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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66639 products of "Inhibitors"

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  • Dihydrokainic acid

    CAS:
    <p>EAAT2(GLT1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptake</p>
    Formula:C10H17NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:215.25
  • Nrf2 activator-2


    <p>Compound O15, an Osthole derivative, is a potent Nrf2 agonist with an EC50 of 2.9 μM; it inhibits Keap1-Nrf2 binding and Nrf2 ubiquitination.</p>
    Formula:C20H17BrO3
    Color and Shape:Solid
    Molecular weight:385.25
  • Sagopilone

    CAS:
    <p>Sagopilone: synthetic epothilone, inhibits cell division and induces apoptosis, effective in MDR tumors, not P-gp substrate.</p>
    Formula:C30H41NO6S
    Color and Shape:Solid
    Molecular weight:543.71
  • BRD0418

    CAS:
    <p>BRD0418 acts as an upregulator of TRIB1 expression by leading to reprogramming of hepatic lipoprotein metabolism from adipogenesis to clearance it.</p>
    Formula:C29H32N2O5
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:488.57
  • LasR-IN-1


    <p>LasR-IN-1 (9g) strongly inhibits LasR, potent vs E. coli, with a 28.13 μM MIC against P. aeruginosa.</p>
    Formula:C23H21N3O2
    Color and Shape:Solid
    Molecular weight:371.43
  • hDHODH-IN-10


    <p>hDHODH-IN-10: selective oral inhibitor of hDHODH (IC50: 10.9 nM); blocks cancer cell growth, aids cancer research.</p>
    Formula:C21H15ClF4N2O4
    Color and Shape:Solid
    Molecular weight:470.8
  • FAK-IN-3


    <p>FAK-IN-3 inhibits FAK, reduces PA-1 cell migration/invasion, and tumor growth, with no major side effects.</p>
    Formula:C28H28N6O4
    Color and Shape:Solid
    Molecular weight:512.56
  • CU-2010

    CAS:
    <p>CU-2010 is a synthetic compound that reduces blood loss and aids recovery post-cardiac surgery.</p>
    Formula:C37H42N6O6S
    Color and Shape:Solid
    Molecular weight:698.83
  • BMS-986339

    CAS:
    <p>BMS-986339: oral, potent FXR agonist; binds to His298/ASN287; for PBC, PSC, NASH, anti-fibrosis research.</p>
    Formula:C35H41F4N3O4
    Color and Shape:Solid
    Molecular weight:643.71
  • Lepidozin G


    <p>Lepidozin G blocks cancer growth (IC50=4.2-5.7μM) and triggers apoptosis in PC-3 cells via mitochondria.</p>
    Formula:C30H48O4
    Color and Shape:Solid
    Molecular weight:472.7
  • SZ1676

    CAS:
    <p>SZ1676 is a derivative of SZ1677, which is an agent of neuromuscular blocking.</p>
    Formula:C37H59BrN2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:707.78
  • PARP10/15-IN-2

    CAS:
    <p>PARP10/15-IN-2 (Compound 8h) blocks PARP10/15, has IC50s: 0.15μM/0.37μM, cell-permeable, prevents apoptosis.</p>
    Formula:C15H11FN2O3
    Color and Shape:Solid
    Molecular weight:286.26
  • EBI-1051

    CAS:
    <p>EBI-1051 is a highly potent and orally efficacious inhibitor of MEK (IC50: 3.9 nM).</p>
    Formula:C18H15F2IN2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:504.22
  • MtMetAP1-IN-1


    <p>MtMetAP1-IN-1 is an inhibitor of methionine aminopeptidase 1 ( MetAP1 ). MtMetAP1-IN-1 shows antimycobacterial activity.</p>
    Formula:C15H10BrN5O2S
    Color and Shape:Solid
    Molecular weight:404.24
  • Complex III-IN-1


