Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,523 products)
- Apoptosis(5,792 products)
- Cell Cycle/Checkpoint(4,449 products)
- Chromatin/Epigenetics(2,238 products)
- Cytoskeletal Signaling(1,383 products)
- DNA Damage/DNA Repair(2,825 products)
- Endocrinology/Hormones(3,507 products)
- Enzyme(3,640 products)
- GPCR/G-Protein(8,333 products)
- Immunology and Inflammation(3,526 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(404 products)
- MAPK Signaling(1,202 products)
- Membrane Transporter/Ion Channel(2,790 products)
- Metabolism(9,448 products)
- Microbiology/Virology(6,981 products)
- Neuroscience(9,926 products)
- Other Inhibitors(37,926 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,400 products)
- Proteases/Proteasome(1,597 products)
- Stem Cell and Derivatives(831 products)
- Tyrosine Kinase/Adaptors(2,016 products)
- Ubiquitination(1,650 products)
Show 16 more subcategories
Found 66641 products of "Inhibitors"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
COX-2-IN-29
<p>COX-2-IN-29 is a selective inhibitor of orally active COX-2 (IC50: 0.005 μM).</p>Formula:C22H23FN2O6S2Color and Shape:SolidMolecular weight:494.56Diguanosine 5′-triphosphate lithium
<p>Diguanosine 5′-triphosphate (Gp3G) lithium is a dinucleoside triphosphate and a virus-specific oligonucleotide.Diguanosine 5′-triphosphate lithium is required</p>Formula:C20H27N10O18P3·xLiColor and Shape:SolidBACE1-IN-4
CAS:<p>BACE1-IN-4 is a potent and highly selective BACE1 inhibitor (IC50: 3.8 nM; Ki: 1.9 nM), more selective at BACE1 over BACE2.</p>Formula:C21H23F2N5O4S2Purity:98%Color and Shape:SolidMolecular weight:511.57Cortistatin A
CAS:<p>Cortistatin A is a potent and selective mediator-associated kinase CDK8 and its paralogue CDK19 inhibitor.</p>Formula:C30H36N2O3Purity:98%Color and Shape:SolidMolecular weight:472.62Lumirubin
CAS:<p>Lumirubin is a water-soluble photoproduct of bilirubin formed in vivo during phototherapy.</p>Formula:C33H36N4O6Color and Shape:SolidMolecular weight:584.66AMPK Activator SC4
CAS:<p>SC4 is a potent, direct AMPK activator. SC4 preferentially activates α2 complexes and stimulates skeletal muscle glucose uptake.</p>Formula:C26H18ClN3O4Color and Shape:SolidMolecular weight:471.89PRN694
CAS:<p>PRN694 is a potent, irreversible ITK/RLK inhibitor with IC50s: 0.3/1.4 nM; offers lasting effector cell suppression.</p>Formula:C28H35F2N5O2SPurity:98%Color and Shape:SolidMolecular weight:543.67Inupadenant HCl
CAS:<p>Inupadenant (EOS-850) is a selective A2a receptor antagonist, targeting immunosuppression in tumors.</p>Formula:C25H27ClF2N8O4S2Color and Shape:SolidMolecular weight:641.11MsbA-IN-1
<p>MsbA-IN-1: Potent MsbA inhibitor (IC50: 4 nM), anti-E. coli (MIC: 79 μM), penetrates Gram-negative bacteria.</p>Formula:C23H18Cl2FNO3Color and Shape:SolidMolecular weight:446.3Myxothiazol
CAS:<p>Myxothiazol blocks mitochondrial complex III and triggers SESN2, a gene important for stress response.</p>Formula:C25H33N3O3S2Color and Shape:SolidMolecular weight:487.68sEH inhibitor-2
<p>SEH inhibitor-2 is an orally active sEH blocker (IC50=0.9 nM) with predicted 71.2-88.4% absorption, potentially aiding cardiovascular health.</p>Formula:C23H18N4O3Color and Shape:SolidMolecular weight:398.41Cav 2.2/3.2 blocker 1
<p>Compound 9e is a Cav 2.2/3.2 blocker; IC50: 1.22 μM & 80 μM, respectively; penetrates CNS.</p>Formula:C28H30N2O3Color and Shape:SolidMolecular weight:442.55AAK1-IN-2 TFA
<p>AAK1-IN-2 TFA (compound (S)-31) is a selective and potent AAK1 inhibitor (IC50: 5.8 nM) that can cross the blood-brain barrier.</p>Formula:C24H22F6N4O4Color and Shape:SolidMolecular weight:544.45L 739749
CAS:<p>L 739749 is a CAAX peptidomimetic. It is also an inhibitor of farnesyl-protein transferase.</p>Formula:C24H41N3O6S2Purity:98%Color and Shape:SolidMolecular weight:531.73HCV-IN-7
CAS:<p>HCV-IN-7: potent oral HCV NS5A inhibitor, pan-genotypic, IC50s 3-47 pM, good pharmacokinetics, favorable liver uptake.</p>Formula:C40H48N8O6SPurity:98%Color and Shape:SolidMolecular weight:768.92CDK9-IN-13
<p>CDK9-IN-13 is a potent and selective CDK inhibitor (IC50<3 nM). CDK9-IN-13 has a very short half-life in rodents.</p>Formula:C27H35N5O2Color and Shape:SolidMolecular weight:461.6trans-RdRP-IN-5
<p>Trans-RdRP-IN-5 is a potent inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), with applications in influenza virus research.</p>Formula:C23H21N3O5Color and Shape:SolidMolecular weight:419.43JNJ-1250132
