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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66639 products of "Inhibitors"

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  • KCa2 channel modulator 2


    <p>Compound 2q is a potent, subtype-selective K/Ca 2 modulator, effective on human K Ca 2.3 and rat K Ca 2.2a with EC50s of 0.60 μM and 0.64 μM.</p>
    Formula:C16H15ClFN5
    Color and Shape:Solid
    Molecular weight:331.78
  • Latrunculins A

    CAS:
    <p>Latrunculins A is a novel marine toxin, disrupts microfilament organization in cultured cells.</p>
    Formula:C22H31NO6S
    Color and Shape:Solid
    Molecular weight:437.55
  • TP-6076

    CAS:
    <p>TP-6076 is a fluorocycline antibiotic, inhibiting bacterial protein synthesis, exhibiting great antimicrobial activity against carbapenem-resistant A.</p>
    Formula:C28H32F3N3O7
    Color and Shape:Solid
    Molecular weight:579.56
  • 5(S),6(S)-DiHETE

    CAS:
    <p>5(S),6(S)-DiHETE: a 5,6-dihydroxy acid from LTA4 hydrolysis, lacks leukotriene activity.</p>
    Formula:C20H32O4
    Color and Shape:Solid
    Molecular weight:336.47
  • CXCR2 antagonist 4


    <p>CXCR2 antagonist 4 inhibits CXCR2 (IC50: 0.13 μM) and CXCL8-induced calcium rise (IC50: 27 μM), promising for cancer research.</p>
    Formula:C15H14F2N4OS2
    Color and Shape:Solid
    Molecular weight:368.42
  • Odiparcil

    CAS:
    <p>Odiparcil is an orally active beta-d-thioxyloside analog.</p>
    Formula:C15H16O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.35
  • Ketomethylenebestatin

    CAS:
    <p>Ketomethylenebestatin, a weaker carba-analog of aminopeptidase inhibitor bestatin, is 10x less potent.</p>
    Formula:C17H25NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:307.38
  • Ep vinyl quinidine

    CAS:
    <p>3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.</p>
    Formula:C20H24N2O2
    Color and Shape:Solid
    Molecular weight:324.42
  • CXCR2 antagonist 5


    <p>CXCR2 antagonist 5 (compound 25) binds strongly (IC50=0.013μM) and mobilizes calcium (IC50=0.1μM).</p>
    Formula:C15H14F2N4O2S
    Color and Shape:Solid
    Molecular weight:352.36
  • Anticancer agent 54


    <p>Anticancer agent 54 blocks cell cycle in G0/G1, induces apoptosis, and fights cancer via DNA embedding and ROS.</p>
    Formula:C33H36N6
    Color and Shape:Solid
    Molecular weight:516.68
  • Ganoderic acid R

    CAS:
    <p>Ganoderic acid R: potent anticancer, induces apoptosis, cytotoxic to MDR and sensitive tumor cells.</p>
    Formula:C34H50O6
    Color and Shape:Solid
    Molecular weight:554.76
  • SB 258741 hydrochloride


    <p>SB 258741 hydrochloride is a potent antagonist of the 5-HT 7 receptor, designed specifically for studying schizophrenia [1].</p>
    Formula:C19H31ClN2O2S
    Color and Shape:Solid
    Molecular weight:386.98
  • Dicetrorelix pamoate

    CAS:
    <p>Cetrorelix pamoate is a synthetic decapeptide that acts as a GnRH antagonist, inhibiting the release of LH and FSH from the pituitary.</p>
    Formula:C163H200Cl2N34O34
    Color and Shape:Solid
    Molecular weight:3250.49
  • PI3Kα-IN-8


    <p>PI3Kα-IN-8 is a selective inhibitor of PI3Kα (IC50: 0.012 μM).</p>
    Formula:C26H27BrN4O2
    Color and Shape:Solid
    Molecular weight:507.42
  • DNDI-8219

