Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,846 products)
- Apoptosis(6,332 products)
- Cell Cycle/Checkpoint(4,887 products)
- Chromatin/Epigenetics(2,615 products)
- Cytoskeletal Signaling(1,577 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,753 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,025 products)
- Immunology and Inflammation(3,926 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,258 products)
- Membrane Transporter/Ion Channel(3,160 products)
- Metabolism(10,133 products)
- Microbiology/Virology(7,625 products)
- Neuroscience(10,540 products)
- Other Inhibitors(35,857 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(731 products)
- Tyrosine Kinase/Adaptors(1,991 products)
- Ubiquitination(1,727 products)
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Found 66513 products of "Inhibitors"
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AMG-548 dihydrochloride
AMG-548 dihydrochloride, an oral p38α inhibitor (Ki: 0.5 nM), selectively targets p38β, γ, δ, inhibits TNFα (IC50: 3 nM), and suppresses Wnt signaling.Formula:C29H29Cl2N5OColor and Shape:SolidMolecular weight:534.48CS-003 Free base
CAS:CS-003: Triple neurokinin receptor antagonist; Ki=2.3 nM (NK1), 0.54 nM (NK2), 0.74 nM (NK3); treats respiratory diseases.Formula:C34H38Cl2N2O6SPurity:98%Color and Shape:SolidMolecular weight:673.65Tabimorelin hemifumarate
CAS:orally active ghrelin receptor (GHS-R1a) agonistFormula:C32H40N403C4H404Purity:98%Color and Shape:SolidMolecular weight:586.72Antiallergic agent-1
Antiallergic agent-1, an Src family kinase inhibitor, is a new and valuable lead compound with potential as an anti-allergic agent.Formula:C27H19F6N5OColor and Shape:SolidMolecular weight:543.46LY309887
CAS:LY309887 is a potent inhibitor of glycinamide ribonucleotide formyltransferase (Ki: 6.5 nM). It also has antitumor activity.Formula:C19H23N5O6SColor and Shape:SolidMolecular weight:449.48PF-06372222
CAS:PF-06372222: a small-molecule that modulates GCGR and antagonizes GLP-1R, affecting insulin and glucagon.Formula:C26H28F3N5O3Purity:98%Color and Shape:SolidMolecular weight:515.53Antileishmanial agent-4
Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].Formula:C17H18N4O4Color and Shape:SolidMolecular weight:342.35Protopine hydrochloride
CAS:Protopine inhibits thromboxane, lowers intracellular calcium, and reduces cell adhesion by altering adhesive factors.Formula:C20H20ClNO5Purity:98%Color and Shape:Prisms From Alc SolidMolecular weight:389.83Tasidotin hydrochloride
CAS:Tasidotin hydrochloride, a dolastatin 15 analog, inhibits microtubule assembly and dynamics.Formula:C32H59ClN6O5Purity:98%Color and Shape:SolidMolecular weight:643.30TTA-P1
CAS:TTA-P1: potent T-type calcium channel inhibitor; impacts neuron firing, hormone secretion, cell growth; potential in absence epilepsy research.Formula:C19H27Cl2FN2OColor and Shape:SolidMolecular weight:389.33Lafadofensine (D-(-)-Mandelic acid)
Lafadofensine D-(-)-Mandelic acid is a monoamines reuptake inhibitor with adequate effects when administered short-term.Formula:C32H32F2N2O6Color and Shape:SolidMolecular weight:578.6ONO-8809
CAS:ONO-8809: Thromboxane A2 antagonist, reduces airway hyperresponse, macrophage accumulation, and MMP-9 in SHRSP brains.Formula:C30H46BrNO4SPurity:98%Color and Shape:SolidMolecular weight:596.66U92016A hydrochloride
