Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,849 products)
- Apoptosis(6,366 products)
- Cell Cycle/Checkpoint(4,907 products)
- Chromatin/Epigenetics(2,623 products)
- Cytoskeletal Signaling(1,585 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,759 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,051 products)
- Immunology and Inflammation(3,945 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,162 products)
- Metabolism(10,149 products)
- Microbiology/Virology(7,672 products)
- Neuroscience(10,549 products)
- Other Inhibitors(35,857 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,693 products)
- Stem Cell and Derivatives(734 products)
- Tyrosine Kinase/Adaptors(1,991 products)
- Ubiquitination(1,743 products)
Show 16 more subcategories
Found 66517 products of "Inhibitors"
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A-9758
CAS:A-9758: RORγt selective inverse agonist, IC50 5nM, inhibits IL-17A, Th17, and treats psoriasis.Formula:C25H23Cl2F3N2O3Purity:98%Color and Shape:SolidMolecular weight:527.36Antidepressant agent 2
Antidepressant agent 2 showed significant antidepressant effects with a MED value of 0.1 mg/kg.Formula:C21H22ClFN2O3SColor and Shape:SolidMolecular weight:436.93JAK3 covalent inhibitor-1
CAS:JAK3 Covalent Inhibitor-1 is a compound characterized by its potent and selective inhibition of Janus kinase 3 (JAK3), possessing an IC50 of 11 nM andFormula:C22H17FN6O2SPurity:98%Color and Shape:SolidMolecular weight:448.47MEK1/2-IN-2
MEK1/2-IN-2 is a potent, ATP-competitive MEK1/2 inhibitor that exhibits equal inhibitory effects on wild-type MEK1/2 and a group of MEK1/2 mutant cells.Formula:C28H22ClFN6OColor and Shape:SolidMolecular weight:512.97AZ-3
CAS:AZ-3 is a potent and selective JAK1 inhibitor (IC50: 34 nM).Formula:C20H28FN7Purity:98%Color and Shape:SolidMolecular weight:385.48EGFR/BRAF-IN-1
EGFR/BRAF-IN-1 inhibits EGFR/BRAF (BRAFV600E IC50: 45 nM, GI50: 35 nM) and has antioxidant properties.Formula:C26H28ClN3O4Color and Shape:SolidMolecular weight:481.97HIV-1 inhibitor-13
HIV-1 inhibitor-13: oral NNRTI, IC50=0.14μM for HIV-1 RT, effective on resistant strains (EC50=2.85-18nM).Formula:C30H32N6O3Color and Shape:SolidMolecular weight:524.61VEGFR-2-IN-26
CAS:VEGFR-2-IN-26 inhibits VEGFR-2 (IC50: 15.5 nM), combating various cancers' cell growth.Formula:C24H19F3N6O2Color and Shape:SolidMolecular weight:480.44Menin-MLL inhibitor 26
CAS:Menin-MLL inhibitor 26: Active reference, inhibits cell growth, used in leukemia research.Formula:C27H29F3N6O3SColor and Shape:SolidMolecular weight:574.62AT-IAP
CAS:AT-IAP is an effective dual antagonist of XIAP and cIAP1.Formula:C29H40FN5O2Purity:98%Color and Shape:SolidMolecular weight:509.66Onfasprodil
CAS:Onfasprodil, NR2B inhibitor & GABA regulator, potential for Alzheimer's research. (Patent CN111481543A)Formula:C20H23FN2O3Color and Shape:SolidMolecular weight:358.41TAK-024
CAS:TAK-024 is an inhibitor of platelet(IC50s of 31, 79 and 51 nM in human, monkey and guinea pig, respectively).Formula:C27H34N10O6Purity:98%Color and Shape:SolidMolecular weight:594.62Kahweol linoleate
CAS:Kahweol linoleate, a semi-synthetic from coffee, blocks osteoclast creation, fights cancerous cells, prevents DNA damage, and reduces oxidative stress.Formula:C38H56O4Color and Shape:SolidMolecular weight:576.85Trichostatin A S-isomer
