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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66513 products of "Inhibitors"

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  • YM-60828 dihydrochloride

    CAS:
    YM-60828 dihydrochloride is a Factor Xa (FXa) inhibitor and anticoagulant used in the treatment of venous thromboembolic disease.
    Formula:C27H33Cl2N5O5S
    Color and Shape:Solid
    Molecular weight:610.55

    Ref: TM-T70184

    5mg
    1,791.00€
    10mg
    2,412.00€
    25mg
    3,582.00€
    50mg
    4,834.00€
    100mg
    6,525.00€
  • PCTR1

    CAS:
    PCTR1, derived from DHA, hastens inflammation resolution and boosts macrophage function, reducing PGE2, PGD2, and TXB2 in mice.
    Formula:C32H47N3O9S
    Color and Shape:Solid
    Molecular weight:649.8

    Ref: TM-T37300

    10µg
    500.00€
    25µg
    1,153.00€
    50µg
    2,223.00€
    100µg
    3,898.00€
  • MB-07344 sodium


    "MB-07344 sodium is a TR-β agonist with a 2.17 nM Ki, boosts Atorvastatin's cholesterol-lowering effects in various animals."
    Formula:C19H25NaO5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:387.36

    Ref: TM-T11954L

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • SPR-00305

    CAS:
    SPR-00305 is a novel potent inhibitor of the mvfr pathway
    Formula:C24H19ClN2O3
    Color and Shape:Solid
    Molecular weight:418.87

    Ref: TM-T70030

    25mg
    2,448.00€
    50mg
    3,222.00€
    100mg
    4,410.00€
  • 2-Methylsorbinol

    CAS:
    2-Methylsorbinol is a bioactive chemical.
    Formula:C12H11FN2O3
    Color and Shape:Solid
    Molecular weight:250.23

    Ref: TM-T29357

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • ERK1/2 inhibitor 6

    CAS:
    ERK1/2 inhibitor 6 - potent cancer/inflammation treatment from WO2021063335A1.
    Formula:C27H29ClFN7O5
    Color and Shape:Solid
    Molecular weight:586.01

    Ref: TM-T64147

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MAP3K14-IN-173

    CAS:
    MAP3K14-IN-173 is a potent MAP3K14 kinase inhibitor.
    Formula:C29H31N7O2
    Color and Shape:Solid
    Molecular weight:509.60

    Ref: TM-T69894

    25mg
    2,583.00€
    50mg
    3,402.00€
    100mg
    4,680.00€
  • c-Myc inhibitor 4


    Potent oral c-Myc inhibitor 4 reduces the proto-oncogene linked to tumor development.
    Formula:C26H33FN6O3
    Color and Shape:Solid
    Molecular weight:496.58

    Ref: TM-T63359

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (Z)-Lanoconazole


    (Z)-Lanoconazole, an imidazole antifungal for dermatophytosis and onychomycosis, inhibits fungal ergosterol production.
    Formula:C14H10ClN3S2
    Color and Shape:Solid
    Molecular weight:319.83

    Ref: TM-T60853

    2mg
    51.00€
  • Bleomycin Free Base

    CAS:
    Bleomycin Free Base, a glycopeptide antibiotic, halts DNA function and treats solid tumors.
    Formula:C55H84N17O21S3
    Color and Shape:Solid
    Molecular weight:1415.55

    Ref: TM-T71445

    25mg
    8,658.00€
    50mg
    11,502.00€
    100mg
    16,830.00€
  • GSK866

    CAS:
    GSK866 is a selective glucocorticoid receptor agonist (SEGRA).
    Formula:C23H21Cl2F4N5O3
    Color and Shape:Solid
    Molecular weight:562.34

    Ref: TM-T68224

    25mg
    2,313.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • SARS-CoV-2 nsp14-IN-2


    SARS-CoV-2 nsp14-IN-2: Strong Nsp14 methyltransferase inhibitor (IC50: 0.09 μM), potential for COVID-19 research.
    Formula:C21H21N5O5S
    Color and Shape:Solid
    Molecular weight:455.49