CAS:U92016A hydrochloride: potent, orally active 5-HT1A agonist, metabolically stable, high intrinsic activity, Ki=0.2 nM.Formula:C19H26ClN3Color and Shape:SolidMolecular weight:331.89ATM Inhibitor-3
ATM Inhibitor-3 selectively inhibits ATM (IC50: 0.71 nM), targets PI3K kinase family, and is metabolically stable.Formula:C25H29FN6O3Color and Shape:SolidMolecular weight:480.53Tyk2-IN-3
CAS:Tyk2-IN-3 is an inhibitor of Tyk2 pseudokinase (IC50: 485 nM).Formula:C25H24N6O3S2Purity:98%Color and Shape:SolidMolecular weight:520.63AMG-25
CAS:AMG-25 (c-Kit-IN-5-1) is a c-Kit inhibitor that inhibits c-Kit, KDR, p38, Lck, and Src, and can be used for the study of mast cell-associated fibrotic diseases.Formula:C23H17N5O2Purity:98.16%Color and Shape:SolidMolecular weight:395.41CCG258208
CAS:GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).Formula:C24H25FN4O4Purity:98%Color and Shape:SolidMolecular weight:452.48Carmegliptin dihydrochloride
CAS:Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.Formula:C20H30Cl2FN3O3Color and Shape:SolidMolecular weight:450.384'-Ethynyl-2'-deoxyadenosine
CAS:4'-E-dA is a potent nucleoside RT inhibitor for drug-resistant HIV (EC50: 98 nM in MT-4 cells).Formula:C12H13N5O3Purity:98%Color and Shape:SolidMolecular weight:275.26ATM Inhibitor-1
CAS:ATM Inhibitor-1 is a highly potent, selective and orally active ATM inhibito (IC50: 0.7 nM) anti-tumor activity.Formula:C27H36N6O3Purity:98%Color and Shape:SolidMolecular weight:492.61S-8510 phosphate
CAS:S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).Formula:C12H13N4O6PPurity:98%Color and Shape:SolidMolecular weight:340.23Topoisomerase I/II inhibitor 4
Topoisomerase I/II inhibitor 4 halts cell growth and spread, induces apoptosis, and is used in liver cancer research.Formula:C27H21N5O6Color and Shape:SolidMolecular weight:511.49BRD-K98645985
CAS:BRD-K98645985: BAF inhibitor, binds ARID1A, reverses HIV-1 latency, EC50 ~2.37μM, alters nucleosome placement.Formula:C33H43N5O4Purity:98%Color and Shape:SolidMolecular weight:573.73KT2-962
CAS:KT2-962 is a TXA2/prostaglandin endoperoxide receptor antagonist.Formula:C23H27ClNNaO5S2Color and Shape:SolidMolecular weight:520.04Nedocromil sodium
CAS:Nedocromil sodium is a pharmacologic stabilizer of mast cells, has been shown to normalize cytokine levels and attenuate cardiac remodeling.Formula:C19H17NNaO7Purity:98%Color and Shape:SolidMolecular weight:394.335Antitumor agent-42
Antitumor agent-42 inhibits microtubule multimerisation and NO release, exhibiting anti-angiogenic, colony-forming and apoptosis-inducing effects.Formula:C24H19BrN2O8SColor and Shape:SolidMolecular weight:575.39Longicoricin
CAS:Longicoricin is a monotetrahydrofuran Annonaceous acetogenin from Asimina longifolia.Formula:C37H68O6Color and Shape:SolidMolecular weight:608.93Coleon-U-quinone
CAS:Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.Formula:C20H24O5Color and Shape:SolidMolecular weight:344.4Rpi 856 C
CAS:Rpi 856 C is a retrovirus protease inhibitor from Streptomyces that is effective against HIV-1 and HTLV-1 proteases.Formula:C39H56N6O10Purity:98%Color and Shape:SolidMolecular weight:768.90Piperazinomycin
CAS:Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.