CAS:Trichostatin A S-isomer, a HDAC 1, 3, 4, 6, 10 inhibitor with IC50 ~20 nM, has wide-ranging epigenetic effects.Formula:C17H22N2O3Purity:98%Color and Shape:SolidMolecular weight:302.37PARP-1-IN-1
PARP-1-IN-1: Selective, oral PARP-1 inhibitor with 0.96 nM IC50; well-tolerated and effective in single-dose MDA-MB-436 model.Formula:C23H25FN4OColor and Shape:SolidMolecular weight:392.47Scytonemin
CAS:Scytonemin, a cyanobacterial pigment, inhibits cancer cell growth by decreasing Plk1 activity, especially effective on U266 myeloma cells.Formula:C36H20N2O4Color and Shape:SolidMolecular weight:544.55PPARγ agonist 2
PPARγ agonist 2 is a highly effective compound that acts as a partial agonist for PPARγ.Formula:C24H20O5Color and Shape:SolidMolecular weight:388.41ZLWT-37
ZLWT-37: Oral CDK inhibitor, CDK9 IC50=0.002 µM, CDK2 IC50=0.054 µM; halts HCT116 cells at G2/M, induces apoptosis.Formula:C26H30ClN5OColor and Shape:SolidMolecular weight:464RWJ-445167
CAS:RWJ-445167 is a thrombin and factor Xa dual inhibitor(Ki of 4.0 nM and 230 nM, respectively), with potent antithrombotic activity.Formula:C18H24N6O5SPurity:98%Color and Shape:SolidMolecular weight:436.49AD5075
CAS:AD5075 is a bioactive chemical.Formula:C22H20N2O5SColor and Shape:SolidMolecular weight:424.47GSK945237
CAS:GSK945237 is a type IIA topoisomerase inhibitor, effective on Gram-positive and negative bacteria, with favorable pharmacokinetics and in vivo efficacy.Formula:C24H26FN5O3Color and Shape:SolidMolecular weight:451.49Anticancer agent 26
Anticancer agent 26 is a promising candidate for cancer therapy and deserves further development.Formula:C28H33NO5Color and Shape:SolidMolecular weight:463.57LSD1-IN-18
LSD1-IN-18 inhibits LSD1 (Ki: 0.156 μM, KD: 0.075 μM), blocking THP-1 and MDA-MB-231 cell growth (IC50: 0.16, 0.21 μM).Formula:C31H40N6O2Color and Shape:SolidMolecular weight:528.69BCL6-IN-9
CAS:BCL6-IN-9 (compound 1) is a potent inhibitor of B-cell lymphoma 6 protein (BCL6) (IC50: 3.9 nM) and can be used to study cancer.Formula:C22H18ClF2N5O2Color and Shape:SolidMolecular weight:457.8611-Oxahomoaminopterin
CAS:11-Oxahomoaminopterin exhibits antifolate activity against two folate-requiring microorganisms and inhibited Lactobacillus casei DHFR.Formula:C20H21N7O6Purity:98%Color and Shape:SolidMolecular weight:455.42RMS-07
CAS:RMS-07, a covalent MPS1/TTK inhibitor, has an IC50 of 13.1 nM, targeting a kinase hinge cysteine.Formula:C35H40N8O2Color and Shape:SolidMolecular weight:604.74Antimalarial agent 9
Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.Formula:C28H32BrN3O2Color and Shape:SolidMolecular weight:522.48OncoFAP
CAS:OncoFAP is an ultra-high affinity fibroblast activating protein (FAP) ligand with potential tumour targeting.Formula:C21H19F2N5O5Purity:99.77%Color and Shape:SolidMolecular weight:459.40DDCPPB-Glu
CAS:DDCPPB-Glu is a 6-5 fused ring heterocycle antifolate that shows antitumor activity.Formula:C22H27N5O5Purity:98%Color and Shape:SolidMolecular weight:441.48AD013
AD013 is a selective ACE inhibitor and NEP inhibitor with potential anti-hypertensive and cardioprotective benefits.Formula:C24H28N2O5Color and Shape:SolidMolecular weight:424.49AL 6598
CAS:AL 6598, a prodrug of PGD2 agonist AL 6556, reduces IOP by 53% at 1μg twice daily in monkeys; binds DP receptors with Ki of 3.2μM.Formula:C23H39ClO5Color and Shape:SolidMolecular weight:431.01VEGFR-2-IN-15
