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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66626 products of "Inhibitors"

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  • (Rac)-Nebivolol

    CAS:
    <p>(Rac)-Nebivolol, a racemic β1-adrenergic blocker (IC50=0.8 nM), has vasodilatory properties and mitigates ethanol-induced cardiac harm.</p>
    Formula:C22H25F2NO4
    Color and Shape:Solid
    Molecular weight:405.43
  • AAK1-IN-2 TFA


    <p>AAK1-IN-2 TFA (compound (S)-31) is a selective and potent AAK1 inhibitor (IC50: 5.8 nM) that can cross the blood-brain barrier.</p>
    Formula:C24H22F6N4O4
    Color and Shape:Solid
    Molecular weight:544.45
  • CREB-IN-1 TFA


    <p>CREB-IN-1 TFA: Potent oral CREB inhibitor, IC50 of 0.18 μM, suppresses breast cancer cell growth.</p>
    Color and Shape:Solid
  • Cathepsin C-IN-3


    <p>Cathepsin C-IN-3 is a potent inhibitor of histone C (IC50: 61.79 nM) and also inhibits THP-1 cells (IC50: 101.5 nM) and U937 cells (IC50: 86.5 nM).</p>
    Formula:C28H21F3N6OS
    Color and Shape:Solid
    Molecular weight:546.57
  • PD-1/PD-L1-IN-17


    <p>PD-1/PD-L1-IN-17 (Compound P20) is a potent PD-1/PD-L1 inhibitor (IC50: 26.8 nM).</p>
    Formula:C23H20ClN3O4
    Color and Shape:Solid
    Molecular weight:437.88
  • MK-8876

    CAS:
    <p>MK-8876 is an Inhibitor of HCV NS5B Site D.</p>
    Formula:C32H24F2N4O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:614.62
  • ZK 93426 hydrochloride

    CAS:
    <p>benzodiazepine receptor antagonist,competitive</p>
    Formula:C18H21ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.82
  • CDK9-IN-13


    <p>CDK9-IN-13 is a potent and selective CDK inhibitor (IC50&lt;3 nM). CDK9-IN-13 has a very short half-life in rodents.</p>
    Formula:C27H35N5O2
    Color and Shape:Solid
    Molecular weight:461.6
  • Macropa-NCS

    CAS:
    <p>Macropa-NCS is a macropa bifunctional analog with antitumor activity and can be used to study prostate cancer.</p>
    Formula:C27H35N5O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:589.66
  • C108297

    CAS:
    <p>C108297: glucocorticoid modulator, combats diet obesity/inflammation, reduces appetite/lipid storage, boosts fat burn.</p>
    Formula:C30H36FN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.69
  • AFM-30a hydrochloride


    <p>AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.</p>
    Formula:C24H28ClFN6O3
    Color and Shape:Solid
    Molecular weight:502.97
  • CB 30900

    CAS:
    <p>CB30900 is a novel and effective thymidylate synthase inhibitor.</p>
    Formula:C31H32FN5O9
    Color and Shape:Solid
    Molecular weight:637.61
  • PF-06726304 acetate

    CAS:
    <p>PF-06726304 acetate is a selective inhibitor of EZH2, with robust antitumor growth activity.</p>
    Formula:C24H25Cl2N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:506.38
  • Vanin-1-IN-3


    <p>Vanin-1-IN-3 (OMP-7) is a vanin-1 inhibitor with an IC 50 of 0.038 μM [1].</p>
    Formula:C17H22F3NO5
    Color and Shape:Solid
    Molecular weight:377.36
  • AKN-028 acetate


    <p>AKN-028 acetate: an oral TK inhibitor for AML research, targets FLT3 with IC50 of 6 nM, inhibits autophosphorylation, and induces apoptosis.</p>
    Formula:C19H18N6O2
    Color and Shape:Solid
    Molecular weight:362.39
  • Mu opioid receptor antagonist 2


    <p>Compound 25: potent, selective MOR antagonist, crosses blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM), for OUD research.</p>
    Formula:C25H28N2O4S
    Color and Shape:Solid
    Molecular weight:452.57
  • METTL3-IN-2

    CAS:
    <p>METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.</p>
    Formula:C25H26N8O
    Color and Shape:Solid
    Molecular weight:454.53
  • HIV-1 inhibitor-52

    CAS:
    <p>HIV-1 inhibitor-52: potent, broad-spectrum with EC50s 1.6-6.4 nM against various HIV-1 strains.</p>
    Formula:C46H72FNO5S
    Color and Shape:Solid
    Molecular weight:770.13
  • MAO-B-IN-10