    CAS:
    <p>DNDI-8219 is an antitubercular agent. It has potent antileishmanial effects.</p>
    Formula:C13H10F3N3O5
    Color and Shape:Solid
    Molecular weight:345.23
  • PF-07202954

    CAS:
    <p>PF-07202954, a weakly basic diacylglycerol O-acyltransferase 2 (DGAT2) inhibitor, exhibits an inhibition concentration half-maximum (IC50) of 10 nM against</p>
    Formula:C22H23FN6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.45
  • GNE-431

    CAS:
    <p>GNE-431: potent, selective noncovalent Btk inhibitor, IC50=3.2 nM; effective against C481R, T474I, T474M mutants, may counter ibrutinib resistance.</p>
    Formula:C30H32N10O2
    Color and Shape:Solid
    Molecular weight:564.64
  • Ganciclovir monophosphonate

    CAS:
    <p>Ganciclovir monophosphate treats CMV, inhibiting replication in human/animal strains (IC50: 0.01μM).</p>
    Formula:C10H16N5O6P
    Color and Shape:Solid
    Molecular weight:333.24
  • HMG499

    CAS:
    <p>HMG499 inhibits HMG-CoA reductase (IC50: 0.41μM), reduces statin-induced HMGCR, lowers cholesterol, and lessens atherosclerosis.</p>
    Formula:C33H54O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.78
  • COX-1/2-IN-2


    <p>COX-1/2-IN-2, a potent dual inhibitor, has IC50s: COX-1 at 9.7μM &amp; COX-2 at 4.6μM.</p>
    Formula:C15H10ClIN2O
    Color and Shape:Solid
    Molecular weight:396.61
  • COX-2/PI3K-IN-2


    <p>COX-2/PI3K-IN-2 (5f): anti-inflammatory &amp; anti-cancer, selectively inhibits COX-2 (Ki=3.02nM), potently blocks PI3K (IC50=2.78nM).</p>
    Formula:C16H17N5O2
    Color and Shape:Solid
    Molecular weight:311.34
  • Carbodine

    CAS:
    <p>Carbodine is an antiviral targeting CTP synthetase, effective against influenza A0/PR-8/34 and A2/Aichi/2/68.</p>
    Formula:C10H15N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:241.24
  • Danshenxinkun D

    CAS:
    <p>Danshenxinkun D has antituberculosis H_(37)Rv activity in vitro.</p>
    Formula:C21H20O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:336.38
  • Etamicastat

    CAS:
    <p>Etamicastat can be used in the research of cardiovascular diseases.</p>
    Formula:C14H15F2N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:311.35
  • Tabimorelin hemifumarate

    CAS:
    <p>orally active ghrelin receptor (GHS-R1a) agonist</p>
    Formula:C32H40N403C4H404
    Purity:98%
    Color and Shape:Solid
    Molecular weight:586.72
  • RSV-IN-5

    CAS:
    <p>RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM &amp; 8.1 nM. Potent anti-RSV.</p>
    Formula:C28H37N7O2
    Color and Shape:Solid
    Molecular weight:503.64
  • Dehatrine

    CAS:
    <p>Dehatrine: alkaloid from Beilschmiedia madang, inhibits Plasmodium falciparum K1 growth.</p>
    Formula:C37H38N2O6
    Color and Shape:Solid
    Molecular weight:606.71
  • UTPγS trisodium salt

    CAS:
    <p>P2Y2 and P2Y4 receptor agonist</p>
    Formula:C9H12N2Na3O14P3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:566.15
  • Mibefradil dihydrochloride hydrate

    CAS:
    <p>Mibefradil dihydrochloride hydrate is a long-acting antihypertensive blocking high-voltage L calcium channels.</p>
    Formula:C29H42Cl2FN3O4
    Color and Shape:Solid
    Molecular weight:586.57
  • DMGF