    Ref: TM-T62819

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MsbA-IN-5


    MsbA-IN-5 (compound 40) is a potent and highly selective inhibitor of MsbA (IC50: 2 nM). MsbA-IN-5 can be used in Gram-negative studies.
    Formula:C23H19Cl2N5O
    Color and Shape:Solid
    Molecular weight:452.34

    Ref: TM-T62753

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PI3K-IN-35

    CAS:
    PI3K-IN-35 (6l) selectively inhibits PI3K-α, β, δ (IC50: 13.98, 7.22, 10.94 μM), blocks G2/M phase, induces apoptosis, and is useful in leukemia research.
    Formula:C25H23N7O2
    Color and Shape:Solid
    Molecular weight:453.5

    Ref: TM-T62779

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Uprosertib hydrochloride

    CAS:
    Uprosertib hydrochloride is a potent and selective inhibitor of pan-Akt (IC50: 180/328/38 nM for Akt1/Akt2/Akt3, respectively).
    Formula:C18H17Cl3F2N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:465.71

    Ref: TM-T15428

    25mg
    2,448.00€
    50mg
    3,222.00€
    100mg
    4,410.00€
  • P2X receptor-1


    P2X receptor-1 is a potential inhibitor of P2X receptor for the treatment of pain and inflammation.
    Formula:C14H14ClN3O3S2
    Color and Shape:Solid
    Molecular weight:371.86

    Ref: TM-T61490

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Haspin-IN-1


    Haspin-IN-1 blocks haspin (IC50: 119 nM) and inhibits CLK1, DYRK1A, CDK9 with potential as an anticancer drug.
    Formula:C12H8N4O2S
    Color and Shape:Solid
    Molecular weight:272.28

    Ref: TM-T60477

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • OICR-9429-N-C2-NH2

    CAS:
    OICR-9429-N-C2-NH2, a ligand for WDR5, intermediate 2, serves as a crucial compound in the synthesis of PROTACs.
    Formula:C31H38F3N7O2
    Color and Shape:Solid
    Molecular weight:597.687

    Ref: TM-T39977

    25mg
    1,639.00€
  • MtTMPK-IN-2

    CAS:
    MtTMPK-IN-2 inhibits M. tuberculosis TMPK (IC50: 1.1 μM), Mtb H37Rv (MIC: 12.5 μM), and is cytotoxic in MRC-5 cells (EC50: 6.1 μM).
    Formula:C23H24ClN3O3
    Color and Shape:Solid
    Molecular weight:425.91

    Ref: TM-T62305

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • rel-MDM2/4-p53-IN-3


    rel-MDM2/4-p53-IN-3 inhibits MDM2/4-p53 PPI, IC50: MDM2 18.5nM, MDM4 14.8nM, targets cancer research.
    Formula:C25H24Cl2FN3O3
    Color and Shape:Solid
    Molecular weight:504.38

    Ref: TM-T63438

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Chitin synthase inhibitor 9


    CHS inhibitor 9: a broad-spectrum antifungal for studying fungal infections.
    Formula:C24H25N3O6
    Color and Shape:Solid
    Molecular weight:451.47

    Ref: TM-T62739

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DH376

    CAS:
    DH376 inhibits DAGLα in a time and dose dependent manner in mouse brain. DH376 shows picomolar activity.
    Formula:C31H28F2N4O3
    Color and Shape:Solid
    Molecular weight:542.58

    Ref: TM-T27161

    25mg
    2,313.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • Fandosentan

    CAS:
    Fandosentan is an endothelin receptor antagonist.
    Formula:C25H18F3NO6S
    Color and Shape:Solid
    Molecular weight:517.47

    Ref: TM-T69791

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • KRAS G12C inhibitor 50

    CAS:
    KRAS G12C inhibitor 50 is a KRAS G12C inhibitor (IC50: 46.7 nM).
    Formula:C31H34N8O2
    Color and Shape:Solid
    Molecular weight:550.65

    Ref: TM-T63891

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • LRRK2-IN-5


    LRRK2-IN-5 is an oral, BBB-penetrating selective inhibitor for LRRK2 with IC50s: 1.2μM (GS) and 16μM (WT); halts LRRK2 autophosphorylation.
    Formula:C24H26F2N4O2S
    Color and Shape:Solid
    Molecular weight:472.55

