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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66618 products of "Inhibitors"

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  • Gemilukast

    CAS:
    <p>Gemilukast (ONO-6950) is a cysteinyl leukotriene 1 and 2 receptor inhibitor that inhibits bronchoconstriction and is used in the treatment of asthma.</p>
    Formula:C36H37F2NO5
    Purity:98.27% - 99.5%
    Color and Shape:Solid
    Molecular weight:601.68
  • PIM-1/HDAC-IN-1


    <p>PIM-1/HDAC-IN-1 (4d): inhibits PIM-1 (IC50: 343.87nM), HDAC1 (63.65nM), HDAC6 (62.39nM); induces apoptosis in MCF-7 cells.</p>
    Formula:C22H19N3O3
    Color and Shape:Solid
    Molecular weight:373.4
  • CXCR2 antagonist 6


    <p>CXCR2 antagonist 6: strong CXCR2 affinity (IC50=0.044 μM), hinders calcium mobilization (IC50=0.66 μM).</p>
    Formula:C17H16F2N4OS
    Color and Shape:Solid
    Molecular weight:362.4
  • RSV-IN-5

    CAS:
    <p>RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM &amp; 8.1 nM. Potent anti-RSV.</p>
    Formula:C28H37N7O2
    Color and Shape:Solid
    Molecular weight:503.64
  • PARP1-IN-5


    <p>PARP1-IN-5 is a potent, selective, orally active, low-toxicity PARP-1 inhibitor with an IC50 value of 14.7 nM. PARP1-IN-5 can be used in cancer research.</p>
    Formula:C25H24N2O5S
    Color and Shape:Solid
    Molecular weight:464.53
  • Y1 receptor antagonist 1

    CAS:
    <p>Y1 receptor antagonist 1 is an antagonist of neuropeptide Y1 receptor.</p>
    Formula:C28H33N5O3
    Purity:98.17%
    Color and Shape:Solid
    Molecular weight:487.59
  • Silvestrol

    CAS:
    <p>Silvestrol is a eukaryotic translation initiation factor 4A inhibitor. Silvestrol causes autophagy and caspase-mediated apoptosis.</p>
    Formula:C34H38O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:654.66
  • GP-1681

    CAS:
    <p>GP-1681, a G-protein coupled receptor (GPCR) agonist, is used potentially for the treatment of influenza infection.</p>
    Formula:C24H30NaO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:421.48
  • LY 235959

    CAS:
    <p>LY 235959 is a NMDA receptor antagonist.</p>
    Formula:C11H20NO5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:277.25
  • S100A2-p53-IN-1

    CAS:
    <p>S100A2-p53-IN-1 inhibits S100A2-p53 in pancreatic cancer, stunting MiaPaCa-2 cell growth at 1.2-3.4 μM.</p>
    Formula:C20H20F6N2O4S
    Color and Shape:Solid
    Molecular weight:498.44
  • AZD 4407

    CAS:
    <p>AZD 4407 is a potent inhibitor of 5-lipoxygenase.</p>
    Formula:C19H21NO3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:375.5
  • CGS 22652

    CAS:
    <p>CGS 22652 has thromboxane receptor antagonism combined with thromboxane synthase inhibition.</p>
    Formula:C22H29ClN2O4S
    Color and Shape:Solid
    Molecular weight:452.99
  • Dup-714

    CAS:
    <p>Dup-714 is a thrombin inhibitor.</p>
    Formula:C21H33BN6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:460.33
  • (-)-Cevimeline hydrochloride hemihydrate


    <p>(-)-Cevimeline HCl hemihydrate, a muscarinic agonist, treats Sjogren's xerostomia. Quick absorption, species-dependent metabolism.</p>
    Formula:C10H19ClNO1·5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:244.78
  • P2X receptor-1


    <p>P2X receptor-1 is a potential inhibitor of P2X receptor for the treatment of pain and inflammation.</p>
    Formula:C14H14ClN3O3S2
    Color and Shape:Solid
    Molecular weight:371.86
  • Deleobuvir

    CAS:
    <p>Deleobuvir(BI207127) is an inhibitor of non-nucleoside hepatitis C virus NS5B polymerase for the treatment of hepatitis C.</p>
    Formula:C34H33BrN6O3
    Color and Shape:Solid
    Molecular weight:653.57
  • BMS-986143