    CAS:
    <p>DMGF, a biflavonoid from Taxus, induces apoptosis, autophagy, and inhibits B16F10 cell motility and MMP-2 expression, hindering melanoma metastasis.</p>
    Formula:C32H22O10
    Color and Shape:Solid
    Molecular weight:566.51
  • MAP3K14-IN-173

    CAS:
    <p>MAP3K14-IN-173 is a potent MAP3K14 kinase inhibitor.</p>
    Formula:C29H31N7O2
    Color and Shape:Solid
    Molecular weight:509.60
  • C5aR-IN-3

    CAS:
    <p>C5aR-IN-3, a potent C5aR inhibitor, may treat autoimmune and inflammatory diseases.</p>
    Formula:C36H40FN5O3
    Color and Shape:Solid
    Molecular weight:609.73
  • Antitumor agent-72

    CAS:
    <p>Antitumor agent-72 (compound 6w) is a potent anticancer agent that exhibits its anticancer activity by inducing apoptosis via caspase-3 activation and PARP</p>
    Formula:C25H20ClNO6
    Color and Shape:Solid
    Molecular weight:465.88
  • FK-906 HCl

    CAS:
    <p>FK-906 HCl is a human renin inhibitor used for the long-term treatment of patients with essential hypertension.</p>
    Formula:C40H64ClN7O7
    Color and Shape:Solid
    Molecular weight:790.44
  • Carbonic anhydrase inhibitor 9


    <p>Carbonic anhydrase inhibitor 9 targets hCA II and IX with Ki of 56.4 and 56.9 nM respectively; shows antiproliferative activity.</p>
    Formula:C22H20BrN5O4S
    Color and Shape:Solid
    Molecular weight:530.39
  • trans-Doxercalciferol

    CAS:
    <p>trans-Doxercalciferol is an isomer of Doxercalciferol. Doxercalciferol is an activator of the Vitamin D receptor and prevents renal disease.</p>
    Formula:C28H44O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.65
  • ONO-AE1-259 lysine

    CAS:
    <p>ONO-AE1-259 is a highly selective agonist of prostaglandin e2 receptor (ep2)</p>
    Formula:C28H49ClN2O6
    Color and Shape:Solid
    Molecular weight:545.15
  • PCSK9-IN-16

    CAS:
    <p>PCSK9-IN-16, holds potential for research into hypercholesterolemia and other cardiovascular diseases [1].</p>
    Formula:C16H20N6O2S3
    Color and Shape:Solid
    Molecular weight:424.56
  • HBV-IN-12

    CAS:
    <p>HBV-IN-12: strong HBsAg &amp; HBV DNA inhibitor; EC50 0.001-0.05 μM &amp; 0.001-0.02 μM respectively. (WO2021204252A1)</p>
    Formula:C23H27NO8
    Color and Shape:Solid
    Molecular weight:445.46
  • hDDAH-1-IN-2 sulfate


    <p>hDDAH-1-IN-2: selective oral hDDAH-1 inhibitor with low cell toxicity.</p>
    Formula:C8H24N4O10S2
    Color and Shape:Solid
    Molecular weight:400.43
  • Wikstrol A

    CAS:
    <p>Wikstrol A: antifungal, anti-mitotic, anti-HIV agent with various IC50/MDC values (67.8-131 µM) and deforms P. oryzae mycelia.</p>
    Formula:C30H22O10
    Color and Shape:Solid
    Molecular weight:542.49
  • JAK1/TYK2-IN-3


    <p>JAK1/TYK2-IN-3, orally active, selectively inhibits TYK2 (IC50: 6 nM), JAK1 (37 nM), JAK2 (140 nM), JAK3 (362 nM), and has anti-inflammatory effects.</p>
    Color and Shape:Solid
  • CN-716 HCl

    CAS:
    <p>cn-716 is a novel Zika virus (ZIKV) NS2B-NS3pro protease inhibitor.</p>
    Formula:C22H33BCl2N6O4
    Color and Shape:Solid
    Molecular weight:527.25
  • A2A receptor antagonist 2