Formula:C18H20N2O2Color and Shape:SolidMolecular weight:296.36Bomedemstat hydrochloride
Bomedemstat (IMG-7289) hydrochloride, an oral LSD1 inhibitor, has anticancer properties, blocking cell growth and triggering apoptosis.Formula:C28H35ClFN7O2Color and Shape:SolidMolecular weight:556.0813(R)-HODE
CAS:13(R)-HODE, produced from linoleic acid, inhibits platelet aggregation (IC50=2.7μM) and is found in bovine endothelial cells.Formula:C18H32O3Color and Shape:SolidMolecular weight:296.44BTK-IN-15
BTK-IN-15: Oral BTK inhibitor, IC50 0.7 nM, induces cancer cell apoptosis, selective with anti-tumor effects.Formula:C28H24FN5O2Color and Shape:SolidMolecular weight:481.52Ambelline
CAS:Ambelline has antitumor activity.Formula:C18H21NO5Purity:98%Color and Shape:SolidMolecular weight:331.36Epolactaene
CAS:Epolactaene: neuritogenic, inhibits mammalian DNA polymerases & human DNA topoisomerase II.Formula:C21H27NO6Color and Shape:SolidMolecular weight:389.44Artemisiane E
CAS:Artemisiane E is a potent PI3K/AKT pathway inhibitor with an IC 50 of 8.9 μM .Formula:C20H22O5Color and Shape:SolidMolecular weight:342.39ATM Inhibitor-2
ATM Inhibitor -2 is a potent and selective inhibitor of ATM (IC50<1 nM).Formula:C26H31N7O3Color and Shape:SolidMolecular weight:489.57PDE4-IN-6
PDE4-IN-6: Potent PDE4 inhibitor, IC50 - 0.125μM (B), 0.43μM (D), anti-inflammatory, for arthritis research.Formula:C25H20FNO5SColor and Shape:SolidMolecular weight:465.49Pamiparib maleate
CAS:Pamiparib (BGB-290) is a selective PARP inhibitor that blocks DNA repair and promotes apoptosis.Formula:C44H42F2N8O14Purity:98%Color and Shape:SolidMolecular weight:944.859GSK579289A
CAS:GSK579289A is an inhibitor of benzimidazole thiophene.Formula:C26H27ClN4O3SPurity:98%Color and Shape:SolidMolecular weight:511.048-Deazafolic acid
CAS:8-Deazafolic acid inhibits folate-dependent bacteria S. faecium & L. casei, and fights lymphoid leukemia L1210 in mice.Formula:C20H20N6O6Purity:98%Color and Shape:SolidMolecular weight:440.41TRPC4/5-IN-1
TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.Formula:C21H21N3OColor and Shape:SolidMolecular weight:331.41Cortistatin A
CAS:Cortistatin A is a potent and selective mediator-associated kinase CDK8 and its paralogue CDK19 inhibitor.Formula:C30H36N2O3Purity:98%Color and Shape:SolidMolecular weight:472.626-trans-12-epi-Leukotriene B4
CAS:6-trans-12-epi-Leukotriene B4, a metabolite of arachidonic acid, serves as a potent anti-inflammatory agent.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47TNP-470
CAS:TNP-470 is a methionine aminopeptidase-2 inhibitor. TNP-470 is also an angiogenesis inhibitor.Formula:C19H28ClNO6Purity:98%Color and Shape:SolidMolecular weight:401.88Antitubercular agent-23
Antitubercular agent-23 combats Candida albicans (MIC: 1.1 μg/ml) and M. tuberculosis (MIC: 1 μg/ml).Formula:C20H22FN5O8SColor and Shape:SolidMolecular weight:511.48Mal-PEG4-VA-PBD
CAS:Mal-PEG4-VA-PBD is a drug-linker conjugate for Antibody-Drug Conjugates (ADCs), comprising the antitumor antibiotic Pyrrolobenzodiazepine (PBD), connectedFormula:C68H79N9O17Purity:98%Color and Shape:SolidMolecular weight:1294.41SID 26681509 quarterhydrate
SID 26681509 is a selective inhibitor of cathepsin L (IC50: 56 nM) and blocks Plasmodium falciparum (IC50: 15.4 μM) and Leishmania major (IC50: 12.5 μM).Formula:C27H35N5O6SColor and Shape:SolidMolecular weight:544.16ChE/Aβ1-42-IN-1
