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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66639 products of "Inhibitors"

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  • DNA-PK-IN-9


    <p>DNA-PK-IN-9 (YK6) is a potent DNA-PK inhibitor with an IC50 of 10.47 nM, important in cancer research.</p>
    Formula:C21H21N5O2
    Color and Shape:Solid
    Molecular weight:375.42
  • AChE/BChE-IN-1


    <p>AChE/BChE-IN-1: dual AChE/BChE inhibitor, IC50 of 1.06 nM/7.3 nM, crosses blood-brain barrier, with antioxidant properties for Alzheimer's research.</p>
    Formula:C32H35ClN6O3
    Color and Shape:Solid
    Molecular weight:587.11
  • cis-RdRP-IN-5


    <p>Cis-RdRP-IN-5 is an effective inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), employed in influenza virus research.</p>
    Formula:C23H21N3O5
    Color and Shape:Solid
    Molecular weight:419.43
  • Antidepressant agent 2


    <p>Antidepressant agent 2 showed significant antidepressant effects with a MED value of 0.1 mg/kg.</p>
    Formula:C21H22ClFN2O3S
    Color and Shape:Solid
    Molecular weight:436.93
  • IRAK4-IN-12


    <p>IRAK4-IN-12 (compound 37) is a potent inhibitor of IRAK4 (IC50: 0.015 μM) with cellular pIRAK4 potency (IC50: 0.5 μM).</p>
    Formula:C24H31FN8O
    Color and Shape:Solid
    Molecular weight:466.55
  • AFP-07 free acid

    CAS:
    <p>AFP 07 free acid is a 7,7-difluoroprostacyclin derivative. It also acts as a selective and highly potent agonist for the IP receptor.</p>
    Formula:C22H30F2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.47
  • WAY-855

    CAS:
    <p>WAY-855 is an EAAT2-preferring, nonsubstrate inhibitor of high-affinity glutamate uptake.</p>
    Formula:C9H11NO4
    Color and Shape:Solid
    Molecular weight:197.19
  • L 702007

    CAS:
    <p>L 702007 is an inhibitor of HIV-1 reverse transcriptase.</p>
    Formula:C18H25N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.41
  • GKA50 quarterhydrate


    <p>GKA50 quarterhydrate: glucokinase activator, EC50 of 33 nM, boosts insulin, cuts glucose in rats.</p>
    Formula:C26H30N2O7
    Color and Shape:Solid
    Molecular weight:469.01
  • SR121566A

    CAS:
    <p>SR121566A is a novel non-peptide antagonist of Glycoprotein IIb/IIIa (GP IIb-IIIa).</p>
    Formula:C20H25N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.51
  • Teslexivir

    CAS:
    <p>Teslexivir is a topical antiviral agent that is an effective and selective inhibitor of the interaction between two essential viral proteins, E1 and E2.</p>
    Formula:C35H36BrN3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:642.58
  • hMAO-B/MB-COMT-IN-2


    <p>Dual inhibitor hMAO-B/MB-COMT-IN-2 targets hMAO-B (IC50: 4.27μM) &amp; MB-COMT (IC50: 2.69μM), aids in neurodegenerative research.</p>
    Formula:C17H18N2O3
    Color and Shape:Solid
    Molecular weight:298.34
  • Dihydrokainic acid

    CAS:
    <p>EAAT2(GLT1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptake</p>
    Formula:C10H17NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:215.25
  • CDK7-IN-17

    CAS:
    <p>CDK7-IN-17, a pyrimidine-based CDK7 inhibitor, shows promise for various cancers, especially with abnormal transcription.</p>
    Formula:C24H26F3N6OP
    Color and Shape:Solid
    Molecular weight:502.47
  • J-104132

    CAS:
    <p>J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.</p>
    Formula:C31H33NO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.60
  • GPR84 antagonist 1


    <p>GPR84 antagonist 1 is a highly selective, high-affinity competitive antagonist of human GPR84.</p>
    Formula:C26H22N4O2
    Color and Shape:Solid
    Molecular weight:422.48
  • MSX-3 free acid

    CAS:
    <p>MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.</p>
    Formula:C21H23N4O7P
    Color and Shape:Solid
    Molecular weight:474.40
  • Fusarochromanone