    <p>A2A receptor antagonist 2 is a highly selective and potent antagonist of the adenosine A2Areceptor (IC50: 8.3 nM).</p>
    Formula:C25H28FN7O3
    Color and Shape:Solid
    Molecular weight:493.53
  • Pociredir

    CAS:
    <p>Pociredir (FTX-6058), a potent EED inhibitor (KD=0.163 nM), may help in SCD research.</p>
    Formula:C22H18FN5O2
    Color and Shape:Solid
    Molecular weight:403.41
  • TLR4/NF-κB/MAPK-IN-1

    CAS:
    <p>TLR4/NF-κB/MAPK-IN-1 is a novel antineuroinflammatory agent that functions by inhibiting the TLR4/NF-κB/MAPK pathways.</p>
    Formula:C19H25BrO6
    Color and Shape:Solid
    Molecular weight:429.3
  • CVS-1578

    CAS:
    <p>CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.</p>
    Formula:C20H30N6O5S
    Color and Shape:Solid
    Molecular weight:466.55
  • Belotecan

    CAS:
    <p>Belotecan (CKD-602) inhibits DNA topoisomerase I, blocks cell cycle, induces apoptosis, and is a camptothecin-derived anticancer agent.</p>
    Formula:C25H27N3O4
    Color and Shape:Solid
    Molecular weight:433.5
  • Ro 0437626

    CAS:
    <p>P2X1 purinergic receptor antagonist</p>
    Formula:C27H35N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:525.66
  • Antifungal agent 38


    <p>Antifungal agent 38, a heterocyclic disulfide, shrinks hyphae and damages cell membranes, causing leakage.</p>
    Formula:C8H12N2S2
    Color and Shape:Solid
    Molecular weight:200.32
  • α5β1 integrin agonist-1

    CAS:
    <p>α5β1 integrin agonist-1 is an α5β1 integrin agonist that selectively delivers 5-FU to tumour cells and induces tumour cell death.</p>
    Formula:C24H26FN5O9
    Color and Shape:Solid
    Molecular weight:547.49
  • QPX7728 methoxy acetoxy methy ester

    CAS:
    <p>QPX7728 methoxy acetoxy methy ester is an inhibitor of boronic acid β-lactamase.</p>
    Formula:C14H14BFO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.07
  • Intoplicine

    CAS:
    <p>Intoplicine is an inhibitor of DNA topoisomerase I and II.</p>
    Formula:C21H24N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.44
  • LY3325656

    CAS:
    <p>LY3325656, a GPR142 agonist with anti-diabetic properties, progresses to phase 1 trials for Type 2 diabetes.</p>
    Formula:C21H23F3N6O2
    Color and Shape:Solid
    Molecular weight:448.44
  • (±)-ANAP hydrochloride (1185251-08-4 free base)


    <p>(±)-ANAP hydrochloride is the amino acid analog of prodan. It can be used as a fluorescent probes and enhance environmental sensitivity.</p>
    Formula:C15H17ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:308.76
  • Pol I-IN-1


    <p>Pol I-IN-1 is a powerful inhibitor of RNA polymerase I (Pol I), specifically targeting the large catalytic subunit RPA194, demonstrating an inhibition</p>
    Formula:C23H22N4O2
    Color and Shape:Solid
    Molecular weight:386.45
  • Fandosentan

    CAS:
    <p>Fandosentan is an endothelin receptor antagonist.</p>
    Formula:C25H18F3NO6S
    Color and Shape:Solid
    Molecular weight:517.47
  • CB1/2 agonist 1


    <p>Potent CB1/2 agonist 1; crosses blood-brain barrier; anti-inflammatory, analgesic; for multiple sclerosis research.</p>
    Formula:C21H24BrFN2O2
    Color and Shape:Solid
    Molecular weight:435.33
  • Tofacitinib Prodrug-1


