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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66513 products of "Inhibitors"

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  • AMG-548 dihydrochloride


    AMG-548 dihydrochloride, an oral p38α inhibitor (Ki: 0.5 nM), selectively targets p38β, γ, δ, inhibits TNFα (IC50: 3 nM), and suppresses Wnt signaling.
    Formula:C29H29Cl2N5O
    Color and Shape:Solid
    Molecular weight:534.48

    Ref: TM-T63762

    25mg
    825.00€
    50mg
    1,071.00€
    100mg
    1,755.00€
  • CS-003 Free base

    CAS:
    CS-003: Triple neurokinin receptor antagonist; Ki=2.3 nM (NK1), 0.54 nM (NK2), 0.74 nM (NK3); treats respiratory diseases.
    Formula:C34H38Cl2N2O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:673.65

    Ref: TM-T10892

    25mg
    3,078.00€
    50mg
    3,853.00€
    100mg
    5,040.00€
  • Tabimorelin hemifumarate

    CAS:
    orally active ghrelin receptor (GHS-R1a) agonist
    Formula:C32H40N403C4H404
    Purity:98%
    Color and Shape:Solid
    Molecular weight:586.72

    Ref: TM-T23413

    10mg
    1,251.00€
  • Antiallergic agent-1


    Antiallergic agent-1, an Src family kinase inhibitor, is a new and valuable lead compound with potential as an anti-allergic agent.
    Formula:C27H19F6N5O
    Color and Shape:Solid
    Molecular weight:543.46

    Ref: TM-T63825

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LY309887

    CAS:
    LY309887 is a potent inhibitor of glycinamide ribonucleotide formyltransferase (Ki: 6.5 nM). It also has antitumor activity.
    Formula:C19H23N5O6S
    Color and Shape:Solid
    Molecular weight:449.48

    Ref: TM-T15813

    25mg
    1,260.00€
    50mg
    1,639.00€
    100mg
    2,530.00€
  • PF-06372222

    CAS:
    PF-06372222: a small-molecule that modulates GCGR and antagonizes GLP-1R, affecting insulin and glucagon.
    Formula:C26H28F3N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:515.53

    Ref: TM-T24620

    25mg
    1,963.00€
    50mg
    2,710.00€
    100mg
    3,447.00€
  • Antileishmanial agent-4


    Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].
    Formula:C17H18N4O4
    Color and Shape:Solid
    Molecular weight:342.35

    Ref: TM-T61100

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Protopine hydrochloride

    CAS:
    Protopine inhibits thromboxane, lowers intracellular calcium, and reduces cell adhesion by altering adhesive factors.
    Formula:C20H20ClNO5
    Purity:98%
    Color and Shape:Prisms From Alc Solid
    Molecular weight:389.83

    Ref: TM-TMA1944

    500µg
    304.00€
    1mg
    530.00€
  • Tasidotin hydrochloride

    CAS:
    Tasidotin hydrochloride, a dolastatin 15 analog, inhibits microtubule assembly and dynamics.
    Formula:C32H59ClN6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:643.30

    Ref: TM-T16997

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • TTA-P1

    CAS:
    TTA-P1: potent T-type calcium channel inhibitor; impacts neuron firing, hormone secretion, cell growth; potential in absence epilepsy research.
    Formula:C19H27Cl2FN2O
    Color and Shape:Solid
    Molecular weight:389.33

    Ref: TM-T61747

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Lafadofensine (D-(-)-Mandelic acid)


    Lafadofensine D-(-)-Mandelic acid is a monoamines reuptake inhibitor with adequate effects when administered short-term.
    Formula:C32H32F2N2O6
    Color and Shape:Solid
    Molecular weight:578.6

    Ref: TM-T64088

    25mg
    973.00€
    50mg
    1,269.00€
    100mg
    1,998.00€
  • ONO-8809

    CAS:
    ONO-8809: Thromboxane A2 antagonist, reduces airway hyperresponse, macrophage accumulation, and MMP-9 in SHRSP brains.
    Formula:C30H46BrNO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:596.66

