leukocyte interaction.</p>
    Formula:C23H32O4
    Color and Shape:Solid
    Molecular weight:372.50
  • ATP synthase inhibitor 2

    CAS:
    <p>ATP synthase inhibitor 2 blocks P. aeruginosa ATP synthase; IC50=10 μg/mL, fully inhibits at 128 μg/mL.</p>
    Formula:C21H22N2O3S
    Color and Shape:Solid
    Molecular weight:382.48
  • ARG1-IN-1

    CAS:
    ARG1-IN-1 is a human arginase 1 inhibitor with an IC 50 of 29 nM.
    Formula:C11H21BN2O4
    Color and Shape:Solid
    Molecular weight:256.11
  • T-Type calcium channel inhibitor 2


    <p>Compound 6g inhibits T-type Ca channels (IC50: Cav3.1-31μM, Cav3.2-83μM), cytotoxic to A549 (IC50: 5μM) &amp; HCT-116 cells (IC50: 6.4μM).</p>
    Formula:C36H39FN4OS
    Color and Shape:Solid
    Molecular weight:594.78
  • Salacinol

    CAS:
    <p>Salacinol is a naturally occurring alpha-glucosidase inhibitor isolated from an Ayurvedic traditional medicine Salacia reticulata.</p>
    Formula:C9H18O9S2
    Color and Shape:Solid
    Molecular weight:334.37
  • MDL-27788

    CAS:
    <p>MDL-27788 is a tricyclic inhibitor.</p>
    Formula:C24H26N2O5S
    Color and Shape:Solid
    Molecular weight:454.54
  • BW-10

    CAS:
    <p>BW-10 potently inhibits bombesin evoked release of gastrointestinal hormones in vitro and in vivo.</p>
    Formula:C57H72N14O8
    Color and Shape:Solid
    Molecular weight:1081.27
  • PD-1/PD-L1-IN-17


    <p>PD-1/PD-L1-IN-17 (Compound P20) is a potent PD-1/PD-L1 inhibitor (IC50: 26.8 nM).</p>
    Formula:C23H20ClN3O4
    Color and Shape:Solid
    Molecular weight:437.88
  • Ganciclovir monophosphonate

    CAS:
    <p>Ganciclovir monophosphate treats CMV, inhibiting replication in human/animal strains (IC50: 0.01μM).</p>
    Formula:C10H16N5O6P
    Color and Shape:Solid
    Molecular weight:333.24
  • UNC7467

    CAS:
    <p>UNC7467, potent IP6K2/1/6 inhibitor (4.9/8.9/1320 nM); lowers inositol pyrophosphates, minimal impact on other inositol phosphates; for obesity research.</p>
    Formula:C20H13NO3
    Purity:98.28% - 98.64%
    Color and Shape:Soild
    Molecular weight:315.32
  • Galectin-8-IN-1


    <p>Galectin-8-IN-1 selectively binds galectin-8N with 48 μM affinity, 15x more than galectin-3.</p>
    Formula:C16H18N2O6
    Color and Shape:Solid
    Molecular weight:334.32
  • WIN 66306

    CAS:
    <p>WIN 66306: Cyclic heptapeptide, blocks NK1/NK2 receptors, inhibits substance P-triggered contractions in guinea pig ileum.</p>
    Formula:C41H52N8O9
    Color and Shape:Solid
    Molecular weight:800.9
  • Antibacterial agent 63

    CAS:
    <p>Aztreonam-siderophore conjugate 63 is an antibacterial agent that exhibits efficacy against Gram-negative bacteria through the linkage of aztreonam to a</p>
    Formula:C35H43N9O14S2
    Color and Shape:Solid
    Molecular weight:877.9
  • Symplostatin 1

    CAS:
    <p>Symplostatin 1 is a dolastatin 10 analog from the marine cyanobacterium Symploca hydnoides.</p>
    Formula:C43H70N6O6S
    Color and Shape:Solid
    Molecular weight:799.12
  • RdRP-IN-5