    CAS:
    <p>Fusarochromanone (FC-101) is a mycotoxin produced by Fusarium oxysporum with potent antiangiogenic, anticancer and antimalarial activities.</p>
    Formula:C15H20N2O4
    Purity:95.31% - 96%
    Color and Shape:Solid
    Molecular weight:292.33
  • Tofacitinib Prodrug-1


    <p>Tofacitinib Prodrug-1: an oral prodrug reducing Tofacitinib's side effects, treats ulcerative colitis in mice effectively with low toxicity.</p>
    Formula:C36H39ClN10O7
    Color and Shape:Solid
    Molecular weight:759.21
  • MTL-CEBPA


    <p>MTL-CEPBA is a small activating RNA that targets C/EBPα upregulation and exhibits anti-inflammatory and anti-cancer effects.</p>
    Color and Shape:Solid
  • MI-1851

    CAS:
    <p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>
    Formula:C34H53N15O6
    Color and Shape:Solid
    Molecular weight:767.88
  • PCSK9-IN-16

    CAS:
    <p>PCSK9-IN-16, holds potential for research into hypercholesterolemia and other cardiovascular diseases [1].</p>
    Formula:C16H20N6O2S3
    Color and Shape:Solid
    Molecular weight:424.56
  • PPARγ phosphorylation inhibitor 1


    <p>PPARγ phosphorylation inhibitor 1 (Compound 10) is a potent PPARγ binding agent (IC50: 24 nM) with antidiabetic effects.</p>
    Formula:C22H14Cl2N2O4
    Color and Shape:Solid
    Molecular weight:441.26
  • (±)-J 113397

    CAS:
    <p>(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM).</p>
    Formula:C24H37N3O2
    Color and Shape:Solid
    Molecular weight:399.57
  • TAK-915

    CAS:
    <p>TAK-915: potent, brain-ready PDE2A inhibitor, 0.61 nM IC50, 4100x selectivity over PDE1A.</p>
    Formula:C19H18F4N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:458.36
  • SARS-CoV-2-IN-6


    <p>SARS-CoV-2-IN-6 is an inhibitor of SARS-CoV-2 3CLpro with the IC 50 value of 73 nM.</p>
    Formula:C17H13ClN2O2
    Color and Shape:Solid
    Molecular weight:312.75
  • Dazucorilant

    CAS:
    <p>Dazucorilant (CORT113176), a selective non-steroidal GR modulator, has high affinity with a K i &lt;1 nM, useful for neurological research.</p>
    Formula:C29H22F4N4O3S
    Color and Shape:Solid
    Molecular weight:582.57
  • BAY-899

    CAS:
    <p>BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.</p>
    Formula:C25H19F2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.45
  • PIKfyve-IN-1


    <p>PIKfyve-IN-1: potent, cell-active inhibitor for PIKfyve research, IC50=6.9 nM.</p>
    Formula:C20H21N5
    Color and Shape:Solid
    Molecular weight:331.41
  • MetRS-IN-1

    CAS:
    <p>MetRS-IN-1 (Compound 27) is an inhibitor of E. coli methionyl-tRNA synthetase (MetRS) with an IC50 value of 237 nM [1].</p>
    Formula:C15H13N3O4S
    Color and Shape:Solid
    Molecular weight:331.35
  • AHR antagonist 5 hemimaleate


    <p>Potent oral AHR antagonist with IC50 &lt; 0.5 μM, hinders tumor growth with anti-PD-1.</p>
    Formula:C29H28FN7O4
    Color and Shape:Solid
    Molecular weight:499.55
  • Antibacterial agent 112


    <p>Compound 112: Powerful antibacterial, MIC 1250 μM against B. subtilis, E. coli, E. faecalis, S. typhimurium, S. aureus; also an HIV-1 antibody.</p>
    Formula:C35H23N5O5
    Color and Shape:Solid
    Molecular weight:593.59
  • LIT-001 free base

    CAS:
    <p>LIT-001, a nonpeptide OT-R agonist, enhances mouse autism-like behavior, with EC50=55 nM and Ki=226 nM.</p>
    Formula:C28H33N7O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.67
  • Lafadofensine (D-(-)-Mandelic acid)


    <p>Lafadofensine D-(-)-Mandelic acid is a monoamines reuptake inhibitor with adequate effects when administered short-term.</p>
    Formula:C32H32F2N2O6
    Color and Shape:Solid
    Molecular weight:578.6
  • Zetomipzomib

