
Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,523 products)
- Apoptosis(5,792 products)
- Cell Cycle/Checkpoint(4,449 products)
- Chromatin/Epigenetics(2,238 products)
- Cytoskeletal Signaling(1,383 products)
- DNA Damage/DNA Repair(2,825 products)
- Endocrinology/Hormones(3,507 products)
- Enzyme(3,640 products)
- GPCR/G-Protein(8,333 products)
- Immunology and Inflammation(3,526 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(404 products)
- MAPK Signaling(1,202 products)
- Membrane Transporter/Ion Channel(2,790 products)
- Metabolism(9,448 products)
- Microbiology/Virology(6,981 products)
- Neuroscience(9,926 products)
- Other Inhibitors(37,926 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,400 products)
- Proteases/Proteasome(1,597 products)
- Stem Cell and Derivatives(831 products)
- Tyrosine Kinase/Adaptors(2,016 products)
- Ubiquitination(1,650 products)
Show 16 more subcategories
Found 66641 products of "Inhibitors"
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Stauprimide
CAS:<p>Stauprimide inhibits MYC by blocking NME2, reducing MYC transcription in ESCs.</p>Formula:C35H28N4O5Purity:98%Color and Shape:SolidMolecular weight:584.62GnRH-R antagonist 1
CAS:<p>Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.</p>Formula:C31H28F5N7O6SPurity:98%Color and Shape:SolidMolecular weight:721.65XO/COX/LOX-IN-1
<p>XO/COX/LOX-IN-1 targets XO/COX/LOX, used in research of inflammation, cancer, and metabolic disorders.</p>Formula:C24H20N4O2SColor and Shape:SolidMolecular weight:428.51Cilazapril HCl
CAS:<p>Cilazapril, also known as Ro 31 2848, is a potent ACE inhibitor used for hypertension.</p>Formula:C22H32ClN3O5Color and Shape:SolidMolecular weight:453.96Trypanothione synthetase-IN-4
<p>Trypanothione synthetase-IN-4, an L. infantum inhibitor, has potent anti-leishmanicidal properties (EC50: 0.6 μM).</p>Formula:C29H52INO2Color and Shape:SolidMolecular weight:573.63SCP1-IN-2
<p>SCP1-IN-2: potent, selective SCP1 inhibitor; induces REST degradation, hinders its activity, may study REST-driven glioblastoma growth.</p>Formula:C19H17F3N2O6S2Color and Shape:SolidMolecular weight:490.47AZD-4121 tert-butylammonium
CAS:<p>AZD-4121 tert-butylammonium is an oral cholesterol absorption inhibitor targeting NPC1L1 for the treatment of dyslipidaemia.</p>Formula:C40H50F2N4O7SColor and Shape:SolidMolecular weight:768.91LSD1-IN-21
<p>LSD1-IN-21: potent LSD1 inhibitor, crosses blood-brain barrier, IC50 of 0.956 μM; lowers TNF-α, anti-cancer, anti-inflammatory.</p>Formula:C24H25N5O2SColor and Shape:SolidMolecular weight:447.55ZIKV-IN-4
<p>ZIKV-IN-4 is a low cytotoxic, acid-stable anti-ZIKV agent with an EC50 value of 3.49 μM. ZIKV-IN-4 exhibited potent inhibition of ZIKV NS5 MTase.</p>Formula:C33H37NO4Color and Shape:SolidMolecular weight:511.65MI-1851
CAS:<p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>Formula:C34H53N15O6Color and Shape:SolidMolecular weight:767.88KY-02327 acetate
<p>KY-02327 acetate inhibits Dvl-CXXC5, stabilizes Wnt/β-catenin signaling, and enhances osteoblast differentiation.</p>Formula:C22H31N3O6Color and Shape:SolidMolecular weight:433.59(R)-HETE
CAS:<p>9(R)-HETE, 50% of racemic mix, activates RXRγ 1.5x at 300 nM; identified by HPLC comparison.</p>Formula:C20H32O3Color and Shape:SolidMolecular weight:320.47ADH-6