    Ref: TM-T63057

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • S1P1 agonist 5


    Selective oral S1P1 agonist 5 inhibits lymphocyte drainage, potential for MS research.
    Formula:C23H24ClN2NaO4
    Color and Shape:Solid
    Molecular weight:450.89

    Ref: TM-T62732

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CVS-1578

    CAS:
    CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.
    Formula:C20H30N6O5S
    Color and Shape:Solid
    Molecular weight:466.55

    Ref: TM-T70110

    25mg
    2,313.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • BRD7929

    CAS:
    BRD7929 is a multistage antimalarial inhibitor for single-dose treatment of malaria in mouse models.
    Formula:C33H38N4O2
    Color and Shape:Solid
    Molecular weight:522.68

    Ref: TM-T70215

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • AS2521780

    CAS:
    AS2521780 is an inhibitor of PKCθ (IC50: 0.48 nM).
    Formula:C30H41N7OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:547.76

    Ref: TM-T14328

    25mg
    2,718.00€
    50mg
    3,582.00€
    100mg
    4,950.00€
  • DS01080522


    DS01080522: PRKACA inhibitor, IC50: kinase 0.8 nM, CREB 66 nM; potential for cancer research.
    Formula:C23H20Cl2N4O3
    Color and Shape:Solid
    Molecular weight:471.34

    Ref: TM-T63041

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Antifungal agent 38


    Antifungal agent 38, a heterocyclic disulfide, shrinks hyphae and damages cell membranes, causing leakage.
    Formula:C8H12N2S2
    Color and Shape:Solid
    Molecular weight:200.32

    Ref: TM-T60236

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CH-38083

    CAS:
    CH-38083 is a selective and effective alpha-2 adrenoceptors antagonist.
    Formula:C18H24ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:337.84

    Ref: TM-T23878

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Topoisomerase II inhibitor 6


    Topoisomerase II inhibitor 6, a potent tryptanthrin derivative, blocks G2 phase in CCRF-CEM cells, induces DNA breaks, and may be used for cancer research.
    Formula:C19H18N4O2
    Color and Shape:Solid
    Molecular weight:334.37

    Ref: TM-T61017

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CM-352

    CAS:
    CM-352 is a metalloproteinase inhibitor that reduces brain damage and improves functional recovery in rat models of cerebral hemorrhage.
    Formula:C24H29N3O6S
    Purity:97.24%
    Color and Shape:Solid
    Molecular weight:487.57

    Ref: TM-T70470

    1mg
    374.00€
    5mg
    793.00€
    10mg
    973.00€
    25mg
    1,279.00€
  • Arterolane

    CAS:
    Arterolane is an antimalarial compound. For against P. falciparum Ro73 and W2, the IC50s are both 1.1 nM.
    Formula:C22H36N2O4
    Color and Shape:Solid
    Molecular weight:392.53

    Ref: TM-T14325

    1mL*10mM (DMSO)
    311.00€
    5mg
    313.00€
    25mg
    888.00€
    50mg
    1,224.00€
    100mg
    1,972.00€
  • BI 224436

    CAS:
    BI 224436 is an inhibitor of HIV-1 noncatalytic site integrase. With EC50 values of less than 15 nM against different HIV-1 laboratory strains.
    Formula:C27H26N2O4
    Color and Shape:Solid
    Molecular weight:442.51

    Ref: TM-T14559

    1mg
    4,618.00€
    5mg
    8,883.00€
  • FGFR4-IN-9


    FGFR4-IN-9 is a selective inhibitor of FGFR4 (IC50: 75.3 nM) that effectively inhibits the growth and angiogenesis of hepatocellular carcinoma cells.
    Formula:C24H22ClF3N4O4
    Color and Shape:Solid
    Molecular weight:522.9

    Ref: TM-T63662

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ADU-S100 disodium salt

    CAS:
    ADU-S100 (MIW815) disodium salt is an activator of stimulator of interferon genes (STING).
    Formula:C20H22N10Na2O10P2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:734.51