    CAS:
    <p>KZR-616: Immunoproteasome inhibitor targeting LMP7 (IC50: 39/57 nM) &amp; LMP2 (IC50: 131/179 nM), potential in autoimmune disease research.</p>
    Formula:C30H42N4O8
    Color and Shape:Solid
    Molecular weight:586.68
  • PTP1B-IN-18


    <p>PTP1B-IN-18 is an orally active, fully mixed protein tyrosine phosphatase 1B (PTP1B) inhibitor (Ki: 35.2 μM).PTP1B-IN-18 can be used to study type 2 diabetes.</p>
    Formula:C26H19N3O4S
    Color and Shape:Solid
    Molecular weight:469.51
  • GSK268


    <p>GSK268 is a BET inhibitor.</p>
    Formula:C26H27N5O3
    Color and Shape:Solid
    Molecular weight:457.53
  • IAB15

    CAS:
    <p>IAB15 is a potent inhibitor of T-type calcium channel that can be used in the research of epilepsy [1].</p>
    Formula:C15H14F3NO2
    Color and Shape:Solid
    Molecular weight:297.27
  • (S)-ZG197


    <p>(S)-ZG197 is a compound that acts as a highly selective activator of the Staphylococcus aureus Caseinolytic Protease P (Sa ClpP), demonstrating efficacy at a</p>
    Formula:C28H35F3N4O3
    Color and Shape:Solid
    Molecular weight:532.6
  • GSK789

    CAS:
    <p>GSK789 is a selective inhibitor of the first bromodomains (BD1) of the bromo and extra terminal domain (BET) proteins.</p>
    Formula:C26H33N5O3
    Color and Shape:Solid
    Molecular weight:463.57
  • EED ligand 1


    <p>EED ligand 1: potent PRC2 inhibitor targeting EED subunit.</p>
    Formula:C19H19FN8O
    Color and Shape:Solid
    Molecular weight:394.41
  • KUS121

    CAS:
    <p>KUS121: VCP ATPase activity inhibitor (IC50=330 nM), protects cells from ER stress, assists in cerebral ischemia, and preserves vision in retinitis pigmentosa.</p>
    Formula:C22H17FN4NaO3S
    Color and Shape:Solid
    Molecular weight:459.45
  • Ro 0437626

    CAS:
    <p>P2X1 purinergic receptor antagonist</p>
    Formula:C27H35N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:525.66
  • Aurora A inhibitor 1

    CAS:
    <p>Aurora A inhibitor 1: potent, selective, targets cancer-linked Aurora A overexpression, potential for cancer research. (WO2021147974A1, 49)</p>
    Formula:C25H28ClF2N5O2
    Color and Shape:Solid
    Molecular weight:503.97
  • Y1 receptor antagonist 1

    CAS:
    <p>Y1 receptor antagonist 1 is an antagonist of neuropeptide Y1 receptor.</p>
    Formula:C28H33N5O3
    Purity:98.17%
    Color and Shape:Solid
    Molecular weight:487.59
  • KRAS G12C inhibitor 33

    CAS:
    <p>KRAS G12C inhibitor 33 is a KRAS G12C inhibitor that can be used to study cancer.</p>
    Formula:C30H33N7O3
    Color and Shape:Solid
    Molecular weight:539.63
  • SPR-00305

    CAS:
    <p>SPR-00305 is a novel potent inhibitor of the mvfr pathway</p>
    Formula:C24H19ClN2O3
    Color and Shape:Solid
    Molecular weight:418.87
  • Alkannin

    CAS:
    <p>Alkannin: potent, tumor-specific PKM2 inhibitor; non-inhibitory to PKM1/PKL; potential anticancer agent.</p>
    Formula:C16H16O5
    Color and Shape:Solid
    Molecular weight:288.3
  • ChemR23-IN-3


    <p>ChemR23-IN-3 is a potent thiazole-based ChemR23 inhibitor with an IC 80 value of 12 nM.</p>
    Formula:C31H33N5O5S2
    Color and Shape:Solid
    Molecular weight:619.75
  • COX-1/2-IN-2


    <p>COX-1/2-IN-2, a potent dual inhibitor, has IC50s: COX-1 at 9.7μM &amp; COX-2 at 4.6μM.</p>
    Formula:C15H10ClIN2O
    Color and Shape:Solid
    Molecular weight:396.61
  • Dicetrorelix pamoate

