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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66639 products of "Inhibitors"

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  • CEP-7055

    CAS:
    <p>CEP-18770: oral proteasome inhibitor; blocks NF-kappaB; may cause cancer cell apoptosis; less toxic than bortezomib in normal cells.</p>
    Formula:C32H35N3O4
    Color and Shape:Solid
    Molecular weight:525.64
  • Haspin-IN-1


    <p>Haspin-IN-1 blocks haspin (IC50: 119 nM) and inhibits CLK1, DYRK1A, CDK9 with potential as an anticancer drug.</p>
    Formula:C12H8N4O2S
    Color and Shape:Solid
    Molecular weight:272.28
  • NTU281

    CAS:
    <p>NTU281 inhibits transglutaminase-2, lowers creatinine in diabetic rats, reduces proteinuria, and fights glomerulosclerosis.</p>
    Formula:C25H31N2O6S
    Color and Shape:Solid
    Molecular weight:487.59
  • U 80215

    CAS:
    <p>U 80215 is an enzyme-competitive inhibitor.</p>
    Formula:C42H60N8O6S
    Color and Shape:Solid
    Molecular weight:805.04
  • Lunacalcipol

    CAS:
    <p>Lunacalcipol is used for the treatment of Secondary Hyperparathyroidism.</p>
    Formula:C28H42O4S
    Color and Shape:Solid
    Molecular weight:474.7
  • Anti-inflammatory agent 9


    <p>Benzimidazothiazole-derived Compound 28 from tilomisole targets COX-2, has potent anti-inflammatory effects &amp; is orally bioavailable.</p>
    Formula:C18H15N5O2S
    Color and Shape:Solid
    Molecular weight:365.41
  • Ep vinyl quinidine

    CAS:
    <p>3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.</p>
    Formula:C20H24N2O2
    Color and Shape:Solid
    Molecular weight:324.42
  • Encephalitic alphavirus-IN-1


    <p>Alphavirus-IN-1 blocks VEEV (EC50: 0.24 μM) &amp; EEEV (EC50: 0.16 μM), non-toxic, stable in mice plasma.</p>
    Formula:C27H25FN6O2
    Color and Shape:Solid
    Molecular weight:484.52
  • FCE-27262

    CAS:
    <p>FCE-27262 is a prostaglandin H2/thromboxane A2 receptor antagonist.</p>
    Formula:C23H31N3O3
    Color and Shape:Solid
    Molecular weight:397.51
  • NBD-14189

    CAS:
    <p>NBD-14189: Potent HIV-1 entry blocker, binds gp120, IC50: 89 nM, strong antiviral (EC50 &lt;200 nM).</p>
    Formula:C18H16F4N4O2S
    Color and Shape:Solid
    Molecular weight:428.40
  • U75302

    CAS:
    <p>U75302 is an antagonist of thymosin beta-4 (TB4) receptor with a Ki value of 159 nM on guinea pig lung membranes.</p>
    Formula:C22H35NO3
    Purity:98%
    Color and Shape:Light Yellow Oil
    Molecular weight:361.52
  • KRAS G12D inhibitor 11

    CAS:
    <p>KRAS G12D inhibitor 11 targets KRAS G12D in cancer research (patent WO2021108683A1, compound 52).</p>
    Formula:C29H38BN5O3
    Color and Shape:Solid
    Molecular weight:515.45
  • MDK-3298

    CAS:
    <p>MDK-3298 is a reversible covalent inhibitor of Mcl-1, a target of protein-protein interaction (PPI).</p>
    Formula:C35H32BN3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:617.46
  • ROPA

    CAS:
    <p>ROPA, a potent PKCalpha and PKCgamma activator, promotes tumor growth through PKC-activation.</p>
    Formula:C28H32O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:464.55
  • BAY-693

