Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,846 products)
- Apoptosis(6,332 products)
- Cell Cycle/Checkpoint(4,887 products)
- Chromatin/Epigenetics(2,615 products)
- Cytoskeletal Signaling(1,577 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,753 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,025 products)
- Immunology and Inflammation(3,926 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,258 products)
- Membrane Transporter/Ion Channel(3,160 products)
- Metabolism(10,133 products)
- Microbiology/Virology(7,625 products)
- Neuroscience(10,540 products)
- Other Inhibitors(35,857 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(731 products)
- Tyrosine Kinase/Adaptors(1,991 products)
- Ubiquitination(1,727 products)
Show 16 more subcategories
Found 66513 products of "Inhibitors"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
A 70450
CAS:A 70450, an inhibitor of aspartyl proteinase, can be used as an antifungal agent and may have a role in HIV protease inhibition therapy.Formula:C42H71ClN6O5Purity:98%Color and Shape:SolidMolecular weight:775.50AChE/GSK-3β-IN-1
CAS:AChE/GSK-3β-IN-1 is a potent dual AChE/GSK-3β inhibitor that crosses the blood-brain barrier and acts on hAChE (IC50: 1.2 nM), hBChE (IC50: 149.8 nM) and hGSK-Formula:C31H35N7O3SColor and Shape:SolidMolecular weight:585.72E 5090
CAS:E5090 is a novel orally active inhibitor of IL-1 generation. It also has anti-inflammatory properties.Formula:C19H20O5Purity:98%Color and Shape:SolidMolecular weight:328.36CI 922
CAS:CI 922 is an anaphylaxis mediator release inhibitor. It inhibits the activation of human neutrophils.Formula:C26H30N10O6Color and Shape:SolidMolecular weight:578.58PF-07054894
CAS:PF-07054894: potent CCR6 antagonist, targets GPCR, for inflammatory bowel disease research.Formula:C24H30N6O4Color and Shape:SolidMolecular weight:466.53(R)-ONO-2952
(R)-ONO-2952 is the R-enantiomer of ONO-2952. ONO-2952 is selective and oral effective TSPO antagonist, with Kis of 0.330-9.30 nM inhibiting rat and human TSPO.Formula:C22H20ClFN2O2Color and Shape:SolidMolecular weight:398.86Protease-Activated Receptor-1 antagonist 2
Selective, orally active PAR-1 antagonist with an IC50 of 7 nM, potential for cardiovascular disease studies.Color and Shape:SolidATR-IN-17
CAS:ATR-IN-17 is a potent inhibitor of ATR kinase with good anti-cancer effects in LoVo cells (IC50: 1 nM).Formula:C22H28N6O2SColor and Shape:SolidMolecular weight:440.56UAWJ9-36-1
CAS:UAWJ9-36-1: potent broad-spectrum coronavirus Protease inhibitor; IC50 = 51 nM.Formula:C23H29N3O5Color and Shape:SolidMolecular weight:427.495-HT7R antagonist 1
5-HT7R antagonist 1 is a G protein-biased antagonist with Ki of 6.5 nM for 5-HT 7R.Formula:C14H18Cl2N4Color and Shape:SolidMolecular weight:313.23PAD-IN-2
CAS:PAD-IN-2, potent PAD4 inhibitor, IC50 <1 μM; targets autoimmune/cancer disorders.Formula:C27H28ClN5O2Color and Shape:SolidMolecular weight:490HPK1-IN-3
HPK1-IN-3: Selective HPK1 inhibitor, ATP-competitive, IC50=0.25nM; boosts IL-2 in PBMCs, EC50=108nM.Formula:C23H22F4N6O2Color and Shape:SolidMolecular weight:490.45Carbonic anhydrase inhibitor 5