CAS:<p>ADH-6, a tripyridylamide, disrupts mutant p53 aggregates in cancer cells, reviving its function and inducing apoptosis.</p>Formula:C29H36N8O9Color and Shape:SolidMolecular weight:640.64CCR5 antagonist 1
CAS:<p>CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.</p>Formula:C39H46ClF2N5O3SPurity:98%Color and Shape:SolidMolecular weight:738.33LT-850-166
<p>LT-850-166 is a potent inhibitor of FLT3 and has shown efficacy in overcoming a wide range of FLT3 mutations.</p>Formula:C30H29Cl2N7OColor and Shape:SolidMolecular weight:574.5A 70450
CAS:<p>A 70450, an inhibitor of aspartyl proteinase, can be used as an antifungal agent and may have a role in HIV protease inhibition therapy.</p>Formula:C42H71ClN6O5Purity:98%Color and Shape:SolidMolecular weight:775.50P053
CAS:<p>P053: potent, selective CerS1 inhibitor, IC50 = 0.5µM, curbs muscle fat oxidation, affects body fat.</p>Formula:C18H21Cl2NO2Purity:98%Color and Shape:SolidMolecular weight:354.27L 689065
CAS:<p>L 689065 is a 5-lipoxygenase inhibitor.</p>Formula:C35H33ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:597.17AZ-PFKFB3-67 quarterhydrate
<p>AZ-PFKFB3-67 quarterhydrate inhibits PFKFB3 (IC50: 11 nM), PFKFB2 (159 nM), and PFKFB1 (1130 nM).</p>Formula:C26H27N5O4Color and Shape:SolidMolecular weight:460.01Belatacept
CAS:<p>Belatacept (BMS 224818), a T-cell costimulation inhibitor, targets CD80/86 for transplant immunosuppression.</p>Color and Shape:LiquidGSK-3β inhibitor 7
<p>GSK-3β inhibitor 7 is a GSK-3β inhibitor (IC50: 5.25 μM).</p>Formula:C27H23BrN4O2SColor and Shape:SolidMolecular weight:547.47BI-207524
CAS:<p>BI-207524 is a novel NS5B Thumb Pocket 1 Inhibitor with Improved Potency for the Potential Treatment of Chronic Hepatitis C Virus Infection.</p>Formula:C35H36ClN5O5Color and Shape:SolidMolecular weight:642.14Amdinocillin methylacetate
CAS:<p>Amdinocillin methylacetate is a Synthetic penicillin.</p>Formula:C18H27N3O4SColor and Shape:SolidMolecular weight:381.49BMS-986163
CAS:<p>BMS-986163, a prodrug, quickly becomes BMS-986169, a GluN2B inhibitor (Ki=4 nM, IC50=24 nM).</p>Formula:C23H28FN2O5PPurity:98%Color and Shape:SolidMolecular weight:462.45MA242 free base
CAS:<p>MA242 free base is a dual MDM2/NFAT1 inhibitor that triggers apoptosis in pancreatic cancer cells.</p>Formula:C24H20ClN3O3SColor and Shape:SolidMolecular weight:465.95Chitin synthase inhibitor 12
<p>Chitin synthase inhibitor 12: potent CHS blocker (IC50: 0.16 mM), broad-spectrum antifungal, effective against resistant strains. Useful in IFI research.</p>Formula:C23H21ClFN3O5Color and Shape:SolidMolecular weight:473.88HCV-IN-38
<p>Potent oral HCV inhibitor HCV-IN-38 has 15 nM EC50, 431 SI, high efficacy, and low toxicity.</p>Formula:C22H24ClF3N4O4Color and Shape:SolidMolecular weight:500.9GSK-2878175
CAS:<p>GSK-2878175, a NS5B inhibitor, is used potentially for the treatment of HCV infection.</p>Formula:C27H23BClFN2O6SPurity:98%Color and Shape:SolidMolecular weight:568.81Transthyretin-IN-1
<p>Transthyretin-IN-1 inhibits TTR fibril formation, aiding Alzheimer’s research.</p>Formula:C10H9Br2NO4Color and Shape:SolidMolecular weight:366.99Galidesivir
CAS:<p>Galidesivir (BCX4430) is an antiviral compound that inhibits viral RNA-dependent RNA polymerase (RdRp) activity and reduces lung infections in infected animals.</p>Formula:C11H15N5O3Purity:96.73% - 99.13%Color and Shape:SolidMolecular weight:265.27EF1502 free base
