
Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,542 products)
- Apoptosis(5,816 products)
- Cell Cycle/Checkpoint(4,466 products)
- Chromatin/Epigenetics(2,252 products)
- Cytoskeletal Signaling(1,381 products)
- DNA Damage/DNA Repair(2,830 products)
- Endocrinology/Hormones(3,518 products)
- Enzyme(3,640 products)
- GPCR/G-Protein(8,362 products)
- Immunology and Inflammation(3,540 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(405 products)
- MAPK Signaling(1,201 products)
- Membrane Transporter/Ion Channel(2,809 products)
- Metabolism(9,462 products)
- Microbiology/Virology(7,003 products)
- Neuroscience(9,942 products)
- Other Inhibitors(37,827 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,399 products)
- Proteases/Proteasome(1,598 products)
- Stem Cell and Derivatives(830 products)
- Tyrosine Kinase/Adaptors(2,012 products)
- Ubiquitination(1,651 products)
Show 16 more subcategories
Found 66618 products of "Inhibitors"
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Gemilukast
CAS:<p>Gemilukast (ONO-6950) is a cysteinyl leukotriene 1 and 2 receptor inhibitor that inhibits bronchoconstriction and is used in the treatment of asthma.</p>Formula:C36H37F2NO5Purity:98.27% - 99.5%Color and Shape:SolidMolecular weight:601.68PIM-1/HDAC-IN-1
<p>PIM-1/HDAC-IN-1 (4d): inhibits PIM-1 (IC50: 343.87nM), HDAC1 (63.65nM), HDAC6 (62.39nM); induces apoptosis in MCF-7 cells.</p>Formula:C22H19N3O3Color and Shape:SolidMolecular weight:373.4CXCR2 antagonist 6
<p>CXCR2 antagonist 6: strong CXCR2 affinity (IC50=0.044 μM), hinders calcium mobilization (IC50=0.66 μM).</p>Formula:C17H16F2N4OSColor and Shape:SolidMolecular weight:362.4RSV-IN-5
CAS:<p>RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM & 8.1 nM. Potent anti-RSV.</p>Formula:C28H37N7O2Color and Shape:SolidMolecular weight:503.64PARP1-IN-5
<p>PARP1-IN-5 is a potent, selective, orally active, low-toxicity PARP-1 inhibitor with an IC50 value of 14.7 nM. PARP1-IN-5 can be used in cancer research.</p>Formula:C25H24N2O5SColor and Shape:SolidMolecular weight:464.53Y1 receptor antagonist 1
CAS:<p>Y1 receptor antagonist 1 is an antagonist of neuropeptide Y1 receptor.</p>Formula:C28H33N5O3Purity:98.17%Color and Shape:SolidMolecular weight:487.59Silvestrol
CAS:<p>Silvestrol is a eukaryotic translation initiation factor 4A inhibitor. Silvestrol causes autophagy and caspase-mediated apoptosis.</p>Formula:C34H38O13Purity:98%Color and Shape:SolidMolecular weight:654.66GP-1681
CAS:<p>GP-1681, a G-protein coupled receptor (GPCR) agonist, is used potentially for the treatment of influenza infection.</p>Formula:C24H30NaO5Purity:98%Color and Shape:SolidMolecular weight:421.48LY 235959
CAS:<p>LY 235959 is a NMDA receptor antagonist.</p>Formula:C11H20NO5PPurity:98%Color and Shape:SolidMolecular weight:277.25S100A2-p53-IN-1
CAS:<p>S100A2-p53-IN-1 inhibits S100A2-p53 in pancreatic cancer, stunting MiaPaCa-2 cell growth at 1.2-3.4 μM.</p>Formula:C20H20F6N2O4SColor and Shape:SolidMolecular weight:498.44AZD 4407
CAS:<p>AZD 4407 is a potent inhibitor of 5-lipoxygenase.</p>Formula:C19H21NO3S2Purity:98%Color and Shape:SolidMolecular weight:375.5CGS 22652
CAS:<p>CGS 22652 has thromboxane receptor antagonism combined with thromboxane synthase inhibition.</p>Formula:C22H29ClN2O4SColor and Shape:SolidMolecular weight:452.99Dup-714
