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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66641 products of "Inhibitors"

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  • Stauprimide

    CAS:
    <p>Stauprimide inhibits MYC by blocking NME2, reducing MYC transcription in ESCs.</p>
    Formula:C35H28N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:584.62
  • GnRH-R antagonist 1

    CAS:
    <p>Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.</p>
    Formula:C31H28F5N7O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:721.65
  • XO/COX/LOX-IN-1


    <p>XO/COX/LOX-IN-1 targets XO/COX/LOX, used in research of inflammation, cancer, and metabolic disorders.</p>
    Formula:C24H20N4O2S
    Color and Shape:Solid
    Molecular weight:428.51
  • Cilazapril HCl

    CAS:
    <p>Cilazapril, also known as Ro 31 2848, is a potent ACE inhibitor used for hypertension.</p>
    Formula:C22H32ClN3O5
    Color and Shape:Solid
    Molecular weight:453.96
  • Trypanothione synthetase-IN-4


    <p>Trypanothione synthetase-IN-4, an L. infantum inhibitor, has potent anti-leishmanicidal properties (EC50: 0.6 μM).</p>
    Formula:C29H52INO2
    Color and Shape:Solid
    Molecular weight:573.63
  • SCP1-IN-2


    <p>SCP1-IN-2: potent, selective SCP1 inhibitor; induces REST degradation, hinders its activity, may study REST-driven glioblastoma growth.</p>
    Formula:C19H17F3N2O6S2
    Color and Shape:Solid
    Molecular weight:490.47
  • AZD-4121 tert-butylammonium

    CAS:
    <p>AZD-4121 tert-butylammonium is an oral cholesterol absorption inhibitor targeting NPC1L1 for the treatment of dyslipidaemia.</p>
    Formula:C40H50F2N4O7S
    Color and Shape:Solid
    Molecular weight:768.91
  • LSD1-IN-21


    <p>LSD1-IN-21: potent LSD1 inhibitor, crosses blood-brain barrier, IC50 of 0.956 μM; lowers TNF-α, anti-cancer, anti-inflammatory.</p>
    Formula:C24H25N5O2S
    Color and Shape:Solid
    Molecular weight:447.55
  • ZIKV-IN-4


    <p>ZIKV-IN-4 is a low cytotoxic, acid-stable anti-ZIKV agent with an EC50 value of 3.49 μM. ZIKV-IN-4 exhibited potent inhibition of ZIKV NS5 MTase.</p>
    Formula:C33H37NO4
    Color and Shape:Solid
    Molecular weight:511.65
  • MI-1851

    CAS:
    <p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>
    Formula:C34H53N15O6
    Color and Shape:Solid
    Molecular weight:767.88
  • KY-02327 acetate


    <p>KY-02327 acetate inhibits Dvl-CXXC5, stabilizes Wnt/β-catenin signaling, and enhances osteoblast differentiation.</p>
    Formula:C22H31N3O6
    Color and Shape:Solid
    Molecular weight:433.5
  • 9(R)-HETE

    CAS:
    <p>9(R)-HETE, 50% of racemic mix, activates RXRγ 1.5x at 300 nM; identified by HPLC comparison.</p>
    Formula:C20H32O3
    Color and Shape:Solid
    Molecular weight:320.47
  • ADH-6

    CAS:
    <p>ADH-6, a tripyridylamide, disrupts mutant p53 aggregates in cancer cells, reviving its function and inducing apoptosis.</p>
    Formula:C29H36N8O9
    Color and Shape:Solid
    Molecular weight:640.64
  • CCR5 antagonist 1

    CAS:
    <p>CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.</p>
    Formula:C39H46ClF2N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:738.33
  • LT-850-166


    <p>LT-850-166 is a potent inhibitor of FLT3 and has shown efficacy in overcoming a wide range of FLT3 mutations.</p>
    Formula:C30H29Cl2N7O
    Color and Shape:Solid
    Molecular weight:574.5
  • A 70450

    CAS:
    <p>A 70450, an inhibitor of aspartyl proteinase, can be used as an antifungal agent and may have a role in HIV protease inhibition therapy.</p>
    Formula:C42H71ClN6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:775.50
  • P053

    CAS:
    <p>P053: potent, selective CerS1 inhibitor, IC50 = 0.5µM, curbs muscle fat oxidation, affects body fat.</p>
    Formula:C18H21Cl2NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:354.27
  • L 689065