    Ref: TM-T28251

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • U92016A hydrochloride

    CAS:
    U92016A hydrochloride: potent, orally active 5-HT1A agonist, metabolically stable, high intrinsic activity, Ki=0.2 nM.
    Formula:C19H26ClN3
    Color and Shape:Solid
    Molecular weight:331.89

    Ref: TM-T60990

    1mg
    128.00€
  • ATM Inhibitor-3


    ATM Inhibitor-3 selectively inhibits ATM (IC50: 0.71 nM), targets PI3K kinase family, and is metabolically stable.
    Formula:C25H29FN6O3
    Color and Shape:Solid
    Molecular weight:480.53

    Ref: TM-T63171

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tyk2-IN-3

    CAS:
    Tyk2-IN-3 is an inhibitor of Tyk2 pseudokinase (IC50: 485 nM).
    Formula:C25H24N6O3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:520.63

    Ref: TM-T13233

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • AMG-25

    CAS:
    AMG-25 (c-Kit-IN-5-1) is a c-Kit inhibitor that inhibits c-Kit, KDR, p38, Lck, and Src, and can be used for the study of mast cell-associated fibrotic diseases.
    Formula:C23H17N5O2
    Purity:98.16%
    Color and Shape:Solid
    Molecular weight:395.41

    Ref: TM-T22256

    2mg
    449.00€
  • CCG258208

    CAS:
    GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).
    Formula:C24H25FN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:452.48

    Ref: TM-T13714

    25mg
    2,313.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • Carmegliptin dihydrochloride

    CAS:
    Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.
    Formula:C20H30Cl2FN3O3
    Color and Shape:Solid
    Molecular weight:450.38

    Ref: TM-T68652

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • 4'-Ethynyl-2'-deoxyadenosine

    CAS:
    4'-E-dA is a potent nucleoside RT inhibitor for drug-resistant HIV (EC50: 98 nM in MT-4 cells).
    Formula:C12H13N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:275.26

    Ref: TM-T10141

    25mg
    2,268.00€
    50mg
    2,772.00€
    100mg
    3,420.00€
  • ATM Inhibitor-1

    CAS:
    ATM Inhibitor-1 is a highly potent, selective and orally active ATM inhibito (IC50: 0.7 nM) anti-tumor activity.
    Formula:C27H36N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:492.61

    Ref: TM-T10396

    25mg
    2,808.00€
    50mg
    3,492.00€
    100mg
    4,500.00€
  • S-8510 phosphate

    CAS:
    S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).
    Formula:C12H13N4O6P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:340.23

    Ref: TM-T12792

    25mg
    2,583.00€
    50mg
    3,402.00€
    100mg
    4,680.00€
  • Topoisomerase I/II inhibitor 4


    Topoisomerase I/II inhibitor 4 halts cell growth and spread, induces apoptosis, and is used in liver cancer research.
    Formula:C27H21N5O6
    Color and Shape:Solid
    Molecular weight:511.49

    Ref: TM-T63526

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BRD-K98645985

    CAS:
    BRD-K98645985: BAF inhibitor, binds ARID1A, reverses HIV-1 latency, EC50 ~2.37μM, alters nucleosome placement.
    Formula:C33H43N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:573.73

    Ref: TM-T10605

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • KT2-962

    CAS:
    KT2-962 is a TXA2/prostaglandin endoperoxide receptor antagonist.
    Formula:C23H27ClNNaO5S2
    Color and Shape:Solid
    Molecular weight:520.04

    Ref: TM-T71035

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • Nedocromil sodium

    CAS:
    Nedocromil sodium is a pharmacologic stabilizer of mast cells, has been shown to normalize cytokine levels and attenuate cardiac remodeling.
    Formula:C19H17NNaO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:394.335

    Ref: TM-T19472

    5mg
    148.00€
    10mg
    268.00€
    25mg
    617.00€
    50mg
    1,018.00€
  • Antitumor agent-42