    <p>Complex III-IN-1 inhibits complex III, has antifungal properties, and an EC50 of 18.53 mg/L against S. sclerotiorum.</p>
    Formula:C14H20ClNO2S2
    Color and Shape:Solid
    Molecular weight:333.9
  • MsbA-IN-2


    <p>MsbA-IN-2 is a potent inhibitor of the lipopolysaccharide transporter MsbA and is able to act on E. coli MsbA (IC50: 2 nM).</p>
    Formula:C23H19Cl2NO3
    Color and Shape:Solid
    Molecular weight:428.31
  • (S)-Butaprost free acid

    CAS:
    <p>(S)-Butaprost (free acid) is a potent and highly selective EP2 receptor agonist[1].</p>
    Formula:C23H38O5
    Color and Shape:Solid
    Molecular weight:394.54
  • CY208-243 Mandelate

    CAS:
    <p>CY208-243 is a D1 agonist boosting memory in T-maze, enhances adenylate cyclase (EC50=125nM), and alters monkey electroretinogram.</p>
    Formula:C27H26N2O3
    Color and Shape:Solid
    Molecular weight:426.52
  • PLP_Snyder530


    <p>PLP_Snyder530, a potent PL pro inhibitor, halts SARS-CoV-2 by triggering protease conformation changes.</p>
    Formula:C24H24N2O2
    Color and Shape:Solid
    Molecular weight:372.46
  • Tubulin inhibitor 14


    <p>Tubulin inhibitor 14 blocks NQO2 and microtubule formation, disrupts blood vessels, and may target tumors; IC50 of 1.0 μM.</p>
    Formula:C15H9F2NO
    Color and Shape:Solid
    Molecular weight:257.23
  • MS8815

    CAS:
    <p>MS8815 is a selective EZH2 PROTAC degrader with IC50 of 8.6 nM, used in triple-negative breast cancer research.</p>
    Formula:C65H87N9O8S
    Color and Shape:Solid
    Molecular weight:1154.51
  • Tubulin polymerization-IN-9

    CAS:
    <p>Tubulin-IN-9 inhibits tubulin (IC50: 1.82 μM), halts K562 cells in G2/M, induces apoptosis, and has anti-cancer effects.</p>
    Formula:C19H19NO5Se
    Color and Shape:Solid
    Molecular weight:420.32
  • Naltalimide

    CAS:
    <p>Naltalimide: µ-opioid receptor partial agonist, improves bladder storage by affecting spinal cord reflex.</p>
    Formula:C28H28N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.53
  • Myxothiazol

    CAS:
    <p>Myxothiazol blocks mitochondrial complex III and triggers SESN2, a gene important for stress response.</p>
    Formula:C25H33N3O3S2
    Color and Shape:Solid
    Molecular weight:487.68
  • Avibactam sodium dihydrate


    <p>Avibactam sodium dihydrate (NXL-104) is a reversible covalent inhibitor for CTX-M-15 and TEM-1 β-lactamases with IC50s of 5 nM and 8 nM.</p>
    Formula:C7H14N3NaO8S
    Color and Shape:Solid
    Molecular weight:323.26
  • Indoluidin E


    <p>Indoluidin E selectively inhibits DHODH and has an inhibitory effect on cancer cell growth.</p>
    Formula:C28H30N4O2
    Color and Shape:Solid
    Molecular weight:454.56
  • LA-810

    CAS:
    <p>LA-810 is a nitrous oxide donor.</p>
    Formula:C15H25N5O7S
    Color and Shape:Solid
    Molecular weight:419.45
  • CK156

    CAS:
    <p>CK156 inhibits DAPK with high selectivity; IC50: 182 nM (DRAK1), 34 μM (CK2a1), 39 μM (CK2a2); key in autoimmune/inflammation research.</p>
    Formula:C21H25N5O3
    Color and Shape:Solid
    Molecular weight:395.45
  • Macbecin I