    CAS:
    <p>L 689065 is a 5-lipoxygenase inhibitor.</p>
    Formula:C35H33ClN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:597.17
  • AZ-PFKFB3-67 quarterhydrate


    <p>AZ-PFKFB3-67 quarterhydrate inhibits PFKFB3 (IC50: 11 nM), PFKFB2 (159 nM), and PFKFB1 (1130 nM).</p>
    Formula:C26H27N5O4
    Color and Shape:Solid
    Molecular weight:460.01
  • Belatacept

    CAS:
    <p>Belatacept (BMS 224818), a T-cell costimulation inhibitor, targets CD80/86 for transplant immunosuppression.</p>
    Color and Shape:Liquid
  • GSK-3β inhibitor 7


    <p>GSK-3β inhibitor 7 is a GSK-3β inhibitor (IC50: 5.25 μM).</p>
    Formula:C27H23BrN4O2S
    Color and Shape:Solid
    Molecular weight:547.47
  • BI-207524

    CAS:
    <p>BI-207524 is a novel NS5B Thumb Pocket 1 Inhibitor with Improved Potency for the Potential Treatment of Chronic Hepatitis C Virus Infection.</p>
    Formula:C35H36ClN5O5
    Color and Shape:Solid
    Molecular weight:642.14
  • Amdinocillin methylacetate

    CAS:
    <p>Amdinocillin methylacetate is a Synthetic penicillin.</p>
    Formula:C18H27N3O4S
    Color and Shape:Solid
    Molecular weight:381.49
  • BMS-986163

    CAS:
    <p>BMS-986163, a prodrug, quickly becomes BMS-986169, a GluN2B inhibitor (Ki=4 nM, IC50=24 nM).</p>
    Formula:C23H28FN2O5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:462.45
  • MA242 free base

    CAS:
    <p>MA242 free base is a dual MDM2/NFAT1 inhibitor that triggers apoptosis in pancreatic cancer cells.</p>
    Formula:C24H20ClN3O3S
    Color and Shape:Solid
    Molecular weight:465.95
  • Chitin synthase inhibitor 12


    <p>Chitin synthase inhibitor 12: potent CHS blocker (IC50: 0.16 mM), broad-spectrum antifungal, effective against resistant strains. Useful in IFI research.</p>
    Formula:C23H21ClFN3O5
    Color and Shape:Solid
    Molecular weight:473.88
  • HCV-IN-38


    <p>Potent oral HCV inhibitor HCV-IN-38 has 15 nM EC50, 431 SI, high efficacy, and low toxicity.</p>
    Formula:C22H24ClF3N4O4
    Color and Shape:Solid
    Molecular weight:500.9
  • GSK-2878175

    CAS:
    <p>GSK-2878175, a NS5B inhibitor, is used potentially for the treatment of HCV infection.</p>
    Formula:C27H23BClFN2O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:568.81
  • Transthyretin-IN-1


    <p>Transthyretin-IN-1 inhibits TTR fibril formation, aiding Alzheimer’s research.</p>
    Formula:C10H9Br2NO4
    Color and Shape:Solid
    Molecular weight:366.99
  • Galidesivir

    CAS:
    <p>Galidesivir (BCX4430) is an antiviral compound that inhibits viral RNA-dependent RNA polymerase (RdRp) activity and reduces lung infections in infected animals.</p>
    Formula:C11H15N5O3
    Purity:96.73% - 99.13%
    Color and Shape:Solid
    Molecular weight:265.27
  • EF1502 free base

    CAS:
    <p>EF1502 is a potent and selective GABA transporter inhibitor.</p>
    Formula:C22H26N2O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.58
  • Aquayamycin

    CAS:
    <p>Aquayamycin is an anthraquinone derivative and inhibitor of the enzyme tyrosine hydroxylase..</p>
    Formula:C25H26O10
    Color and Shape:Solid
    Molecular weight:486.47
  • IRAK4-IN-11


    <p>IRAK4-IN-11 (compound 6) is a potent inhibitor of IRAK4 with an IC 50 of 0.008 μM. IRAK4-IN-11 exhibits cell pIRAK4 potencies with an IC 50 of 0.19 μM [1].</p>
    Formula:C16H19N7O
    Color and Shape:Solid
    Molecular weight:325.37
  • DSM705 hydrochloride