    CAS:
    <p>BAY-693 is a ERK5 negative control agent with IC50 (ERK5) = 6400 nM. Its analog, BAY-885, is a potent and selective ERK5 (MAPK7) inhibitor with IC50 of 40 nM</p>
    Formula:C26H30F3N7O2
    Color and Shape:Solid
    Molecular weight:529.56
  • AZD-4121 tert-butylammonium

    CAS:
    <p>AZD-4121 tert-butylammonium is an oral cholesterol absorption inhibitor targeting NPC1L1 for the treatment of dyslipidaemia.</p>
    Formula:C40H50F2N4O7S
    Color and Shape:Solid
    Molecular weight:768.91
  • JAK3-IN-7

    CAS:
    <p>JAK3-IN-7 is a potent and selective JAK3 inhibitor (IC50&lt;0.01 μM) for the treatment of rejection in organ transplantation, graft-versus-host reaction after</p>
    Formula:C17H20N6O
    Purity:98.81%
    Color and Shape:Solid
    Molecular weight:324.38
  • Notch inhibitor 1

    CAS:
    <p>Notch inhibitor 1 blocks Notch 1/3 (IC50: 7.8/8.5 nM) and aids cancer research.</p>
    Formula:C26H25F7N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:574.49
  • AZD-3199 dihydrobromide

    CAS:
    <p>AZD-3199 dihydrobromide is a β2 adrenergic receptor agonist potentially for the treatment of asthma and chronic obstructive.</p>
    Formula:C32H44Br2N4O4S
    Color and Shape:Solid
    Molecular weight:740.59
  • Aspochalasin M

    CAS:
    <p>Aspochalasin M shows moderate activity on HL-60 cells (IC50=20.0 μ M). Aspochalasin M has research potential in leukemia diseases.</p>
    Formula:C24H35NO4
    Color and Shape:Solid
    Molecular weight:401.54
  • LRRK2-IN-3

    CAS:
    <p>LRRK2-IN-3: potent, selective oral LRRK2 blocker, BBB-penetrant, IC50 of 0.6 nM in hPBMCs, for Parkinson's research.</p>
    Formula:C25H29ClF2N6O2
    Color and Shape:Solid
    Molecular weight:518.99
  • CB 30900

    CAS:
    <p>CB30900 is a novel and effective thymidylate synthase inhibitor.</p>
    Formula:C31H32FN5O9
    Color and Shape:Solid
    Molecular weight:637.61
  • LY367385 hydrochloride

    CAS:
    <p>LY367385 hydrochloride: selective mGluR1a antagonist, IC50 = 8.8 μM, neuroprotective, anticonvulsant, antiepileptic.</p>
    Formula:C10H12ClNO4
    Color and Shape:Solid
    Molecular weight:245.66
  • Streptonigrin (racemate)

    CAS:
    <p>Streptonigrin: aminoquinone antibiotic; antitumor, antibacterial; blocks β-Catenin/Tcf, cytotoxic; alters hamster chromosomes; (-)-isomer, CAS#3930-19-6.</p>
    Formula:C25H22N4O8
    Color and Shape:Solid
    Molecular weight:506.46
  • MDL-43291

    CAS:
    <p>MDL-43291 is a leukotriene receptor antagonist.</p>
    Formula:C25H42O4S
    Color and Shape:Solid
    Molecular weight:438.66
  • P-gp inhibitor 2

    CAS:
    <p>Potent P-gp inhibitor 2 reverses Doxorubicin resistance in colorectal carcinoma cells with IC50 of 0.22 µM.</p>
    Formula:C29H26N2O6
    Color and Shape:Solid
    Molecular weight:498.53
  • A1AR antagonist 1


    <p>Compound 18g, a potent A1AR blocker with Ki: 2.08 nM (hA1), 6.91 nM (hA2A), 31.2 nM (hA2B).</p>
    Formula:C18H14N4O
    Color and Shape:Solid
    Molecular weight:302.33
  • 6-trans-12-epi-Leukotriene B4

    CAS:
    <p>6-trans-12-epi-Leukotriene B4, a metabolite of arachidonic acid, serves as a potent anti-inflammatory agent.</p>
    Formula:C20H32O4
    Color and Shape:Solid
    Molecular weight:336.47
  • TIM-3-IN-1