CAS:<p>EF1502 is a potent and selective GABA transporter inhibitor.</p>Formula:C22H26N2O2S2Purity:98%Color and Shape:SolidMolecular weight:414.58Aquayamycin
CAS:<p>Aquayamycin is an anthraquinone derivative and inhibitor of the enzyme tyrosine hydroxylase..</p>Formula:C25H26O10Color and Shape:SolidMolecular weight:486.47IRAK4-IN-11
<p>IRAK4-IN-11 (compound 6) is a potent inhibitor of IRAK4 with an IC 50 of 0.008 μM. IRAK4-IN-11 exhibits cell pIRAK4 potencies with an IC 50 of 0.19 μM [1].</p>Formula:C16H19N7OColor and Shape:SolidMolecular weight:325.37DSM705 hydrochloride
<p>DSM705 hydrochloride: potent antimalarial, pyrrole-based DHODH inhibitor effective against Plasmodium, non-toxic to mammalian DHODH.</p>Formula:C19H20ClF3N6OColor and Shape:SolidMolecular weight:440.85Norbinaltorphimine dihydrochloride
CAS:<p>Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.</p>Formula:C40H45Cl2N3O6Purity:98.17% - 99.88%Color and Shape:SolidMolecular weight:734.71Musettamycin
CAS:<p>Musettamycin triggers erythroid differentiation in blood cells, acts like anthracycline antibiotics, but only inhibits gram-positive bacteria.</p>Formula:C36H45NO14Color and Shape:SolidMolecular weight:715.74Tubulin polymerization-IN-33
<p>Tubulin-IN-33, an oxazoloisoindole, hinders microtubule assembly; effective against NCI cancer cells.</p>Formula:C27H28N2O6Color and Shape:SolidMolecular weight:476.525-HT7R antagonist 1
<p>5-HT7R antagonist 1 is a G protein-biased antagonist with Ki of 6.5 nM for 5-HT 7R.</p>Formula:C14H18Cl2N4Color and Shape:SolidMolecular weight:313.23MtTMPK-IN-1
<p>MtTMPK-IN-1 inhibits MtTMPK with 2.5 μM IC50, shows moderate anti-tuberculosis activity, and is low in cytotoxicity.</p>Formula:C22H24N4O3Color and Shape:SolidMolecular weight:392.459(S),10(S),13(S)-TriHOME
CAS:<p>9(S),10(S),13(S)-TriHOME is an oxylipin derived from linoleic acid. It has been detected in beer and in bronchoalveolar lavage fluid (BALF) from female smokers.</p>Formula:C18H34O5Color and Shape:SolidMolecular weight:330.46(S)-3-Hydroxy Midostaurin
CAS:<p>(S)-3-Hydroxy Midostaurin is a potent inhibitor of kinases(IC50 of <400 nM for 13 kinases (VEGFR-2, TRK-A, FLT3, et)).</p>Formula:C35H30N4O5Purity:98%Color and Shape:SolidMolecular weight:586.64BTK-IN-16
CAS:<p>BTK-IN-16 is a potential inhibitor of wild-type BTK and C481S mutants.BTK-IN-16 can be used to study various autoimmune diseases and cancers caused by BTK.</p>Formula:C15H14N4O2Purity:99.04%Color and Shape:SoildMolecular weight:282.3VEGFR-2-IN-12
<p>VEGFR-2-IN-12 (compound 6g), a 2-oxoquinoxalinyl-1,2,4-triazole, is a potent inhibitor of VEGFR-2 (IC50: 0.037 μM). VEGFR-2-IN-12 has anti-tumour effects.</p>Formula:C22H24N6O3SColor and Shape:SolidMolecular weight:452.53SLC4011540
<p>SLC4011540 is a potent and selective SphK1/2 dual inhibitor with Ki value of 120 nM and 90 nM respectively.</p>Formula:C24H23ClF3N7OSColor and Shape:SolidMolecular weight:550Tabimorelin hemifumarate
CAS:<p>orally active ghrelin receptor (GHS-R1a) agonist</p>Formula:C32H40N403C4H404Purity:98%Color and Shape:SolidMolecular weight:586.72CCR4 antagonist 2
CAS:<p>CCR4 antagonist 2 (Compound 31) is a novel potent, orally bioavailable small molecule antagonists of CC chemokine receptor 4 (CCR4) that inhibits Treg</p>Formula:C26H28Cl2N6OPurity:98%Color and Shape:SolidMolecular weight:511.45NITD-688