    Ref: TM-T10252

    50mg
    3,718.00€
    100mg
    5,571.00€
    200mg
    8,362.00€
  • Enpp-1-IN-7


    Enpp-1-IN-7: potent enpp-1 inhibitor, broad specificity, potential in cancer/infectious disease research. (WO2021203772A1)
    Formula:C18H19N7O4S
    Color and Shape:Solid
    Molecular weight:429.45

    Ref: TM-T62368

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Antiviral agent 15


    Compound 15f, a Clofazimine derivative, inhibits rabies (EC50: 1.45 μM) and SARS-CoV-2 (EC50: 14.6 μM).
    Formula:C27H24FN5O
    Color and Shape:Solid
    Molecular weight:453.51

    Ref: TM-T62780

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tubulin polymerization-IN-34


    "Tubulin-IN-34 inhibits oxazolylisoindole microtubule assembly, selective for VL51 lymphoma."
    Formula:C31H35N3O6
    Color and Shape:Solid
    Molecular weight:545.63

    Ref: TM-T63849

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LHC-165

    CAS:
    LHC-165 is an agonist of TLR7. It also has the potential to treat solid tumors.
    Formula:C29H32F2N3O7P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:603.55

    Ref: TM-T15751

    25mg
    2,583.00€
    50mg
    3,402.00€
    100mg
    4,680.00€
  • KPH2f

    CAS:
    KPH2f: dual URAT1/GLUT9 inhibitor, orally active, IC50: 0.24μM (URAT1), 9.37μM (GLUT9), minimal OAT1/ABCG2 impact.
    Formula:C24H16N3NaO2S
    Color and Shape:Solid
    Molecular weight:433.46

    Ref: TM-T62432

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 9-cis-β-Carotene

    CAS:
    9-cis-β-Carotene, a precursor of retinal, is cleaved by beta-carotene oxygenase 1 (BCMO1) to produce 9-cis-retinal.
    Formula:C40H56
    Purity:98%
    Color and Shape:Solid
    Molecular weight:536.87

    Ref: TM-T13524

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Complex III-IN-1


    Complex III-IN-1 inhibits complex III, has antifungal properties, and an EC50 of 18.53 mg/L against S. sclerotiorum.
    Formula:C14H20ClNO2S2
    Color and Shape:Solid
    Molecular weight:333.9

    Ref: TM-T61009

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CP-608039

    CAS:
    CP-608039 is a selective adenosine A3 receptor agonist for both human A3 and human A1 receptors.
    Formula:C23H25ClN8O5
    Color and Shape:Solid
    Molecular weight:528.95

    Ref: TM-T31068

    25mg
    2,448.00€
    50mg
    3,222.00€
    100mg
    4,410.00€
  • α-Glucosidase-IN-19


    Alpha-Glucosidase-IN-19 (Compound 6B) is an orally active alpha-glucosidase inhibitor (IC50: 3.63 μM) with antidiabetic effects.
    Formula:C31H25NOS
    Color and Shape:Solid
    Molecular weight:459.6

    Ref: TM-T62891

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RMG8-8


    RMG8-8 shows the excellent efficacy against C. neoformans (1.56 μg/mL).
    Formula:C41H78N8O5
    Color and Shape:Solid
    Molecular weight:763.11

    Ref: TM-T73480

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • Tubulin polymerization-IN-9

    CAS:
    Tubulin-IN-9 inhibits tubulin (IC50: 1.82 μM), halts K562 cells in G2/M, induces apoptosis, and has anti-cancer effects.
    Formula:C19H19NO5Se
    Color and Shape:Solid
    Molecular weight:420.32

    Ref: TM-T62217

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Nrf2 activator-6

    CAS:
    Nrf2 activator-6, a tetrahydroisoquinoline, inhibits Kelch-Nrf2 at 5 nM IC50 (WO2021214470A1).
    Formula:C31H37ClFN5O5
    Color and Shape:Solid
    Molecular weight:614.11