    <p>DSM705 hydrochloride: potent antimalarial, pyrrole-based DHODH inhibitor effective against Plasmodium, non-toxic to mammalian DHODH.</p>
    Formula:C19H20ClF3N6O
    Color and Shape:Solid
    Molecular weight:440.85
  • Norbinaltorphimine dihydrochloride

    CAS:
    <p>Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.</p>
    Formula:C40H45Cl2N3O6
    Purity:98.17% - 99.88%
    Color and Shape:Solid
    Molecular weight:734.71
  • Musettamycin

    CAS:
    <p>Musettamycin triggers erythroid differentiation in blood cells, acts like anthracycline antibiotics, but only inhibits gram-positive bacteria.</p>
    Formula:C36H45NO14
    Color and Shape:Solid
    Molecular weight:715.74
  • Tubulin polymerization-IN-33


    <p>Tubulin-IN-33, an oxazoloisoindole, hinders microtubule assembly; effective against NCI cancer cells.</p>
    Formula:C27H28N2O6
    Color and Shape:Solid
    Molecular weight:476.52
  • 5-HT7R antagonist 1


    <p>5-HT7R antagonist 1 is a G protein-biased antagonist with Ki of 6.5 nM for 5-HT 7R.</p>
    Formula:C14H18Cl2N4
    Color and Shape:Solid
    Molecular weight:313.23
  • MtTMPK-IN-1


    <p>MtTMPK-IN-1 inhibits MtTMPK with 2.5 μM IC50, shows moderate anti-tuberculosis activity, and is low in cytotoxicity.</p>
    Formula:C22H24N4O3
    Color and Shape:Solid
    Molecular weight:392.45
  • 9(S),10(S),13(S)-TriHOME

    CAS:
    <p>9(S),10(S),13(S)-TriHOME is an oxylipin derived from linoleic acid. It has been detected in beer and in bronchoalveolar lavage fluid (BALF) from female smokers.</p>
    Formula:C18H34O5
    Color and Shape:Solid
    Molecular weight:330.46
  • (S)-3-Hydroxy Midostaurin

    CAS:
    <p>(S)-3-Hydroxy Midostaurin is a potent inhibitor of kinases(IC50 of &lt;400 nM for 13 kinases (VEGFR-2, TRK-A, FLT3, et)).</p>
    Formula:C35H30N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:586.64
  • BTK-IN-16

    CAS:
    <p>BTK-IN-16 is a potential inhibitor of wild-type BTK and C481S mutants.BTK-IN-16 can be used to study various autoimmune diseases and cancers caused by BTK.</p>
    Formula:C15H14N4O2
    Purity:99.04%
    Color and Shape:Soild
    Molecular weight:282.3
  • VEGFR-2-IN-12


    <p>VEGFR-2-IN-12 (compound 6g), a 2-oxoquinoxalinyl-1,2,4-triazole, is a potent inhibitor of VEGFR-2 (IC50: 0.037 μM). VEGFR-2-IN-12 has anti-tumour effects.</p>
    Formula:C22H24N6O3S
    Color and Shape:Solid
    Molecular weight:452.53
  • SLC4011540


    <p>SLC4011540 is a potent and selective SphK1/2 dual inhibitor with Ki value of 120 nM and 90 nM respectively.</p>
    Formula:C24H23ClF3N7OS
    Color and Shape:Solid
    Molecular weight:550
  • Tabimorelin hemifumarate

    CAS:
    <p>orally active ghrelin receptor (GHS-R1a) agonist</p>
    Formula:C32H40N403C4H404
    Purity:98%
    Color and Shape:Solid
    Molecular weight:586.72
  • CCR4 antagonist 2

    CAS:
    <p>CCR4 antagonist 2 (Compound 31) is a novel potent, orally bioavailable small molecule antagonists of CC chemokine receptor 4 (CCR4) that inhibits Treg</p>
    Formula:C26H28Cl2N6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:511.45
  • NITD-688

    CAS:
    <p>NITD-688 is a pan-serotype inhibitor targeting the dengue virus NS4B protein, effective through oral administration.</p>
    Formula:C25H32N4O3S2
    Color and Shape:Solid
    Molecular weight:500.68
  • MLKL-IN-1


    <p>MLKL-IN-1 is a covalent inhibitor of MLKL with a Kd value of 50 μM.</p>
    Formula:C19H20N2O3
    Color and Shape:Solid
    Molecular weight:324.37
  • MK2-IN-4