    Antitumor agent-42 inhibits microtubule multimerisation and NO release, exhibiting anti-angiogenic, colony-forming and apoptosis-inducing effects.
    Formula:C24H19BrN2O8S
    Color and Shape:Solid
    Molecular weight:575.39

    Ref: TM-T64071

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Longicoricin

    CAS:
    Longicoricin is a monotetrahydrofuran Annonaceous acetogenin from Asimina longifolia.
    Formula:C37H68O6
    Color and Shape:Solid
    Molecular weight:608.93

    Ref: TM-T32863

    25mg
    2,313.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • Coleon-U-quinone

    CAS:
    Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.
    Formula:C20H24O5
    Color and Shape:Solid
    Molecular weight:344.4

    Ref: TM-T72735

    25mg
    2,313.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • Rpi 856 C

    CAS:
    Rpi 856 C is a retrovirus protease inhibitor from Streptomyces that is effective against HIV-1 and HTLV-1 proteases.
    Formula:C39H56N6O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:768.90

    Ref: TM-T26128

    25mg
    To inquire
    50mg
    To inquire
    100mg
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  • Piperazinomycin

    CAS:

    Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.

    Formula:C18H20N2O2
    Color and Shape:Solid
    Molecular weight:296.36

    Ref: TM-T68604

    25mg
    5,391.00€
    50mg
    7,082.00€
    100mg
    9,505.00€
  • Bomedemstat hydrochloride


    Bomedemstat (IMG-7289) hydrochloride, an oral LSD1 inhibitor, has anticancer properties, blocking cell growth and triggering apoptosis.
    Formula:C28H35ClFN7O2
    Color and Shape:Solid
    Molecular weight:556.08

    Ref: TM-T63935

    25mg
    6,083.00€
    50mg
    7,892.00€
  • 13(R)-HODE

    CAS:
    13(R)-HODE, produced from linoleic acid, inhibits platelet aggregation (IC50=2.7μM) and is found in bovine endothelial cells.
    Formula:C18H32O3
    Color and Shape:Solid
    Molecular weight:296.44

    Ref: TM-T37973

    25µg
    273.00€
    50µg
    472.00€
    100µg
    818.00€
    250µg
    1,863.00€
  • BTK-IN-15


    BTK-IN-15: Oral BTK inhibitor, IC50 0.7 nM, induces cancer cell apoptosis, selective with anti-tumor effects.
    Formula:C28H24FN5O2
    Color and Shape:Solid
    Molecular weight:481.52

    Ref: TM-T63182

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ambelline

    CAS:
    Ambelline has antitumor activity.
    Formula:C18H21NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.36

    Ref: TM-T25075

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Epolactaene

    CAS:
    Epolactaene: neuritogenic, inhibits mammalian DNA polymerases & human DNA topoisomerase II.
    Formula:C21H27NO6
    Color and Shape:Solid
    Molecular weight:389.44

    Ref: TM-T70284

    25mg
    2,718.00€
    50mg
    3,582.00€
    100mg
    4,950.00€
  • Artemisiane E

    CAS:
    Artemisiane E is a potent PI3K/AKT pathway inhibitor with an IC 50 of 8.9 μM .
    Formula:C20H22O5
    Color and Shape:Solid
    Molecular weight:342.39

    Ref: TM-T72903

    25mg
    3,529.00€
    50mg
    4,663.00€
    100mg
    6,570.00€
  • ATM Inhibitor-2


    ATM Inhibitor -2 is a potent and selective inhibitor of ATM (IC50<1 nM).
    Formula:C26H31N7O3
    Color and Shape:Solid
    Molecular weight:489.57

    Ref: TM-T63279

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PDE4-IN-6


    PDE4-IN-6: Potent PDE4 inhibitor, IC50 - 0.125μM (B), 0.43μM (D), anti-inflammatory, for arthritis research.
    Formula:C25H20FNO5S
    Color and Shape:Solid
    Molecular weight:465.49

    Ref: TM-T62969

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Pamiparib maleate

    CAS:
    Pamiparib (BGB-290) is a selective PARP inhibitor that blocks DNA repair and promotes apoptosis.
    Formula:C44H42F2N8O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:944.859