    CAS:
    <p>RdRP-IN-5 (compound 20), a potent inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), has potential application in influenza research [1].</p>
    Formula:C23H21N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:419.43
  • J-113397

    CAS:
    J-113397 is a potent and selective NOP receptor antagonist (IC50 = 2.3 nM).
    Formula:C24H37N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.57
  • ZIKV-IN-4


    <p>ZIKV-IN-4 is a low cytotoxic, acid-stable anti-ZIKV agent with an EC50 value of 3.49 μM. ZIKV-IN-4 exhibited potent inhibition of ZIKV NS5 MTase.</p>
    Formula:C33H37NO4
    Color and Shape:Solid
    Molecular weight:511.65
  • WQ3810

    CAS:
    <p>WQ3810 is an orally active fluoroquinolone, has potent antibacterial activities.</p>
    Formula:C22H22F3N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:461.44
  • L 668750

    CAS:
    <p>L 668750 is an inhibitor of platelet-activating factor.</p>
    Formula:C25H34O9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.6
  • MY-875


    <p>MY-875 inhibits microtubule formation, binds like colchicine (IC50: 0.92 μM), activates Hippo pathway, and induces apoptosis with anticancer properties.</p>
    Formula:C21H25NO6
    Color and Shape:Solid
    Molecular weight:387.43
  • DNA-PK-IN-2

    CAS:
    <p>DNA-PK-IN-2 is an inhibitor of the DNA-PK enzyme complex, useful in cancer research.</p>
    Formula:C20H23N5O3
    Color and Shape:Solid
    Molecular weight:381.43
  • AVE-1330A sodium

    CAS:
    <p>AVE-1330A sodium is a beta-Lactamase inhibitor.</p>
    Formula:C7H10N3NaO6S
    Color and Shape:Solid
    Molecular weight:287.23
  • GRPR antagonist-2


    <p>GRPR antagonist-2 blocks GRPR, kills some cancer cells, effective on HGC-27 (IC50: 0.77 μM) &amp; Pan02 (IC50: 2.5 μM).</p>
    Formula:C28H32F3N5O4
    Color and Shape:Solid
    Molecular weight:559.58
  • KC-11404

    CAS:
    <p>KC-11404 is an LTB4 inhibitor for the treatment of b-cell leukemias and lymphomas, potently inhibiting histamine, platelet activating factor and 5-lipoxygenase.</p>
    Formula:C28H38N4O
    Color and Shape:Solid
    Molecular weight:446.63
  • Saprisartan potassium

    CAS:
    <p>Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.</p>
    Formula:C25H21BrF3KN4O4S
    Color and Shape:Solid
    Molecular weight:649.52
  • CHF-6366

    CAS:
    <p>CHF-6366: M3 antagonist &amp; β2 agonist (pKi 10.4/11.4), mild Ca channel blocker, used in COPD study.</p>
    Formula:C42H48N6O8
    Color and Shape:Solid
    Molecular weight:764.87
  • BMS 310705

    CAS:
    <p>BMS 310705, an Epothilone B analog, targets ovarian/renal/bladder/lung cancer, inducing apoptosis via mitochondria.</p>
    Formula:C27H42N2O6S
    Color and Shape:Solid
    Molecular weight:522.70
  • Kahweol Acetate

    CAS:
    <p>Kahweol Acetate, a semi-synthetic coffee bean derivative, inhibits osteoclasts, cancer cells, DNA damage, and oxidative stress.</p>
    Formula:C22H28O4
    Color and Shape:Solid
    Molecular weight:356.46
  • Cacospongionolide B

    CAS:
    <p>Cacospongionolide B from Fasciospongia cavernosa inhibits secretory phospholipase A2, curbing inflammation.</p>
    Formula:C25H36O4
    Color and Shape:Solid
    Molecular weight:400.55
  • MEIS-IN-1