CAS:<p>Dup-714 is a thrombin inhibitor.</p>Formula:C21H33BN6O5Purity:98%Color and Shape:SolidMolecular weight:460.33(-)-Cevimeline hydrochloride hemihydrate
<p>(-)-Cevimeline HCl hemihydrate, a muscarinic agonist, treats Sjogren's xerostomia. Quick absorption, species-dependent metabolism.</p>Formula:C10H19ClNO1·5SPurity:98%Color and Shape:SolidMolecular weight:244.78P2X receptor-1
<p>P2X receptor-1 is a potential inhibitor of P2X receptor for the treatment of pain and inflammation.</p>Formula:C14H14ClN3O3S2Color and Shape:SolidMolecular weight:371.86Deleobuvir
CAS:<p>Deleobuvir(BI207127) is an inhibitor of non-nucleoside hepatitis C virus NS5B polymerase for the treatment of hepatitis C.</p>Formula:C34H33BrN6O3Color and Shape:SolidMolecular weight:653.57BMS-986143
CAS:<p>BMS-986143: oral BTK inhibitor, IC50=0.26 nM, potential for autoimmune research, also targets TEC, BLK, BMX, TXK, YES1, ITK.</p>Formula:C31H24Cl2N4O4Color and Shape:SolidMolecular weight:587.45Cap-dependent endonuclease-IN-17
CAS:<p>CEN inhibitor IN-17 targets influenza A/H3N2; IC50: 1.29 μM. From patent CN112898346A, DSC701.</p>Formula:C24H20F2N3O7PSColor and Shape:SolidMolecular weight:563.47Tubulin polymerization-IN-35
<p>Tubulin-IN-35 inhibits oxazolylisoindole microtubule formation, targeting VL51 marginal zone lymphoma.</p>Formula:C31H35N3O5Color and Shape:SolidMolecular weight:529.63MAFP
CAS:MAFP (Methyl Arachidonyl Fluorophosphonate) is an effective irreversible inhibitor of anandamide amidase.Formula:C21H36FO2PColor and Shape:SolidMolecular weight:370.48UH 301
CAS:<p>UH 301 is a 5-HT1A receptor antagonist.</p>Formula:C16H24FNOColor and Shape:SolidMolecular weight:265.37Carbonic anhydrase inhibitor 2
CAS:<p>Compound 7c inhibits carbonic anhydrase II, lowering intraocular pressure in glaucomatous rabbits.</p>Formula:C12H16N4O6SColor and Shape:SolidMolecular weight:344.342R,4S-Sacubitril
CAS:<p>2R,4S-Sacubitril (Sacubitril Enantiomer) is the impurity of Sacubitril which is a neprilysin inhibitor.</p>Formula:C24H28NO51CaPurity:98%Color and Shape:SolidMolecular weight:430.49FGFR4-IN-10
<p>FGFR4-IN-10 (compound 5a) is a potent, selective FGFR4 inhibitor with IC50 of 70.7 nM, sparing FGFR1-3.</p>Formula:C20H19F3N6O3Color and Shape:SolidMolecular weight:448.4Spicamycin
CAS:<p>Spicamycin can be used as a potent inducer of differentiation of human myeloid leukemia cells (HL-60) and murine myeloid leukemia cells (M1).</p>Formula:C30H51N7O7Color and Shape:SolidMolecular weight:621.77Keap1-Nrf2-IN-4
<p>Keap1-Nrf2-IN-4 hinders MGC-803 cell growth (IC50=2.55μM), migration, and induces apoptosis with low toxicity.</p>Formula:C26H34N2OColor and Shape:SolidMolecular weight:390.56Arterolane
CAS:<p>Arterolane is an antimalarial compound. For against P. falciparum Ro73 and W2, the IC50s are both 1.1 nM.</p>Formula:C22H36N2O4Color and Shape:SolidMolecular weight:392.53Cilazapril HCl
CAS:<p>Cilazapril, also known as Ro 31 2848, is a potent ACE inhibitor used for hypertension.</p>Formula:C22H32ClN3O5Color and Shape:SolidMolecular weight:453.96Tubulin polymerization-IN-33
<p>Tubulin-IN-33, an oxazoloisoindole, hinders microtubule assembly; effective against NCI cancer cells.</p>Formula:C27H28N2O6Color and Shape:SolidMolecular weight:476.52PD 136450