Potent hCA inhibitor: targets hCA II, IX & XII with IC50s of 42.9, 47.6, & 6.7 nM respectively.Formula:C24H20ClN3O3SColor and Shape:SolidMolecular weight:465.95Flusoxolol
CAS:Flusoxolol is a beta-adrenoceptor partial agonist.Formula:C22H30FNO4Color and Shape:SolidMolecular weight:391.48B-3852
CAS:B-3852 is a Bradykinin inhibitor.Formula:C55H74F3N15O11Color and Shape:SolidMolecular weight:1178.27GID4 Ligand 2
GID4 Ligand 2 (compound 67) is a selective binder for GID4 with IC50 of 18.9 μM and Kd of 17 μM. GID4 Ligand 2 can be used for the synthesis of PROTACs [1].Formula:C15H16N2Color and Shape:SolidMolecular weight:224.3DNA crosslinker 4 dihydrochloride
CAS:DNA Crosslinker 4 binds DNA's minor groove, inhibits NCI-H460, A2780, MCF-7 cancer cells, and is used in cancer research.Formula:C16H24Cl2N8OColor and Shape:SolidMolecular weight:415.32BAY-7598
CAS:BAY-7598 is a potent, selective, and orally bioavailable MMP12 inhibitor (IC50s: 0.085, 0.67, and 1.1 nM for human/murine/rat MMP12).Formula:C28H31N3O6Purity:98%Color and Shape:SolidMolecular weight:505.56Pyridoxatin
CAS:Pyridoxatin: fungal metabolite; blocks TBARS production, prevents AAPH-induced hemolysis, and acts against C. albicans.Formula:C15H21NO3Color and Shape:SolidMolecular weight:263.33Amdinocillin methylacetate
CAS:Amdinocillin methylacetate is a Synthetic penicillin.Formula:C18H27N3O4SColor and Shape:SolidMolecular weight:381.49Everafenib
Everafenib: potent BRAF inhibitor, crosses blood-brain barrier, hinders MAPK, effective on V600EBRAF cells, outperforms other drugs in trials.Formula:C20H23ClFN5O2S2Color and Shape:SolidMolecular weight:484.01KRAS G12C inhibitor 20
CAS:KRAS G12C inhibitor 20 is a KRAS G12C inhibitor.Formula:C33H37ClFN7O3Color and Shape:SolidMolecular weight:634.14Teslexivir
CAS:Teslexivir is a topical antiviral agent that is an effective and selective inhibitor of the interaction between two essential viral proteins, E1 and E2.Formula:C35H36BrN3O4Purity:98%Color and Shape:SolidMolecular weight:642.58SphK2-IN-1
CAS:SphK2-IN-1 is an SphK2 inhibitor with an IC50 value of 0.359 μM. SphK2-IN-1 can be used to study cancer, inflammation, neurological and cardiovascular diseases.Formula:C23H22ClF3N8OColor and Shape:SolidMolecular weight:518.92IRAK4-IN-15
CAS:IRAK4-IN-15: selective IRAK4 inhibitor, IC50 0.002 μM, good PK, low clearance, synergizes with Acalabrutinib in MyD88/CD79 mutant ABC-DLBCL.Formula:C25H29FN10Color and Shape:SolidMolecular weight:488.56XR8-89
CAS:XR8-89, a potent PLpro inhibitor (IC50=0.1μM), blocks SARS-CoV-2 replication; useful for research.Formula:C29H36N4O2SColor and Shape:SolidMolecular weight:504.69Anticancer agent 53
CAS:Anticancer agent 53 exhibits potent in vitro cytotoxicity, triggers apoptosis, halts S/G2/M cycle, and has antitumor effects without toxicity.Formula:C31H25FN4O6SColor and Shape:SolidMolecular weight:600.62Complex III-IN-2
Complex III-IN-2 inhibits complex III, with antifungal EC50: 29.31 mg/L vs R. solani, 29.98 mg/L vs S. sclerotiorum.Formula:C15H21ClN2O2SColor and Shape:SolidMolecular weight:328.86KDOAM-25 trihydrochloride