CAS:<p>NITD-688 is a pan-serotype inhibitor targeting the dengue virus NS4B protein, effective through oral administration.</p>Formula:C25H32N4O3S2Color and Shape:SolidMolecular weight:500.68MLKL-IN-1
<p>MLKL-IN-1 is a covalent inhibitor of MLKL with a Kd value of 50 μM.</p>Formula:C19H20N2O3Color and Shape:SolidMolecular weight:324.37MK2-IN-4
CAS:<p>MK2-IN-4 is a MAPKAPK2 (MK2) inhibitor (IC50: 45 nM). MK2-IN-4 can be used in cancer, inflammation and immunology studies.</p>Formula:C25H24N4O2Color and Shape:SolidMolecular weight:412.48ROPA
CAS:<p>ROPA, a potent PKCalpha and PKCgamma activator, promotes tumor growth through PKC-activation.</p>Formula:C28H32O6Purity:98%Color and Shape:SolidMolecular weight:464.55Ep vinyl quinidine
CAS:<p>3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.</p>Formula:C20H24N2O2Color and Shape:SolidMolecular weight:324.42Topoisomerase II inhibitor 5
<p>Topoisomerase II inhibitor 5 (Compound E24) is a DNAtopoisomerase II inhibitor with anticancer effects.</p>Formula:C26H27N5O4Color and Shape:SolidMolecular weight:473.52Revexepride
CAS:<p>Revexepride, a 5-HT4 agonist, may boost CYP3A4, used for treating GERD.</p>Formula:C21H32ClN3O4Purity:98%Color and Shape:SolidMolecular weight:425.95KRAS inhibitor-13
CAS:<p>KRAS inhibitor-13 blocks KRAS G12C (IC50: 0.883 μM) and p-ERK in some cancer cells; promising for pancreatic, colorectal, lung cancer research.</p>Formula:C25H19ClFN3O2SColor and Shape:SolidMolecular weight:479.95PF-06726304 acetate
CAS:<p>PF-06726304 acetate is a selective inhibitor of EZH2, with robust antitumor growth activity.</p>Formula:C24H25Cl2N3O5Purity:98%Color and Shape:SolidMolecular weight:506.38DMGF
CAS:<p>DMGF, a biflavonoid from Taxus, induces apoptosis, autophagy, and inhibits B16F10 cell motility and MMP-2 expression, hindering melanoma metastasis.</p>Formula:C32H22O10Color and Shape:SolidMolecular weight:566.51Antitumor agent-48
<p>Antitumor agent-48, a 2,3-dehydrosilybin derivative, exhibits cytotoxicity on MCF-7, NCI-H1299, HepG2, HT29 cells; IC50 ranging 8.06-16.51 µM.</p>Formula:C35H34N2O14Color and Shape:SolidMolecular weight:706.65AChE-IN-22
<p>AChE-IN-22 (10q) selectively inhibits AChE (IC50: 0.88 μM), less on BuChE (IC50: 10 μM), targets CAS and PAS, useful in Alzheimer's research.</p>Formula:C21H20N4O5SColor and Shape:SolidMolecular weight:440.47M3258
CAS:<p>LMP7-IN-1 may used in the research of inflammatory and autoimmune diseases, neurodegenerative diseases, proliferative diseases and cancer, is an inhibitor of</p>Formula:C17H20BNO5Purity:98%Color and Shape:SolidMolecular weight:329.16Trichostatin A S-isomer
CAS:<p>Trichostatin A S-isomer, a HDAC 1, 3, 4, 6, 10 inhibitor with IC50 ~20 nM, has wide-ranging epigenetic effects.</p>Formula:C17H22N2O3Purity:98%Color and Shape:SolidMolecular weight:302.37ONO-5334
CAS:<p>ONO-5334: selective cathepsin K inhibitor, potential for osteoporosis study; Ki: 0.10 nM (human), 0.049 nM (rabbit), 0.85 nM (rat).</p>Formula:C21H34N4O4SPurity:98.22% - 99.60%Color and Shape:SolidMolecular weight:438.58Ro 24-4383
CAS:<p>Ro 24-4383 is a carbamate-linked dual-action antibacterial agent.</p>Formula:C32H31FN8O10S2Purity:98%Color and Shape:SolidMolecular weight:770.76IL-17 modulator 1 disodium