    <p>MAO-B-IN-10: Potent, selective MAO-B inhibitor; crosses blood-brain barrier; IC50 5.3 μM; reduces Aβ aggregation 58.2%, disaggregates 43.3%.</p>
    Formula:C23H26N2O4
    Color and Shape:Solid
    Molecular weight:394.46
  • L 156903

    CAS:
    <p>L 156903 is a bioactive chemical. It also inhibits the binding of neurotensin to brain tissue.</p>
    Formula:C35H41N7O5S
    Color and Shape:Solid
    Molecular weight:671.81
  • Atorvastatin 3-Deoxyhept-2E-Enoic Acid

    CAS:
    Atorvastatin 3-Deoxyhept-2E-Enoic Acid, an impurity in Atorvastatin, lowers blood lipids as an HMG-CoA reductase inhibitor.
    Formula:C33H33FN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:540.62
  • PDHK-IN-5


    <p>PDHK-IN-5, potent PDHK2 (0.006 μM IC50) &amp; PDHK4 (0.0329 μM IC50) inhibitor, may be explored for cancer and diabetes treatment.</p>
    Formula:C30H31N5O2
    Color and Shape:Solid
    Molecular weight:493.6
  • Antibacterial agent 113


    <p>Antibacterial agent 113 targets multiple bacteria including P. aeruginosa and E. coli, showing efficacy at MIC 15625 μM.</p>
    Formula:C29H18ClN5O
    Color and Shape:Solid
    Molecular weight:487.94
  • Irinotecan Carboxylate Sodium Salt

    CAS:
    <p>Irinotecan Carboxylate Sodium Salt is a DNA topoisomerase inhibitor.</p>
    Formula:C33H39N4NaO7
    Color and Shape:Solid
    Molecular weight:626.68
  • Anticancer agent 12


    <p>Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity.</p>
    Formula:C16H17BrN4O2S
    Color and Shape:Solid
    Molecular weight:409.3
  • CEP-7055

    CAS:
    <p>CEP-18770: oral proteasome inhibitor; blocks NF-kappaB; may cause cancer cell apoptosis; less toxic than bortezomib in normal cells.</p>
    Formula:C32H35N3O4
    Color and Shape:Solid
    Molecular weight:525.64
  • KUSC-5037


    <p>KUSC-5037 inhibits HIF-1 (IC50 = 1.2 μM) and mitochondrial complex V/FoF1ATP synthase.</p>
    Formula:C18H17F3N6O2
    Color and Shape:Solid
    Molecular weight:406.13651
  • VEGFR-2-IN-15


    <p>VEGFR-2-IN-15 (Compound 14b) is a potent inhibitor of VEGFR-2. VEGFR-2-IN-15 inhibits the growth of HepG2 cells in the Pre-G1 phase and induces apoptosis.</p>
    Formula:C23H18ClN3O4S
    Color and Shape:Solid
    Molecular weight:467.92
  • Dexnebivolol

    CAS:
    <p>Dexnebivolol (R67138), a ß-adrenergic antagonist, is Nebivolol's enantiomer with β1 blocking and vasodilation properties.</p>
    Formula:C22H25F2NO4
    Color and Shape:Solid
    Molecular weight:405.43
  • BRD4 Inhibitor-17


    <p>BRD4 Inhibitor-17: Potent with 0.33 μM IC50; modulates gene expression, may counter arsenic toxicity.</p>
    Formula:C16H16FN3O3S
    Color and Shape:Solid
    Molecular weight:349.38
  • Cilengitide hydrochloride

    CAS:
    <p>Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.</p>
    Formula:C27H41ClN8O7
    Color and Shape:Solid
    Molecular weight:625.12
  • p38-α MAPK-IN-5

    CAS:
    <p>p38-α MAPK-IN-5: potent p38α inhibitor, IC50s: 0.1 nM (α), 0.2 nM (β), 944 nM (γ), 4100 nM (δ); anti-inflammatory, promising for asthma/COPD research.</p>
    Formula:C37H49N11O2
    Color and Shape:Solid
    Molecular weight:679.86
  • YW3-56

    CAS:
    <p>YW3-56 is a potent peptidylarginine deiminase (PAD) inhibitor, with an IC50 of 1-5 μM for PAD4.</p>
    Formula:C27H32ClN5O2
    Color and Shape:Solid
    Molecular weight:494.03
  • U 80215