    Ref: TM-T72697

    25mg
    3,529.00€
    50mg
    4,663.00€
    100mg
    6,570.00€
  • Fonsartan free acid

    CAS:
    Fonsartan: Angiotensin receptor blocker, halts angiotensin II effects on rat vascular cells.
    Formula:C26H32N4O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:544.69

    Ref: TM-T27347

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Thiomuscimol hydrobromide

    CAS:
    Thiomuscimol hydrobromide is an agonist of GABAA receptor.
    Formula:C4H6N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:130.17

    Ref: TM-T28965

    500µg
    144.00€
    1mg
    245.00€
    5mg
    607.00€
    10mg
    888.00€
  • LY3325656

    CAS:
    LY3325656, a GPR142 agonist with anti-diabetic properties, progresses to phase 1 trials for Type 2 diabetes.
    Formula:C21H23F3N6O2
    Color and Shape:Solid
    Molecular weight:448.44

    Ref: TM-T70005

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • (RS)-AMPA monohydrate

    CAS:
    (RS)-AMPA monohydrate, potent glutamate analogue, selectively activates L-glutamic acid without affecting kainic acid or NMDA receptors.
    Formula:C7H12N2O5
    Color and Shape:Solid
    Molecular weight:204.182

    Ref: TM-T60242

    25mg
    797.00€
    50mg
    1,035.00€
    100mg
    1,566.00€
  • K-14585

    CAS:
    K-14585 blocks PAR(2), reduces NFkappaB activity, and IL-8 response, but alone can boost IL-8.
    Formula:C51H56Cl2N8O4
    Color and Shape:Solid
    Molecular weight:915.95

    Ref: TM-T27708

    5mg
    3,931.00€
  • MEIS-IN-3


    MEIS-IN-3 is a potent inhibitor of MEIS.
    Formula:C25H26N2O4
    Color and Shape:Solid
    Molecular weight:418.48

    Ref: TM-T62194

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • HOE-288

    CAS:
    HOE-288 is a converting enzyme (CE) inhibitor.
    Formula:C27H38N2O5
    Color and Shape:Solid
    Molecular weight:470.60

    Ref: TM-T68309

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • 7(Z),11(Z)-Nonacosadiene

    CAS:
    7(Z),11(Z)-Nonacosadiene, a female fly pheromone, spurs male courtship; it's a C29 diene made by a female-specific elongase.
    Formula:C29H56
    Color and Shape:Solid
    Molecular weight:404.75

    Ref: TM-T37921

    10mg
    1,288.00€
    50mg
    5,805.00€
  • MK2-IN-4

    CAS:
    MK2-IN-4 is a MAPKAPK2 (MK2) inhibitor (IC50: 45 nM). MK2-IN-4 can be used in cancer, inflammation and immunology studies.
    Formula:C25H24N4O2
    Color and Shape:Solid
    Molecular weight:412.48

    Ref: TM-T62110

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Calphostin I

    CAS:
    Calphostins, from Cladosporium fungus, inhibit PKC. Notably, calphostin C is a potent biochemical tool.
    Formula:C44H38O15
    Color and Shape:Solid
    Molecular weight:806.76

    Ref: TM-T71135

    25mg
    2,718.00€
    50mg
    3,582.00€
    100mg
    4,950.00€
  • D-Cl-amidine hydrochloride


    D-Cl-amidine hydrochloride is a potent and highly selective inhibitor of PAD1. It exhibits excellent tolerance and does not induce significant toxicity [1].
    Formula:C14H20Cl2N4O2
    Color and Shape:Solid
    Molecular weight:347.24

    Ref: TM-T61155

    100mg
    1,341.00€
  • CGP 22979

    CAS:
    CGP 22979 is a renal selective vasodilator prodrug.
    Formula:C16H24N4O4
    Color and Shape:Solid
    Molecular weight:336.39

    Ref: TM-T30821

    25mg
    2,448.00€
    50mg
    3,222.00€
    100mg
    4,410.00€
  • MRS-2339

    CAS:
    MRS-2339 is a P2X receptor activator.
    Formula:C12H15ClN5O6P
    Color and Shape:Solid
    Molecular weight:391.70