    Ref: TM-T28293

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • GSK579289A

    CAS:
    GSK579289A is an inhibitor of benzimidazole thiophene.
    Formula:C26H27ClN4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:511.04

    Ref: TM-T27484

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • 8-Deazafolic acid

    CAS:
    8-Deazafolic acid inhibits folate-dependent bacteria S. faecium & L. casei, and fights lymphoid leukemia L1210 in mice.
    Formula:C20H20N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.41

    Ref: TM-T24990

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • TRPC4/5-IN-1


    TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.
    Formula:C21H21N3O
    Color and Shape:Solid
    Molecular weight:331.41

    Ref: TM-T60981

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cortistatin A

    CAS:
    Cortistatin A is a potent and selective mediator-associated kinase CDK8 and its paralogue CDK19 inhibitor.
    Formula:C30H36N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.62

    Ref: TM-T23909

    25mg
    To inquire
    50mg
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    100mg
    To inquire
  • 6-trans-12-epi-Leukotriene B4

    CAS:
    6-trans-12-epi-Leukotriene B4, a metabolite of arachidonic acid, serves as a potent anti-inflammatory agent.
    Formula:C20H32O4
    Color and Shape:Solid
    Molecular weight:336.47

    Ref: TM-T72144

    25µg
    273.00€
    50µg
    467.00€
    100µg
    872.00€
  • TNP-470

    CAS:
    TNP-470 is a methionine aminopeptidase-2 inhibitor. TNP-470 is also an angiogenesis inhibitor.
    Formula:C19H28ClNO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.88

    Ref: TM-T17110

    5mg
    298.00€
    10mg
    565.00€
    25mg
    1,288.00€
  • Antitubercular agent-23


    Antitubercular agent-23 combats Candida albicans (MIC: 1.1 μg/ml) and M. tuberculosis (MIC: 1 μg/ml).
    Formula:C20H22FN5O8S
    Color and Shape:Solid
    Molecular weight:511.48

    Ref: TM-T63525

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Mal-PEG4-VA-PBD

    CAS:
    Mal-PEG4-VA-PBD is a drug-linker conjugate for Antibody-Drug Conjugates (ADCs), comprising the antitumor antibiotic Pyrrolobenzodiazepine (PBD), connected
    Formula:C68H79N9O17
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1294.41

    Ref: TM-T18289

    1mg
    795.00€
    5mg
    2,242.00€
    10mg
    3,025.00€
    25mg
    4,491.00€
    50mg
    6,058.00€
    100mg
    8,190.00€
  • SID 26681509 quarterhydrate


    SID 26681509 is a selective inhibitor of cathepsin L (IC50: 56 nM) and blocks Plasmodium falciparum (IC50: 15.4 μM) and Leishmania major (IC50: 12.5 μM).
    Formula:C27H35N5O6S
    Color and Shape:Solid
    Molecular weight:544.16

    Ref: TM-T63831

    25mg
    1,359.00€
    50mg
    1,770.00€
    100mg
    2,657.00€
  • ChE/Aβ1-42-IN-1


    ChE/Aβ1-42-IN-1 (compound 28) is a potent aggregation inhibitor of ChE and Aβ 1-42 with excellent BBB permeability.
    Formula:C19H24N2O3
    Color and Shape:Solid
    Molecular weight:328.41

    Ref: TM-T60940

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MtTMPK-IN-2

    CAS:
    MtTMPK-IN-2 inhibits M. tuberculosis TMPK (IC50: 1.1 μM), Mtb H37Rv (MIC: 12.5 μM), and is cytotoxic in MRC-5 cells (EC50: 6.1 μM).
    Formula:C23H24ClN3O3
    Color and Shape:Solid
    Molecular weight:425.91