    CAS:
    <p>U 80215 is an enzyme-competitive inhibitor.</p>
    Formula:C42H60N8O6S
    Color and Shape:Solid
    Molecular weight:805.04
  • Agosterol A

    CAS:
    <p>Agosterol A is isolated from marine sponge Spongia.</p>
    Formula:C33H52O8
    Color and Shape:Solid
    Molecular weight:576.76
  • LY2934747

    CAS:
    <p>LY2934747 is a novel, potent, and systemically bioavailable mGlu2/3 receptor agonist, exhibiting both antipsychotic and analgesic properties in vivo.</p>
    Formula:C10H13NO4
    Color and Shape:Solid
    Molecular weight:211.21
  • SP4206

    CAS:
    SP4206 is an interaction inhibitor of IL-2/IL-2Rα (IL-2 and IL-2Rα with Kd of 70 nM and 10 nM,respectively)
    Formula:C30H37Cl2N7O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:662.56
  • Kendomycin

    CAS:
    <p>Kendomycin is a proteasome inhibitor and endothelin receptor antagonist. It induces apoptosis in lymphoma.</p>
    Formula:C29H42O6
    Color and Shape:Solid
    Molecular weight:486.64
  • AKT-IN-3

    CAS:
    AKT-IN-3: potent oral Akt inhibitor with low hERG blockage. IC50: 1.4-1.7 nM for Akt1-3. Inhibits AGC kinases like PKA, PKC.
    Formula:C23H23Cl2F2N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:526.36
  • Lp-PLA2-IN-6

    CAS:
    <p>Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.</p>
    Formula:C25H21F5N4O3
    Color and Shape:Solid
    Molecular weight:520.45
  • A1AR antagonist 1


    <p>Compound 18g, a potent A1AR blocker with Ki: 2.08 nM (hA1), 6.91 nM (hA2A), 31.2 nM (hA2B).</p>
    Formula:C18H14N4O
    Color and Shape:Solid
    Molecular weight:302.33
  • SB-423557

    CAS:
    SB-423557 is an orally active antagonist of calcium-sensing receptor (CaR) with IC50 of 520 nM
    Formula:C28H36N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:464.60
  • SCH-900822

    CAS:
    <p>SCH-900822 is a potent and selective glucagon receptor antagonist.</p>
    Formula:C34H43Cl2N7O2
    Color and Shape:Solid
    Molecular weight:652.66
  • TEI-9063

    CAS:
    <p>TEI-9063 is a stable and highly specific prostacyclin analogue of prostacyclin receptor in mast cell tumor p-815 cells.</p>
    Formula:C23H38O4
    Color and Shape:Solid
    Molecular weight:378.55
  • AL 6598

    CAS:
    <p>AL 6598, a prodrug of PGD2 agonist AL 6556, reduces IOP by 53% at 1μg twice daily in monkeys; binds DP receptors with Ki of 3.2μM.</p>
    Formula:C23H39ClO5
    Color and Shape:Solid
    Molecular weight:431.01
  • Antitumor agent-78


    <p>Antitumor agent-78 blocks GPx-4, raises COX2, triggers apoptosis, halts EMT, and stifles cancer cell growth and migration.</p>
    Color and Shape:Soild
  • LY 292728

    CAS:
    <p>LY 292728 is a highly potent antagonist of leukotriene B4 receptor.</p>
    Formula:C34H29FO9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:600.59
  • 11-trans Leukotriene E4

    CAS:
    <p>Slow isomerization of the C-11 double bond of LTE4 leads to the formation of 11-trans LTE4. 11-trans LTE4 is equipotent to LTE4 in contracting guinea pig ileum.</p>
    Formula:C23H37NO5S
    Color and Shape:Solid
    Molecular weight:439.61
  • TX2-121-1

    CAS:
    <p>TX2-121-1 targets HER3 for proteasome-mediated degradation to inhibit HER3-dependent signalling and growth.</p>
    Formula:C42H52N8O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:716.91
  • Resolvin D1 methyl ester

    CAS:
    <p>Resolvin D1, from docosahexaenoic acid via 15-/5-lipoxygenase, curbs acute inflammation; EC50 ~30 nM. Its methyl ester may enhance bioavailability.</p>
    Formula:C23H34O5
    Color and Shape:Solid
    Molecular weight:390.51
  • AS2521780

    CAS:
    AS2521780 is an inhibitor of PKCθ (IC50: 0.48 nM).
    Formula:C30H41N7OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:547.76
  • IRAK4-IN-11