VEGFR-2-IN-15 (Compound 14b) is a potent inhibitor of VEGFR-2. VEGFR-2-IN-15 inhibits the growth of HepG2 cells in the Pre-G1 phase and induces apoptosis.Formula:C23H18ClN3O4SColor and Shape:SolidMolecular weight:467.92JAK3-IN-7
CAS:JAK3-IN-7 is a potent and selective JAK3 inhibitor (IC50<0.01 μM) for the treatment of rejection in organ transplantation, graft-versus-host reaction afterFormula:C17H20N6OPurity:98.81%Color and Shape:SolidMolecular weight:324.38BMS-751324
CAS:BMS-751324: p38α MAPK inhibitor with carbamyl-methyl, esters, phosphate from HPA. Reduces rat arthritis swelling and TNFα.Formula:C32H35N6O10PColor and Shape:SolidMolecular weight:694.63Dyrk1A-IN-1
Dyrk1A-IN-1 is a triple inhibitor of Dyrk1A kinase activity, aggregation of tau and α-syn oligomers, with an IC50 value of 119 nM for Dyrk1A kinase.Formula:C23H20N4O3SColor and Shape:SolidMolecular weight:432.49cis-RdRP-IN-5
Cis-RdRP-IN-5 is an effective inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), employed in influenza virus research.Formula:C23H21N3O5Color and Shape:SolidMolecular weight:419.43Prohibitin ligand 1
Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.Formula:C20H22N2OColor and Shape:SolidMolecular weight:306.4PDHK-IN-5
PDHK-IN-5, potent PDHK2 (0.006 μM IC50) & PDHK4 (0.0329 μM IC50) inhibitor, may be explored for cancer and diabetes treatment.Formula:C30H31N5O2Color and Shape:SolidMolecular weight:493.6CDK4-IN-1
CAS:CDK4 inhibitor is a novel and specific CDK4/Cyclin D1 inhibitor with an IC50 of 10 nM; 1500 and 500 fold than CDK1/Cyclin B (IC50>15 uM) and CDK2/Cyclin A (IC50Formula:C22H29ClN8Purity:98%Color and Shape:SolidMolecular weight:440.97DSM705 hydrochloride
DSM705 hydrochloride: potent antimalarial, pyrrole-based DHODH inhibitor effective against Plasmodium, non-toxic to mammalian DHODH.Formula:C19H20ClF3N6OColor and Shape:SolidMolecular weight:440.85Anti-inflammatory agent 13
Pentacyclic triterpene, Anti-inflammatory 13 inhibits DAMP/PAMP inflammation models.Formula:C30H48O4Color and Shape:SolidMolecular weight:472.7Samuraciclib hydrochloride hydrate
Samuraciclib (CT7001) is a potent oral CDK7 inhibitor (IC50: 41 nM) with anti-breast cancer properties.Formula:C22H35ClN6O3Color and Shape:SolidMolecular weight:521.7RORγt modulator 5
CAS:RORγt modulator 5, a potent RORγt modulator, exhibits a dissociation constant (K_i) of <100 nM.Formula:C27H22F5N3O6SColor and Shape:SolidMolecular weight:611.54Oiligodendrocyte differentiation promoter 1
CAS:Oiligodendrocyte differentiation promoter 1 is a promoter of oiligodendrocyte differentiation .Formula:C25H25Cl2NO5Purity:98%Color and Shape:SolidMolecular weight:490.38UB 165
CAS:Subtype-selective nicotinic agonistFormula:C13H15ClN2Purity:98%Color and Shape:SolidMolecular weight:234.72NMDA receptor antagonist-3
NMDA antagonist-3: recovery rate 40% at 100 μM, low toxicity in SH-SY5Y, human stem cells.Formula:C13H19N3O6Color and Shape:SolidMolecular weight:313.31Dyrk1A-IN-2
Dyrk1A-IN-2 is a DYRK1A inhibitor (EC50: 37 nM). dyrk1A-IN-2 exhibits efficient promotion of human β-cell replication, as well as low cytotoxicity.Formula:C27H32N6O4Color and Shape:SolidMolecular weight:504.58Atorvastatin 3-Deoxyhept-2E-Enoic Acid