    CAS:
    <p>MK2-IN-4 is a MAPKAPK2 (MK2) inhibitor (IC50: 45 nM). MK2-IN-4 can be used in cancer, inflammation and immunology studies.</p>
    Formula:C25H24N4O2
    Color and Shape:Solid
    Molecular weight:412.48
  • ROPA

    CAS:
    <p>ROPA, a potent PKCalpha and PKCgamma activator, promotes tumor growth through PKC-activation.</p>
    Formula:C28H32O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:464.55
  • Ep vinyl quinidine

    CAS:
    <p>3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.</p>
    Formula:C20H24N2O2
    Color and Shape:Solid
    Molecular weight:324.42
  • Topoisomerase II inhibitor 5


    <p>Topoisomerase II inhibitor 5 (Compound E24) is a DNAtopoisomerase II inhibitor with anticancer effects.</p>
    Formula:C26H27N5O4
    Color and Shape:Solid
    Molecular weight:473.52
  • Revexepride

    CAS:
    <p>Revexepride, a 5-HT4 agonist, may boost CYP3A4, used for treating GERD.</p>
    Formula:C21H32ClN3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:425.95
  • KRAS inhibitor-13

    CAS:
    <p>KRAS inhibitor-13 blocks KRAS G12C (IC50: 0.883 μM) and p-ERK in some cancer cells; promising for pancreatic, colorectal, lung cancer research.</p>
    Formula:C25H19ClFN3O2S
    Color and Shape:Solid
    Molecular weight:479.95
  • PF-06726304 acetate

    CAS:
    <p>PF-06726304 acetate is a selective inhibitor of EZH2, with robust antitumor growth activity.</p>
    Formula:C24H25Cl2N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:506.38
  • DMGF

    CAS:
    <p>DMGF, a biflavonoid from Taxus, induces apoptosis, autophagy, and inhibits B16F10 cell motility and MMP-2 expression, hindering melanoma metastasis.</p>
    Formula:C32H22O10
    Color and Shape:Solid
    Molecular weight:566.51
  • Antitumor agent-48


    <p>Antitumor agent-48, a 2,3-dehydrosilybin derivative, exhibits cytotoxicity on MCF-7, NCI-H1299, HepG2, HT29 cells; IC50 ranging 8.06-16.51 µM.</p>
    Formula:C35H34N2O14
    Color and Shape:Solid
    Molecular weight:706.65
  • AChE-IN-22


    <p>AChE-IN-22 (10q) selectively inhibits AChE (IC50: 0.88 μM), less on BuChE (IC50: 10 μM), targets CAS and PAS, useful in Alzheimer's research.</p>
    Formula:C21H20N4O5S
    Color and Shape:Solid
    Molecular weight:440.47
  • M3258

    CAS:
    <p>LMP7-IN-1 may used in the research of inflammatory and autoimmune diseases, neurodegenerative diseases, proliferative diseases and cancer, is an inhibitor of</p>
    Formula:C17H20BNO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.16
  • Trichostatin A S-isomer

    CAS:
    <p>Trichostatin A S-isomer, a HDAC 1, 3, 4, 6, 10 inhibitor with IC50 ~20 nM, has wide-ranging epigenetic effects.</p>
    Formula:C17H22N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.37
  • ONO-5334

    CAS:
    <p>ONO-5334: selective cathepsin K inhibitor, potential for osteoporosis study; Ki: 0.10 nM (human), 0.049 nM (rabbit), 0.85 nM (rat).</p>
    Formula:C21H34N4O4S
    Purity:98.22% - 99.60%
    Color and Shape:Solid
    Molecular weight:438.58
  • Ro 24-4383

    CAS:
    <p>Ro 24-4383 is a carbamate-linked dual-action antibacterial agent.</p>
    Formula:C32H31FN8O10S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:770.76
  • IL-17 modulator 1 disodium

    CAS:
    <p>Potent, orally active IL-17 Modulator 1 (disodium) from patent WO 2020127685, used in psoriasis and arthritis research.</p>
    Formula:C28H37N6NaO6P
    Color and Shape:Solid
    Molecular weight:607.604
  • Calphostin B

    CAS:
    <p>Calphostins, PKC inhibitors from Cladosporium fungus, include A, B, C, D, I; C is most potent.</p>
    Formula:C37H34O11
    Color and Shape:Solid
    Molecular weight:654.66
  • LPM4870108