    CAS:
    <p>BMS-986143: oral BTK inhibitor, IC50=0.26 nM, potential for autoimmune research, also targets TEC, BLK, BMX, TXK, YES1, ITK.</p>
    Formula:C31H24Cl2N4O4
    Color and Shape:Solid
    Molecular weight:587.45
  • Cap-dependent endonuclease-IN-17

    CAS:
    <p>CEN inhibitor IN-17 targets influenza A/H3N2; IC50: 1.29 μM. From patent CN112898346A, DSC701.</p>
    Formula:C24H20F2N3O7PS
    Color and Shape:Solid
    Molecular weight:563.47
  • Tubulin polymerization-IN-35


    <p>Tubulin-IN-35 inhibits oxazolylisoindole microtubule formation, targeting VL51 marginal zone lymphoma.</p>
    Formula:C31H35N3O5
    Color and Shape:Solid
    Molecular weight:529.63
  • MAFP

    CAS:
    MAFP (Methyl Arachidonyl Fluorophosphonate) is an effective irreversible inhibitor of anandamide amidase.
    Formula:C21H36FO2P
    Color and Shape:Solid
    Molecular weight:370.48
  • UH 301

    CAS:
    <p>UH 301 is a 5-HT1A receptor antagonist.</p>
    Formula:C16H24FNO
    Color and Shape:Solid
    Molecular weight:265.37
  • Carbonic anhydrase inhibitor 2

    CAS:
    <p>Compound 7c inhibits carbonic anhydrase II, lowering intraocular pressure in glaucomatous rabbits.</p>
    Formula:C12H16N4O6S
    Color and Shape:Solid
    Molecular weight:344.34
  • 2R,4S-Sacubitril

    CAS:
    <p>2R,4S-Sacubitril (Sacubitril Enantiomer) is the impurity of Sacubitril which is a neprilysin inhibitor.</p>
    Formula:C24H28NO51Ca
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.49
  • FGFR4-IN-10


    <p>FGFR4-IN-10 (compound 5a) is a potent, selective FGFR4 inhibitor with IC50 of 70.7 nM, sparing FGFR1-3.</p>
    Formula:C20H19F3N6O3
    Color and Shape:Solid
    Molecular weight:448.4
  • Spicamycin

    CAS:
    <p>Spicamycin can be used as a potent inducer of differentiation of human myeloid leukemia cells (HL-60) and murine myeloid leukemia cells (M1).</p>
    Formula:C30H51N7O7
    Color and Shape:Solid
    Molecular weight:621.77
  • Keap1-Nrf2-IN-4


    <p>Keap1-Nrf2-IN-4 hinders MGC-803 cell growth (IC50=2.55μM), migration, and induces apoptosis with low toxicity.</p>
    Formula:C26H34N2O
    Color and Shape:Solid
    Molecular weight:390.56
  • Arterolane

    CAS:
    <p>Arterolane is an antimalarial compound. For against P. falciparum Ro73 and W2, the IC50s are both 1.1 nM.</p>
    Formula:C22H36N2O4
    Color and Shape:Solid
    Molecular weight:392.53
  • Cilazapril HCl

    CAS:
    <p>Cilazapril, also known as Ro 31 2848, is a potent ACE inhibitor used for hypertension.</p>
    Formula:C22H32ClN3O5
    Color and Shape:Solid
    Molecular weight:453.96
  • Tubulin polymerization-IN-33


    <p>Tubulin-IN-33, an oxazoloisoindole, hinders microtubule assembly; effective against NCI cancer cells.</p>
    Formula:C27H28N2O6
    Color and Shape:Solid
    Molecular weight:476.52
  • PD 136450

    CAS:
    <p>PD-136,450: partial stomach secretory agonist, full pancreas agonist in rats; potential acid-reducing drug, adjuvant for gastrin-sensitive tumors.</p>
    Formula:C35H40N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:612.72
  • Luffariellolide

    CAS:
    <p>Luffariellolide is a terpene compound obtained from the marine sponge Hyrtios communis that is an HSF-PLA2 inhibitor and a RAR agonist.</p>
    Formula:C25H38O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.57
  • I-BET282E


    <p>I-BET282E inhibits eight BET bromodomains (pIC50 6.4-7.7) with selectivity for other bromodomain proteins.</p>
    Formula:C26H34N4O7S
    Color and Shape:Solid
    Molecular weight:546.64
  • β-Glucuronidase/hCAII-IN-2