CAS:<p>PD-136,450: partial stomach secretory agonist, full pancreas agonist in rats; potential acid-reducing drug, adjuvant for gastrin-sensitive tumors.</p>Formula:C35H40N4O6Purity:98%Color and Shape:SolidMolecular weight:612.72Luffariellolide
CAS:<p>Luffariellolide is a terpene compound obtained from the marine sponge Hyrtios communis that is an HSF-PLA2 inhibitor and a RAR agonist.</p>Formula:C25H38O3Purity:98%Color and Shape:SolidMolecular weight:386.57I-BET282E
<p>I-BET282E inhibits eight BET bromodomains (pIC50 6.4-7.7) with selectivity for other bromodomain proteins.</p>Formula:C26H34N4O7SColor and Shape:SolidMolecular weight:546.64β-Glucuronidase/hCAII-IN-2
<p>β-Glucuronidase/hCAII-IN-2 is a potent inhibitor of β-glucuronidase and hCA II, and their IC50 values were 670.7 μM and 21.77 μM, respectively.</p>Formula:C31H23NO8Color and Shape:SolidMolecular weight:537.52NS2B/NS3-IN-3
CAS:<p>NS2B/NS3-IN-3 (Compd 66) is an inhibitor of Flavivirus NS2B-NS3 protease [1] .</p>Formula:C19H21N3O2Color and Shape:SolidMolecular weight:323.39STING agonist-7
<p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>Formula:C17H12N4O4Color and Shape:SolidMolecular weight:336.3AX15910
<p>AX15910 is a potent inhibitor of BRD4 and ERK5.</p>Formula:C32H38N6O3Color and Shape:SolidMolecular weight:554.7CK2-IN-3
<p>CK2-IN-3: potent, selective CK2 inhibitor; Kd=12 nM, IC50: 1.51 μM (CK2α), 7.64 μM (CK2α'). For cancer research.</p>Formula:C22H26N4O7Color and Shape:SolidMolecular weight:458.46DLK-IN-1
CAS:DLK-IN-1: Oral DLK (MAP3K12) inhibitor, Ki=3nM, effective in Alzheimer's model, CNS permeable, well-tolerated with sustained brain levels.Formula:C20H24F3N5O2Color and Shape:SolidMolecular weight:423.43XIAP/cIAP1 antagonist-1
<p>Potent oral XIAP/cIAP1 inhibitor with EC50s: XIAP 5.1 nM, cIAP1 0.32 nM; curbs tumor growth in vivo.</p>Color and Shape:SolidSR121566A
CAS:SR121566A is a novel non-peptide antagonist of Glycoprotein IIb/IIIa (GP IIb-IIIa).Formula:C20H25N5O4SPurity:98%Color and Shape:SolidMolecular weight:431.51J-104132
CAS:<p>J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.</p>Formula:C31H33NO7Purity:98%Color and Shape:SolidMolecular weight:531.60NCATS-SM4487
CAS:<p>NCATS-SM4487 is a highly selective inhibitor of GALK1 (IC50: 0.05 μM).</p>Formula:C25H24ClFN8O2Color and Shape:SolidMolecular weight:522.96FLT3-IN-13
<p>FLT3-IN-13 inhibits topoisomerase II/FLT3 in leukemia with IC50 of 2.26 μM, causes G2/M arrest, and promotes apoptosis.</p>Formula:C20H14N4O2Color and Shape:SolidMolecular weight:342.35PARP-1-IN-1
<p>PARP-1-IN-1: Selective, oral PARP-1 inhibitor with 0.96 nM IC50; well-tolerated and effective in single-dose MDA-MB-436 model.</p>Formula:C23H25FN4OColor and Shape:SolidMolecular weight:392.47PPARγ agonist 2
<p>PPARγ agonist 2 is a highly effective compound that acts as a partial agonist for PPARγ.</p>Formula:C24H20O5Color and Shape:SolidMolecular weight:388.41GSK945237
CAS:<p>GSK945237 is a type IIA topoisomerase inhibitor, effective on Gram-positive and negative bacteria, with favorable pharmacokinetics and in vivo efficacy.</p>Formula:C24H26FN5O3Color and Shape:SolidMolecular weight:451.49Dyrk1A-IN-1
<p>Dyrk1A-IN-1 is a triple inhibitor of Dyrk1A kinase activity, aggregation of tau and α-syn oligomers, with an IC50 value of 119 nM for Dyrk1A kinase.</p>Formula:C23H20N4O3SColor and Shape:SolidMolecular weight:432.49PF-06380101