    <p>LPM4870108: Potent, oral pan-Trk inhibitor, selective over ALK, with anti-tumor effects. TrkC IC50=0.2nM, TrkA IC50=2.4nM.</p>
    Formula:C20H19FN6O3
    Color and Shape:Solid
    Molecular weight:410.4
  • CCT369260

    CAS:
    <p>CCT369260 (compound 1), an orally active inhibitor targeting B-cell lymphoma 6 (BCL6), demonstrates anti-tumor efficacy with an IC50 value of 520 nM [1].</p>
    Formula:C24H31ClF2N6O2
    Color and Shape:Solid
    Molecular weight:508.99
  • DI-404

    CAS:
    <p>DI-404: Potent DCN1-UBC12 inhibitor, selectivity blocks cullin 3 neddylation, Kd=6.9 nM.</p>
    Formula:C35H45ClN6O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:713.29
  • FTO-IN-5

    CAS:
    <p>FTO-IN-5 is a potent, selective inhibitor targeting the fat mass obesity-associated protein (FTO).</p>
    Formula:C23H18Cl2N6O6
    Color and Shape:Solid
    Molecular weight:545.33
  • E7090 succinate

    CAS:
    <p>E7090 succinate inhibits FGFR1, FGFR2, and FGFR3 with IC50: 0.71, 0.50, 1.2 nM; less so FGFR4 at 120 nM.</p>
    Formula:C76H92N10O24
    Color and Shape:Solid
    Molecular weight:1529.60
  • MIV-150

    CAS:
    <p>MIV-150 is a nonnucleoside inhibitor of reverse transcriptase (NNRT). MIV-150 also blocking HIV-1 and HIV-2 infections (EC50&lt;1 nM against HIV-1/HIV-2MN).</p>
    Formula:C19H17FN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.36
  • HIF-1/2α-IN-1


    <p>HIF-1/2α-IN-1, an orally active compound, functions as an inhibitor of HIF-2α.</p>
    Formula:C17H16N6O4
    Color and Shape:Solid
    Molecular weight:368.35
  • BPTF-IN-BZ1


    <p>BPTF-IN-BZ1 is a BPTF inhibitor that possesses a high potency with a Kd of 6.3 nM.</p>
    Formula:C13H15ClN4O
    Color and Shape:Solid
    Molecular weight:278.74
  • CDK7/12-IN-1

    CAS:
    <p>CDK7/12-IN-1 is a selective CDK7 (IC50: 3 nM) and CDK12 (IC50: 277 nM) inhibitor, effective against tumor growth.</p>
    Formula:C25H34N8O
    Color and Shape:Solid
    Molecular weight:462.59
  • KRAS G12C inhibitor 56

    CAS:
    <p>KRAS G12C inhibitor 56, a powerful inhibitor of SOS1 with an inhibitory concentration (IC50) of 1.6 nM, holds promise for use in cancer research.</p>
    Formula:C32H39N7O4S
    Color and Shape:Solid
    Molecular weight:617.76
  • GSK2578999A

    CAS:
    <p>GSK2578999A is a betulin derivative with antitumor activity.</p>
    Formula:C46H62ClNO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:776.44
  • TRβ agonist 1

    CAS:
    <p>TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.</p>
    Formula:C29H25FN2O8
    Color and Shape:Solid
    Molecular weight:548.52
  • Xeruborbactam

    CAS:
    <p>QPX7728 is an of ultra-broad-spectrum boronic acid beta-lactamase.</p>
    Formula:C10H8BFO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:221.98
  • Murizatoclax

    CAS:
    <p>AMG 397 is an oral MCL1 inhibitor .</p>
    Formula:C42H57ClN4O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:765.44
  • Balanol

    CAS:
    <p>Balanol is an ATP-competitive Protein Kinase C and Protein Kinase A inhibitor.</p>
    Formula:C28H26N2O10
    Color and Shape:Solid
    Molecular weight:550.51
  • GGTI298

    CAS:
    <p>GGTI298 is a potent GGTase I inhibitor; IC50 3μM for Rap1A, &gt;20μM for Ha-Ras.</p>
    Formula:C27H33N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:479.63
  • FGFR1 inhibitor-6


    <p>FGFR1 inhibitor-6, IC50: 16.31 nM, blocks cell cycle at pro-G1/G2/M and induces apoptosis.</p>
    Formula:C27H19N5O4S2
    Color and Shape:Solid
    Molecular weight:541.6
  • KRAS G12D inhibitor 16