CAS:<p>Potent, orally active IL-17 Modulator 1 (disodium) from patent WO 2020127685, used in psoriasis and arthritis research.</p>Formula:C28H37N6NaO6PColor and Shape:SolidMolecular weight:607.604Calphostin B
CAS:<p>Calphostins, PKC inhibitors from Cladosporium fungus, include A, B, C, D, I; C is most potent.</p>Formula:C37H34O11Color and Shape:SolidMolecular weight:654.66LPM4870108
<p>LPM4870108: Potent, oral pan-Trk inhibitor, selective over ALK, with anti-tumor effects. TrkC IC50=0.2nM, TrkA IC50=2.4nM.</p>Formula:C20H19FN6O3Color and Shape:SolidMolecular weight:410.4CCT369260
CAS:<p>CCT369260 (compound 1), an orally active inhibitor targeting B-cell lymphoma 6 (BCL6), demonstrates anti-tumor efficacy with an IC50 value of 520 nM [1].</p>Formula:C24H31ClF2N6O2Color and Shape:SolidMolecular weight:508.99DI-404
CAS:<p>DI-404: Potent DCN1-UBC12 inhibitor, selectivity blocks cullin 3 neddylation, Kd=6.9 nM.</p>Formula:C35H45ClN6O6SPurity:98%Color and Shape:SolidMolecular weight:713.29FTO-IN-5
CAS:<p>FTO-IN-5 is a potent, selective inhibitor targeting the fat mass obesity-associated protein (FTO).</p>Formula:C23H18Cl2N6O6Color and Shape:SolidMolecular weight:545.33E7090 succinate
CAS:<p>E7090 succinate inhibits FGFR1, FGFR2, and FGFR3 with IC50: 0.71, 0.50, 1.2 nM; less so FGFR4 at 120 nM.</p>Formula:C76H92N10O24Color and Shape:SolidMolecular weight:1529.60MIV-150
CAS:<p>MIV-150 is a nonnucleoside inhibitor of reverse transcriptase (NNRT). MIV-150 also blocking HIV-1 and HIV-2 infections (EC50<1 nM against HIV-1/HIV-2MN).</p>Formula:C19H17FN4O3Purity:98%Color and Shape:SolidMolecular weight:368.36HIF-1/2α-IN-1
<p>HIF-1/2α-IN-1, an orally active compound, functions as an inhibitor of HIF-2α.</p>Formula:C17H16N6O4Color and Shape:SolidMolecular weight:368.35BPTF-IN-BZ1
<p>BPTF-IN-BZ1 is a BPTF inhibitor that possesses a high potency with a Kd of 6.3 nM.</p>Formula:C13H15ClN4OColor and Shape:SolidMolecular weight:278.74CDK7/12-IN-1
CAS:<p>CDK7/12-IN-1 is a selective CDK7 (IC50: 3 nM) and CDK12 (IC50: 277 nM) inhibitor, effective against tumor growth.</p>Formula:C25H34N8OColor and Shape:SolidMolecular weight:462.59KRAS G12C inhibitor 56
CAS:<p>KRAS G12C inhibitor 56, a powerful inhibitor of SOS1 with an inhibitory concentration (IC50) of 1.6 nM, holds promise for use in cancer research.</p>Formula:C32H39N7O4SColor and Shape:SolidMolecular weight:617.76GSK2578999A
CAS:<p>GSK2578999A is a betulin derivative with antitumor activity.</p>Formula:C46H62ClNO7Purity:98%Color and Shape:SolidMolecular weight:776.44TRβ agonist 1
CAS:<p>TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.</p>Formula:C29H25FN2O8Color and Shape:SolidMolecular weight:548.52Xeruborbactam
CAS:<p>QPX7728 is an of ultra-broad-spectrum boronic acid beta-lactamase.</p>Formula:C10H8BFO4Purity:98%Color and Shape:SolidMolecular weight:221.98Murizatoclax
CAS:<p>AMG 397 is an oral MCL1 inhibitor .</p>Formula:C42H57ClN4O5SPurity:98%Color and Shape:SolidMolecular weight:765.44Balanol
CAS:<p>Balanol is an ATP-competitive Protein Kinase C and Protein Kinase A inhibitor.</p>Formula:C28H26N2O10Color and Shape:SolidMolecular weight:550.51GGTI298
CAS:<p>GGTI298 is a potent GGTase I inhibitor; IC50 3μM for Rap1A, >20μM for Ha-Ras.</p>Formula:C27H33N3O3SPurity:98%Color and Shape:SolidMolecular weight:479.63FGFR1 inhibitor-6