    <p>β-Glucuronidase/hCAII-IN-2 is a potent inhibitor of β-glucuronidase and hCA II, and their IC50 values were 670.7 μM and 21.77 μM, respectively.</p>
    Formula:C31H23NO8
    Color and Shape:Solid
    Molecular weight:537.52
  • NS2B/NS3-IN-3

    CAS:
    <p>NS2B/NS3-IN-3 (Compd 66) is an inhibitor of Flavivirus NS2B-NS3 protease [1] .</p>
    Formula:C19H21N3O2
    Color and Shape:Solid
    Molecular weight:323.39
  • STING agonist-7


    <p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>
    Formula:C17H12N4O4
    Color and Shape:Solid
    Molecular weight:336.3
  • AX15910


    <p>AX15910 is a potent inhibitor of BRD4 and ERK5.</p>
    Formula:C32H38N6O3
    Color and Shape:Solid
    Molecular weight:554.7
  • CK2-IN-3


    <p>CK2-IN-3: potent, selective CK2 inhibitor; Kd=12 nM, IC50: 1.51 μM (CK2α), 7.64 μM (CK2α'). For cancer research.</p>
    Formula:C22H26N4O7
    Color and Shape:Solid
    Molecular weight:458.46
  • DLK-IN-1

    CAS:
    DLK-IN-1: Oral DLK (MAP3K12) inhibitor, Ki=3nM, effective in Alzheimer's model, CNS permeable, well-tolerated with sustained brain levels.
    Formula:C20H24F3N5O2
    Color and Shape:Solid
    Molecular weight:423.43
  • XIAP/cIAP1 antagonist-1


    <p>Potent oral XIAP/cIAP1 inhibitor with EC50s: XIAP 5.1 nM, cIAP1 0.32 nM; curbs tumor growth in vivo.</p>
    Color and Shape:Solid
  • SR121566A

    CAS:
    SR121566A is a novel non-peptide antagonist of Glycoprotein IIb/IIIa (GP IIb-IIIa).
    Formula:C20H25N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.51
  • J-104132

    CAS:
    <p>J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.</p>
    Formula:C31H33NO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.60
  • NCATS-SM4487

    CAS:
    <p>NCATS-SM4487 is a highly selective inhibitor of GALK1 (IC50: 0.05 μM).</p>
    Formula:C25H24ClFN8O2
    Color and Shape:Solid
    Molecular weight:522.96
  • FLT3-IN-13


    <p>FLT3-IN-13 inhibits topoisomerase II/FLT3 in leukemia with IC50 of 2.26 μM, causes G2/M arrest, and promotes apoptosis.</p>
    Formula:C20H14N4O2
    Color and Shape:Solid
    Molecular weight:342.35
  • PARP-1-IN-1


    <p>PARP-1-IN-1: Selective, oral PARP-1 inhibitor with 0.96 nM IC50; well-tolerated and effective in single-dose MDA-MB-436 model.</p>
    Formula:C23H25FN4O
    Color and Shape:Solid
    Molecular weight:392.47
  • PPARγ agonist 2


    <p>PPARγ agonist 2 is a highly effective compound that acts as a partial agonist for PPARγ.</p>
    Formula:C24H20O5
    Color and Shape:Solid
    Molecular weight:388.41
  • GSK945237

    CAS:
    <p>GSK945237 is a type IIA topoisomerase inhibitor, effective on Gram-positive and negative bacteria, with favorable pharmacokinetics and in vivo efficacy.</p>
    Formula:C24H26FN5O3
    Color and Shape:Solid
    Molecular weight:451.49
  • Dyrk1A-IN-1


    <p>Dyrk1A-IN-1 is a triple inhibitor of Dyrk1A kinase activity, aggregation of tau and α-syn oligomers, with an IC50 value of 119 nM for Dyrk1A kinase.</p>
    Formula:C23H20N4O3S
    Color and Shape:Solid
    Molecular weight:432.49
  • PF-06380101

    CAS:
    <p>PF-06380101, a potent auristatin analog and Dolastatin 10 derivative, shows strong anti-tumor activity and unique ADME attributes.</p>
    Formula:C39H62N6O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:743.01
  • KT2-962

    CAS:
    <p>KT2-962 is a TXA2/prostaglandin endoperoxide receptor antagonist.</p>
    Formula:C23H27ClNNaO5S2
    Color and Shape:Solid
    Molecular weight:520.04
  • Carmegliptin dihydrochloride