    CAS:
    <p>MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.</p>
    Formula:C24H21F3N2O4
    Color and Shape:Solid
    Molecular weight:458.43
  • Antibacterial agent 99

    CAS:
    <p>Compound 7b (Antibacterial agent 99) is an effective agent with antibacterial, antifungal properties and no haemolytic activity.</p>
    Formula:C27H27BrN2
    Color and Shape:Solid
    Molecular weight:459.42
  • BAY-091

    CAS:
    <p>BAY-091 is a novel potent and highly selective PIP4K2A kinase inhibitor.</p>
    Formula:C26H21FN4O2
    Purity:97.66% - 99.23%
    Color and Shape:Soild
    Molecular weight:440.47
  • MB-07344 sodium


    <p>"MB-07344 sodium is a TR-β agonist with a 2.17 nM Ki, boosts Atorvastatin's cholesterol-lowering effects in various animals."</p>
    Formula:C19H25NaO5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:387.36
  • Latrunculins A

    CAS:
    Latrunculins A is a novel marine toxin, disrupts microfilament organization in cultured cells.
    Formula:C22H31NO6S
    Color and Shape:Solid
    Molecular weight:437.55
  • Pociredir

    CAS:
    <p>Pociredir (FTX-6058), a potent EED inhibitor (KD=0.163 nM), may help in SCD research.</p>
    Formula:C22H18FN5O2
    Color and Shape:Solid
    Molecular weight:403.41
  • Massarilactone H

    CAS:
    <p>Massarilactone H, a polyketide, is a neuraminidase inhibitor, with an IC 50 of 8.18 µM .</p>
    Formula:C11H12O5
    Color and Shape:Solid
    Molecular weight:224.21
  • Karenitecin

    CAS:
    <p>Karenitecin (Cositecan) is an inhibitor of topoisomerase I. It has potent anti-cancer activity.</p>
    Formula:C25H28N2O4Si
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.59
  • Rivenprost

    CAS:
    <p>Rivenprost, selective EP4 agonist (Ki: 0.7 nM), promotes bone growth, osteoblast differentiation, and aids wound healing.</p>
    Formula:C24H34O6S
    Color and Shape:Solid
    Molecular weight:450.59
  • Antiviral agent 6


    <p>Antiviral agent 6 showed excellent anti-TSWV effects in vivo (EC50: 188 mg/L).</p>
    Formula:C23H27BrN2O3S2
    Color and Shape:Solid
    Molecular weight:523.51
  • PptT-IN-2


    <p>PptT-IN-2 inhibits PptT enzyme crucial in tuberculosis, with 2.5 μM IC50, showing potential in TB research.</p>
    Formula:C22H29N5O2
    Color and Shape:Solid
    Molecular weight:395.5
  • PF-9404C

    CAS:
    <p>PF-9404C: S-S diastereoisomer, beta-blocker with vasodilation, boosts cyclic GMP in rat aorta cells from 3 to 53 pmol/mg protein.</p>
    Formula:C16H25N3O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:403.38
  • 5-HT1A antagonist 1


    <p>Compound 6f is a potent, selective 5-HT1A receptor blocker (Ki: 35 nM), useful in CNS disorder research.</p>
    Formula:C23H29ClN6O2
    Color and Shape:Solid
    Molecular weight:456.97
  • K252d

    CAS:
    <p>K252d: indolocarbazole alkaloid in Nocardiopsis; inhibits PKC in rat brain and bovine heart phosphodiesterase.</p>
    Formula:C26H23N3O5
    Color and Shape:Solid
    Molecular weight:457.48
  • Tazide


    <p>Tazide is an antitumor agent [1].</p>
    Formula:C12H16N4O
    Color and Shape:Solid
    Molecular weight:232.28
  • TGR5 Receptor Agonist 3