    CAS:
    <p>Cetrorelix pamoate is a synthetic decapeptide that acts as a GnRH antagonist, inhibiting the release of LH and FSH from the pituitary.</p>
    Formula:C163H200Cl2N34O34
    Color and Shape:Solid
    Molecular weight:3250.49
  • AM-6494

    CAS:
    <p>AM-6494 is a potent and orally active BACE1 inhibitor (IC50: 0.4 nM) with in vivo selectivity over BACE2 (IC50: 18.6 nM).</p>
    Formula:C22H21F2N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:473.5
  • S1P1 agonist 5


    <p>Selective oral S1P1 agonist 5 inhibits lymphocyte drainage, potential for MS research.</p>
    Formula:C23H24ClN2NaO4
    Color and Shape:Solid
    Molecular weight:450.89
  • MALT1-IN-5

    CAS:
    <p>MALT1-IN-5 is a potent inhibitor of the MALT1 protease and can be used in cancer research.</p>
    Formula:C17H17ClF2N6O3
    Color and Shape:Solid
    Molecular weight:426.80
  • Lu 26-046

    CAS:
    <p>Lu 26-046 is a muscarinic receptor agonist.</p>
    Formula:C10H12N2OS
    Color and Shape:Solid
    Molecular weight:208.28
  • BET-IN-6

    CAS:
    <p>BET-IN-6: Potent BRD2/4 inhibitor and ligand for PROTAC BRD2/BRD4 degrader-1 synthesis.</p>
    Formula:C22H20N2O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.47
  • Tzc 5665

    CAS:
    <p>Tzc 5665 is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory action.</p>
    Formula:C31H38ClN5O7
    Color and Shape:Solid
    Molecular weight:628.12
  • (RS)-AMPA hydrobromide

    CAS:
    AMPAR agonist
    Formula:C7H11BrN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.08
  • D4R antagonist-1


    <p>Potent, selective D4R antagonist; IC50 = 6.87 µM; potential in Parkinson’s disease research.</p>
    Formula:C21H25F2NO2
    Color and Shape:Solid
    Molecular weight:361.43
  • Omaciclovir

    CAS:
    <p>Omaciclovir (ABT-091) is a herpesvirus herpesvirus replication inhibitor with antiviral activity that is used in the study of herpesvirus infections.</p>
    Formula:C10H15N5O3
    Purity:99.46% - 99.46%
    Color and Shape:Solid
    Molecular weight:253.26
  • SM-433 hydrochloride


    <p>SM-433 hydrochloride, a Smac mimetic &amp; IAP inhibitor, binds XIAP BIR3; potent IC50 &lt;1 μM. (Patent WO2008128171A2)</p>
    Formula:C32H44ClN5O4
    Color and Shape:Solid
    Molecular weight:598.18
  • Antitubercular agent-29


    <p>Compound 6xa inhibits drug-resistant tuberculosis with MICs 0.03 μg/mL for DS-Mtb and 0.03-0.06 for DR-Mtb, SI&gt;40 for Vero cells.</p>
    Formula:C20H12ClN3O5
    Color and Shape:Solid
    Molecular weight:409.78
  • Antitumor agent-47


    <p>Antitumor agent-47, a silibinin derivative, shows cytotoxicity in NCI-H1299 (IC50: 8.07µM) and HT29 (IC50: 6.27µM) cells.</p>
    Formula:C30H27NO11
    Color and Shape:Solid
    Molecular weight:577.54
  • ATM Inhibitor-3


    <p>ATM Inhibitor-3 selectively inhibits ATM (IC50: 0.71 nM), targets PI3K kinase family, and is metabolically stable.</p>
    Formula:C25H29FN6O3
    Color and Shape:Solid
    Molecular weight:480.53
  • Lentiginosine

    CAS:
    <p>Lentiginosine is a selective amyloglucosidase inhibitor.</p>
    Formula:C8H15NO2
    Color and Shape:Solid
    Molecular weight:157.21
  • DHU-Se1


    <p>DHU-Se1: potent anti-inflammatory, releases reactive selenium from macrophages, inhibits iNOS/TNF-α, blocks M0 to M1 polarization.</p>
    Formula:C23H23N3OSSe
    Color and Shape:Solid
    Molecular weight:468.47
  • PD 113271