CAS:<p>PF-06380101, a potent auristatin analog and Dolastatin 10 derivative, shows strong anti-tumor activity and unique ADME attributes.</p>Formula:C39H62N6O6SPurity:98%Color and Shape:SolidMolecular weight:743.01KT2-962
CAS:<p>KT2-962 is a TXA2/prostaglandin endoperoxide receptor antagonist.</p>Formula:C23H27ClNNaO5S2Color and Shape:SolidMolecular weight:520.04Carmegliptin dihydrochloride
CAS:<p>Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.</p>Formula:C20H30Cl2FN3O3Color and Shape:SolidMolecular weight:450.38[D-Leu-4]-OB3
CAS:[D-Leu-4]-OB3 suppresses the expression of genes associated with inflammation, proliferation, and metastasis, as well as the expression of PD-L1.Formula:C29H50N8O12SColor and Shape:SolidMolecular weight:734.82HIF-1/2α-IN-1
<p>HIF-1/2α-IN-1, an orally active compound, functions as an inhibitor of HIF-2α.</p>Formula:C17H16N6O4Color and Shape:SolidMolecular weight:368.35Antifungal agent 16
<p>Antifungal agent 16 has antimicrobial activity comparable to that of ciprofloxacin and has higher antifungal activity than fluconazole.</p>Formula:C27H21N5O2SColor and Shape:SolidMolecular weight:479.55Netupitant metabolite Monohydroxy Netupitant
CAS:Monohydroxy Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.Formula:C30H32F6N4O2Purity:98%Color and Shape:SolidMolecular weight:594.59Mesulergine hydrochloride
CAS:<p>5-HT2A and 2C receptor antagonist</p>Formula:C18H27ClN4O2SPurity:98%Color and Shape:SolidMolecular weight:398.95Fandosentan
CAS:<p>Fandosentan is an endothelin receptor antagonist.</p>Formula:C25H18F3NO6SColor and Shape:SolidMolecular weight:517.47BMS-986118
CAS:BMS-986118 is a GPR40 full agonist targeting type II diabetes, prompting insulin release without hypoglycemia risk.Formula:C25H28ClF3N4O4Purity:98%Color and Shape:SolidMolecular weight:540.96NLRP3/AIM2-IN-1
<p>NLRP3/AIM2-IN-1 is an inhibitor of thermal sepsis (IC50 = 3.136 ± 0.7667 μM).</p>Formula:C15H16BNO4Color and Shape:SolidMolecular weight:285.1SHP2 IN-1
CAS:<p>SHP2 IN-1 is an allergic SHP2 (PTPN11) inhibitor(IC50 : 3 nM).</p>Formula:C18H22Cl2N6OSPurity:98%Color and Shape:SolidMolecular weight:441.38LSD1-IN-16
<p>LSD1-IN-16 (4b) inhibits LSD1, MAO-A/B; IC50: 0.015-0.366 μM. Halts prostate cancer cell growth; IC50: 15.2 μM.</p>Formula:C20H18N2OSColor and Shape:SolidMolecular weight:334.43HDAC6-IN-9
CAS:<p>HDAC6-IN-9 is a γ-secretase modulator that can significantly reduce the level of Aβ42 in mouse brain and can be used to study neurological diseases.</p>Formula:C19H16N2O3Purity:98.84%Color and Shape:SolidMolecular weight:320.34DYRK1-IN-1
CAS:<p>DYRK1-IN-1: Selective DYRK1A inhibitor with IC50 of 220 nM, good permeability, CNS penetrant for research, no P-glycoprotein issues.</p>Formula:C12H12N6Color and Shape:SolidMolecular weight:240.26SARS 3CLpro-IN-1
CAS:<p>SARS 3CLpro-IN-1: stereospecific SARS 3CL protease inhibitor, octahydroisochromene class, IC50 = 95 μM.</p>Formula:C22H38N4O2Color and Shape:SolidMolecular weight:390.56VEGFR-2-IN-11
<p>VEGFR-2-IN-11 is a potent inhibitor of VEGFR-2 (IC50: 60.27 nM) with an IC50 value of 60.27 nM, which induces apoptosis and has anticancer activity.</p>Formula:C29H22BrN5SColor and Shape:SolidMolecular weight:552.49Irinotecan Carboxylate Sodium Salt
CAS:<p>Irinotecan Carboxylate Sodium Salt is a DNA topoisomerase inhibitor.</p>Formula:C33H39N4NaO7Color and Shape:SolidMolecular weight:626.68CBP/p300-IN-16