    CAS:
    <p>Hsp90 inhibitor</p>
    Formula:C30H42N2O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:558.66
  • GNE-616

    CAS:
    <p>GNE-616: a potent, stable, oral Nav1.7 inhibitor; Ki: 0.79 nM, Kd: 0.38 nM; for chronic pain.</p>
    Formula:C24H23F4N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:537.53
  • MCB-3681

    CAS:
    <p>MCB-3681, active against gram-positive bacterium, is the antibacterial Oxaquin's active substance.</p>
    Formula:C31H32F2N4O8
    Color and Shape:Solid
    Molecular weight:626.6
  • DC1SMe

    CAS:
    <p>DC1, a CC-1065-like ADC cytotoxin, is used in cancer-targeting antibody-drug conjugates. DC1Sme, a derivative, has IC50s: 22-250 pm in various cancer cells.</p>
    Formula:C35H30ClN5O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:684.23
  • mPGES-1-IN-1


    <p>MPGES-1, potential anti-inflammatory drug target, has IC50 of 0.03 μM with mPGES-1-IN-1.</p>
    Formula:C21H14N4O2S
    Color and Shape:Solid
    Molecular weight:386.43
  • Resolvin D1 methyl ester

    CAS:
    <p>Resolvin D1, from docosahexaenoic acid via 15-/5-lipoxygenase, curbs acute inflammation; EC50 ~30 nM. Its methyl ester may enhance bioavailability.</p>
    Formula:C23H34O5
    Color and Shape:Solid
    Molecular weight:390.51
  • SSM3 TFA

    CAS:
    <p>SSM3 TFA is a potent furin inhibitor, blocking furin-dependent cell surface processing of anthrax protective antigen-83 in vitro..</p>
    Formula:C22H32N12O2
    Color and Shape:Solid
    Molecular weight:496.57
  • Ceclazepide

    CAS:
    <p>Ceclazepide is an antagonist of cholecystokinin receptor.</p>
    Formula:C30H32N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:556.61
  • PPARγ phosphorylation inhibitor 1


    <p>PPARγ phosphorylation inhibitor 1 (Compound 10) is a potent PPARγ binding agent (IC50: 24 nM) with antidiabetic effects.</p>
    Formula:C22H14Cl2N2O4
    Color and Shape:Solid
    Molecular weight:441.26
  • AMG-548 dihydrochloride


    <p>AMG-548 dihydrochloride, an oral p38α inhibitor (Ki: 0.5 nM), selectively targets p38β, γ, δ, inhibits TNFα (IC50: 3 nM), and suppresses Wnt signaling.</p>
    Formula:C29H29Cl2N5O
    Color and Shape:Solid
    Molecular weight:534.48
  • Verrucarin A

    CAS:
    <p>Verrucarin A, a mycotoxin from Myrothecium verrucaria, inhibits protein synthesis, leukemia growth, and triggers apoptosis.</p>
    Formula:C27H34O9
    Color and Shape:Solid
    Molecular weight:502.55
  • 2-Methylsorbinol

    CAS:
    <p>2-Methylsorbinol is a bioactive chemical.</p>
    Formula:C12H11FN2O3
    Color and Shape:Solid
    Molecular weight:250.23
  • PDE4B-IN-3


    <p>PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.</p>
    Formula:C30H35N3O4S2
    Color and Shape:Solid
    Molecular weight:565.75
  • OncoFAP

    CAS:
    <p>OncoFAP is an ultra-high affinity fibroblast activating protein (FAP) ligand with potential tumour targeting.</p>
    Formula:C21H19F2N5O5
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:459.40
  • RMS-07

    CAS:
    <p>RMS-07, a covalent MPS1/TTK inhibitor, has an IC50 of 13.1 nM, targeting a kinase hinge cysteine.</p>
    Formula:C35H40N8O2
    Color and Shape:Solid
    Molecular weight:604.74
  • (+)-Cevimeline hydrochloride hemihydrate