    <p>IRAK4-IN-11 (compound 6) is a potent inhibitor of IRAK4 with an IC 50 of 0.008 μM. IRAK4-IN-11 exhibits cell pIRAK4 potencies with an IC 50 of 0.19 μM [1].</p>
    Formula:C16H19N7O
    Color and Shape:Solid
    Molecular weight:325.37
  • PDE4B-IN-3


    <p>PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.</p>
    Formula:C30H35N3O4S2
    Color and Shape:Solid
    Molecular weight:565.75
  • Freselestat

    CAS:
    <p>Freselestat (ONO-6818) inhibits neutrophil elastase, reduces interleukin 8, C5B-9, and inflammation in cardiopulmonary bypass.</p>
    Formula:C23H28N6O4
    Color and Shape:Solid
    Molecular weight:452.51
  • ATR-IN-7

    CAS:
    <p>ATR-IN-7 is a potent inhibitor of ATR.</p>
    Formula:C21H22FN7O
    Color and Shape:Solid
    Molecular weight:407.44
  • CDK8-IN-9


    <p>CDK8-IN-9, potent CDK8 inhibitor (IC50: 48.6 nM), curbs tumor growth, useful for colorectal cancer research.</p>
    Color and Shape:Solid
  • L-threo-Sphingosine C-18

    CAS:
    <p>L-threo-Sphingosine C-18 is a protein kinase C inhibitor.</p>
    Formula:C18H37NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.49
  • ROS1-IN-1


    <p>ROS1-IN-1, a potent ROS1 kinase inhibitor, has an IC50 of 0.097 μM.</p>
    Formula:C17H15ClN6S
    Color and Shape:Solid
    Molecular weight:370.86
  • RWJ-56110

    CAS:
    <p>protease-activated receptor-1 (PAR1) antagonist</p>
    Formula:C41H43Cl2F2N7O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:790.73
  • VEGFR-2-IN-11


    <p>VEGFR-2-IN-11 is a potent inhibitor of VEGFR-2 (IC50: 60.27 nM) with an IC50 value of 60.27 nM, which induces apoptosis and has anticancer activity.</p>
    Formula:C29H22BrN5S
    Color and Shape:Solid
    Molecular weight:552.49
  • Menin-MLL inhibitor 4

    CAS:
    Menin-MLL inhibitor 4 has antitumor activity.Menin-MLL inhibitor 4 is an inhibitor of Menin- MLL (mixed-lineage leukemia protein) interaction .
    Formula:C32H38FN7O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:587.69
  • MK-8825

    CAS:
    <p>MK-8825 is a CGRP receptor antagonist.</p>
    Formula:C31H30F2N6O3
    Color and Shape:Solid
    Molecular weight:572.61
  • Tenellin

    CAS:
    <p>Tenellin is a fungal metabolite that inhibits Mg2+-, Ca2+-, and Na+/K+-ATPase activities in erythrocytes. Tenellin is cytotoxic to Sf9 and Sf21 insect cells.</p>
    Formula:C21H23NO5
    Color and Shape:Solid
    Molecular weight:369.41
  • Gusperimus

    CAS:
    <p>Gusperimus was synthesized by chemical modification of spergualin and in combination with cyclosporine A to prevent diabetes in susceptible NOD mice.</p>
    Formula:C17H37N7O3
    Color and Shape:Solid
    Molecular weight:387.52
  • Anti-MRSA agent 6


    <p>Anti-MRSA agent 6 (compound 3q6) is a potent anti-methicillin-resistant Staphylococcus aureus (anti-MRSA) agent with low cytoxicity for MCF-7, A549 cells [1].</p>
    Formula:C16H11F2N3
    Color and Shape:Solid
    Molecular weight:283.28
  • Aplaviroc

    CAS:
    <p>Aplaviroc (AK 602), a SDP derivative, is a CCR5 antagonist. With IC50s of 0.1-0.4 nM for HIV-1Ba-L, HIV-1JRFL and HIV-1MOKW.</p>
    Formula:C33H43N3O6
    Purity:97.98% - 98.26%
    Color and Shape:Solid
    Molecular weight:577.71
  • G-744

    CAS:
    <p>G-744 is a selective and orally active inhibitor of Btk (IC50: 2 nM).</p>
    Formula:C29H29N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:527.64
  • MtDTBS-IN-1


    <p>MtDTBS-IN-1 is a notably potent binder (K_D = 57 nM) and inhibitor (K_i = 5 μM) of MtDTBS.</p>
    Formula:C16H16N4O5
    Color and Shape:Solid
    Molecular weight:344.32
  • trans-Doxercalciferol