    Ref: TM-T69255

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • SOS1-IN-9


    SOS1-IN-9 is a potent inhibitor of SOS1 that acts on KRAS G12C-SOS1 (IC50: 116.5 nM).
    Formula:C22H28F3N5O
    Color and Shape:Solid
    Molecular weight:435.49

    Ref: TM-T62478

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CD73-IN-13


    CD73-IN-13, a potent CD73 inhibitor, may be developed for tumor-related disease treatment.
    Formula:C13H11F3N4O2
    Color and Shape:Solid
    Molecular weight:312.25

    Ref: TM-T60779

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • β-Secretase Inhibitor III


    β-Secretase Inhibitor III is a highly selective inhibitor of BACE1 with a Ki value of 0.13 nM.
    Formula:C20H20F2N4O3S
    Color and Shape:Solid
    Molecular weight:434.46

    Ref: TM-T62455

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cdc7-IN-10

    CAS:
    Cdc7-IN-10 is a potent inhibitor of Cdc7 (IC50 ≤ 1 nM) and can be used in studies of proliferative diseases.
    Formula:C20H22F2N4O2S
    Color and Shape:Solid
    Molecular weight:420.48

    Ref: TM-T62230

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • NLRP3-IN-8

    CAS:
    NLRP3-IN-8, orally active inflammasome blocker, IC50 of 1.23μM, stable (t1/2 = 138.63min), non-toxic (IC50 >100μM).
    Formula:C23H20N2O6
    Color and Shape:Solid
    Molecular weight:420.41

    Ref: TM-T62221

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LSD1-IN-22


    LSD1-IN-22: potent LSD1 inhibitor, K_i 98 nM, curbs cancer cell growth.
    Formula:C9H8BrF2N
    Color and Shape:Solid
    Molecular weight:248.07

    Ref: TM-T60362

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • COX-2/PI3K-IN-2


    COX-2/PI3K-IN-2 (5f): anti-inflammatory & anti-cancer, selectively inhibits COX-2 (Ki=3.02nM), potently blocks PI3K (IC50=2.78nM).
    Formula:C16H17N5O2
    Color and Shape:Solid
    Molecular weight:311.34

    Ref: TM-T60769

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BChE-IN-3


    BChE-IN-3: Selective, pseudo-irreversible BChE inhibitor (IC50: 56.9 nM); borderline reversible AChE inhibitor.
    Formula:C26H41N3O2
    Color and Shape:Solid
    Molecular weight:427.62

    Ref: TM-T62336

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ABT 491 Hydrochloride

    CAS:
    ABT-491 hydrochloride is an active platelet activator receptor (PAF-R) antagonist with good selectivity and oral administration.
    Formula:C28H23ClFN5O2
    Color and Shape:Solid
    Molecular weight:515.97

    Ref: TM-T29524

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • Leukotriene B4 dimethyl amide

    CAS:
    LTB4 dimethyl amide: inhibits human neutrophil degranulation and rat lysozyme release; antagonizes LTB4 receptor on guinea pig lung membranes (Ki = 130 nM).
    Formula:C22H37NO3
    Color and Shape:Solid
    Molecular weight:363.53

    Ref: TM-T37618

    25µg
    567.00€
    50µg
    1,063.00€
    100µg
    2,008.00€
  • 5(S),6(S)-DiHETE

    CAS:
    5(S),6(S)-DiHETE: a 5,6-dihydroxy acid from LTA4 hydrolysis, lacks leukotriene activity.
    Formula:C20H32O4
    Color and Shape:Solid
    Molecular weight:336.47

    Ref: TM-T37653

    25mg
    2,718.00€
    50mg
    3,582.00€
    100mg
    4,950.00€
  • WQ3810 TFA


    WQ3810 TFA is an orally available fluoroquinolone with antimicrobial activity against Mycobacterium tuberculosis and inhibits the DNA rotamase activity of
    Formula:C24H23F6N5O5
    Purity:99.52%
    Color and Shape:Soild
    Molecular weight:575.46