    <p>(+)-Cevimeline HCl hemihydrate is a muscarinic agonist for dry mouth in Sjogren's with rapid absorption, differing metabolism in species.</p>
    Formula:C10H19ClNO1·5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:244.78
  • BCL6-IN-9

    CAS:
    <p>BCL6-IN-9 (compound 1) is a potent inhibitor of B-cell lymphoma 6 protein (BCL6) (IC50: 3.9 nM) and can be used to study cancer.</p>
    Formula:C22H18ClF2N5O2
    Color and Shape:Solid
    Molecular weight:457.86
  • SML-10-70-1

    CAS:
    <p>SML-10-70-1 is a Novel Active Site Inhibitor of Oncogenic K-Ras G12C.</p>
    Formula:C25H42ClN7O13P2
    Color and Shape:Solid
    Molecular weight:746.04
  • Suloctidil HCl

    CAS:
    <p>Suloctidil HCl is a peripheral vascular dilator.</p>
    Formula:C20H36ClNOS
    Color and Shape:Solid
    Molecular weight:374.02
  • ODN 2088

    CAS:
    <p>ODN 2088 is a potent inhibitor of TLR3, TLR7 and TLR9 that is non-cytotoxic and shows inhibition of the release of IFN-α and IL-6.</p>
    Color and Shape:Solid
  • ABD957

    CAS:
    <p>ABD957: covalent ABHD17 depalmitoylases inhibitor, IC50 0.21µM for ABHD17B, blocks N-Ras, halts NRAS-mutant AML cell growth.</p>
    Formula:C27H36F3N7O5S
    Color and Shape:Solid
    Molecular weight:627.68
  • BI-44370

    CAS:
    <p>BI-44370, a CGRP (calcitonin gene-related peptide) receptor antagonist, can be used to treat migraines and other chronic pain.</p>
    Formula:C35H47N5O6
    Color and Shape:Solid
    Molecular weight:633.78
  • EGFR/HER2/DHFR-IN-1


    <p>Potent EGFR/HER2/DHFR inhibitor for MCF-7 breast cancer; IC50: 0.153/0.108/0.291 μM; arrests G1/S phase, triggers apoptosis.</p>
    Formula:C14H11BrN4O2S
    Color and Shape:Solid
    Molecular weight:379.23
  • TGR5 Receptor Agonist 3

    CAS:
    <p>TGR5 Receptor Agonist 3 is a GPBAR1 agonist with EC50 of 16.4 nM (hTGR5) &amp; 209 nM (mTGR5), ensures gallbladder safety and reduces filling.</p>
    Formula:C29H27N3O6
    Color and Shape:Solid
    Molecular weight:513.54
  • LY 190388

    CAS:
    <p>LY 190388 is a penicillamine-containing enkephalin analog used as an mu receptor agonist with analgesia activity.</p>
    Formula:C30H41N5O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:615.74
  • LSD1/2-IN-4


    <p>LSD1/2-IN-4, a PCPA derivative, inhibits LSD1 (Ki 0.11 μM) &amp; LSD2 (Ki 130 μM), potentially useful in T-cell leukemia research.</p>
    Formula:C9H8BrF2N
    Color and Shape:Solid
    Molecular weight:248.07
  • CDK8-IN-5

    CAS:
    <p>CDK8-IN-5: potent CDK8 inhibitor, IC50=72 nM, boosts IL-10 by 43%, may aid inflammatory bowel disease research.</p>
    Formula:C26H22N2O4
    Color and Shape:Solid
    Molecular weight:426.46
  • β-Glucuronidase-IN-2


    <p>β-Glucuronidase-IN-2 is a potent inhibitor of E.</p>
    Formula:C21H17Cl3O7
    Color and Shape:Solid
    Molecular weight:487.71
  • PDE4-IN-14