    CAS:
    <p>KRAS G12D inhibitor 16 targets KRAS G12D with IC50 of 0.7 nM and mutant form at 0.35 μM, useful in various cancer studies.</p>
    Formula:C32H39IN6O3
    Color and Shape:Solid
    Molecular weight:682.59
  • Carbonic anhydrase inhibitor 9


    <p>Carbonic anhydrase inhibitor 9 targets hCA II and IX with Ki of 56.4 and 56.9 nM respectively; shows antiproliferative activity.</p>
    Formula:C22H20BrN5O4S
    Color and Shape:Solid
    Molecular weight:530.39
  • MDL-27088

    CAS:
    <p>MDL-27088 is an angiotensin-covering enzyme inhibitor.</p>
    Formula:C25H28N2O5
    Color and Shape:Solid
    Molecular weight:436.50
  • Ici D1542

    CAS:
    <p>Ici D1542: potent TXS inhibitor &amp; TXA2 receptor antagonist, effective thromboxane blocker in vitro.</p>
    Formula:C25H30N2O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:470.51
  • GSK-1264

    CAS:
    <p>GSK-1264: allosteric HIV integrase inhibitor, halts viral replication &amp; abnormal protein multimerization.</p>
    Formula:C26H28FNO5
    Color and Shape:Solid
    Molecular weight:453.5
  • Alentemol hydrobromide

    CAS:
    <p>Alentemol hydrobromide is a Dopamine agonist.</p>
    Formula:C19H26BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:364.32
  • HDAC2-IN-1


    <p>HDAC2-IN-1 is an oral HDAC2 inhibitor (IC50: 0.5 μM), crosses the blood-brain barrier, and inhibits HDAC1 and HDAC8.</p>
    Formula:C22H23ClN4OS
    Color and Shape:Solid
    Molecular weight:426.96
  • Purine phosphoribosyltransferase-IN-1


    <p>Compound (S,R)-48 inhibits Pf, Pv, &amp; Tbr PRT with Ki of 50, 20, 2 nM.</p>
    Formula:C11H15N5Na4O10P2
    Color and Shape:Solid
    Molecular weight:531.17
  • RN941

    CAS:
    <p>RN941 is a highly potent Bruton's tyrosine kinase (BTK) inhibitor.</p>
    Formula:C34H34FN7O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:639.68
  • DNDI-8219

    CAS:
    <p>DNDI-8219 is an antitubercular agent. It has potent antileishmanial effects.</p>
    Formula:C13H10F3N3O5
    Color and Shape:Solid
    Molecular weight:345.23
  • L 668750

    CAS:
    <p>L 668750 is an inhibitor of platelet-activating factor.</p>
    Formula:C25H34O9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.6
  • Acyline

    CAS:
    <p>Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.</p>
    Formula:C80H102ClN15O14
    Color and Shape:Solid
    Molecular weight:1533.21
  • PHGDH-IN-2


    <p>PHGDH-IN-2: potent PHGDH inhibitor, IC50=5.2μM; hinders PHGDH cancer cell growth &amp; serine synthesis in MDA-MB-468.</p>
    Formula:C22H20N4O3S
    Color and Shape:Solid
    Molecular weight:420.48
  • Lysyllysyllysine

    CAS:
    <p>Lysyllysyllysine is a cationic moiety. It may be used in the construction of gene delivery vectors and DNA nanoparticles.</p>
    Formula:C18H38N6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.53
  • KNT-127

    CAS:
    <p>KNT-127 is an agonist of δ-Opioid receptor.</p>
    Formula:C24H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:372.46
  • ML-SI1

    CAS:
    <p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>
    Formula:C23H26Cl2N2O3
    Color and Shape:Solid
    Molecular weight:449.37
  • (±)-HIP-B

    CAS:
    <p>(±)-HIP-B is an excitatory amino acid transporter blocker.</p>
    Formula:C6H8N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:172.14
  • GSK3368715

    CAS:
    <p>GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50s</p>
    Formula:C20H38N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:366.54
  • MRTX-EX185


    <p>MRTX-EX185 inhibits GDP-KRAS/G12D; IC50=90 nM on G12D. It also binds GDP-HRAS.</p>
    Formula:C33H33FN6O2
    Color and Shape:Solid
    Molecular weight:564.65