    <p>Tofacitinib Prodrug-1: an oral prodrug reducing Tofacitinib's side effects, treats ulcerative colitis in mice effectively with low toxicity.</p>
    Formula:C36H39ClN10O7
    Color and Shape:Solid
    Molecular weight:759.21
  • PrCP-7414

    CAS:
    <p>PrCP-7414 is a potent PrCP inhibitor, CAS# 1252037-41-4, named after the CAS number's last four digits.</p>
    Formula:C31H33Cl2N5O2
    Color and Shape:Solid
    Molecular weight:578.53
  • PEN-866

    CAS:
    <p>PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.</p>
    Formula:C49H49N7O9
    Color and Shape:Solid
    Molecular weight:879.95
  • AT1R antagonist 2


    <p>AT1R antagonist 2 is a potent AT1R selective ligand with good AT1R affinity (Ki: 26 nM).</p>
    Formula:C29H37N5O4S2
    Color and Shape:Solid
    Molecular weight:583.77
  • CREB-IN-1 TFA


    <p>CREB-IN-1 TFA: Potent oral CREB inhibitor, IC50 of 0.18 μM, suppresses breast cancer cell growth.</p>
    Color and Shape:Solid
  • Kri 1314

    CAS:
    <p>Kri 1314 is a cyclohexyl-norstatine-containing dipeptide renin inhibitor which has potential for the treatment of hypertension.</p>
    Formula:C38H51N5O7
    Color and Shape:Solid
    Molecular weight:689.84
  • Napsagatran hydrate

    CAS:
    <p>Napsagatran hydrate is a novel and specific inhibitor of thrombin.</p>
    Formula:C26H36N6O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:576.66
  • Autophagy-IN-1


    <p>Autophagy-IN-1 blocks autophagy in cancer cells, hinders tumor growth in mice, and aids in studying colorectal cancer.</p>
    Formula:C23H25NO7
    Color and Shape:Solid
    Molecular weight:427.45
  • Topoisomerase I/II inhibitor 4


    <p>Topoisomerase I/II inhibitor 4 halts cell growth and spread, induces apoptosis, and is used in liver cancer research.</p>
    Formula:C27H21N5O6
    Color and Shape:Solid
    Molecular weight:511.49
  • Cav 3.2 inhibitor 3


    <p>Cav 3.2 inhibitor 3 is a potent inhibitor of the Cav3.2 T-type Ca2+channel (IC50: 0.1534 μM) and has a low binding affinity for D2 receptors.</p>
    Formula:C32H37N3O2
    Color and Shape:Solid
    Molecular weight:495.66
  • LSD1-IN-16


    <p>LSD1-IN-16 (4b) inhibits LSD1, MAO-A/B; IC50: 0.015-0.366 μM. Halts prostate cancer cell growth; IC50: 15.2 μM.</p>
    Formula:C20H18N2OS
    Color and Shape:Solid
    Molecular weight:334.43
  • (R)-ZG197


    <p>(R)-ZG197: Activates Sa ClpP (EC50=1.5μM) &amp; Hs ClpP (EC50=31.4μM); selective for Sa ClpP.</p>
    Formula:C28H35F3N4O3
    Color and Shape:Solid
    Molecular weight:532.6
  • NBTIs-IN-4


    <p>NBTIs-IN-4, a broad-spectrum Gram-positive antibacterial, inhibits DNA rotamases/topoisomerase IV, with low resistance.</p>
    Formula:C22H24FN5O5S
    Color and Shape:Solid
    Molecular weight:489.52
  • Topoisomerase I/II inhibitor 3


    <p>Topoisomerase I/II inhibitor 3 suppresses cell growth and induces apoptosis in liver cancer by blocking PI3K/Akt/mTOR.</p>
    Formula:C24H24N2O4
    Color and Shape:Solid
    Molecular weight:404.46
  • IRAK4-IN-15