KDOAM-25 trihydrochloride selectively inhibits KDM5 enzymes, boosts H3K4 methylation, and suppresses MM1S cell growth.Formula:C15H28Cl3N5O2Color and Shape:SolidMolecular weight:416.77Cyclic-di-GMP sodium
c-di-GMP sodium: STING activator, regulates bacteria biofilm, motility, virulence.Formula:C20H24N10NaO14P2Color and Shape:SolidMolecular weight:713.08464Haspin-IN-1
Haspin-IN-1 blocks haspin (IC50: 119 nM) and inhibits CLK1, DYRK1A, CDK9 with potential as an anticancer drug.Formula:C12H8N4O2SColor and Shape:SolidMolecular weight:272.28Dinordrin I diacetate
CAS:Dinordrin I diacetate is an implantation inhibitor and hormone.Formula:C25H32O4Purity:98%Color and Shape:SolidMolecular weight:396.52HMG499
CAS:HMG499 inhibits HMG-CoA reductase (IC50: 0.41μM), reduces statin-induced HMGCR, lowers cholesterol, and lessens atherosclerosis.Formula:C33H54O3Purity:98%Color and Shape:SolidMolecular weight:498.78Omesdafexor
CAS:Omesdafexor is an FXR agonist that can be used to study diseases caused by liver disease or metabolic inflammation.Formula:C34H43N3O3Color and Shape:SolidMolecular weight:541.72OUN58101
CAS:OUN58101, also MDK-8101/BI-D, is an RSV L-protein inhibitor with no formal name, first reported in patent WO 2005042530.Formula:C32H36N6O6Color and Shape:SolidMolecular weight:600.66Topoisomerase II inhibitor 6
Topoisomerase II inhibitor 6, a potent tryptanthrin derivative, blocks G2 phase in CCRF-CEM cells, induces DNA breaks, and may be used for cancer research.Formula:C19H18N4O2Color and Shape:SolidMolecular weight:334.37Bcl-2-IN-8
Bcl-2-IN-8: potent, hinders cell growth/migration, induces apoptosis, promising in triple-negative breast cancer research.Formula:C36H44O6Color and Shape:SolidMolecular weight:572.73BMS-751324
CAS:BMS-751324: p38α MAPK inhibitor with carbamyl-methyl, esters, phosphate from HPA. Reduces rat arthritis swelling and TNFα.Formula:C32H35N6O10PColor and Shape:SolidMolecular weight:694.63Colistin adjuvant-2
Colistin adjuvant-2 is a compound that acts as a potentiation agent for colistin, effectively enhancing its activity against Gram-negative bacteria [1].Formula:C14H7Cl2F3N2OColor and Shape:SolidMolecular weight:347.12Homodestcardin
CAS:Homodestcardin: cyclic depsipeptide from T. roseum with immunosuppressant properties; inhibits mouse T cell proliferation.Formula:C32H55N5O7Color and Shape:SolidMolecular weight:621.81KPH2f
CAS:KPH2f: dual URAT1/GLUT9 inhibitor, orally active, IC50: 0.24μM (URAT1), 9.37μM (GLUT9), minimal OAT1/ABCG2 impact.Formula:C24H16N3NaO2SColor and Shape:SolidMolecular weight:433.46KIRA9
KIRA9 inhibits IRE1 with a 4.8 μM IC50, blocking ER-stress-induced mRNA decay and apoptosis by fully binding IRE1's ATP site.Formula:C27H27F3N6O3SColor and Shape:SolidMolecular weight:572.6Pociredir
CAS:Pociredir (FTX-6058), a potent EED inhibitor (KD=0.163 nM), may help in SCD research.Formula:C22H18FN5O2Color and Shape:SolidMolecular weight:403.41DYRKs-IN-1
CAS:DYRKs-IN-1 has antitumor activity.