    CAS:
    <p>trans-Doxercalciferol is an isomer of Doxercalciferol. Doxercalciferol is an activator of the Vitamin D receptor and prevents renal disease.</p>
    Formula:C28H44O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.65
  • BM635 mesylate


    <p>BM635 mesylate inhibits MmpL3; kills Divergent bacterium with 0.6 µM MIC50; boosts bioavailability.</p>
    Formula:C26H33FN2O4S
    Color and Shape:Solid
    Molecular weight:488.61
  • B026

    CAS:
    <p>B026: Oral p300/CBP HAT inhibitor, IC50: p300 1.8 nM, CBP 9.5 nM; targets AR+ prostate cancer cells.</p>
    Formula:C27H23F4N5O4
    Color and Shape:Solid
    Molecular weight:557.5
  • Lamivudine, (+/-)-trans-

    CAS:
    <p>Lamivudine, a drug for HIV-1 and HBV, inhibits reverse transcriptase and resembles zalcitabine.</p>
    Formula:C8H11N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:229.26
  • Azonafide-PEABA

    CAS:
    <p>Azonafide-PEABA is a drug moiety with cytotoxic [1].</p>
    Formula:C32H33N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:551.64
  • Acetomycin

    CAS:
    <p>Acetomycin, a γ-lactone from S. ramulosus, halts HCT-8 colon and L1210 leukemia cell growth.</p>
    Formula:C10H14O5
    Color and Shape:Solid
    Molecular weight:214.22
  • AD013


    <p>AD013 is a selective ACE inhibitor and NEP inhibitor with potential anti-hypertensive and cardioprotective benefits.</p>
    Formula:C24H28N2O5
    Color and Shape:Solid
    Molecular weight:424.49
  • Geissoschizoline

    CAS:
    <p>Geissoschizoline inhibits human AChE/BChE (IC50: 20.40/10.21 µM) and has anti-inflammatory properties.</p>
    Formula:C19H26N2O
    Color and Shape:Solid
    Molecular weight:298.42
  • ETX0282

    CAS:
    <p>ETX0282, oral class A/C β-lactamase inhibitor, developed by Entasis with cefpodoxime for bacterial infections.</p>
    Formula:C13H18FN3O5
    Color and Shape:Solid
    Molecular weight:315.30
  • Ro-24-4736

    CAS:
    <p>Ro 24-4736 is an effective and selective platelet-activating factor antagonist.</p>
    Formula:C31H20ClN5OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:546.04
  • Anticancer agent 45


    <p>Anticancer agent 46, potent and selective, induces apoptosis, is cytotoxic to cancer cells, with low toxicity to human lymphocytes.</p>
    Formula:C22H14ClN3O6S2
    Color and Shape:Solid
    Molecular weight:515.95
  • Fandosentan

    CAS:
    <p>Fandosentan is an endothelin receptor antagonist.</p>
    Formula:C25H18F3NO6S
    Color and Shape:Solid
    Molecular weight:517.47
  • Autophagy-IN-1


    <p>Autophagy-IN-1 blocks autophagy in cancer cells, hinders tumor growth in mice, and aids in studying colorectal cancer.</p>
    Formula:C23H25NO7
    Color and Shape:Solid
    Molecular weight:427.45
  • SARS 3CLpro-IN-1

    CAS:
    <p>SARS 3CLpro-IN-1: stereospecific SARS 3CL protease inhibitor, octahydroisochromene class, IC50 = 95 μM.</p>
    Formula:C22H38N4O2
    Color and Shape:Solid
    Molecular weight:390.56
  • Asukamycin

    CAS:
    <p>Asukamycin, from S. nodosus asukaensis, is a polyketide antibiotic inhibiting tumor cells by activating caspases 8 and 3.</p>
    Formula:C31H34N2O7
    Color and Shape:Solid
    Molecular weight:546.61
  • Anticancer agent 30


    <p>Anticancer agent 30 (6f-Z), a 3-arylidene-2-oxindole, selectively inhibits CDK2, showing potent anticancer potential.</p>
    Formula:C22H15ClFNO
    Color and Shape:Solid
    Molecular weight:363.81
  • (2R,3S)-Azelaprag

    CAS:
    <p>(2R,3S)-N-(4-(2,6-dimethoxyphenyl)-5-(5-methylpyridin-3-yl)-4H-1,2,4-triazol-3-yl)-3-(5-methylpyrimidin-2-yl)butane-2-sulfonamide is an Apelin receptor agonist</p>
    Formula:C25H29N7O4S
    Purity:97.47% - >99.99%
    Color and Shape:Soild
    Molecular weight:523.61
  • LDHA-IN-5