    Ref: TM-T62305

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SHR902275

    CAS:
    SHR902275: potent RAF inhibitor, hits RAS mutations, oral use. cRAF IC50=1.6 nM, bRAFwt IC50=10 nM, bRAFV600E IC50=5.7 nM, hinders cell growth.
    Formula:C26H23F3N4O4
    Color and Shape:Solid
    Molecular weight:512.48

    Ref: TM-T63542

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LH secretion antagonist 1

    CAS:
    LH secretion antagonist 1 is an antagonist of luteinizing hormone secretion with analgesic activity.
    Formula:C18H24ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.84

    Ref: TM-T10064

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • RS 2135

    CAS:
    RS 2135 is a novel class I antiarrhythmic agent to inhibit ischemia-induced ventricular arrhythmias.
    Formula:C18H21ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.83

    Ref: TM-T26136

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Retelliptine

    CAS:
    Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.
    Formula:C25H32N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:404.55

    Ref: TM-T28521

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • TGR5 Receptor Agonist 3

    CAS:
    TGR5 Receptor Agonist 3 is a GPBAR1 agonist with EC50 of 16.4 nM (hTGR5) & 209 nM (mTGR5), ensures gallbladder safety and reduces filling.
    Formula:C29H27N3O6
    Color and Shape:Solid
    Molecular weight:513.54

    Ref: TM-T63554

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • EED ligand 1


    EED ligand 1: potent PRC2 inhibitor targeting EED subunit.
    Formula:C19H19FN8O
    Color and Shape:Solid
    Molecular weight:394.41

    Ref: TM-T61825

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ZLHQ-5f


    ZLHQ-5f inhibits CDK2/Topo I, with IC50 of 0.145μM for CDK2/CycA2, and promotes apoptosis by arresting HCT116 cells in S phase.
    Formula:C28H25N5O2
    Color and Shape:Solid
    Molecular weight:463.53

    Ref: TM-T62934

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MsbA-IN-2


    MsbA-IN-2 is a potent inhibitor of the lipopolysaccharide transporter MsbA and is able to act on E. coli MsbA (IC50: 2 nM).
    Formula:C23H19Cl2NO3
    Color and Shape:Solid
    Molecular weight:428.31

    Ref: TM-T62339

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • IRE1α kinase-IN-4

    CAS:
    IRE1α kinase-IN-4 (compound 6) is a potent inhibitor of IRE1α, exhibiting a Ki value of 140 nM. It acts as an ATP-competitive ligand for IRE1α [1].
    Formula:C29H31N7O2
    Color and Shape:Solid
    Molecular weight:509.6

    Ref: TM-T63511

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ATM Inhibitor-4


    ATM Inhibitor -4: selective, potent (IC50: 0.32 nM), inhibits PI3K family, stable, stops mTOR at 1 μM.
    Formula:C26H29FN6O3
    Color and Shape:Solid
    Molecular weight:492.55

    Ref: TM-T63317

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LSD1-IN-13 hydrochloride

    CAS:
    LSD1-IN-13 hydrochloride (7e) is an oral LSD1 inhibitor (IC50: 24.43 nM), promoting differentiation in AML cell lines.
    Formula:C23H30ClN3O2S
    Color and Shape:Solid
    Molecular weight:448.02

    Ref: TM-T62679

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • ITK inhibitor 6

    CAS:
    ITK inhibitor 6 selectively targets ITK, BTK, JAK3, EGFR, LCK, blocks PLCγ1 and ERK1/2 phosphorylation, and inhibits cell proliferation.
    Formula:C28H24F2N4O2
    Color and Shape:Solid
    Molecular weight:486.51

    Ref: TM-T63229

    100mg
    To inquire
    25mg
    6,418.00€
    50mg
    10,350.00€
  • Antibacterial agent 80


    Antibacterial agent 80 (compound 20) has antibacterial activity [1].
    Formula:C14H21N3S2
    Color and Shape:Solid
    Molecular weight:295.47

    Ref: TM-T60634

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SM-433 hydrochloride


    SM-433 hydrochloride, a Smac mimetic & IAP inhibitor, binds XIAP BIR3; potent IC50 <1 μM. (Patent WO2008128171A2)
    Formula:C32H44ClN5O4
    Color and Shape:Solid
    Molecular weight:598.18