<p>CBP/p300-IN-16 (compound 1) is a potent inhibitor of EP300/CBP HAT, acting on HAT EP300 (IC50: 0.61 μM) and LK2 H3K27 (IC50: 2.24 μM).</p>Formula:C26H31N3O4Color and Shape:SolidMolecular weight:449.54CDK4-IN-1
CAS:<p>CDK4 inhibitor is a novel and specific CDK4/Cyclin D1 inhibitor with an IC50 of 10 nM; 1500 and 500 fold than CDK1/Cyclin B (IC50>15 uM) and CDK2/Cyclin A (IC50</p>Formula:C22H29ClN8Purity:98%Color and Shape:SolidMolecular weight:440.97(R)-CSN5i-3
CAS:<p>(R)-CSN5i-3 is CSN5i-3 of the R configuration.</p>Formula:C28H29F2N5O2Purity:99.76% - 99.97%Color and Shape:SolidMolecular weight:505.56Rodatristat
CAS:<p>Rodatristat is an effective tryptophan hydroxylase 1 and TPH2 inhibitor (IC50s: 33 nM and 7 nM, respectively).</p>Formula:C27H27ClF3N5O3Purity:98%Color and Shape:SolidMolecular weight:561.98TAS05567
CAS:<p>TAS05567 is a potent, highly selective, and ATP-competitive Syk inhibitor (IC50: 0.37 nM).</p>Formula:C21H29N9O2Purity:98%Color and Shape:SolidMolecular weight:439.51Nafarelin acetate hydrate
CAS:<p>Nafarelin: a GnRH agonist used to treat endometriosis, precocious puberty, and control IVF. Delivered as a nasal spray. Marketed as Synarel by Pfizer.</p>Formula:C66H83N17O13·xC2H4O2·xH2OColor and Shape:SolidMolecular weight:1400.563ROPA
CAS:<p>ROPA, a potent PKCalpha and PKCgamma activator, promotes tumor growth through PKC-activation.</p>Formula:C28H32O6Purity:98%Color and Shape:SolidMolecular weight:464.55Minnelide
CAS:Minnelide is a prodrug of triptolide,and shows potent antitumor activity in a number of tumor types.Formula:C21H25Na2O10PPurity:98.49% - 99.59%Color and Shape:SolidMolecular weight:514.37Sulprostone
CAS:<p>EP3 and EP1 receptor agonist</p>Formula:C23H31NO7SPurity:98%Color and Shape:White To Off-White SolidMolecular weight:465.56HDAC-IN-34
<p>HDAC-IN-34 inhibits HDAC1 (IC50: 0.022 μM) & HDAC6 (IC50: 0.45 μM), binds DNA causing damage, and halts HCT-116 cell growth (IC50: 1.41 μM).</p>Formula:C24H26N6O3Color and Shape:SolidMolecular weight:446.5SGE-516
CAS:<p>SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.</p>Formula:C23H35N3O2Purity:98%Color and Shape:SolidMolecular weight:385.54AZD0424
CAS:<p>AZD0424: oral Src/Abl kinase inhibitor; potential anticancer; induces apoptosis, cell cycle arrest in lymphoma.</p>Formula:C25H29ClN6O5Purity:98%Color and Shape:SolidMolecular weight:528.99Rezatapopt
CAS:<p>Rezatapopt (PC14586) is a p53 reactivator with antitumor activity for the study of locally advanced or metastatic solid tumors.</p>Formula:C28H31F4N5O2Purity:98.12%Color and Shape:SolidMolecular weight:545.57CDK2-IN-9
<p>CDK2-IN-9: potent CDK2 inhibitor (IC50: 0.63 μM), anti-proliferative, arrests S/G2M cell cycle, induces apoptosis, promising for melanoma study.</p>Formula:C21H16ClN3O4SColor and Shape:SolidMolecular weight:441.89SSR-182289A (Free)
CAS:SSR-182289A (Free) is a thrombin inhibitor.Formula:C30H33F2N5O4SPurity:98%Color and Shape:SolidMolecular weight:597.68KT5926
CAS:<p>KT5926 selectively inhibits myosin light chain kinase and NGF-dependent neurite growth; it's a K-252a analogue.</p>Formula:C30H27N3O6Purity:98%Color and Shape:SolidMolecular weight:525.55LY 245769
CAS:<p>LY 245769 is an inhibitor of leukotriene E4 (LTE4).</p>Formula:C25H33F3N8OSPurity:98%Color and Shape:SolidMolecular weight:550.64CTX-712