    CAS:
    <p>Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.</p>
    Formula:C20H30Cl2FN3O3
    Color and Shape:Solid
    Molecular weight:450.38
  • [D-Leu-4]-OB3

    CAS:
    [D-Leu-4]-OB3 suppresses the expression of genes associated with inflammation, proliferation, and metastasis, as well as the expression of PD-L1.
    Formula:C29H50N8O12S
    Color and Shape:Solid
    Molecular weight:734.82
  • HIF-1/2α-IN-1


    <p>HIF-1/2α-IN-1, an orally active compound, functions as an inhibitor of HIF-2α.</p>
    Formula:C17H16N6O4
    Color and Shape:Solid
    Molecular weight:368.35
  • Antifungal agent 16


    <p>Antifungal agent 16 has antimicrobial activity comparable to that of ciprofloxacin and has higher antifungal activity than fluconazole.</p>
    Formula:C27H21N5O2S
    Color and Shape:Solid
    Molecular weight:479.55
  • Netupitant metabolite Monohydroxy Netupitant

    CAS:
    Monohydroxy Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.
    Formula:C30H32F6N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:594.59
  • Mesulergine hydrochloride

    CAS:
    <p>5-HT2A and 2C receptor antagonist</p>
    Formula:C18H27ClN4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:398.95
  • Fandosentan

    CAS:
    <p>Fandosentan is an endothelin receptor antagonist.</p>
    Formula:C25H18F3NO6S
    Color and Shape:Solid
    Molecular weight:517.47
  • BMS-986118

    CAS:
    BMS-986118 is a GPR40 full agonist targeting type II diabetes, prompting insulin release without hypoglycemia risk.
    Formula:C25H28ClF3N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:540.96
  • NLRP3/AIM2-IN-1


    <p>NLRP3/AIM2-IN-1 is an inhibitor of thermal sepsis (IC50 = 3.136 ± 0.7667 μM).</p>
    Formula:C15H16BNO4
    Color and Shape:Solid
    Molecular weight:285.1
  • SHP2 IN-1

    CAS:
    <p>SHP2 IN-1 is an allergic SHP2 (PTPN11) inhibitor(IC50 : 3 nM).</p>
    Formula:C18H22Cl2N6OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.38
  • LSD1-IN-16


    <p>LSD1-IN-16 (4b) inhibits LSD1, MAO-A/B; IC50: 0.015-0.366 μM. Halts prostate cancer cell growth; IC50: 15.2 μM.</p>
    Formula:C20H18N2OS
    Color and Shape:Solid
    Molecular weight:334.43
  • HDAC6-IN-9

    CAS:
    <p>HDAC6-IN-9 is a γ-secretase modulator that can significantly reduce the level of Aβ42 in mouse brain and can be used to study neurological diseases.</p>
    Formula:C19H16N2O3
    Purity:98.84%
    Color and Shape:Solid
    Molecular weight:320.34
  • DYRK1-IN-1

    CAS:
    <p>DYRK1-IN-1: Selective DYRK1A inhibitor with IC50 of 220 nM, good permeability, CNS penetrant for research, no P-glycoprotein issues.</p>
    Formula:C12H12N6
    Color and Shape:Solid
    Molecular weight:240.26
  • SARS 3CLpro-IN-1

    CAS:
    <p>SARS 3CLpro-IN-1: stereospecific SARS 3CL protease inhibitor, octahydroisochromene class, IC50 = 95 μM.</p>
    Formula:C22H38N4O2
    Color and Shape:Solid
    Molecular weight:390.56
  • VEGFR-2-IN-11


    <p>VEGFR-2-IN-11 is a potent inhibitor of VEGFR-2 (IC50: 60.27 nM) with an IC50 value of 60.27 nM, which induces apoptosis and has anticancer activity.</p>
    Formula:C29H22BrN5S
    Color and Shape:Solid
    Molecular weight:552.49
  • Irinotecan Carboxylate Sodium Salt

    CAS:
    <p>Irinotecan Carboxylate Sodium Salt is a DNA topoisomerase inhibitor.</p>
    Formula:C33H39N4NaO7
    Color and Shape:Solid
    Molecular weight:626.68
  • CBP/p300-IN-16


    <p>CBP/p300-IN-16 (compound 1) is a potent inhibitor of EP300/CBP HAT, acting on HAT EP300 (IC50: 0.61 μM) and LK2 H3K27 (IC50: 2.24 μM).</p>
    Formula:C26H31N3O4
    Color and Shape:Solid
    Molecular weight:449.54
  • CDK4-IN-1