    Ref: TM-T13346L

    1mg
    411.00€
    5mg
    954.00€
  • Diarylalkane derivative 1

    CAS:
    Diarylalkane derivative 1 is used for the research of pancreatitis.
    Formula:C34H51NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:537.77

    Ref: TM-T13662

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • PARP1-IN-12


    PARP1-IN-12: potent PARP1 inhibitor, IC50 2.99 nM, triggers cell apoptosis, G2/M arrest, induces DSBs in BRCA-deficient cells.
    Formula:C43H56FN5O5
    Color and Shape:Solid
    Molecular weight:741.93

    Ref: TM-T73023

    25mg
    2,448.00€
    50mg
    3,222.00€
    100mg
    4,410.00€
  • IL-17 modulator 5

    CAS:
    IL-17 modulator 5 is a IL-17 inhibitor, with an IC 50 of 1 nM .
    Formula:C28H23F6N9O2
    Color and Shape:Solid
    Molecular weight:631.53

    Ref: TM-T72598

    25mg
    2,583.00€
    50mg
    3,402.00€
    100mg
    4,680.00€
  • TP-6076

    CAS:
    TP-6076 is a fluorocycline antibiotic, inhibiting bacterial protein synthesis, exhibiting great antimicrobial activity against carbapenem-resistant A.
    Formula:C28H32F3N3O7
    Color and Shape:Solid
    Molecular weight:579.56

    Ref: TM-T70429

    25mg
    4,609.00€
    50mg
    6,103.00€
    100mg
    8,730.00€
  • EFdA-TP tetrasodium

    CAS:
    EFdA-TP tetrasodium is a potent HIV-1 inhibitor that blocks DNA synthesis as an ICT or DCT.
    Formula:C12H11FN5Na4O12P3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:621.12

    Ref: TM-T72461

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • ATR-IN-11


    ATR-IN-11, a potent ATR kinase inhibitor, shows promise as a lead for DNA damage response-targeted cancer drugs.
    Formula:C25H30N6O2
    Color and Shape:Solid
    Molecular weight:446.54

    Ref: TM-T62651

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • QPX7728 methoxy acetoxy methy ester

    CAS:
    QPX7728 methoxy acetoxy methy ester is an inhibitor of boronic acid β-lactamase.
    Formula:C14H14BFO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:324.07

    Ref: TM-T12602

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Dup-714

    CAS:
    Dup-714 is a thrombin inhibitor.
    Formula:C21H33BN6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:460.33

    Ref: TM-T27220

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Gemilukast

    CAS:
    Gemilukast (ONO-6950) is a cysteinyl leukotriene 1 and 2 receptor inhibitor that inhibits bronchoconstriction and is used in the treatment of asthma.
    Formula:C36H37F2NO5
    Purity:98.27% - 99.5%
    Color and Shape:Solid
    Molecular weight:601.68

    Ref: TM-T11388

    1mg
    109.00€
    5mg
    260.00€
    1mL*10mM (DMSO)
    344.00€
    10mg
    447.00€
    25mg
    865.00€
    50mg
    1,341.00€
    100mg
    2,385.00€
  • GLS1 Inhibitor-5


    GLS1 Inhibitor-5 (24y): Selective, oral glutaminase 1 inhibitor; IC50 68 nM; induces apoptosis; anti-tumor.
    Color and Shape:Solid

    Ref: TM-T64259

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ChE/Aβ1-42-IN-1


    ChE/Aβ1-42-IN-1 (compound 28) is a potent aggregation inhibitor of ChE and Aβ 1-42 with excellent BBB permeability.
    Formula:C19H24N2O3
    Color and Shape:Solid
    Molecular weight:328.41

    Ref: TM-T60940

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GABAA receptor agonist 1


    Compound 3e, a potent GABAA agonist, targets GABA sites and has potential anti-depressive effects in mice.
    Formula:C20H30O3
    Color and Shape:Solid
    Molecular weight:318.45

    Ref: TM-T60842

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tylophorinidine

    CAS:
    Tylophorinidine is an antifungal agent that has shown to inhibit cell growth.
    Formula:C22H23NO4
    Color and Shape:Solid
    Molecular weight:365.42