    CAS:
    <p>IRAK4-IN-15: selective IRAK4 inhibitor, IC50 0.002 μM, good PK, low clearance, synergizes with Acalabrutinib in MyD88/CD79 mutant ABC-DLBCL.</p>
    Formula:C25H29FN10
    Color and Shape:Solid
    Molecular weight:488.56
  • β-Glucuronidase/hCAII-IN-2


    <p>β-Glucuronidase/hCAII-IN-2 is a potent inhibitor of β-glucuronidase and hCA II, and their IC50 values were 670.7 μM and 21.77 μM, respectively.</p>
    Formula:C31H23NO8
    Color and Shape:Solid
    Molecular weight:537.52
  • PARP-1/HDAC-IN-1

    CAS:
    <p>PARP-1/HDAC-IN-1 is a PARP-1 and HDAC6 inhibitor with anticancer, antimigratory, and antiangiogenic activities and is used in tumor research.</p>
    Formula:C22H18N4O4
    Purity:95.94%
    Color and Shape:Solid
    Molecular weight:402.4
  • 8(S),15(S)-DiHETE

    CAS:
    <p>8(S),15(S)-DiHETE, from 15(S)-HETE's oxidation by 15-LO, triggers eosinophil movement at 1.5 μM; it counteracts pain and LTB4 effects.</p>
    Formula:C20H32O4
    Color and Shape:Solid
    Molecular weight:336.47
  • BMS-248360

    CAS:
    <p>BMS-248360: Oral dual hAT1/hETA antagonist with Kis of 10nM &amp; 1.9nM, respectively; treats hypertension.</p>
    Formula:C36H45N5O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:659.84
  • Antiproliferative agent-3


    <p>Antiproliferative agent-3 (comp 4) exhibits potent growth inhibitory effects against MCF-7 cells with IC 50 of 0.19 nM [1].</p>
    Formula:C11H12N2O5S
    Color and Shape:Solid
    Molecular weight:284.29
  • Naldemedine tosylate

    CAS:
    <p>Naldemedine (S-297995) tosylate, a PAMORA, targets μ-, δ-, κ-opioid receptors, aiding OIC research, may bind to SARS-CoV2's 3CL pro.</p>
    Formula:C39H42N4O9S
    Color and Shape:Solid
    Molecular weight:742.84
  • GS-9160

    CAS:
    <p>GS-9160 is a novel and potent inhibitor of human immunodeficiency virus type 1 (HIV-1) integrase (IN) that specifically targets the process of strand transfer.</p>
    Formula:C20H18FN3O4S
    Color and Shape:Solid
    Molecular weight:415.44
  • (Rac)-PT2399

    CAS:
    <p>(Rac)-PT2399 is a potent and specific inhibitor of hypoxia-inducible factor 2a (HIF-2α)(IC50 of 0.01 μM).</p>
    Formula:C17H10F5NO4S
    Color and Shape:Solid
    Molecular weight:419.32
  • NS2B/NS3-IN-3

    CAS:
    <p>NS2B/NS3-IN-3 (Compd 66) is an inhibitor of Flavivirus NS2B-NS3 protease [1] .</p>
    Formula:C19H21N3O2
    Color and Shape:Solid
    Molecular weight:323.39
  • L 156903

    CAS:
    <p>L 156903 is a bioactive chemical. It also inhibits the binding of neurotensin to brain tissue.</p>
    Formula:C35H41N7O5S
    Color and Shape:Solid
    Molecular weight:671.81
  • PF-06795071

    CAS:
    <p>PF-06795071 is an effective and selective covalent inhibitor of MAGL (IC50: 3 nM).</p>
    Formula:C18H17F4N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.34
  • PqsR-IN-1