ChE/Aβ1-42-IN-1 (compound 28) is a potent aggregation inhibitor of ChE and Aβ 1-42 with excellent BBB permeability.Formula:C19H24N2O3Color and Shape:SolidMolecular weight:328.41MtTMPK-IN-2
CAS:MtTMPK-IN-2 inhibits M. tuberculosis TMPK (IC50: 1.1 μM), Mtb H37Rv (MIC: 12.5 μM), and is cytotoxic in MRC-5 cells (EC50: 6.1 μM).Formula:C23H24ClN3O3Color and Shape:SolidMolecular weight:425.91SHR902275
CAS:SHR902275: potent RAF inhibitor, hits RAS mutations, oral use. cRAF IC50=1.6 nM, bRAFwt IC50=10 nM, bRAFV600E IC50=5.7 nM, hinders cell growth.Formula:C26H23F3N4O4Color and Shape:SolidMolecular weight:512.48LH secretion antagonist 1
CAS:LH secretion antagonist 1 is an antagonist of luteinizing hormone secretion with analgesic activity.Formula:C18H24ClNO2Purity:98%Color and Shape:SolidMolecular weight:321.84RS 2135
CAS:RS 2135 is a novel class I antiarrhythmic agent to inhibit ischemia-induced ventricular arrhythmias.Formula:C18H21ClN2O2Purity:98%Color and Shape:SolidMolecular weight:332.83Retelliptine
CAS:Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.Formula:C25H32N4OPurity:98%Color and Shape:SolidMolecular weight:404.55TGR5 Receptor Agonist 3
CAS:TGR5 Receptor Agonist 3 is a GPBAR1 agonist with EC50 of 16.4 nM (hTGR5) & 209 nM (mTGR5), ensures gallbladder safety and reduces filling.Formula:C29H27N3O6Color and Shape:SolidMolecular weight:513.54EED ligand 1
EED ligand 1: potent PRC2 inhibitor targeting EED subunit.Formula:C19H19FN8OColor and Shape:SolidMolecular weight:394.41ZLHQ-5f
ZLHQ-5f inhibits CDK2/Topo I, with IC50 of 0.145μM for CDK2/CycA2, and promotes apoptosis by arresting HCT116 cells in S phase.Formula:C28H25N5O2Color and Shape:SolidMolecular weight:463.53MsbA-IN-2
MsbA-IN-2 is a potent inhibitor of the lipopolysaccharide transporter MsbA and is able to act on E. coli MsbA (IC50: 2 nM).Formula:C23H19Cl2NO3Color and Shape:SolidMolecular weight:428.31IRE1α kinase-IN-4
CAS:IRE1α kinase-IN-4 (compound 6) is a potent inhibitor of IRE1α, exhibiting a Ki value of 140 nM. It acts as an ATP-competitive ligand for IRE1α [1].Formula:C29H31N7O2Color and Shape:SolidMolecular weight:509.6ATM Inhibitor-4
ATM Inhibitor -4: selective, potent (IC50: 0.32 nM), inhibits PI3K family, stable, stops mTOR at 1 μM.Formula:C26H29FN6O3Color and Shape:SolidMolecular weight:492.55LSD1-IN-13 hydrochloride
CAS:LSD1-IN-13 hydrochloride (7e) is an oral LSD1 inhibitor (IC50: 24.43 nM), promoting differentiation in AML cell lines.Formula:C23H30ClN3O2SColor and Shape:SolidMolecular weight:448.02ITK inhibitor 6
CAS:ITK inhibitor 6 selectively targets ITK, BTK, JAK3, EGFR, LCK, blocks PLCγ1 and ERK1/2 phosphorylation, and inhibits cell proliferation.Formula:C28H24F2N4O2Color and Shape:SolidMolecular weight:486.51Antibacterial agent 80
Antibacterial agent 80 (compound 20) has antibacterial activity [1].Formula:C14H21N3S2Color and Shape:SolidMolecular weight:295.47SM-433 hydrochloride
SM-433 hydrochloride, a Smac mimetic & IAP inhibitor, binds XIAP BIR3; potent IC50 <1 μM. (Patent WO2008128171A2)Formula:C32H44ClN5O4Color and Shape:SolidMolecular weight:598.18TMX-4113
TMX-4113 has potential to be used in cancer that is a phosphodiesterase 6D(PDE6D) and casein kinase 1α(CK1α) degrader [1].Formula:C12H12N4O2S2Color and Shape:SolidMolecular weight:308.38Antimalarial agent 9
Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.Formula:C28H32BrN3O2Color and Shape:SolidMolecular weight:522.48AGN-204396
CAS:AGN-204396 is an antagonist that selectively blocks the activity of prostamides (prostaglandin-ethanolamides).Formula:C32H44FN3O4Color and Shape:SolidMolecular weight:553.71KRAS G12C inhibitor 37
CAS:KRAS G12C inhibitor 37 targets a key signaling protein, showing promise for cancer research involving KRAS G12C.Formula:C35H39F3N8O2Color and Shape:SolidMolecular weight:660.73Antitumor agent-54
Compound C11 inhibits 14-3-3η protein (KD: 35 μM), targets liver cancer cells, blocks G1-S phase, and induces apoptosis.Formula:C29H32N2O3Color and Shape:SolidMolecular weight:456.58KFA1982
CAS:KFA1982 is a novel and potent factor Xa inhibitor.Formula:C28H34ClN3O9S2Color and Shape:SolidMolecular weight:656.17RSK4-IN-1
CAS:RSK4-IN-1 is a compound exhibiting potent inhibition of RSK4, demonstrated by an IC50 value of 9.5 nM.Formula:C19H20F2N4O3Color and Shape:SolidMolecular weight:390.38MB725
CAS:MB725 is a strong and selective inducer of viability reduction in several cancer cell lines containing the oncogenic p53-Y220C mutation.Formula:C18H21IN4O2SColor and Shape:SolidMolecular weight:484.35RXR antagonist 1
RXR antagonist 1 is a Retinoid X Receptor (RXR) modulator that exhibits high RXR antagonism (pA2: 8.06). RXR antagonist 1 can be used to study type 2 diabetes.Formula:C28H33F3N2O3Color and Shape:SolidMolecular weight:502.57Antifungal agent 39
CAS:Antifungal agent 39 (Compound 9h) is a broad-spectrum antifungal agent.Formula:C23H22ClN3O5Color and Shape:SolidMolecular weight:455.89GW311616 hydrochloride
CAS:GW-311616 hydrochloride is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).Formula:C19H32ClN3O4SPurity:98%Color and Shape:SolidMolecular weight:433.99CDK5-IN-2
CAS:CDK5-IN-2 (compound 15) is a highly selective CDK5 inhibitor that acts on CDK5/p25 (IC50: 0.2 nM) and CDK2/CycA (IC50: 23 nM).Formula:C29H28FN5OColor and Shape:SolidMolecular weight:481.56PF-00489791
CAS:PF-00489791 (PF4634817) is a long-acting PDE5 inhibitor with hypotensive activity for the study of diabetic nephropathy.Formula:C20H28N8O4SPurity:99.97%Color and Shape:SolidMolecular weight:476.55DMP-728 free base
CAS:DMP-728 free base is a highly potent and selective GPIIbDIIa antagonistFormula:C25H36N8O7Color and Shape:SolidMolecular weight:560.60Menin-MLL inhibitor 4
CAS:Menin-MLL inhibitor 4 has antitumor activity.Menin-MLL inhibitor 4 is an inhibitor of Menin- MLL (mixed-lineage leukemia protein) interaction .Formula:C32H38FN7O3Purity:98%Color and Shape:SolidMolecular weight:587.69BRD-K25923209
CAS:BRD-K25923209 is a novel inhibitor of BAF transcriptional repression.Formula:C29H36N4O3Color and Shape:SolidMolecular weight:488.62JAK3-IN-11
CAS:JAK3-IN-11: potent oral JAK3 inhibitor (IC50=1.7 nM), noncytotoxic, >588-fold selectivity, blocks T-cell growth; useful in autoimmune research.Formula:C23H23N5O2Color and Shape:SolidMolecular weight:401.46MrgprX2 antagonist-6
MrgprX2 antagonist-6 is a potent antiallergic agent with inhibitory effects on mast cell degranulation.Formula:C24H23F3N6O3Color and Shape:SolidMolecular weight:500.47Antiviral agent 7