    <p>TIM-3-IN-1 is a useful tool to enable further studies on the biology of TIM-3 immunoregulation in cancer.</p>
    Formula:C20H16ClN7O3S
    Color and Shape:Solid
    Molecular weight:469.9
  • Ornoprostil

    CAS:
    <p>Ornoprostil, a prostaglandin E1 analogue, acts as a mucosal protectant.</p>
    Formula:C23H38O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.54
  • Antifungal agent 17


    <p>Antifungal agent 17 showed good antifungal activity against B. cinerea (EC50: 2.86 μg/mL).</p>
    Formula:C18H16Br2O2
    Color and Shape:Solid
    Molecular weight:424.13
  • TRPC4/5-IN-1


    <p>TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.</p>
    Formula:C21H21N3O
    Color and Shape:Solid
    Molecular weight:331.41
  • GLPG0492 (R enantiomer)

    CAS:
    <p>GLPG0492 R enantiomer is the R enantiomer of GLPG-0492, a novel selective androgen receptor modulator.</p>
    Formula:C19H14F3N3O3
    Color and Shape:Solid
    Molecular weight:389.33
  • iNOs-IN-1


    <p>iNOs-IN-1 (YPW) is a strong iNOS inhibitor with dose-dependent anti-inflammatory properties, reducing IL-6, iNOS, and NO levels.</p>
    Formula:C25H30N4O5
    Color and Shape:Solid
    Molecular weight:466.53
  • PPARα/γ agonist 1


    <p>PPARα/γ agonist 1 is a potent and dual PPARα/γ partial agonist which is a promising prototype for the research of dyslipidemia and diabetes.</p>
    Formula:C18H19NO2
    Color and Shape:Solid
    Molecular weight:281.35
  • Eilatine

    CAS:
    <p>Eilatine is a novel marine alkaloid inhibits in vitro proliferation of progenitor cells in chronic myeloid leukemia patients.</p>
    Formula:C24H12N4
    Color and Shape:Solid
    Molecular weight:356.38
  • Anticancer agent 53

    CAS:
    <p>Anticancer agent 53 exhibits potent in vitro cytotoxicity, triggers apoptosis, halts S/G2/M cycle, and has antitumor effects without toxicity.</p>
    Formula:C31H25FN4O6S
    Color and Shape:Solid
    Molecular weight:600.62
  • Antibacterial agent 113


    <p>Antibacterial agent 113 targets multiple bacteria including P. aeruginosa and E. coli, showing efficacy at MIC 15625 μM.</p>
    Formula:C29H18ClN5O
    Color and Shape:Solid
    Molecular weight:487.94
  • Monoamine oxidase/Aromatase-IN-1


    <p>Compound 2q: Dual MAO/aromatase inhibitor; IC50: 39 nM (MAO-B), 31 nM (aromatase). Useful in neurological/breast cancer research.</p>
    Formula:C19H19N3O3S
    Color and Shape:Solid
    Molecular weight:369.44
  • β-Glucuronidase-IN-2


    <p>β-Glucuronidase-IN-2 is a potent inhibitor of E.</p>
    Formula:C21H17Cl3O7
    Color and Shape:Solid
    Molecular weight:487.71
  • CCR5 antagonist 1

    CAS:
    <p>CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.</p>
    Formula:C39H46ClF2N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:738.33
  • (±)-HIP-B

    CAS:
    <p>(±)-HIP-B is an excitatory amino acid transporter blocker.</p>
    Formula:C6H8N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:172.14
  • CYP2C1/CYP2C19-IN-2


    <p>CYP2C1/CYP2C19-IN-2 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>
    Formula:C27H28N2O6S
    Color and Shape:Solid
    Molecular weight:508.59
  • Antibiotic LL Z1640-2