    CAS:
    <p>PDE4-IN-14 (Compound 1) serves as an inhibitor of phosphodiesterase 4 (PDE4), applicable in research concerning diseases associated with PDE4, including</p>
    Formula:C19H20F2N4O3S
    Color and Shape:Solid
    Molecular weight:422.45
  • SX 3202

    CAS:
    <p>SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.</p>
    Formula:C17H11BrFN3O4
    Color and Shape:Solid
    Molecular weight:420.19
  • FGFR3-IN-4

    CAS:
    <p>FGFR3-IN-4 is a selective inhibitor targeting FGFR3, demonstrating an IC50 value of under 50 nM.</p>
    Formula:C26H24ClN7O
    Color and Shape:Solid
    Molecular weight:485.97
  • TRPC5-IN-4

    CAS:
    <p>TRPC5-IN-4: Potent, safe inhibitor; IC50 14.07 nM (TRPC5), 65 nM (TRPC4); non-toxic to liver/kidney cells; for CKD research.</p>
    Formula:C18H11ClF4N4O3
    Color and Shape:Solid
    Molecular weight:442.75
  • Minnelide free acid

    CAS:
    <p>Minnelide treats pancreatic cancer, hinders androgen-related prostate growth, shrinks tumors, and improves survival.</p>
    Formula:C21H27O10P
    Color and Shape:Solid
    Molecular weight:470.41
  • CXCR2 antagonist 5


    <p>CXCR2 antagonist 5 (compound 25) binds strongly (IC50=0.013μM) and mobilizes calcium (IC50=0.1μM).</p>
    Formula:C15H14F2N4O2S
    Color and Shape:Solid
    Molecular weight:352.36
  • K252d

    CAS:
    <p>K252d: indolocarbazole alkaloid in Nocardiopsis; inhibits PKC in rat brain and bovine heart phosphodiesterase.</p>
    Formula:C26H23N3O5
    Color and Shape:Solid
    Molecular weight:457.48
  • IDO1-IN-14


    <p>IDO1-IN-14 is an IDO1 enzyme inhibitor with an IC50 of 396.9 nM and suppresses HeLa cell activity with an EC50 of 3393 nM.</p>
    Formula:C18H12Cl2FN3O2
    Color and Shape:Solid
    Molecular weight:392.21
  • MIV-150

    CAS:
    <p>MIV-150 is a nonnucleoside inhibitor of reverse transcriptase (NNRT). MIV-150 also blocking HIV-1 and HIV-2 infections (EC50&lt;1 nM against HIV-1/HIV-2MN).</p>
    Formula:C19H17FN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.36
  • XIAP/cIAP1 antagonist-1


    <p>Potent oral XIAP/cIAP1 inhibitor with EC50s: XIAP 5.1 nM, cIAP1 0.32 nM; curbs tumor growth in vivo.</p>
    Color and Shape:Solid
  • GNTI TFA

    CAS:
    <p>GNTI TFA is a selective kappa opioid receptor antagonist.</p>
    Formula:C31H31F6N5O7
    Color and Shape:Solid
    Molecular weight:699.60
  • GG-43


    <p>GG-43 is a potent inhibitor of LIN28. The IC50 value of GG-43 against human LIN28A is 4 μM [1].</p>
    Formula:C21H21NO3
    Color and Shape:Solid
    Molecular weight:335.4
  • Silvestrol

    CAS:
    <p>Silvestrol is a eukaryotic translation initiation factor 4A inhibitor. Silvestrol causes autophagy and caspase-mediated apoptosis.</p>
    Formula:C34H38O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:654.66
  • Anticancer agent 26


    <p>Anticancer agent 26 is a promising candidate for cancer therapy and deserves further development.</p>
    Formula:C28H33NO5
    Color and Shape:Solid
    Molecular weight:463.57
  • Zanapezil fumarate