Formula:C30H30ClN7O4Purity:98%Color and Shape:SolidMolecular weight:588.06(S)-MALT1-IN-5
CAS:(S)-MALT1-IN-5: Potent MALT1 protease inhibitor, may help in abnormal T/B-cell signalling and MALT1-linked diseases.Formula:C17H17ClF2N6O3Color and Shape:SolidMolecular weight:426.80Pexacerfont
CAS:Pexacerfont (BMS-562086) is a selective antagonist of the corticotropin-releasing factor receptor (IC50: 6.1±0.6 nM for the human CRF1 receptor).Formula:C18H24N6OPurity:99.77%Color and Shape:SolidMolecular weight:340.42CTX-712
CAS:CTX-712 is a potent inhibitor of cdc2-like kinase ( CLK ). CTX-712 inhibits inhibits cancer survival and cancer cell growth.Formula:C19H17FN8O2Color and Shape:SolidMolecular weight:408.39LY3325656
CAS:LY3325656, a GPR142 agonist with anti-diabetic properties, progresses to phase 1 trials for Type 2 diabetes.Formula:C21H23F3N6O2Color and Shape:SolidMolecular weight:448.44BRD-9526
CAS:BRD-9526 is a potent and selective inhibitor of Sonic Hedgehog (Shh).Formula:C26H31Cl2N3O6SPurity:98%Color and Shape:SolidMolecular weight:584.51KT5926
CAS:KT5926 selectively inhibits myosin light chain kinase and NGF-dependent neurite growth; it's a K-252a analogue.Formula:C30H27N3O6Purity:98%Color and Shape:SolidMolecular weight:525.55microRNA-21-IN-1
CAS:microRNA-21-IN-1: microRNA inhibitor, curbs HeLa/HCT-116 growth (IC50: 5.5/2.8 μM), induces HeLa apoptosis, elevates PTEN/EGR1/SLIT2, for cancer research.Formula:C30H37FN6O3Color and Shape:SolidMolecular weight:548.65AMG-369
CAS:AMG-369 (AMG 247) is an S1P1/S1P5 dual agonist that delays the development of experimental autoimmune encephalomyelitis in rats.Formula:C26H22FN3O2SPurity:98.04% - 98.92%Color and Shape:SolidMolecular weight:459.547(Z),11(Z)-Nonacosadiene
CAS:7(Z),11(Z)-Nonacosadiene, a female fly pheromone, spurs male courtship; it's a C29 diene made by a female-specific elongase.Formula:C29H56Color and Shape:SolidMolecular weight:404.75Carumonam Sodium
CAS:Carumonam Sodium is a monobactam, penicillin-binding protein inhibitor. It is used as antibacterials.Formula:C12H12N6Na2O10S2Purity:98%Color and Shape:SolidMolecular weight:510.37Py-MPB-amino-C3-PBD
CAS:Py-MPB-amino-C3-PBD is a cytotoxic agent comprised non-alkylating group,with antimicrobial activity.Formula:C41H44N8O6Purity:98%Color and Shape:SolidMolecular weight:744.84MEIS-IN-1
CAS:MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.Formula:C24H21F3N2O4Color and Shape:SolidMolecular weight:458.43HER2-IN-10
HER2-IN-10 is a psoralen derivative that induces apoptosis. HER2-IN-10 shows anti-breast cancer activity and light-activated cytotoxicity [1].Formula:C15H13NO5Color and Shape:SolidMolecular weight:287.27PDE4B-IN-3
PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.Formula:C30H35N3O4S2Color and Shape:SolidMolecular weight:565.75Tamitinol
CAS:Tamitinol is a neurotropic drug. It has been found to help symptoms of obsessive rumination in conjunction with maprotiline.Formula:C12H20N2OSPurity:98%Color and Shape:SolidMolecular weight:240.37AK-295
CAS:AK 295, also known as CX 295, is a dipeptide inhibitor of alpha-ketoamide calpain.Formula:C26H40N4O6Color and Shape:SolidMolecular weight:504.62SOS1-IN-6
CAS:SOS1-IN-6 (compound 33-P1) is a potent inhibitor of SOS1, acting on SOS1-G12D (IC50: 14.9 nM) and SOS1-G12V (IC50: 73.3 nM).Formula:C26H28F3N3O2Color and Shape:SolidMolecular weight:471.51FAK-IN-4
FAK-IN-4 (Compound 7d) has anticancer activities that can induce cell apoptosis. FAK-IN-4 is potential inhibitor of FAK [1].Formula:C20H22N4OColor and Shape:SolidMolecular weight:334.41Cav 3.2 inhibitor 2