    CAS:
    <p>TGR5 Receptor Agonist 3 is a GPBAR1 agonist with EC50 of 16.4 nM (hTGR5) &amp; 209 nM (mTGR5), ensures gallbladder safety and reduces filling.</p>
    Formula:C29H27N3O6
    Color and Shape:Solid
    Molecular weight:513.54
  • 14α-Demethylase/DNA Gyrase-IN-1


    14α-Demethylase/DNA Gyrase-IN-1 (Compound 7c) is a potent inhibitor of 14α-Demethylase/DNA Gyrase with antibacterial activity.
    Formula:C26H22N4O4
    Color and Shape:Solid
    Molecular weight:454.48
  • LP-284

    CAS:
    <p>LP-284 is a DNA alkylating agent effective against solid tumors and hematologic cancers like MCL.</p>
    Formula:C16H20N2O4
    Color and Shape:Solid
    Molecular weight:304.34
  • EED ligand 1


    <p>EED ligand 1: potent PRC2 inhibitor targeting EED subunit.</p>
    Formula:C19H19FN8O
    Color and Shape:Solid
    Molecular weight:394.41
  • SH498

    CAS:
    <p>SH498 is a novel Bmi-1-mediated anti-tumor agent with significant anti-proliferative effects.</p>
    Formula:C27H25F3N2O4
    Color and Shape:Solid
    Molecular weight:498.49
  • SC13

    CAS:
    <p>SC13, a novel mitragynine analog, exhibits low-efficacy agonism at Mu opioid receptors and provides antinociception while minimizing adverse effects.</p>
    Formula:C26H30N2O5
    Color and Shape:Solid
    Molecular weight:450.53
  • SML-10-70-1

    CAS:
    <p>SML-10-70-1 is a Novel Active Site Inhibitor of Oncogenic K-Ras G12C.</p>
    Formula:C25H42ClN7O13P2
    Color and Shape:Solid
    Molecular weight:746.04
  • MsbA-IN-2


    <p>MsbA-IN-2 is a potent inhibitor of the lipopolysaccharide transporter MsbA and is able to act on E. coli MsbA (IC50: 2 nM).</p>
    Formula:C23H19Cl2NO3
    Color and Shape:Solid
    Molecular weight:428.31
  • CB2 receptor antagonist 1

    CAS:
    <p>Compound 29 is a potent, CB2-selective antagonist/reverse agonist. Derivatives 23 &amp; 24 offer antinociception; 24 activates cannabinoid/TRPV1 receptors.</p>
    Formula:C28H47NO3
    Color and Shape:Solid
    Molecular weight:445.68
  • IRE1α kinase-IN-4

    CAS:
    <p>IRE1α kinase-IN-4 (compound 6) is a potent inhibitor of IRE1α, exhibiting a Ki value of 140 nM. It acts as an ATP-competitive ligand for IRE1α [1].</p>
    Formula:C29H31N7O2
    Color and Shape:Solid
    Molecular weight:509.6
  • Mifepristone methochloride

    CAS:
    <p>Mifepristone methochloride is a glucocorticoid antagonist. This product will be sold for research use only.</p>
    Formula:C30H38ClNO2
    Color and Shape:Solid
    Molecular weight:480.08
  • LSD1-IN-13 hydrochloride

    CAS:
    <p>LSD1-IN-13 hydrochloride (7e) is an oral LSD1 inhibitor (IC50: 24.43 nM), promoting differentiation in AML cell lines.</p>
    Formula:C23H30ClN3O2S
    Color and Shape:Solid
    Molecular weight:448.02
  • Antibacterial agent 110


    <p>Compound 4e, an antibacterial against P. aeruginosa, disrupts cell membranes (MIC: 1 μg/ml).</p>
    Formula:C22H21N5O4S
    Color and Shape:Solid
    Molecular weight:451.5
  • Antibacterial agent 80


    <p>Antibacterial agent 80 (compound 20) has antibacterial activity [1].</p>
    Formula:C14H21N3S2
    Color and Shape:Solid
    Molecular weight:295.47
  • Dictyostatin