CAS:Atorvastatin 3-Deoxyhept-2E-Enoic Acid, an impurity in Atorvastatin, lowers blood lipids as an HMG-CoA reductase inhibitor.Formula:C33H33FN2O4Purity:98%Color and Shape:SolidMolecular weight:540.62APJ receptor agonist 3
CAS:APJ receptor agonist 3 is a highly effective and orally administerable agonist of the APJ receptor, demonstrating a potent EC50 value of 0.027 nM.Formula:C26H29ClN4O5Color and Shape:SolidMolecular weight:512.98PARP10/15-IN-2
CAS:PARP10/15-IN-2 (Compound 8h) blocks PARP10/15, has IC50s: 0.15μM/0.37μM, cell-permeable, prevents apoptosis.Formula:C15H11FN2O3Color and Shape:SolidMolecular weight:286.26Rodatristat
CAS:Rodatristat is an effective tryptophan hydroxylase 1 and TPH2 inhibitor (IC50s: 33 nM and 7 nM, respectively).Formula:C27H27ClF3N5O3Purity:98%Color and Shape:SolidMolecular weight:561.98AKT-IN-11
AKT-IN-11 is one of the most potent antibacterial agents against human hepatocellular carcinoma Bel-7402 cell line (IC50: 1.15 μM).Formula:C27H27ClF3NO4Color and Shape:SolidMolecular weight:521.96Topoisomerase I/II inhibitor 2
Compound 1a inhibits Topoisomerase I/II, shrinks mouse liver tumors, IC50: 6.83/9.82 μM for LM9/Huh7 cells.Formula:C19H16N2O4Color and Shape:SolidMolecular weight:336.34Foroxymithine
CAS:Foroxymithine is an inhibitor of angiotensin-converting enzyme.Formula:C22H37N7O11Purity:98%Color and Shape:SolidMolecular weight:575.57HIV-1 protease-IN-6
HIV-1 protease-IN-6 (17d) strongly inhibits HIV-1 protease (IC50: 21 pM, Ki: 4.7 pM) and effectively targets DRV-resistant mutants.Formula:C27H31FN2O6SColor and Shape:SolidMolecular weight:530.61L 739749
CAS:L 739749 is a CAAX peptidomimetic. It is also an inhibitor of farnesyl-protein transferase.Formula:C24H41N3O6S2Purity:98%Color and Shape:SolidMolecular weight:531.73Agosterol A
CAS:Agosterol A is isolated from marine sponge Spongia.Formula:C33H52O8Color and Shape:SolidMolecular weight:576.76Kallikrein-IN-1
CAS:Kallikrein-IN-1 (Formula A) is an inhibitor of the kinin-releasing enzyme Kallikrein.Formula:C28H26FN5O4Color and Shape:SolidMolecular weight:515.5417β-HSD1-IN-1
17β-HSD1-IN-1 (Compound 1) can be used in the non-small cell lung cancer (NSCLC) research.Formula:C21H21NO3Color and Shape:SolidMolecular weight:335.4TLR7/8 antagonist 1
Compound 16c, an imidazoquinoline, is a TLR7/8 agonist; IC50: 3.91 μM (TLR7), 2.19 μM (TLR8); targets TLR-2050 for disease treatment.Formula:C24H27N5O2Color and Shape:SolidMolecular weight:417.5Cilobamine mesylate
CAS:Cilobamine mesylate is a drug which acts as a norepinephrine-dopamine reuptake inhibitor (NDRI) and has stimulant and antidepressant effects.Formula:C18H27Cl2NO4SColor and Shape:SolidMolecular weight:424.38Falecalcitriol
CAS:Falecalcitriol is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems, which is longer duration of action in vivo.Formula:C27H38F6O3Purity:98%Color and Shape:SolidMolecular weight:524.58ADU-S100 disodium salt
CAS:ADU-S100 (MIW815) disodium salt is an activator of stimulator of interferon genes (STING).Formula:C20H22N10Na2O10P2S2Purity:98%Color and Shape:SolidMolecular weight:734.51EBOV-GP-IN-1
EBOV-GP-IN-1 (Compound 28) is a potent inhibitor of Ebola entry, acting on the Ebola virus envelope glycoprotein (EBOV-GP) (IC50: 0.05 μM).Formula:C25H40ClN3O2Color and Shape:SolidMolecular weight:450.06Ivaltinostat formic