    Ref: TM-T69444

    25mg
    3,123.00€
    50mg
    4,123.00€
    100mg
    5,760.00€
  • PRMT5-IN-1 hydrochloride


    PRMT5 IN-1 hydrochloride is a potent PRMT5 inhibitor (IC50: 11 nM), forms covalent adduct with C449, and converts to an aldehyde in vivo.
    Formula:C19H20Cl2N4O5
    Color and Shape:Solid
    Molecular weight:455.29

    Ref: TM-T62815

    25mg
    8,370.00€
  • Ciluprevir

    CAS:
    Ciluprevir is a selective HCV NS3 protease inhibitor, effective against non-genotype-1 HCV; less potent for genotypes 2/3.
    Formula:C40H50N6O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:774.93

    Ref: TM-T19627

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • AY-22,252

    CAS:
    AY-22,252 is an inhibitor of beef heart & rat brain nucleoside-3',5'- monophosphate phosphodiesterase.
    Formula:C27H37NaO7
    Color and Shape:Solid
    Molecular weight:496.57

    Ref: TM-T69159

    25mg
    2,853.00€
    50mg
    3,763.00€
    100mg
    5,220.00€
  • APJ receptor agonist 3

    CAS:
    APJ receptor agonist 3 is a highly effective and orally administerable agonist of the APJ receptor, demonstrating a potent EC50 value of 0.027 nM.
    Formula:C26H29ClN4O5
    Color and Shape:Solid
    Molecular weight:512.98

    Ref: TM-T63548

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GAT564


    GAT564, an allosteric CB1R modulator, shows EC50s of 87 nM (cAMP) & 320 nM (β-arrestin2) and lowers IOP effectively in glaucoma mice.
    Formula:C20H16N2O2S
    Color and Shape:Solid
    Molecular weight:348.42

    Ref: TM-T61180

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Carbodine

    CAS:
    Carbodine is an antiviral targeting CTP synthetase, effective against influenza A0/PR-8/34 and A2/Aichi/2/68.
    Formula:C10H15N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:241.24

    Ref: TM-T10677

    25mg
    2,853.00€
    50mg
    3,763.00€
    100mg
    5,220.00€
  • 22-HDHA

    CAS:
    22-HDHA is an oxidation product of docosahexaenoic acid .
    Formula:C22H32O3
    Color and Shape:Solid
    Molecular weight:344.49

    Ref: TM-T35997

    25µg
    945.00€
    50µg
    1,765.00€
    100µg
    3,412.00€
  • Holothurinogenin

    CAS:
    Holothurinogenin, as a lanosterol derivative, has toxic to nerve tissue.
    Formula:C30H46O4
    Color and Shape:Solid
    Molecular weight:470.68

    Ref: TM-T32095

    25mg
    8,928.00€
    50mg
    11,862.00€
    100mg
    17,370.00€
  • eIF4A3-IN-6

    CAS:
    eIF4A3-IN-6 is a potent eIF4A inhibitor, potentially used for treating eIF4A-related diseases like cancer. (US20170145026A1)
    Formula:C26H25N3O5
    Color and Shape:Solid
    Molecular weight:459.49

    Ref: TM-T62884

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • ERα degrader 5


    ERα degrader 5 is an orally active, selective estrogen receptor (ER) reducer that acts on ERα (EC50: 1.1 nM). ERα degrader 5 shows anti-tumour effects in vivo.
    Formula:C29H25F4N3O2S
    Color and Shape:Solid
    Molecular weight:555.59

    Ref: TM-T63922

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Aquayamycin

    CAS:
    Aquayamycin is an anthraquinone derivative and inhibitor of the enzyme tyrosine hydroxylase..
    Formula:C25H26O10
    Color and Shape:Solid
    Molecular weight:486.47

    Ref: TM-T69569

    25mg
    6,634.00€
    50mg
    8,802.00€
    100mg
    12,780.00€
  • Homomoschatoline

    CAS:
    Homomoschatoline is an antibacterial isolated from Artabotrys crassifolius.
    Formula:C19H15NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.33

    Ref: TM-T25505

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€