    CAS:
    <p>Zanapezil is an acetylcholinesterase (AChE) inhibitor. Zanapezil increases choline acetyltransferase activity in cultured rat septal cholinergic neurons.</p>
    Formula:C29H36N2O5
    Color and Shape:Solid
    Molecular weight:492.61
  • iNOS/PGE2-IN-1


    <p>iNOS/PGE2-IN-1: iNOS/PGE2 inhibitor, reduces LPS-induced NO, low ulcer risk, anti-inflammatory.</p>
    Formula:C26H22ClN3O4
    Color and Shape:Solid
    Molecular weight:475.92
  • BTK-IN-6


    <p>BTK-IN-6, a potent BTK inhibitor, may treat immune, cardiac, cancer, viral, inflammatory, metabolic, and neurological disorders.</p>
    Formula:C23H22FN5O3
    Color and Shape:Solid
    Molecular weight:435.45
  • (S)-Purvalanol B

    CAS:
    <p>(S)-Purvalanol B is the S enantiomer of Purvalanol B. Purvalanol B is an inhibitor of cyclin-dependent kinase(CDK) .</p>
    Formula:C20H25ClN6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.9
  • HDAC2-IN-1


    <p>HDAC2-IN-1 is an oral HDAC2 inhibitor (IC50: 0.5 μM), crosses the blood-brain barrier, and inhibits HDAC1 and HDAC8.</p>
    Formula:C22H23ClN4OS
    Color and Shape:Solid
    Molecular weight:426.96
  • YK5

    CAS:
    <p>YK5 is an allosteric inhibitor pocket of Hsp70 and represents a previously unknown chemical tool to investigate cellular mechanisms associated with Hsp70.</p>
    Formula:C18H24N8O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.50
  • Revexepride

    CAS:
    <p>Revexepride, a 5-HT4 agonist, may boost CYP3A4, used for treating GERD.</p>
    Formula:C21H32ClN3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:425.95
  • ONO-DI-004

    CAS:
    <p>ONO-DI-004 is a selective EP1 Prostanoid receptor agonist.</p>
    Formula:C24H38O6
    Color and Shape:Solid
    Molecular weight:422.55
  • Dual AChE-MAO B-IN-1


    <p>Dual AChE-MAO B-IN-1: orally active CNS-permeable, safe, stable neuroprotective agent; AChE IC50=550 nM, MAO-B IC50=8.2 nM.</p>
    Formula:C23H25F2NO4
    Color and Shape:Solid
    Molecular weight:417.45
  • Amdinocillin methylacetate

    CAS:
    <p>Amdinocillin methylacetate is a Synthetic penicillin.</p>
    Formula:C18H27N3O4S
    Color and Shape:Solid
    Molecular weight:381.49
  • AChE-IN-10


    <p>AChE-IN-10 (24r) inhibits AChE (IC50=2.4 nM), reducing amyloid buildup, tau phosphorylation, and promotes neuron health.</p>
    Formula:C23H27F2NO4S
    Color and Shape:Solid
    Molecular weight:451.53
  • 2R,4S-Sacubitril

    CAS:
    <p>2R,4S-Sacubitril (Sacubitril Enantiomer) is the impurity of Sacubitril which is a neprilysin inhibitor.</p>
    Formula:C24H28NO51Ca
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.49
  • Cacospongionolide B

    CAS:
    <p>Cacospongionolide B from Fasciospongia cavernosa inhibits secretory phospholipase A2, curbing inflammation.</p>
    Formula:C25H36O4
    Color and Shape:Solid
    Molecular weight:400.55
  • MGAT2-IN-1

    CAS:
    MGAT2-IN-1 is an orally active monoacylglycerol acyltransferase (MGAT2)inhibitor (human and mouse MGAT2 with IC50 of 7.8 and 2.4 nM , respectively).
    Formula:C27H21ClF5N7O3S
    Color and Shape:Solid
    Molecular weight:654.01
  • CHF-6366