Cav 3.2 inhibitor 2 blocks T-type Ca2+ channels (IC50=0.09339 μM) and reduces mouse somatic/visceral pain. Used for intractable pain studies.Formula:C32H37F2N3OColor and Shape:SolidMolecular weight:517.65HIV-1 inhibitor-17
HIV-1 inhibitor-18 blocks HIV-1 capsid, acts on NL4-3 strain (EC50: 2.57 μM), has low cytotoxicity (MT-4 CC50: >8.55).Formula:C32H32N4O5SColor and Shape:SolidMolecular weight:584.69VEGFR-2-IN-14
VEGFR-2-IN-14 (Compound 5) is a potent inhibitor of VEGFR-2, which inhibits the growth of HepG2 cells in the Pre-G1 phase and induces apoptosis.Formula:C24H23N3O3SColor and Shape:SolidMolecular weight:433.52Alkyne-probe 1
Alkyne-probe 1 is usually used as an Alkyne-labeled fluorescent or chemical probe.Formula:C14H23N5O2Purity:98%Color and Shape:SolidMolecular weight:293.36Lasonolide A
CAS:Lasonolide A, an anticancer compound from Forcepia sponge, shows nanomolar growth inhibition and unique cytotoxicity in the NCI 60-cell-line screen.Formula:C41H60O9Color and Shape:SolidMolecular weight:696.91Ro-51
CAS:dual P2X3 and P2X2/3 antagonistFormula:C17H23IN4O4Purity:98%Color and Shape:SolidMolecular weight:474.29CPX-351
CAS:CPX-351 (Vyxeos) is a liposomal encapsulant of cytarabine and Zoerythromycin with potential antitumor activity.Formula:C36H42N4O15Purity:98.95% - 99.763%Color and Shape:SolidMolecular weight:770.74P-gp inhibitor 2
CAS:Potent P-gp inhibitor 2 reverses Doxorubicin resistance in colorectal carcinoma cells with IC50 of 0.22 µM.Formula:C29H26N2O6Color and Shape:SolidMolecular weight:498.53Menin-MLL inhibitor 26
CAS:Menin-MLL inhibitor 26: Active reference, inhibits cell growth, used in leukemia research.Formula:C27H29F3N6O3SColor and Shape:SolidMolecular weight:574.62WQ3810 TFA
WQ3810 TFA is an orally available fluoroquinolone with antimicrobial activity against Mycobacterium tuberculosis and inhibits the DNA rotamase activity ofFormula:C24H23F6N5O5Purity:99.52%Color and Shape:SoildMolecular weight:575.46EB-0156
EB-0156: potent ER α-glucosidase inhibitor, IC50 of 0.0479/ <0.001 μM, N-substituted valerian, broad-spectrum antiviral potential.Formula:C21H32N6O7Color and Shape:SolidMolecular weight:480.51Quinagolide Free Base
CAS:Quinagolide Free Base is a non-ergot dopamine D(2)-agonist.Formula:C20H33N3O3SColor and Shape:SolidMolecular weight:395.56p38-α MAPK-IN-5
CAS:p38-α MAPK-IN-5: potent p38α inhibitor, IC50s: 0.1 nM (α), 0.2 nM (β), 944 nM (γ), 4100 nM (δ); anti-inflammatory, promising for asthma/COPD research.Formula:C37H49N11O2Color and Shape:SolidMolecular weight:679.86Verrucarin A
CAS:Verrucarin A, a mycotoxin from Myrothecium verrucaria, inhibits protein synthesis, leukemia growth, and triggers apoptosis.Formula:C27H34O9Color and Shape:SolidMolecular weight:502.55ART615
ART615 is a related isomer of ART558. ART615 inhibits Polθ by <10% at 12 μM and is able to act as a control for ART558 (IC50:7.9 nM).Formula:C21H21F3N4O2Color and Shape:SolidMolecular weight:418.41RMI-18341
CAS:RMI-18341 is a Testosterone 5 alpha reductase inhibitor.Formula:C22H34N2O2Color and Shape:SolidMolecular weight:358.52KDOAM-25 citrate
CAS:KDOAM-25 citrate inhibits KDM5A/B/C/D (IC50: 71, 19, 69, 69 nM); boosts H3K4 methylation, hinders MM1S cell growth. [1]Formula:C21H33N5O9Purity:98%Color and Shape:SolidMolecular weight:499.51Anticancer agent 80
Anticancer agent 80 (Compound 3c) is an anticancer agent that exhibits a significant dark toxic effect on T47-D (IC50: 10.14 μM).Formula:C19H12BrNO5Color and Shape:SolidMolecular weight:414.21AFM-30a hydrochloride
AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.Formula:C24H28ClFN6O3Color and Shape:SolidMolecular weight:502.97LY593093
CAS:LY593093 is a selective partial orthosteric agonist of M1 muscarinic acetylcholine receptor.Formula:C32H30FN3O2Purity:98%Color and Shape:SolidMolecular weight:507.6Samuraciclib
CAS:Samuraciclib (CT7001) is an oral CDK7 inhibitor with 41 nM IC50, notable for its high selectivity and potency against breast cancer cells.Formula:C22H30N6OColor and Shape:SolidMolecular weight:394.51(RS)-AMPA hydrobromide
CAS:AMPAR agonistFormula:C7H11BrN2O4Purity:98%Color and Shape:SolidMolecular weight:267.08SG3199
CAS:SG3199, a PBD dimer, binds DNA's minor groove, forms covalent cross-links, and is cytotoxic to various human cancer cells.Formula:C33H36N4O6Color and Shape:SolidMolecular weight:584.66Revamilast
CAS:Revamilast, also known as GRC4039, is a phosphodiesterase IV inhibitor for potentially treating of asthma and rheumatoid arthritisFormula:C18H9Cl2F2N3O4Color and Shape:SolidMolecular weight:440.18MK-6913
CAS:MK-6913 is a potent and selective agonist of estrogen receptor β.Formula:C25H27N3O2Purity:98%Color and Shape:SolidMolecular weight:401.5MK-8825
CAS:MK-8825 is a CGRP receptor antagonist.Formula:C31H30F2N6O3Color and Shape:SolidMolecular weight:572.61SHR902275
CAS:SHR902275: potent RAF inhibitor, hits RAS mutations, oral use. cRAF IC50=1.6 nM, bRAFwt IC50=10 nM, bRAFV600E IC50=5.7 nM, hinders cell growth.Formula:C26H23F3N4O4Color and Shape:SolidMolecular weight:512.4820-HEDE
CAS:20-HEDE (WIT 002) is a 20-hydroxyeicosatetraenoic acid (20-HETE) antagonist.Formula:C20H36O3Purity:98%Color and Shape:SolidMolecular weight:324.50KRAS inhibitor-8
CAS:KRAS inhibitor-8 is a potent KRAS G12C inhibitor.Formula:C26H24ClF4N5O3Purity:98%Color and Shape:SolidMolecular weight:565.95Homopteroic Acid
CAS:Homopteroic Acid, a precursor to Homofolic Acid, inhibits L1210 mouse leukemia growth by targeting folate uptake.Formula:C15H14N6O3Color and Shape:SolidMolecular weight:326.31Glycotriosyl glutamine
CAS:Glycotriosyl glutamine is a nephritogenoside analog.Formula:C23H40N2O18Color and Shape:SolidMolecular weight:632.57EF1502 free base
CAS:EF1502 is a potent and selective GABA transporter inhibitor.Formula:C22H26N2O2S2Purity:98%Color and Shape:SolidMolecular weight:414.58STA-1474
CAS:STA-1474, a soluble prodrug of ganetespib (STA-9090), becomes a strong HSP90 inhibitor effective against canine tumors.Formula:C20H21N4O6PColor and Shape:SolidMolecular weight:444.38DMP-728 free base
CAS:DMP-728 free base is a highly potent and selective GPIIbDIIa antagonistFormula:C25H36N8O7Color and Shape:SolidMolecular weight:560.60Odiparcil
CAS:Odiparcil is an orally active beta-d-thioxyloside analog.Formula:C15H16O6SPurity:98%Color and Shape:SolidMolecular weight:324.35EGFR/HER2-IN-5
EGFR/HER2-IN-5: Irreversible, oral dual EGFR inhibitor, IC50 0.6 nM, targets L858R/T790M mutations, anti-tumor in vivo for lung cancer study.Color and Shape:SolidD4R antagonist-1
Potent, selective D4R antagonist; IC50 = 6.87 µM; potential in Parkinson’s disease research.Formula:C21H25F2NO2Color and Shape:SolidMolecular weight:361.43CCW 28-3
CAS:CCW 28-3 is a novel potent covalent BRD4 degrader, degrading BRD4 in a proteasome- and RNF4-dependent manner without inhibiting RNF4 autoubiquitination activityFormula:C44H42Cl2N6O4SColor and Shape:SolidMolecular weight:821.81