    CAS:
    <p>Dictyostatin: potent microtubule stabilizer &amp; anticancer agent with antiproliferative effects; researched for tauopathies.</p>
    Formula:C32H52O6
    Color and Shape:Solid
    Molecular weight:532.75
  • Leukotriene F-4 sulfone

    CAS:
    <p>Leukotriene F-4 sulfone induces vascular permeability changes.</p>
    Formula:C28H44N2O10S
    Color and Shape:Solid
    Molecular weight:600.72
  • ORP-101

    CAS:
    <p>ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.</p>
    Formula:C60H84N2O8
    Color and Shape:Solid
    Molecular weight:961.32
  • Irinotecan Carboxylate Sodium Salt

    CAS:
    <p>Irinotecan Carboxylate Sodium Salt is a DNA topoisomerase inhibitor.</p>
    Formula:C33H39N4NaO7
    Color and Shape:Solid
    Molecular weight:626.68
  • Terguride

    CAS:
    <p>Terguride: treats hyperprolactinemia, blocks 5-HT2A/B, activates dopamine receptors, studied for PAH.</p>
    Formula:C20H28N4O
    Color and Shape:Solid
    Molecular weight:340.46
  • RhlR antagonist 1


    <p>RhlR antagonist 1: IC50 of 26 μM, selective for RhlR, inhibits P. aeruginosa biofilm and virulence factors.</p>
    Formula:C12H10F2O
    Color and Shape:Solid
    Molecular weight:208.2
  • CM-414

    CAS:
    <p>CM-414: HDAC/PDE5 inhibitor, targeting Alzheimer’s, IC50s: PDE5 (60 nM), HDAC1/2/3/6. Reduces Aβ, pTau in mice, boosts cognition.</p>
    Formula:C23H29N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:439.51
  • PF-00489791

    CAS:
    <p>PF-00489791 (PF4634817) is a long-acting PDE5 inhibitor with hypotensive activity for the study of diabetic nephropathy.</p>
    Formula:C20H28N8O4S
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:476.55
  • Tarloxotinib bromide

    CAS:
    Tarloxotinib bromide (TH-4000) is an irreversible inhibitor of EGFR/HER2.
    Formula:C24H24Br2ClN9O3
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:681.77
  • ODN 2088

    CAS:
    <p>ODN 2088 is a potent inhibitor of TLR3, TLR7 and TLR9 that is non-cytotoxic and shows inhibition of the release of IFN-α and IL-6.</p>
    Color and Shape:Solid
  • Guraxetan


    <p>Guraxetan can be used in the synthesis of the antitumour drug Lutetium (177Lu) zadavotide Guraxetan.</p>
    Formula:C20H34N4O9
    Color and Shape:Solid
    Molecular weight:474.51
  • Dihydrophaseic acid

    CAS:
    <p>Dihydrophaseic acid 3'-O-b-D-glucopyranoside (D3G) can increase the proliferation and differentiation of osteoblast cells and enhance bone formation, suggests</p>
    Formula:C15H22O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:282.33
  • Vindeburnol

    CAS:
    <p>Vindeburnol is a cerebral vasodilator vincamine analog that bears neuroprotective properties.</p>
    Formula:C17H20N2O
    Color and Shape:Solid
    Molecular weight:268.35
  • Elacestrant S enantiomer dihydrochloride


    <p>Elacestrant (RAD1901) dihydrochloride, an oral ERR degrader, has IC50 of 48 nM (ERα) and 870 nM (ERβ). Its S enantiomer has low activity.</p>
    Formula:C30H40Cl2N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.56
  • hAChE/Aβ1-42-IN-1

    CAS:
    <p>Compound 16 (hAChE/Aβ1-42-IN-1) is a potent inhibitor targeting both hAChE and Aβ1-42 aggregation, demonstrating considerable safety in hepG2 cell lines and</p>
    Formula:C20H24N6O
    Color and Shape:Solid
    Molecular weight:364.44