    CAS:
    <p>CHF-6366: M3 antagonist &amp; β2 agonist (pKi 10.4/11.4), mild Ca channel blocker, used in COPD study.</p>
    Formula:C42H48N6O8
    Color and Shape:Solid
    Molecular weight:764.87
  • Saprisartan potassium

    CAS:
    <p>Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.</p>
    Formula:C25H21BrF3KN4O4S
    Color and Shape:Solid
    Molecular weight:649.52
  • (R)-BAY-899


    <p>(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.</p>
    Formula:C25H19F2N5O2
    Color and Shape:Solid
    Molecular weight:459.45
  • NS2B/NS3-IN-2


    <p>Potent dengue inhibitor NS2B/NS3-IN-2 (IC50: 6 nM, Ki: 0.66 μM) boosts cell viability, non-toxic.</p>
    Formula:C24H21N3O5S
    Color and Shape:Solid
    Molecular weight:463.51
  • STING agonist-7


    <p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>
    Formula:C17H12N4O4
    Color and Shape:Solid
    Molecular weight:336.3
  • SOS1-IN-6

    CAS:
    <p>SOS1-IN-6 (compound 33-P1) is a potent inhibitor of SOS1, acting on SOS1-G12D (IC50: 14.9 nM) and SOS1-G12V (IC50: 73.3 nM).</p>
    Formula:C26H28F3N3O2
    Color and Shape:Solid
    Molecular weight:471.51
  • Tuberculosis inhibitor 5


    <p>Compound 11i: potent, non-toxic anti-tuberculosis biphenyl analogue.</p>
    Formula:C25H18N2O2S
    Color and Shape:Solid
    Molecular weight:410.49
  • OSI-7904L free acid

    CAS:
    <p>OSI-7904L is a folate-based thymidylate synthase inhibitor. It also has antimalarial and antitumor properties.</p>
    Formula:C27H24N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.5
  • VU0463271 quarterhydrate


    <p>VU0463271 quarterhydrate is a potent KCC2 antagonist, with an IC 50 of 61 nM [1].</p>
    Formula:C19H20N4O2S2
    Color and Shape:Solid
    Molecular weight:387
  • VEGFR-2-IN-25

    CAS:
    <p>VEGFR-2-IN-25 (compound 5d) is a potent inhibitor of VEGFR-2 (IC50: 12.1 nM).</p>
    Formula:C24H22N6O2
    Color and Shape:Solid
    Molecular weight:426.47
  • Homomoschatoline

    CAS:
    <p>Homomoschatoline is an antibacterial isolated from Artabotrys crassifolius.</p>
    Formula:C19H15NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.33
  • FP0429

    CAS:
    <p>FP0429 is an agonist of mGlu4.</p>
    Formula:C10H12N2O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:272.21
  • PTP1B-IN-3 diammonium


    <p>PTP1B-IN-3 diammonium, an oral enzyme inhibitor, has potent antidiabetic and anticancer effects, with a 120 nM IC50.</p>
    Formula:C12H13BrF2N3O3P
    Color and Shape:Solid
    Molecular weight:396.12
  • Autophagy-IN-1


    <p>Autophagy-IN-1 blocks autophagy in cancer cells, hinders tumor growth in mice, and aids in studying colorectal cancer.</p>
    Formula:C23H25NO7
    Color and Shape:Solid
    Molecular weight:427.45
  • NVP-CGM097 sulfate

    CAS:
    <p>NVP-CGM097 sulfate is a potent and selective inhibitor of MDM2 (hMDM2, IC50 of 1.7±0.1 nM).</p>
    Formula:C38H49ClN4O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:757.34
  • HBV-IN-20


    <p>HBV-IN-20 is a potent, orally active HBV inhibitor (EC50: 0.46 μM). HBV-IN-20 is a classical type II CpAM (core protein assembly regulator).</p>
    Color and Shape:Solid