    CAS:
    <p>Antibiotic LL Z1640-2 is an inhibitor against the TAK1 activity.</p>
    Formula:C19H22O7
    Color and Shape:Solid
    Molecular weight:362.38
  • Combretastatin A1 phosphate

    CAS:
    <p>Combretastatin A1 phosphate: potent anti-angiogenic and tumor vascular disruptor, with research potential in pancreatic neuroendocrine tumors.</p>
    Formula:C18H22O12P2
    Color and Shape:Solid
    Molecular weight:492.31
  • hCAII-IN-3


    <p>hCAII-IN-3 inhibits key hCA isoforms with Ki: hCA I (403.8 nM), hCA II (5.1 nM), hCA IX (10.2 nM), hCA XII (5.2 nM); shows anticancer potential.</p>
    Formula:C17H21N3O3S
    Color and Shape:Solid
    Molecular weight:347.43
  • Squalestatin 3

    CAS:
    <p>Squalestatin 3 is an inhibitor of squalene synthase.</p>
    Formula:C25H30O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:538.5
  • IRAK4-IN-18


    <p>IRAK4-IN-18: Potent IRAK4 inhibitor (IC50: 15 nM), reduces IL23 in cells, prevents rat arthritis.</p>
    Formula:C24H25FN6O3
    Color and Shape:Solid
    Molecular weight:464.49
  • LP 12 hydrochloride hydrate


    <p>LP 12 hydrochloride hydrate: potent, selective 5-HT7 agonist (Ki: 0.13 nM); less affinity for D2, 5-HT1A/2A receptors.</p>
    Formula:C32H39N3O·HCl·xH2O
    Color and Shape:Solid
  • cis-4-Br-2,5-F2-PCPA


    <p>cis-4-Br-2,5-F2-PCPA (S1024) blocks LSD1/LSD2 (Ki: 94 nM/8.4 μM), hinders cancer stem cell growth, raises H3K4me2 in CCRF-CEM cells.</p>
    Formula:C9H8BrF2N
    Color and Shape:Solid
    Molecular weight:248.07
  • FCE-24379

    CAS:
    <p>FCE-24379 is a selective antagonist of vascular serotonin receptors that has been shown to lowers blood pressure in hypertensive rats.</p>
    Formula:C20H22N4O2
    Color and Shape:Solid
    Molecular weight:350.41
  • Beloranib

    CAS:
    <p>Beloranib is a fumagillin anticancer drug. Beloranib belongs to an angiogenesis inhibitor.</p>
    Formula:C29H41NO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:499.64
  • BMS-751324

    CAS:
    <p>BMS-751324: p38α MAPK inhibitor with carbamyl-methyl, esters, phosphate from HPA. Reduces rat arthritis swelling and TNFα.</p>
    Formula:C32H35N6O10P
    Color and Shape:Solid
    Molecular weight:694.63
  • Polvitolimod

    CAS:
    <p>Polvitolimod is a TLR7 agonist used to treat infectious disease and cancer.</p>
    Formula:C13H14FN5O4
    Color and Shape:Solid
    Molecular weight:323.28
  • Pexacerfont

    CAS:
    <p>Pexacerfont (BMS-562086) is a selective antagonist of the corticotropin-releasing factor receptor (IC50: 6.1±0.6 nM for the human CRF1 receptor).</p>
    Formula:C18H24N6O
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:340.42
  • TY 11345

    CAS:
    <p>TY 11345 is a proton pump inhibitor.</p>
    Formula:C18H18N3NaO2S
    Color and Shape:Solid
    Molecular weight:363.41
  • NSD2-IN-1

    CAS:
    <p>NSD2-IN-1: potent, selective NSD2-PWWP1 inhibitor, IC50 0.11 μM, induces gene expression changes, apoptosis, cell cycle arrest.</p>
    Formula:C29H31N5
    Color and Shape:Solid
    Molecular weight:449.59
  • Asukamycin