CAS:<p>CTX-712 is a potent inhibitor of cdc2-like kinase ( CLK ). CTX-712 inhibits inhibits cancer survival and cancer cell growth.</p>Formula:C19H17FN8O2Color and Shape:SolidMolecular weight:408.39Antitumor agent-42
<p>Antitumor agent-42 inhibits microtubule multimerisation and NO release, exhibiting anti-angiogenic, colony-forming and apoptosis-inducing effects.</p>Formula:C24H19BrN2O8SColor and Shape:SolidMolecular weight:575.39hCAII-IN-4
CAS:hCAII-IN-4 (Compound 12j) is a potent inhibitor of human carbonic anhydrase II (hCA II), exhibiting an inhibitory concentration (IC50) of 7.78 μM.Formula:C31H23NO9Color and Shape:SolidMolecular weight:553.52JH295 hydrate
<p>JH295 hydrate: potent, irreversible Nek2 inhibitor (IC50 = 770 nM), selective, doesn't target Cdk1, Aurora B or Plk1.</p>Formula:C18H18N4O3Color and Shape:SolidMolecular weight:338.36Bometolol Hydrochloride
CAS:<p>Bometolol Hydrochloride is a beta-adrenergic blocking compound used for the treatment of cardiovascular disease.</p>Formula:C25H33ClN2O7Purity:98%Color and Shape:SolidMolecular weight:508.99CEP-14083
CAS:<p>CEP-14083: potent ALK inhibitor, effective in NPM/ALK T-cell lymphoma, binds ATP site; IC50=11 nmol/L, also inhibits insulin receptor, preclinical efficacy.</p>Formula:C31H30N6O2Color and Shape:SolidMolecular weight:518.61Microtubule inhibitor 2
<p>Microtubule inhibitor 2: potent, selective, oral, induces ferroptosis, strong antitumor effect.</p>Formula:C20H23NO7Color and Shape:SolidMolecular weight:389.4PCSK9-IN-17
CAS:<p>PCSK9-IN-17 is a PCSK9 inhibitor utilized in the research of cholesterol metabolism.</p>Formula:C16H19N5OSColor and Shape:SolidMolecular weight:329.42A1/A3 AR antagonist 1
<p>Compound 10 is a potent dual A1/A3 AR antagonist, with Ki values of 37.6 nM (hA1), 25.4 nM (hA3), and 1.47 nM (rA1), studied in renal, lung, and Alzheimer's.</p>Formula:C24H18N2O3SColor and Shape:SolidMolecular weight:414.48Zaragozic acid C
CAS:<p>Zaragozic acid C is an effective inhibitor of squalene synthase.</p>Formula:C40H50O14Purity:98%Color and Shape:SolidMolecular weight:754.82SH498
CAS:<p>SH498 is a novel Bmi-1-mediated anti-tumor agent with significant anti-proliferative effects.</p>Formula:C27H25F3N2O4Color and Shape:SolidMolecular weight:498.49MtMetAP1-IN-1
<p>MtMetAP1-IN-1 is an inhibitor of methionine aminopeptidase 1 ( MetAP1 ). MtMetAP1-IN-1 shows antimycobacterial activity.</p>Formula:C15H10BrN5O2SColor and Shape:SolidMolecular weight:404.24Ro-51
CAS:<p>dual P2X3 and P2X2/3 antagonist</p>Formula:C17H23IN4O4Purity:98%Color and Shape:SolidMolecular weight:474.29Ceclazepide
CAS:<p>Ceclazepide is an antagonist of cholecystokinin receptor.</p>Formula:C30H32N6O5Purity:98%Color and Shape:SolidMolecular weight:556.61Urease-IN-1
<p>Urease -IN-1 is a urease inhibitor (IC50: 2.21±0.45 μM).</p>Formula:C17H12BrFN4O2SColor and Shape:SolidMolecular weight:435.27AM Toxin II
CAS:<p>AM Toxin II is a Cyclic tetradepsipeptide isolated from Alternaria mali.</p>Formula:C22H29N3O5Color and Shape:SolidMolecular weight:415.49Atiratecan
CAS:<p>Atiratecan (TP300), a CH0793076-based camptothecin prodrug, combats BCRP+/- tumors; doesn't affect AChE.</p>Formula:C31H34N6O6Purity:98%Color and Shape:SolidMolecular weight:586.64CI-988
CAS:<p>CCK2 (CCK-B) receptor antagonist</p>Formula:C35H42N4O6Purity:98%Color and Shape:SolidMolecular weight:614.73