    CAS:
    <p>CDK4 inhibitor is a novel and specific CDK4/Cyclin D1 inhibitor with an IC50 of 10 nM; 1500 and 500 fold than CDK1/Cyclin B (IC50&gt;15 uM) and CDK2/Cyclin A (IC50</p>
    Formula:C22H29ClN8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.97
  • (R)-CSN5i-3

    CAS:
    <p>(R)-CSN5i-3 is CSN5i-3 of the R configuration.</p>
    Formula:C28H29F2N5O2
    Purity:99.76% - 99.97%
    Color and Shape:Solid
    Molecular weight:505.56
  • Rodatristat

    CAS:
    <p>Rodatristat is an effective tryptophan hydroxylase 1 and TPH2 inhibitor (IC50s: 33 nM and 7 nM, respectively).</p>
    Formula:C27H27ClF3N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:561.98
  • TAS05567

    CAS:
    <p>TAS05567 is a potent, highly selective, and ATP-competitive Syk inhibitor (IC50: 0.37 nM).</p>
    Formula:C21H29N9O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:439.51
  • Nafarelin acetate hydrate

    CAS:
    <p>Nafarelin: a GnRH agonist used to treat endometriosis, precocious puberty, and control IVF. Delivered as a nasal spray. Marketed as Synarel by Pfizer.</p>
    Formula:C66H83N17O13·xC2H4O2·xH2O
    Color and Shape:Solid
    Molecular weight:1400.563
  • ROPA

    CAS:
    <p>ROPA, a potent PKCalpha and PKCgamma activator, promotes tumor growth through PKC-activation.</p>
    Formula:C28H32O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:464.55
  • Minnelide

    CAS:
    Minnelide is a prodrug of triptolide,and shows potent antitumor activity in a number of tumor types.
    Formula:C21H25Na2O10P
    Purity:98.49% - 99.59%
    Color and Shape:Solid
    Molecular weight:514.37
  • Sulprostone

    CAS:
    <p>EP3 and EP1 receptor agonist</p>
    Formula:C23H31NO7S
    Purity:98%
    Color and Shape:White To Off-White Solid
    Molecular weight:465.56
  • HDAC-IN-34


    <p>HDAC-IN-34 inhibits HDAC1 (IC50: 0.022 μM) &amp; HDAC6 (IC50: 0.45 μM), binds DNA causing damage, and halts HCT-116 cell growth (IC50: 1.41 μM).</p>
    Formula:C24H26N6O3
    Color and Shape:Solid
    Molecular weight:446.5
  • SGE-516

    CAS:
    <p>SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.</p>
    Formula:C23H35N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:385.54
  • AZD0424

    CAS:
    <p>AZD0424: oral Src/Abl kinase inhibitor; potential anticancer; induces apoptosis, cell cycle arrest in lymphoma.</p>
    Formula:C25H29ClN6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:528.99
  • Rezatapopt

    CAS:
    <p>Rezatapopt (PC14586) is a p53 reactivator with antitumor activity for the study of locally advanced or metastatic solid tumors.</p>
    Formula:C28H31F4N5O2
    Purity:98.12%
    Color and Shape:Solid
    Molecular weight:545.57
  • CDK2-IN-9


    <p>CDK2-IN-9: potent CDK2 inhibitor (IC50: 0.63 μM), anti-proliferative, arrests S/G2M cell cycle, induces apoptosis, promising for melanoma study.</p>
    Formula:C21H16ClN3O4S
    Color and Shape:Solid
    Molecular weight:441.89
  • SSR-182289A (Free)

    CAS:
    SSR-182289A (Free) is a thrombin inhibitor.
    Formula:C30H33F2N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:597.68
  • KT5926

    CAS:
    <p>KT5926 selectively inhibits myosin light chain kinase and NGF-dependent neurite growth; it's a K-252a analogue.</p>
    Formula:C30H27N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:525.55
  • LY 245769

    CAS:
    <p>LY 245769 is an inhibitor of leukotriene E4 (LTE4).</p>
    Formula:C25H33F3N8OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:550.64
  • CTX-712

    CAS:
    <p>CTX-712 is a potent inhibitor of cdc2-like kinase ( CLK ). CTX-712 inhibits inhibits cancer survival and cancer cell growth.</p>
    Formula:C19H17FN8O2
    Color and Shape:Solid
    Molecular weight:408.39
  • Antitumor agent-42