    CAS:
    <p>LDHA-IN-5 is a novel and potent inhibitor targeting both glycolate oxidase (GO) and lactate dehydrogenase A (LDHA), designed for the treatment of primary</p>
    Formula:C27H22FN7O6S3
    Color and Shape:Solid
    Molecular weight:655.7
  • HBV-IN-20


    <p>HBV-IN-20 is a potent, orally active HBV inhibitor (EC50: 0.46 μM). HBV-IN-20 is a classical type II CpAM (core protein assembly regulator).</p>
    Color and Shape:Solid
  • Retelliptine

    CAS:
    Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.
    Formula:C25H32N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:404.55
  • BMS-751324

    CAS:
    <p>BMS-751324: p38α MAPK inhibitor with carbamyl-methyl, esters, phosphate from HPA. Reduces rat arthritis swelling and TNFα.</p>
    Formula:C32H35N6O10P
    Color and Shape:Solid
    Molecular weight:694.63
  • HSP90-IN-9


    <p>HSP90-IN-9: potent HSP90 inhibitor, dose-dependent fungicide, impedes biofilm/morphology with FLC, reverses FLC resistance.</p>
    Color and Shape:Solid
  • cis-4-Br-2,5-F2-PCPA


    <p>cis-4-Br-2,5-F2-PCPA (S1024) blocks LSD1/LSD2 (Ki: 94 nM/8.4 μM), hinders cancer stem cell growth, raises H3K4me2 in CCRF-CEM cells.</p>
    Formula:C9H8BrF2N
    Color and Shape:Solid
    Molecular weight:248.07
  • Dihydro-β-erythroidine hydrobromide

    CAS:
    <p>Dihydro-β-erythroidine hydrobromide(DHβE) is a potent, oral active and competitive antagonist of neuronal nicotinic acetylcholine receptors (nAChRs).</p>
    Formula:C16H22BrNO3
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:356.26
  • NS2B/NS3-IN-2


    <p>Potent dengue inhibitor NS2B/NS3-IN-2 (IC50: 6 nM, Ki: 0.66 μM) boosts cell viability, non-toxic.</p>
    Formula:C24H21N3O5S
    Color and Shape:Solid
    Molecular weight:463.51
  • α-Glucosidase-IN-17

    CAS:
    <p>α-Glucosidase-IN-17 (Compound 12B) is a potent and orally active inhibitor of α-glucosidase, demonstrating antidiabetic activity with an inhibitory</p>
    Formula:C30H27NO2S
    Color and Shape:Solid
    Molecular weight:465.61
  • Carbacyclin

    CAS:
    <p>Carbacyclin, a PGI2 analog, is a prostacyclin (PGI2) receptor agonist and vasodilator with potent inhibitory platelet aggregation.</p>
    Formula:C21H34O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:350.49
  • Metoquizine

    CAS:
    <p>Metoquizine is an anticholinergic compound. It is a muscarinic acetylcholine receptor antagonist that has been used to treat ulcers.</p>
    Formula:C22H27N5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.48
  • AL-GDa62


    <p>AL-GDa62, a gastric cancer treatment lead, has EC50 of 3.2 μM (MCF10A-WT) and 2 μM (MCF10A-CDH1 -/-).</p>
    Formula:C24H28FN3O
    Color and Shape:Solid
    Molecular weight:393.5
  • hCAII-IN-3


    <p>hCAII-IN-3 inhibits key hCA isoforms with Ki: hCA I (403.8 nM), hCA II (5.1 nM), hCA IX (10.2 nM), hCA XII (5.2 nM); shows anticancer potential.</p>
    Formula:C17H21N3O3S
    Color and Shape:Solid
    Molecular weight:347.43
  • L-2'-Fd4C

    CAS:
    <p>L-2'-Fd4C is an L-nucleoside analogue with both anti-human immunodeficiency virus (HIV) and anti-hepatitis B virus (HBV) activity [1].</p>
    Formula:C9H10FN3O3
    Color and Shape:Solid
    Molecular weight:227.19
  • MAFP

    CAS:
    MAFP (Methyl Arachidonyl Fluorophosphonate) is an effective irreversible inhibitor of anandamide amidase.
    Formula:C21H36FO2P
    Color and Shape:Solid
    Molecular weight:370.48