    CAS:
    <p>Asukamycin, from S. nodosus asukaensis, is a polyketide antibiotic inhibiting tumor cells by activating caspases 8 and 3.</p>
    Formula:C31H34N2O7
    Color and Shape:Solid
    Molecular weight:546.61
  • COX-2-IN-7


    <p>COX-2-IN-7: potent, orally active COX-2 inhibitor with higher selectivity than Celecoxib, IC50 6.585 uM, anti-inflammatory, low ulcer risk.</p>
    Formula:C15H13N3O2S2
    Color and Shape:Solid
    Molecular weight:331.41
  • (+)-Sparteine sulfate pentahydrate


    <p>(+)-sparteine (sulfate pentahydrate) is a ganglion blocker that competitively blocks nicotinic acetylcholine receptors in neurons.</p>
    Formula:C15H38N2O9S
    Color and Shape:Solid
    Molecular weight:422.54
  • Fandosentan

    CAS:
    <p>Fandosentan is an endothelin receptor antagonist.</p>
    Formula:C25H18F3NO6S
    Color and Shape:Solid
    Molecular weight:517.47
  • DNA-PK-IN-8

    CAS:
    <p>DNA-PK-IN-8: Potent, selective oral DNA-PK inhibitor, IC50 = 0.8 nM, boosts anti-cancer effects with Doxorubicin.</p>
    Formula:C19H22N8O2
    Color and Shape:Solid
    Molecular weight:394.43
  • Resolvin E2

    CAS:
    <p>RvE2, a bioactive lipid from the SPM family, is made from EPA and reduces inflammatory neutrophil infiltration and helps treat NAFLD and other diseases.</p>
    Formula:C20H30O4
    Color and Shape:Solid
    Molecular weight:334.45
  • Avibactam sodium dihydrate


    <p>Avibactam sodium dihydrate (NXL-104) is a reversible covalent inhibitor for CTX-M-15 and TEM-1 β-lactamases with IC50s of 5 nM and 8 nM.</p>
    Formula:C7H14N3NaO8S
    Color and Shape:Solid
    Molecular weight:323.26
  • Sovesudil hydrochloride


    <p>Sovesudil (PHP-201) HCl: potent local ROCK inhibitor; targets ROCK I/II (IC50: 3.7/2.3 nM); lowers IOP, non-congesting.</p>
    Formula:C23H23ClFN3O3
    Color and Shape:Solid
    Molecular weight:443.9
  • Dyrk1A/B-IN-1


    <p>Dyrk1A/B-IN-1 (3n) is a potent DYRK1A/B inhibitor, cell-permeable, with Ki values of 67.8 nM (1A) and 237.9 nM (1B), IC50s of 1.1 and 0.8 μM.</p>
    Formula:C21H17N3O2S2
    Color and Shape:Solid
    Molecular weight:407.51
  • Menin-MLL inhibitor 26

    CAS:
    <p>Menin-MLL inhibitor 26: Active reference, inhibits cell growth, used in leukemia research.</p>
    Formula:C27H29F3N6O3S
    Color and Shape:Solid
    Molecular weight:574.62
  • NCATS-SM4487

    CAS:
    <p>NCATS-SM4487 is a highly selective inhibitor of GALK1 (IC50: 0.05 μM).</p>
    Formula:C25H24ClFN8O2
    Color and Shape:Solid
    Molecular weight:522.96
  • FLT3-IN-13


    <p>FLT3-IN-13 inhibits topoisomerase II/FLT3 in leukemia with IC50 of 2.26 μM, causes G2/M arrest, and promotes apoptosis.</p>
    Formula:C20H14N4O2
    Color and Shape:Solid
    Molecular weight:342.35
  • PLP_Snyder530


    <p>PLP_Snyder530, a potent PL pro inhibitor, halts SARS-CoV-2 by triggering protease conformation changes.</p>
    Formula:C24H24N2O2
    Color and Shape:Solid
    Molecular weight:372.46
  • SX 3202

    CAS:
    <p>SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.</p>
    Formula:C17H11BrFN3O4
    Color and Shape:Solid
    Molecular weight:420.19
  • Sequoiaflavone