    Ref: TM-T64217

    25mg
    1,414.00€
    50mg
    2,277.00€
  • TMX-4113


    TMX-4113 has potential to be used in cancer that is a phosphodiesterase 6D(PDE6D) and casein kinase 1α(CK1α) degrader [1].
    Formula:C12H12N4O2S2
    Color and Shape:Solid
    Molecular weight:308.38

    Ref: TM-T60740

    25mg
    1,260.00€
    50mg
    1,639.00€
    100mg
    2,538.00€
  • Antimalarial agent 9


    Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.
    Formula:C28H32BrN3O2
    Color and Shape:Solid
    Molecular weight:522.48

    Ref: TM-T63655

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AGN-204396

    CAS:
    AGN-204396 is an antagonist that selectively blocks the activity of prostamides (prostaglandin-ethanolamides).
    Formula:C32H44FN3O4
    Color and Shape:Solid
    Molecular weight:553.71

    Ref: TM-T68576

    25mg
    2,718.00€
    50mg
    3,582.00€
    100mg
    4,950.00€
  • KRAS G12C inhibitor 37

    CAS:
    KRAS G12C inhibitor 37 targets a key signaling protein, showing promise for cancer research involving KRAS G12C.
    Formula:C35H39F3N8O2
    Color and Shape:Solid
    Molecular weight:660.73

    Ref: TM-T72340

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • Antitumor agent-54


    Compound C11 inhibits 14-3-3η protein (KD: 35 μM), targets liver cancer cells, blocks G1-S phase, and induces apoptosis.
    Formula:C29H32N2O3
    Color and Shape:Solid
    Molecular weight:456.58

    Ref: TM-T62835

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • KFA1982

    CAS:
    KFA1982 is a novel and potent factor Xa inhibitor.
    Formula:C28H34ClN3O9S2
    Color and Shape:Solid
    Molecular weight:656.17

    Ref: TM-T69276

    25mg
    2,853.00€
    50mg
    3,763.00€
    100mg
    5,220.00€
  • RSK4-IN-1

    CAS:
    RSK4-IN-1 is a compound exhibiting potent inhibition of RSK4, demonstrated by an IC50 value of 9.5 nM.
    Formula:C19H20F2N4O3
    Color and Shape:Solid
    Molecular weight:390.38

    Ref: TM-T61766

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MB725

    CAS:
    MB725 is a strong and selective inducer of viability reduction in several cancer cell lines containing the oncogenic p53-Y220C mutation.
    Formula:C18H21IN4O2S
    Color and Shape:Solid
    Molecular weight:484.35

    Ref: TM-T33219

    25mg
    2,718.00€
    50mg
    3,582.00€
    100mg
    4,950.00€
  • RXR antagonist 1


    RXR antagonist 1 is a Retinoid X Receptor (RXR) modulator that exhibits high RXR antagonism (pA2: 8.06). RXR antagonist 1 can be used to study type 2 diabetes.
    Formula:C28H33F3N2O3
    Color and Shape:Solid
    Molecular weight:502.57

    Ref: TM-T63415

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Antifungal agent 39

    CAS:
    Antifungal agent 39 (Compound 9h) is a broad-spectrum antifungal agent.
    Formula:C23H22ClN3O5
    Color and Shape:Solid
    Molecular weight:455.89

    Ref: TM-T62823

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GW311616 hydrochloride

    CAS:
    GW-311616 hydrochloride is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).
    Formula:C19H32ClN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.99

    Ref: TM-T11525L

    1mg
    273.00€
    5mg
    818.00€
    10mg
    1,359.00€
  • CDK5-IN-2

    CAS:
    CDK5-IN-2 (compound 15) is a highly selective CDK5 inhibitor that acts on CDK5/p25 (IC50: 0.2 nM) and CDK2/CycA (IC50: 23 nM).
    Formula:C29H28FN5O
    Color and Shape:Solid
    Molecular weight:481.56