Ivaltinostat (CG-200745) is an oral panHDAC inhibitor, inducing apoptosis and enhancing cancer drug sensitivity.Formula:C25H35N3O6Color and Shape:SolidMolecular weight:473.56GSK-3β inhibitor 7
GSK-3β inhibitor 7 is a GSK-3β inhibitor (IC50: 5.25 μM).Formula:C27H23BrN4O2SColor and Shape:SolidMolecular weight:547.47(R)-NVS-ZP7-4
CAS:(R)-NVS-ZP7-4, an R-isomer, inhibits ZIP7 to study ER zinc impact & Notch pathway.Formula:C28H28FN5OSPurity:98%Color and Shape:SolidMolecular weight:501.62Intoplicine
CAS:Intoplicine is an inhibitor of DNA topoisomerase I and II.Formula:C21H24N4OPurity:98%Color and Shape:SolidMolecular weight:348.44BW A868C
CAS:BW A868C is a potent, selective PGD2 antagonist and a BW245C analogue, inert to other prostaglandin receptors.Formula:C25H37N3O5Color and Shape:SolidMolecular weight:459.58SOS1-IN-6
CAS:SOS1-IN-6 (compound 33-P1) is a potent inhibitor of SOS1, acting on SOS1-G12D (IC50: 14.9 nM) and SOS1-G12V (IC50: 73.3 nM).Formula:C26H28F3N3O2Color and Shape:SolidMolecular weight:471.51Sunobinop
CAS:Sunobinop (S 117957) is an opioid receptor-like orphan receptor (ORL1) modulator.Formula:C26H33N3O3Color and Shape:SolidMolecular weight:435.56Neuraminidase-IN-11
Neuraminidase-IN-11 (15e) inhibits H1N1 (IC50: 4.7nM), H5N1 (8.46nM), H5N8 viruses (1.5nM) selectively & potently.
Color and Shape:SolidAnti-TSWV agent 1
Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV).Formula:C22H27ClN4OS3Color and Shape:SolidMolecular weight:495.12Antitubercular agent-11
Antitubercular agent-11 (Compound 1e) is an antitubercular agent with a bulkier electron-donating group (Bu-t) that shows the best MIC value of 0.060 μg/mL [1].Formula:C16H15N3O4Color and Shape:SolidMolecular weight:313.31Hsp90-IN-16
Hsp90-IN-16, a selective HSP90 inhibitor, targets HER2+ cancers with 6 μM IC50 in HCC1954 cells, blocking client proteins and inducing apoptosis.Formula:C30H26FN3O6Color and Shape:SolidMolecular weight:543.54MPro N3
CAS:Mpro inhibitor blocks MHV-A29, HCoV-229E, FOPV (IC50: 2.7–8.8 μM), and SARS-CoV-2 (IC50: 16.8 μM) in plaque assays.Formula:C35H48N6O8Color and Shape:SolidMolecular weight:680.79SC-435 mesylate
CAS:SC-435 is an ileal apical sodium co-dependent bile acid transporter (ASBT). SC-435 inhibits plasma cholesterol.Formula:C37H59N3O7S2Purity:98%Color and Shape:SolidMolecular weight:722.01Chitin synthase inhibitor 9
CHS inhibitor 9: a broad-spectrum antifungal for studying fungal infections.Formula:C24H25N3O6Color and Shape:SolidMolecular weight:451.47CCR5 antagonist 1
CAS:CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.Formula:C39H46ClF2N5O3SPurity:98%Color and Shape:SolidMolecular weight:738.33Cilobamine (free base)
CAS:Cilobamine: a stimulant antidepressant, inhibits norepinephrine-dopamine reuptake, based on dichloroisoprenaline structure.Formula:C17H23Cl2NOColor and Shape:SolidMolecular weight:328.28Nrf2/HO-1 activator 2
Compound 13m, a difluoro derivative, activates Nrf2/HO-1, showing neuroprotective and antioxidant effects, useful in PD research.Formula:C20H16F2O5Color and Shape:SolidMolecular weight:374.33(1R,3S)-THCCA-Asn
(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.Formula:C24H24N4O6Color and Shape:SolidMolecular weight:464.47RORγt Inverse agonist 2
CAS:RORγt Inverse agonist 2 is a selective, orally active inverse agonist of RORγt(EC50 of 119 nM).Formula:C27H25F8NO5SPurity:98%Color and Shape:SolidMolecular weight:627.54DSP-6952