    CAS:
    <p>Sequoiaflavone is a biflavone isolated from Ginkgo biloba.</p>
    Formula:C31H20O10
    Color and Shape:Solid
    Molecular weight:552.48
  • ATM Inhibitor-2


    <p>ATM Inhibitor -2 is a potent and selective inhibitor of ATM (IC50&lt;1 nM).</p>
    Formula:C26H31N7O3
    Color and Shape:Solid
    Molecular weight:489.57
  • BMS-248360

    CAS:
    <p>BMS-248360: Oral dual hAT1/hETA antagonist with Kis of 10nM &amp; 1.9nM, respectively; treats hypertension.</p>
    Formula:C36H45N5O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:659.84
  • Artemisiane E

    CAS:
    <p>Artemisiane E is a potent PI3K/AKT pathway inhibitor with an IC 50 of 8.9 μM .</p>
    Formula:C20H22O5
    Color and Shape:Solid
    Molecular weight:342.39
  • KRAS G12C inhibitor 46

    CAS:
    <p>KRAS G12C inhibitor 46 is a potent inhibitor of KRAS G12C.</p>
    Formula:C32H33F2N7O2
    Color and Shape:Solid
    Molecular weight:585.65
  • Antitumor agent-54


    <p>Compound C11 inhibits 14-3-3η protein (KD: 35 μM), targets liver cancer cells, blocks G1-S phase, and induces apoptosis.</p>
    Formula:C29H32N2O3
    Color and Shape:Solid
    Molecular weight:456.58
  • VEGFR-2-IN-5 hydrochloride


    <p>VEGFR-2-IN-5 hydrochloride is an effective VEGFR2 inhibitor.</p>
    Formula:C19H25ClN8
    Color and Shape:Solid
    Molecular weight:400.91
  • Antitumor agent-48


    <p>Antitumor agent-48, a 2,3-dehydrosilybin derivative, exhibits cytotoxicity on MCF-7, NCI-H1299, HepG2, HT29 cells; IC50 ranging 8.06-16.51 µM.</p>
    Formula:C35H34N2O14
    Color and Shape:Solid
    Molecular weight:706.65
  • VEGFR-2/DHFR-IN-1


    <p>Compound 8b inhibits VEGFR-2/DHFR, combats various bacteria, and fights cancer cells.</p>
    Formula:C20H18ClNO4
    Color and Shape:Solid
    Molecular weight:371.81
  • TEI-9063

    CAS:
    <p>TEI-9063 is a stable and highly specific prostacyclin analogue of prostacyclin receptor in mast cell tumor p-815 cells.</p>
    Formula:C23H38O4
    Color and Shape:Solid
    Molecular weight:378.55
  • PF 03709270

    CAS:
    <p>PF 03709270 is an oral prodrug of sulopenem with broad-spectrum antibacterial effects on gram-positive and gram-negative bacteria.</p>
    Formula:C19H27NO7S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:477.61
  • SCH-900822

    CAS:
    <p>SCH-900822 is a potent and selective glucagon receptor antagonist.</p>
    Formula:C34H43Cl2N7O2
    Color and Shape:Solid
    Molecular weight:652.66
  • ADH-6

    CAS:
    <p>ADH-6, a tripyridylamide, disrupts mutant p53 aggregates in cancer cells, reviving its function and inducing apoptosis.</p>
    Formula:C29H36N8O9
    Color and Shape:Solid
    Molecular weight:640.64
  • KPC-2-IN-2


    <p>KPC-2-IN-2 (6c) inhibits KPC-2 enzyme in Klebsiella pneumoniae (Ki 0.038 μM) and boosts cefotaxime in E. coli KPC-2.</p>
    Formula:C12H10BN3O2S
    Color and Shape:Solid
    Molecular weight:271.1
  • AZD-3409