    <p>PqsR-IN-1, potent PqsR inhibitor, curbs pyocyanin in Pseudomonas aeruginosa with low cytotoxicity.</p>
    Formula:C17H18ClN3OS
    Color and Shape:Solid
    Molecular weight:347.86
  • CDK1-IN-3


    <p>CDK1-IN-3 is a selective inhibitor targeting CDK1 (36.8 nM), CDK2 (305.17 nM), CDK5 (369.37 nM); used in cancer research.</p>
    Formula:C28H25ClF3N5O2
    Color and Shape:Solid
    Molecular weight:555.98
  • CXCR4 modulator-1

    CAS:
    <p>CXCR4 modulator-1 (ZINC72372983) is potent (EC50=100nM) with uses in anti-inflammatory, anticancer, and anti-HIV research.</p>
    Formula:C23H27N5O2
    Color and Shape:Solid
    Molecular weight:405.49
  • (S)-Butaprost free acid

    CAS:
    <p>(S)-Butaprost (free acid) is a potent and highly selective EP2 receptor agonist[1].</p>
    Formula:C23H38O5
    Color and Shape:Solid
    Molecular weight:394.54
  • MtTMPK-IN-8


    <p>MtTMPK-IN-8 inhibits MtbTMPK, has low cytotoxicity, shows 0.78-9.4 μM activity against Mycobacterium, useful for tuberculosis research.</p>
    Formula:C24H24N6O7
    Color and Shape:Solid
    Molecular weight:508.48
  • BW A868C

    CAS:
    BW A868C is a potent, selective PGD2 antagonist and a BW245C analogue, inert to other prostaglandin receptors.
    Formula:C25H37N3O5
    Color and Shape:Solid
    Molecular weight:459.58
  • PTP1B-IN-21


    <p>PTP1B-IN-21 inhibits PTP1B (IC50=1.56μM) selectively over TCPTP, a type 2 diabetes target.</p>
    Formula:C22H22O11
    Color and Shape:Solid
    Molecular weight:462.4
  • ONO-AE1-329

    CAS:
    <p>ONO-AE1-329 is a novel agonist of the prostaglandin PGE2 receptor EP4.</p>
    Formula:C22H30O6S2
    Color and Shape:Solid
    Molecular weight:454.6
  • GNE684

    CAS:
    <p>GNE684 inhibits RIP1; Ki app: 21 nM (human), 189 nM (mouse), 691 nM (rat).</p>
    Formula:C23H24N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.48
  • α-Glucosidase-IN-12


    <p>α-Glucosidase-IN-12 is a potent inhibitor of α-glucosidase (IC50: 10.20 μM).</p>
    Formula:C25H30N4O4S2
    Color and Shape:Solid
    Molecular weight:514.66
  • MEIS-IN-1

    CAS:
    <p>MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.</p>
    Formula:C24H21F3N2O4
    Color and Shape:Solid
    Molecular weight:458.43
  • Antitumor agent-58


    <p>Antitumor agent-58 suppresses tumor growth, colony formation, cell migration, and induces mitochondrial dysfunction in MGC-803 cells.</p>
    Formula:C27H28F3N9S
    Color and Shape:Solid
    Molecular weight:567.63
  • Pralatrexate, (R)-

    CAS:
    <p>Pralatrexate is a high-affinity DHFR inhibitor targeting RFC-1, used in cancer treatment and immunosuppression.</p>
    Formula:C23H23N7O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:477.47
  • TNP-470

    CAS:
    <p>TNP-470 is a methionine aminopeptidase-2 inhibitor. TNP-470 is also an angiogenesis inhibitor.</p>
    Formula:C19H28ClNO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.88
  • Canosimibe

    CAS:
    <p>Canosimibe is a cholesterol absorption inhibitor</p>
    Formula:C44H60FN3O10
    Color and Shape:Solid
    Molecular weight:809.96
  • A25822B

    CAS:
    <p>A25822B is an antifungal agent.</p>
    Formula:C28H45NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.66