CAS:DSP-6952 is a 5-HT4 receptor partial agonist, inhibiting visceral hypersensitivity and ameliorating gastrointestinal dysfunction.Formula:C21H32BrClN4O5Color and Shape:SolidMolecular weight:535.86AR-13324 M1 metabolite
CAS:AR-13324 M1 metabolite is a hydrolysis metabolite of AR-13324 mesylate.Formula:C19H19N3O2Purity:98%Color and Shape:SolidMolecular weight:321.37PRN694
CAS:PRN694 is a potent, irreversible ITK/RLK inhibitor with IC50s: 0.3/1.4 nM; offers lasting effector cell suppression.Formula:C28H35F2N5O2SPurity:98%Color and Shape:SolidMolecular weight:543.67GSK3368715 3HCl
CAS:GSK3368715, a potent inhibitor of type I protein arginine methyltransferases (PRMT), could inhibit PRMT1, 3, 4, 6 and 8 with Kiapp vaules ranging from 1.5 to 81Formula:C20H41Cl3N4O2Purity:98%Color and Shape:SolidMolecular weight:475.92Resolvin E2
CAS:RvE2, a bioactive lipid from the SPM family, is made from EPA and reduces inflammatory neutrophil infiltration and helps treat NAFLD and other diseases.Formula:C20H30O4Color and Shape:SolidMolecular weight:334.45PPI-2458
CAS:PPI-2458, a fumagillin derivative, irreversibly blocks MetAP2, hindering abnormal cell growth and angiogenesis with improved toxicity.Formula:C22H36N2O6Color and Shape:SolidMolecular weight:424.53Nedocromil sodium
CAS:Nedocromil sodium is a pharmacologic stabilizer of mast cells, has been shown to normalize cytokine levels and attenuate cardiac remodeling.Formula:C19H17NNaO7Purity:98%Color and Shape:SolidMolecular weight:394.335Hit 1
Hit 1 is an activator of insulin-degrading enzymes (IDE) (EC50: 5.5 μM) and reduces glucose-stimulated insulin secretion.Formula:C22H24N4O3S2Color and Shape:SolidMolecular weight:456.58Rpi 856 C
CAS:Rpi 856 C is a retrovirus protease inhibitor from Streptomyces that is effective against HIV-1 and HTLV-1 proteases.Formula:C39H56N6O10Purity:98%Color and Shape:SolidMolecular weight:768.90Bafilomycin C1
CAS:vacuolar H+-ATPases (V-ATPases) inhibitorFormula:C39H60O12Purity:98%Color and Shape:Light Tan SolidMolecular weight:720.89CH5447240
CAS:CH5447240: potent hPTHR1 agonist, treats Hypoparathyroidism, EC50 12 nM, 55% oral bioavailability, raises rat serum calcium.Formula:C26H39N5O4SPurity:98%Color and Shape:SolidMolecular weight:517.68BRD7929
CAS:BRD7929 is a multistage antimalarial inhibitor for single-dose treatment of malaria in mouse models.Formula:C33H38N4O2Color and Shape:SolidMolecular weight:522.68CN-716 HCl
CAS:cn-716 is a novel Zika virus (ZIKV) NS2B-NS3pro protease inhibitor.Formula:C22H33BCl2N6O4Color and Shape:SolidMolecular weight:527.25PDE4-IN-5
PDE4-IN-5: potent PDE4 inhibitor, IC50 = 3.1 nM, superb skin penetration, anti-psoriasis effect.Formula:C21H28N2O3Color and Shape:SolidMolecular weight:356.46SARS-CoV-2 nsp14-IN-1
SARS-CoV-2 nsp14-IN-1 inhibits Nsp14 Mtase with an IC50 of 0.061 μM, affecting multiple substrates.Formula:C20H20N6O5SColor and Shape:SolidMolecular weight:456.48Ketomethylenebestatin
CAS:Ketomethylenebestatin, a weaker carba-analog of aminopeptidase inhibitor bestatin, is 10x less potent.Formula:C17H25NO4Purity:98%Color and Shape:SolidMolecular weight:307.38ACSS2-IN-1
CAS:ACSS2-IN-1, a potent ACSS2 inhibitor, has IC50 0.01-<1 nM; useful in cancer research.Formula:C27H25ClN6O2Color and Shape:SolidMolecular weight:500.98