    CAS:
    <p>AZD-3409 is a more potent prenyl transferase inhibitor than lonafarnib with varied IC(50) in cells, acting on gefitinib-resistant breast cancer.</p>
    Formula:C34H41FN4O4S2
    Color and Shape:Solid
    Molecular weight:652.84
  • LHC-165

    CAS:
    <p>LHC-165 is an agonist of TLR7. It also has the potential to treat solid tumors.</p>
    Formula:C29H32F2N3O7P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:603.55
  • NA 382

    CAS:
    <p>NA 382 is a staurosporine derivative that inhibits multidrug resistance.</p>
    Formula:C31H28N4O6
    Color and Shape:Solid
    Molecular weight:552.58
  • DNA crosslinker 4 dihydrochloride

    CAS:
    <p>DNA Crosslinker 4 binds DNA's minor groove, inhibits NCI-H460, A2780, MCF-7 cancer cells, and is used in cancer research.</p>
    Formula:C16H24Cl2N8O
    Color and Shape:Solid
    Molecular weight:415.32
  • Valopicitabine dihydrochloride

    CAS:
    <p>Valopicitabine, a NS5B inhibitor, is used potentially for the treatment of HCV infection.</p>
    Formula:C15H25ClN4O6
    Color and Shape:Solid
    Molecular weight:392.84
  • Anticancer agent 79


    <p>Anticancer agent 79 (3d) has potent activity against breast cancer, with cytotoxic effects on T47-D, IC50=13.64±0.26μM.</p>
    Formula:C20H12F3NO5
    Color and Shape:Solid
    Molecular weight:403.31
  • Antitubercular agent-16


    <p>Compound 5q is a potent antitubercular with low MIC90 values (0.40-23.51 μg/mL) against M. tuberculosis strains, showing minimal cytotoxicity.</p>
    Formula:C21H27N3S
    Color and Shape:Solid
    Molecular weight:353.52
  • CH5447240

    CAS:
    <p>CH5447240: potent hPTHR1 agonist, treats Hypoparathyroidism, EC50 12 nM, 55% oral bioavailability, raises rat serum calcium.</p>
    Formula:C26H39N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:517.68
  • RAD51-IN-8


    <p>RAD51-IN-8 inhibits RAD51-BRCA2 interaction and H4A4 with EC50 of 19 μM; a micromolar PPI inhibitor.</p>
    Formula:C16H14Cl2FN3O2
    Color and Shape:Solid
    Molecular weight:370.21
  • VEGFR-2-IN-14


    <p>VEGFR-2-IN-14 (Compound 5) is a potent inhibitor of VEGFR-2, which inhibits the growth of HepG2 cells in the Pre-G1 phase and induces apoptosis.</p>
    Formula:C24H23N3O3S
    Color and Shape:Solid
    Molecular weight:433.52
  • TLN-232

    CAS:
    <p>TLN-232, a synthetic heptapeptide, may inhibit cancer by targeting M2PK to disrupt tumor cell energy production.</p>
    Formula:C36H49N9O7S2
    Color and Shape:Solid
    Molecular weight:783.96
  • Cyclic-di-GMP sodium


    <p>c-di-GMP sodium: STING activator, regulates bacteria biofilm, motility, virulence.</p>
    Formula:C20H24N10NaO14P2
    Color and Shape:Solid
    Molecular weight:713.08464
  • PF-03715455

    CAS:
    <p>PF-03715455 is a potent p38 MAPK inhibitor, reducing TNFα in blood (IC50=1.7 nM) with selectivity for p38α, and may treat COPD.</p>
    Formula:C35H34ClN7O3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:700.27
  • Antitumor agent-75


    <p>Antitumor agent-75 is a novel and potent antitumor agent.</p>
    Formula:C26H23FN6
    Color and Shape:Solid
    Molecular weight:438.5
  • OUN58101

    CAS:
    <p>OUN58101, also MDK-8101/BI-D, is an RSV L-protein inhibitor with no formal name, first reported in patent WO 2005042530.</p>
    Formula:C32H36N6O6
    Color and Shape:Solid
    Molecular weight:600.66