<p>FGFR1 inhibitor-6, IC50: 16.31 nM, blocks cell cycle at pro-G1/G2/M and induces apoptosis.</p>Formula:C27H19N5O4S2Color and Shape:SolidMolecular weight:541.6KRAS G12D inhibitor 16
CAS:<p>KRAS G12D inhibitor 16 targets KRAS G12D with IC50 of 0.7 nM and mutant form at 0.35 μM, useful in various cancer studies.</p>Formula:C32H39IN6O3Color and Shape:SolidMolecular weight:682.59Carbonic anhydrase inhibitor 9
<p>Carbonic anhydrase inhibitor 9 targets hCA II and IX with Ki of 56.4 and 56.9 nM respectively; shows antiproliferative activity.</p>Formula:C22H20BrN5O4SColor and Shape:SolidMolecular weight:530.39MDL-27088
CAS:<p>MDL-27088 is an angiotensin-covering enzyme inhibitor.</p>Formula:C25H28N2O5Color and Shape:SolidMolecular weight:436.50Ici D1542
CAS:<p>Ici D1542: potent TXS inhibitor & TXA2 receptor antagonist, effective thromboxane blocker in vitro.</p>Formula:C25H30N2O7Purity:98%Color and Shape:SolidMolecular weight:470.51GSK-1264
CAS:<p>GSK-1264: allosteric HIV integrase inhibitor, halts viral replication & abnormal protein multimerization.</p>Formula:C26H28FNO5Color and Shape:SolidMolecular weight:453.5Alentemol hydrobromide
CAS:<p>Alentemol hydrobromide is a Dopamine agonist.</p>Formula:C19H26BrNOPurity:98%Color and Shape:SolidMolecular weight:364.32HDAC2-IN-1
<p>HDAC2-IN-1 is an oral HDAC2 inhibitor (IC50: 0.5 μM), crosses the blood-brain barrier, and inhibits HDAC1 and HDAC8.</p>Formula:C22H23ClN4OSColor and Shape:SolidMolecular weight:426.96Purine phosphoribosyltransferase-IN-1
<p>Compound (S,R)-48 inhibits Pf, Pv, & Tbr PRT with Ki of 50, 20, 2 nM.</p>Formula:C11H15N5Na4O10P2Color and Shape:SolidMolecular weight:531.17RN941
CAS:<p>RN941 is a highly potent Bruton's tyrosine kinase (BTK) inhibitor.</p>Formula:C34H34FN7O5Purity:98%Color and Shape:SolidMolecular weight:639.68DNDI-8219
CAS:<p>DNDI-8219 is an antitubercular agent. It has potent antileishmanial effects.</p>Formula:C13H10F3N3O5Color and Shape:SolidMolecular weight:345.23L 668750
CAS:<p>L 668750 is an inhibitor of platelet-activating factor.</p>Formula:C25H34O9SPurity:98%Color and Shape:SolidMolecular weight:510.6Acyline
CAS:<p>Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.</p>Formula:C80H102ClN15O14Color and Shape:SolidMolecular weight:1533.21PHGDH-IN-2
<p>PHGDH-IN-2: potent PHGDH inhibitor, IC50=5.2μM; hinders PHGDH cancer cell growth & serine synthesis in MDA-MB-468.</p>Formula:C22H20N4O3SColor and Shape:SolidMolecular weight:420.48Lysyllysyllysine
CAS:<p>Lysyllysyllysine is a cationic moiety. It may be used in the construction of gene delivery vectors and DNA nanoparticles.</p>Formula:C18H38N6O4Purity:98%Color and Shape:SolidMolecular weight:402.53KNT-127
CAS:<p>KNT-127 is an agonist of δ-Opioid receptor.</p>Formula:C24H24N2O2Purity:98%Color and Shape:SolidMolecular weight:372.46ML-SI1
CAS:<p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>Formula:C23H26Cl2N2O3Color and Shape:SolidMolecular weight:449.37(±)-HIP-B
CAS:<p>(±)-HIP-B is an excitatory amino acid transporter blocker.</p>Formula:C6H8N2O4Purity:98%Color and Shape:SolidMolecular weight:172.14GSK3368715
CAS:<p>GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50s</p>Formula:C20H38N4O2Purity:98%Color and Shape:SolidMolecular weight:366.54MRTX-EX185
<p>MRTX-EX185 inhibits GDP-KRAS/G12D; IC50=90 nM on G12D. It also binds GDP-HRAS.</p>Formula:C33H33FN6O2Color and Shape:SolidMolecular weight:564.65