    CAS:
    <p>PD 113,271 is an analog of the fermentation products fostriecin with antitumor activity in vitro and in vivo.</p>
    Formula:C19H27O10P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:446.39
  • STA 2

    CAS:
    <p>STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.</p>
    Formula:C21H34O3S
    Color and Shape:Solid
    Molecular weight:366.56
  • LAF-153

    CAS:
    <p>LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.</p>
    Formula:C18H32N2O7
    Color and Shape:Solid
    Molecular weight:388.46
  • EGFR/HER2-IN-5


    <p>EGFR/HER2-IN-5: Irreversible, oral dual EGFR inhibitor, IC50 0.6 nM, targets L858R/T790M mutations, anti-tumor in vivo for lung cancer study.</p>
    Color and Shape:Solid
  • G-479

    CAS:
    <p>G-479, a potent MEK inhibitor and improved analogue of GDC-0623, has distributed polarity enhancing bioactivity.</p>
    Formula:C16H15FIN5O4
    Color and Shape:Solid
    Molecular weight:487.22
  • CE-2072

    CAS:
    <p>CE-2072 is a synthetic host serine proteases inhibitor.</p>
    Formula:C33H41N5O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:603.71
  • SBI-581


    <p>SBI-581: oral, potent TAO3 inhibitor, IC50=42nM, alters TKS5α at RAB11+ vesicles, blocks invadopodia, good mouse pharmacokinetics, anti-tumor.</p>
    Formula:C24H21N3O2
    Color and Shape:Solid
    Molecular weight:383.44
  • Anti-Influenza agent 3


    <p>Compound 11h: Potent, low-toxicity anti-influenza, inhibits M2 ion channels. EC50: 3.29μM (H3N2), 2.45μM (H1N1).</p>
    Formula:C16H22ClNOS
    Color and Shape:Solid
    Molecular weight:311.87
  • NSD2-IN-1

    CAS:
    <p>NSD2-IN-1: potent, selective NSD2-PWWP1 inhibitor, IC50 0.11 μM, induces gene expression changes, apoptosis, cell cycle arrest.</p>
    Formula:C29H31N5
    Color and Shape:Solid
    Molecular weight:449.59
  • JTE 151A

    CAS:
    <p>JTE-151 is a novel RORγ inverse agonist.</p>
    Formula:C26H30ClN3O5
    Color and Shape:Solid
    Molecular weight:499.99
  • Namitecan

    CAS:
    <p>Namitecan is an effective inhibitor of topoisomerase I. It has antitumor property.</p>
    Formula:C23H22N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:434.44
  • Pparδ agonist 5


    <p>Pparδ agonist 5 is a selective, orally active PPARδ agonist with an EC50 of 0.335 μM and better selectivity than GW0742.</p>
    Formula:C23H21F3N2O2S
    Color and Shape:Solid
    Molecular weight:446.49
  • LpxA-IN-1

    CAS:
    <p>LpxA-IN-1, a novel UDP-N-acetylglucosamine acyltransferase (LpxA) inhibitor exhibiting potent activity (IC 50 2 nM), effectively targets Pseudomonas aeruginosa</p>
    Formula:C21H11D7F3N5O3
    Color and Shape:Solid
    Molecular weight:452.44
  • Antibiotic MA 144M1

    CAS:
    <p>Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.</p>
    Formula:C42H55NO15
    Color and Shape:Solid
    Molecular weight:813.88
  • Topo I/COX-2-IN-1


    <p>Topo I/COX-2-IN-1: potent dual inhibitor; IC50 0.24μM (COX-2), 4.42μM (Topo I); anti-cancer; induces apoptosis, halts migration.</p>
    Formula:C21H18ClFN2O3
    Color and Shape:Solid
    Molecular weight:400.83
  • Unoprostone isopropyl

    CAS:
    <p>Unoprostone isopropyl, a prostanoid and synthetic docosanoid, is approved for the treatment of ocular hypertension and open-angle glaucoma.</p>
    Formula:C25H44O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:424.61
  • WQ3810

    CAS:
    <p>WQ3810 is an orally active fluoroquinolone, has potent antibacterial activities.</p>
    Formula:C22H22F3N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:461.44
  • RORγt inverse agonist 29


    <p>RORγt inverse agonist 29 is a potent, selective, orally active RORγt inverse agonist with an IC50 value of 21 nM.</p>
    Formula:C25H24N2O5S
    Color and Shape:Solid
    Molecular weight:464.53
  • Orvepitant