    Ref: TM-T63184

    25mg
    3,492.00€
    50mg
    5,239.00€
    100mg
    7,857.00€
  • PF-00489791

    CAS:
    PF-00489791 (PF4634817) is a long-acting PDE5 inhibitor with hypotensive activity for the study of diabetic nephropathy.
    Formula:C20H28N8O4S
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:476.55

    Ref: TM-T28360

    1mg
    34.00€
    5mg
    62.00€
    10mg
    100.00€
    25mg
    268.00€
  • DMP-728 free base

    CAS:
    DMP-728 free base is a highly potent and selective GPIIbDIIa antagonist
    Formula:C25H36N8O7
    Color and Shape:Solid
    Molecular weight:560.60

    Ref: TM-T70482

    25mg
    2,853.00€
    50mg
    3,763.00€
    100mg
    5,220.00€
  • Menin-MLL inhibitor 4

    CAS:
    Menin-MLL inhibitor 4 has antitumor activity.Menin-MLL inhibitor 4 is an inhibitor of Menin- MLL (mixed-lineage leukemia protein) interaction .
    Formula:C32H38FN7O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:587.69

    Ref: TM-T12002

    25mg
    2,853.00€
    50mg
    3,763.00€
    100mg
    5,220.00€
  • BRD-K25923209

    CAS:
    BRD-K25923209 is a novel inhibitor of BAF transcriptional repression.
    Formula:C29H36N4O3
    Color and Shape:Solid
    Molecular weight:488.62

    Ref: TM-T69692

    25mg
    2,853.00€
    50mg
    3,763.00€
    100mg
    5,220.00€
  • JAK3-IN-11

    CAS:
    JAK3-IN-11: potent oral JAK3 inhibitor (IC50=1.7 nM), noncytotoxic, >588-fold selectivity, blocks T-cell growth; useful in autoimmune research.
    Formula:C23H23N5O2
    Color and Shape:Solid
    Molecular weight:401.46

    Ref: TM-T9811

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MrgprX2 antagonist-6


    MrgprX2 antagonist-6 is a potent antiallergic agent with inhibitory effects on mast cell degranulation.
    Formula:C24H23F3N6O3
    Color and Shape:Solid
    Molecular weight:500.47

    Ref: TM-T63394

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Antiviral agent 7


    Antiviral agent 7 is a peptide-based coating that kills viruses.
    Formula:C29H31F2N3O6
    Color and Shape:Solid
    Molecular weight:555.57

    Ref: TM-T63921

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Nonsteroidal aromatase inhibitor 1


    Compound 13h, a nonsteroidal aromatase inhibitor, has a potent IC50 of 0.09 nM against CYP19A1, showing promise for breast cancer research.
    Formula:C22H16N4O2
    Color and Shape:Solid
    Molecular weight:368.39

    Ref: TM-T61444

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JBIR-22

    CAS:
    JBIR-22 is a natural inhibitor for protein−protein interaction of the homodimer of proteasome assembly factor 3.
    Formula:C23H33NO6
    Color and Shape:Solid
    Molecular weight:419.51

    Ref: TM-T71203

    25mg
    2,448.00€
    50mg
    3,222.00€
    100mg
    4,410.00€
  • KDOAM-25 trihydrochloride (2230731-99-2 free base)


    KDOAM-25 trihydrochloride, a selective KDM5 inhibitor (IC50: 19-71 nM), boosts H3K4 methylation and hinders MM1S cell growth.
    Formula:C15H28Cl3N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:416.77

    Ref: TM-T11750L

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • A1/A3 AR antagonist 1


    Compound 10 is a potent dual A1/A3 AR antagonist, with Ki values of 37.6 nM (hA1), 25.4 nM (hA3), and 1.47 nM (rA1), studied in renal, lung, and Alzheimer's.
    Formula:C24H18N2O3S
    Color and Shape:Solid
    Molecular weight:414.48