    <p>Antitumor agent-42 inhibits microtubule multimerisation and NO release, exhibiting anti-angiogenic, colony-forming and apoptosis-inducing effects.</p>
    Formula:C24H19BrN2O8S
    Color and Shape:Solid
    Molecular weight:575.39
  • hCAII-IN-4

    CAS:
    hCAII-IN-4 (Compound 12j) is a potent inhibitor of human carbonic anhydrase II (hCA II), exhibiting an inhibitory concentration (IC50) of 7.78 μM.
    Formula:C31H23NO9
    Color and Shape:Solid
    Molecular weight:553.52
  • JH295 hydrate


    <p>JH295 hydrate: potent, irreversible Nek2 inhibitor (IC50 = 770 nM), selective, doesn't target Cdk1, Aurora B or Plk1.</p>
    Formula:C18H18N4O3
    Color and Shape:Solid
    Molecular weight:338.36
  • Bometolol Hydrochloride

    CAS:
    <p>Bometolol Hydrochloride is a beta-adrenergic blocking compound used for the treatment of cardiovascular disease.</p>
    Formula:C25H33ClN2O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:508.99
  • CEP-14083

    CAS:
    <p>CEP-14083: potent ALK inhibitor, effective in NPM/ALK T-cell lymphoma, binds ATP site; IC50=11 nmol/L, also inhibits insulin receptor, preclinical efficacy.</p>
    Formula:C31H30N6O2
    Color and Shape:Solid
    Molecular weight:518.61
  • Microtubule inhibitor 2


    <p>Microtubule inhibitor 2: potent, selective, oral, induces ferroptosis, strong antitumor effect.</p>
    Formula:C20H23NO7
    Color and Shape:Solid
    Molecular weight:389.4
  • PCSK9-IN-17

    CAS:
    <p>PCSK9-IN-17 is a PCSK9 inhibitor utilized in the research of cholesterol metabolism.</p>
    Formula:C16H19N5OS
    Color and Shape:Solid
    Molecular weight:329.42
  • A1/A3 AR antagonist 1


    <p>Compound 10 is a potent dual A1/A3 AR antagonist, with Ki values of 37.6 nM (hA1), 25.4 nM (hA3), and 1.47 nM (rA1), studied in renal, lung, and Alzheimer's.</p>
    Formula:C24H18N2O3S
    Color and Shape:Solid
    Molecular weight:414.48
  • Zaragozic acid C

    CAS:
    <p>Zaragozic acid C is an effective inhibitor of squalene synthase.</p>
    Formula:C40H50O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:754.82
  • SH498

    CAS:
    <p>SH498 is a novel Bmi-1-mediated anti-tumor agent with significant anti-proliferative effects.</p>
    Formula:C27H25F3N2O4
    Color and Shape:Solid
    Molecular weight:498.49
  • MtMetAP1-IN-1


    <p>MtMetAP1-IN-1 is an inhibitor of methionine aminopeptidase 1 ( MetAP1 ). MtMetAP1-IN-1 shows antimycobacterial activity.</p>
    Formula:C15H10BrN5O2S
    Color and Shape:Solid
    Molecular weight:404.24
  • Ro-51

    CAS:
    <p>dual P2X3 and P2X2/3 antagonist</p>
    Formula:C17H23IN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:474.29
  • Ceclazepide

    CAS:
    <p>Ceclazepide is an antagonist of cholecystokinin receptor.</p>
    Formula:C30H32N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:556.61
  • Urease-IN-1


    <p>Urease -IN-1 is a urease inhibitor (IC50: 2.21±0.45 μM).</p>
    Formula:C17H12BrFN4O2S
    Color and Shape:Solid
    Molecular weight:435.27
  • AM Toxin II

    CAS:
    <p>AM Toxin II is a Cyclic tetradepsipeptide isolated from Alternaria mali.</p>
    Formula:C22H29N3O5
    Color and Shape:Solid
    Molecular weight:415.49
  • Atiratecan

    CAS:
    <p>Atiratecan (TP300), a CH0793076-based camptothecin prodrug, combats BCRP+/- tumors; doesn't affect AChE.</p>
    Formula:C31H34N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:586.64
  • CI-988

    CAS:
    <p>CCK2 (CCK-B) receptor antagonist</p>
    Formula:C35H42N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:614.73