    CAS:
    <p>Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.</p>
    Formula:C31H35F7N4O2
    Color and Shape:Solid
    Molecular weight:628.62
  • MI-1481

    CAS:
    <p>MI-1481: potent MML1 inhibitor, IC50 3.6 nM; disrupts menin-MLL1, active in MLL leukemia.</p>
    Formula:C29H30F3N7O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:597.65
  • Topo I/COX-2-IN-2


    <p>Compound W10 is a dual inhibitor of Topo I (IC50: 0.90μM) and COX-2 (IC50: 2.31μM), inducing cancer cell apoptosis via mitochondria.</p>
    Formula:C24H25ClN4O
    Color and Shape:Solid
    Molecular weight:420.93
  • CTX-712

    CAS:
    <p>CTX-712 is a potent inhibitor of cdc2-like kinase ( CLK ). CTX-712 inhibits inhibits cancer survival and cancer cell growth.</p>
    Formula:C19H17FN8O2
    Color and Shape:Solid
    Molecular weight:408.39
  • COX-2/PI3K-IN-2


    <p>COX-2/PI3K-IN-2 (5f): anti-inflammatory &amp; anti-cancer, selectively inhibits COX-2 (Ki=3.02nM), potently blocks PI3K (IC50=2.78nM).</p>
    Formula:C16H17N5O2
    Color and Shape:Solid
    Molecular weight:311.34
  • Cap-dependent endonuclease-IN-5

    CAS:
    <p>Cap-dependent endonuclease-IN-5 inhibits CEN and fights influenza with low toxicity and good in vivo properties.</p>
    Formula:C27H21F2N3O4S2
    Color and Shape:Solid
    Molecular weight:553.60
  • Adafosbuvir

    CAS:
    <p>Adafosbuvir has antiviral activity.</p>
    Formula:C22H29FN3O10P
    Color and Shape:Solid
    Molecular weight:545.457
  • GLP-1R agonist 8

    CAS:
    <p>GLP-1R agonist 8 is a potent agonist of GLP-1R (EC50 &lt; 2 nM).</p>
    Formula:C33H32N4O5
    Color and Shape:Solid
    Molecular weight:564.63
  • BM635 hydrochloride


    <p>BM635 hydrochloride, an MmpL3 inhibitor, strongly blocks Divergent bacteriophage H37Rv (MIC50: 0.08 μM), with doubled in vivo potency.</p>
    Formula:C25H30ClFN2O
    Color and Shape:Solid
    Molecular weight:428.97
  • Lp-PLA2-IN-6

    CAS:
    <p>Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.</p>
    Formula:C25H21F5N4O3
    Color and Shape:Solid
    Molecular weight:520.45
  • CHK1-IN-2

    CAS:
    <p>CHK1-IN-2 is an inhibitor of checkpoint kinase 1 (CHK1; IC50: 6 nM).</p>
    Formula:C20H22N4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:366.48
  • PptT-IN-1


    <p>PptT-IN-1, a potent PptT inhibitor (IC50: 2.8 μM), shows promise for tuberculosis research.</p>
    Formula:C18H29N5O2
    Color and Shape:Solid
    Molecular weight:347.46
  • Autophagy-IN-1


    <p>Autophagy-IN-1 blocks autophagy in cancer cells, hinders tumor growth in mice, and aids in studying colorectal cancer.</p>
    Formula:C23H25NO7
    Color and Shape:Solid
    Molecular weight:427.45
  • BU09059

    CAS:
    <p>BU09059 is a potent, selective, short-acting antagonist of the κ-opioid receptor (KOR).</p>
    Formula:C28H37N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:495.61
  • GYKI-53784

    CAS:
    <p>GYKI-53784 (LY 303070) is an effective selective AMPA receptor antagonist.</p>
    Formula:C19H20N4O3
    Color and Shape:Solid
    Molecular weight:352.39
  • PDE4-IN-12


    <p>PDE4-IN-12 is a potent and safe PDE4 ubiquitous inhibitor that acts on PDE4 (IC50: 3.5 nM, SI: 2.71) and PDE7 (IC50: 15 nM, SI: 4.27).</p>
    Formula:C34H35NO6
    Color and Shape:Solid
    Molecular weight:553.64