    Ref: TM-T62134

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • EGFR-IN-58


    EGFR-IN-58 is a potent, selective, ATP-competitive inhibitor of EGFR. EGFR-IN-58 exhibits significant cytotoxicity against melanoma, colon and blood cancers.
    Formula:C31H30FN7O
    Color and Shape:Solid
    Molecular weight:535.61

    Ref: TM-T63774

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TIY-7


    TIY-7 is a selective, orally active inhibitor of the promyosin receptor kinase (TRK) enzyme. TIY-7 exhibited anti-tumour effects in a mouse xenograft model.
    Color and Shape:Solid

    Ref: TM-T64296

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MAO A/HDAC-IN-1


    MAO A/HDAC-IN-1 is an effective monoamine oxidase A (MAO A) and HDAC dual inhibitor, which can be used for glioma research.
    Formula:C21H24ClN3O3
    Color and Shape:Solid
    Molecular weight:401.89

    Ref: TM-T61958

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MALT1-IN-5

    CAS:
    MALT1-IN-5 is a potent inhibitor of the MALT1 protease and can be used in cancer research.
    Formula:C17H17ClF2N6O3
    Color and Shape:Solid
    Molecular weight:426.80

    Ref: TM-T62323

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • AMG-315

    CAS:
    AMG-315: Chiral AEA analogue, potent CB1 agonist (Ki 7.8 nM, EC50 0.6 nM), stable against hydrolyzing/oxidative enzymes.
    Formula:C24H41NO2
    Color and Shape:Solid
    Molecular weight:375.59

    Ref: TM-T69740

    25mg
    2,718.00€
    50mg
    3,582.00€
    100mg
    4,950.00€
  • CLK1/2-IN-1

    CAS:
    CLK1/2-IN-1 is a CLK1 and CLK2 inhibitor and it also inhibits SRPK1 and SRPK2.
    Formula:C21H20F3N7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:443.42

    Ref: TM-T23896

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Furaprevir

    CAS:
    Furaprevir is an HCV NS3/4A Inhibitor
    Formula:C47H56N6O10S
    Color and Shape:Solid
    Molecular weight:897.05

    Ref: TM-T70655

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • CDK9-IN-13


    CDK9-IN-13 is a potent and selective CDK inhibitor (IC50<3 nM). CDK9-IN-13 has a very short half-life in rodents.
    Formula:C27H35N5O2
    Color and Shape:Solid
    Molecular weight:461.6

    Ref: TM-T62919

    25mg
    1,108.00€
    50mg
    1,449.00€
    100mg
    2,385.00€
  • Monlunabant

    CAS:
    Monlunabant ((S)-MRI-1891), a solid dispersion compound, functions as an inhibitor of the cannabinoid CB1 receptor [1].
    Formula:C26H22ClF3N6O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:591.00

    Ref: TM-T79137

    5mg
    131.00€
    10mg
    197.00€
    25mg
    393.00€
    50mg
    595.00€
  • Vimirogant

    CAS:
    Vimirogant is a RORγ inhibitor (Ki: <100 nM).
    Formula:C27H35F3N4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:552.65

    Ref: TM-T16787

    25mg
    4,185.00€
    50mg
    5,494.00€
    100mg
    7,375.00€
  • TAK-024

    CAS:
    TAK-024 is an inhibitor of platelet(IC50s of 31, 79 and 51 nM in human, monkey and guinea pig, respectively).
    Formula:C27H34N10O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:594.62

    Ref: TM-T13065

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • EGFR/HER2-IN-7


    EGFR/HER2-IN-7: Potent, selective dual inhibitor for MCF-7 cancer; IC50: EGFR 0.18μM, HER2 0.146μM, DHFR 0.907μM.
    Formula:C19H21N3O2S
    Color and Shape:Solid
    Molecular weight:355.45

    Ref: TM-T61272

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AT-IAP

    CAS:
    AT-IAP is an effective dual antagonist of XIAP and cIAP1.
    Formula:C29H40FN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:509.66

    Ref: TM-T23760

    100mg
    To inquire
    10mg
    4,050.00€
    25mg
    6,238.00€
    50mg
    9,360.00€