Antiviral agent 7 is a peptide-based coating that kills viruses.Formula:C29H31F2N3O6Color and Shape:SolidMolecular weight:555.57Nonsteroidal aromatase inhibitor 1
Compound 13h, a nonsteroidal aromatase inhibitor, has a potent IC50 of 0.09 nM against CYP19A1, showing promise for breast cancer research.Formula:C22H16N4O2Color and Shape:SolidMolecular weight:368.39JBIR-22
CAS:JBIR-22 is a natural inhibitor for protein−protein interaction of the homodimer of proteasome assembly factor 3.Formula:C23H33NO6Color and Shape:SolidMolecular weight:419.51KDOAM-25 trihydrochloride (2230731-99-2 free base)
KDOAM-25 trihydrochloride, a selective KDM5 inhibitor (IC50: 19-71 nM), boosts H3K4 methylation and hinders MM1S cell growth.Formula:C15H28Cl3N5O2Purity:98%Color and Shape:SolidMolecular weight:416.77A1/A3 AR antagonist 1
Compound 10 is a potent dual A1/A3 AR antagonist, with Ki values of 37.6 nM (hA1), 25.4 nM (hA3), and 1.47 nM (rA1), studied in renal, lung, and Alzheimer's.Formula:C24H18N2O3SColor and Shape:SolidMolecular weight:414.48EGFR-IN-58
EGFR-IN-58 is a potent, selective, ATP-competitive inhibitor of EGFR. EGFR-IN-58 exhibits significant cytotoxicity against melanoma, colon and blood cancers.Formula:C31H30FN7OColor and Shape:SolidMolecular weight:535.61TIY-7
TIY-7 is a selective, orally active inhibitor of the promyosin receptor kinase (TRK) enzyme. TIY-7 exhibited anti-tumour effects in a mouse xenograft model.Color and Shape:SolidMAO A/HDAC-IN-1
MAO A/HDAC-IN-1 is an effective monoamine oxidase A (MAO A) and HDAC dual inhibitor, which can be used for glioma research.Formula:C21H24ClN3O3Color and Shape:SolidMolecular weight:401.89MALT1-IN-5
CAS:MALT1-IN-5 is a potent inhibitor of the MALT1 protease and can be used in cancer research.Formula:C17H17ClF2N6O3Color and Shape:SolidMolecular weight:426.80AMG-315
CAS:AMG-315: Chiral AEA analogue, potent CB1 agonist (Ki 7.8 nM, EC50 0.6 nM), stable against hydrolyzing/oxidative enzymes.Formula:C24H41NO2Color and Shape:SolidMolecular weight:375.59CLK1/2-IN-1
CAS:CLK1/2-IN-1 is a CLK1 and CLK2 inhibitor and it also inhibits SRPK1 and SRPK2.Formula:C21H20F3N7OPurity:98%Color and Shape:SolidMolecular weight:443.42Furaprevir
CAS:Furaprevir is an HCV NS3/4A InhibitorFormula:C47H56N6O10SColor and Shape:SolidMolecular weight:897.05CDK9-IN-13
CDK9-IN-13 is a potent and selective CDK inhibitor (IC50<3 nM). CDK9-IN-13 has a very short half-life in rodents.Formula:C27H35N5O2Color and Shape:SolidMolecular weight:461.6Monlunabant
CAS:Monlunabant ((S)-MRI-1891), a solid dispersion compound, functions as an inhibitor of the cannabinoid CB1 receptor [1].Formula:C26H22ClF3N6O3SPurity:98%Color and Shape:SolidMolecular weight:591.00Vimirogant
CAS:Vimirogant is a RORγ inhibitor (Ki: <100 nM).Formula:C27H35F3N4O3SPurity:98%Color and Shape:SolidMolecular weight:552.65TAK-024
CAS:TAK-024 is an inhibitor of platelet(IC50s of 31, 79 and 51 nM in human, monkey and guinea pig, respectively).Formula:C27H34N10O6Purity:98%Color and Shape:SolidMolecular weight:594.62EGFR/HER2-IN-7
EGFR/HER2-IN-7: Potent, selective dual inhibitor for MCF-7 cancer; IC50: EGFR 0.18μM, HER2 0.146μM, DHFR 0.907μM.Formula:C19H21N3O2SColor and Shape:SolidMolecular weight:355.45AT-IAP
CAS:AT-IAP is an effective dual antagonist of XIAP and cIAP1.Formula:C29H40FN5O2Purity:98%Color and Shape:SolidMolecular weight:509.66