CAS:<p>JNJ-1250132 is a steroidal progesterone receptor modulator that inhibits binding of the receptor to DNA in vitro.</p>Formula:C33H41NO4Color and Shape:SolidMolecular weight:515.68SB-612111 hydrochloride
<p>SB-612111 is a potent ORL-1 antagonist, with high affinity (Ki: 0.33 nM) and µ-receptor activity (Ki: 57.6 nM), blocking Nociceptin-induced pain.</p>Formula:C24H30Cl3NOColor and Shape:SolidMolecular weight:454.86Tubulosine
CAS:<p>Tubulosine is an anticancer agent that inhibits cancer cell growth.</p>Formula:C29H37N3O3Color and Shape:SolidMolecular weight:475.62ABT 491 Hydrochloride
CAS:<p>ABT-491 hydrochloride is an active platelet activator receptor (PAF-R) antagonist with good selectivity and oral administration.</p>Formula:C28H23ClFN5O2Color and Shape:SolidMolecular weight:515.97FAK-IN-2
<p>FAK-IN-2: potent oral FAK inhibitor, IC50 35 nM, reduces tumor growth, migration, and induces cell death.</p>Formula:C28H31ClN8O3Color and Shape:SolidMolecular weight:563.05NI-Pano
<p>NI-Pano (CH-03) is a novel hypoxia-activated KDAC inhibitor capable of O2-dependent release of the compound panobinostat.</p>Formula:C26H28N6O4Color and Shape:SolidMolecular weight:488.54ACHN-975
CAS:<p>ACHN-975: potent LpxC inhibitor with subnanomolar activity; targets many gram-negative bacteria; MIC ≤1 μg/mL.</p>Formula:C20H23N3O4Purity:98%Color and Shape:SolidMolecular weight:369.41NB-216
CAS:<p>NB-216 is a macrocyclic peptidic BACE-1 inhibitor.</p>Formula:C35H45N3O4Color and Shape:SolidMolecular weight:571.75SF0166
CAS:<p>SF0166: potent αvβ3 antagonist, IC50: 0.6 nM. Blocks cell adhesion, IC50: 7.6 pM-76 nM. Reduces neovascularization in mice.</p>Formula:C23H27F2N5O4Color and Shape:SolidMolecular weight:475.49Anti-inflammatory agent 12
<p>Pentacyclic triterpene, anti-inflammatory agent 12, inhibits LPS inflammation (IC50: 2.22 μM). May benefit inflammatory disease studies.</p>Formula:C30H50O4Color and Shape:SolidMolecular weight:474.72BI-685509
CAS:<p>BI-685509: potent, oral sGC activator, boosts cGMP, enhances NO pathways, for CKD/DKD research.</p>Formula:C34H38N4O5Color and Shape:SolidMolecular weight:582.69Dyrk1A/α-synuclein-IN-1
<p>Dyrk1A/α-synuclein-IN-1 (Compound b1) is a dual inhibitor of Dyrk1A (IC50: 177 nM) and α-synuclein aggregation (IC50: 10.5 μM).</p>Formula:C20H21N5O3SColor and Shape:SolidMolecular weight:411.48CAII-IN-1
<p>CAII-IN-1 (3n) is a selective bovine CA-II inhibitor with 10.3 μM IC50, used in carbonic anhydrase disorder studies.</p>Formula:C19H21FN4SColor and Shape:SolidMolecular weight:356.46Tezampanel hydrate
CAS:<p>Tezampanel is used for the treatment of migraine, neuropathic pain.</p>Formula:C13H23N5O3Color and Shape:SolidMolecular weight:297.35Ambelline
CAS:<p>Ambelline has antitumor activity.</p>Formula:C18H21NO5Purity:98%Color and Shape:SolidMolecular weight:331.36AZ12971554
<p>AZ12971554: Human thrombin inhibitor, Ki=0.3nM; APTT IC50=0.68µM; ECT IC50=0.16µM.</p>Formula:C20H17ClFN7O3Color and Shape:SolidMolecular weight:457.85ODN 2088
CAS:<p>ODN 2088 is a potent inhibitor of TLR3, TLR7 and TLR9 that is non-cytotoxic and shows inhibition of the release of IFN-α and IL-6.</p>Color and Shape:SolidBMS-901715
CAS:<p>BMS-901715 is an effective and selective inhibitor of adapter protein-2 associated kinase 1 (AAK1; IC50: 3.3 nM).</p>Formula:C22H28N10OPurity:98%Color and Shape:SolidMolecular weight:448.52Cyclic-di-GMP sodium
<p>c-di-GMP sodium: STING activator, regulates bacteria biofilm, motility, virulence.</p>Formula:C20H24N10NaO14P2Color and Shape:SolidMolecular weight:713.08464WW437
<p>WW437 is a histone deacetylase (HDAC) inhibitor that exhibits potent anti-breast cancer activity both in vitro and in vivo.</p>Formula:C23H27N5O4Color and Shape:SolidMolecular weight:437.49Osanetant HCl
CAS:<p>Osanetant HCl is the (R)-enantiomer; neurokinin-3 receptor antagonist</p>Formula:C35H42Cl3N3O2Color and Shape:SolidMolecular weight:643.09Lp-PLA2-IN-6
CAS:<p>Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.</p>Formula:C25H21F5N4O3Color and Shape:SolidMolecular weight:520.45PS-519
CAS:<p>PS-519 is a human tissue plasminogen activator and proteasome inhibitor.</p>Formula:C12H19NO4Color and Shape:SolidMolecular weight:241.28Antiallergic agent-1
<p>Antiallergic agent-1, an Src family kinase inhibitor, is a new and valuable lead compound with potential as an anti-allergic agent.</p>Formula:C27H19F6N5OColor and Shape:SolidMolecular weight:543.46Antitumor agent-78
<p>Antitumor agent-78 blocks GPx-4, raises COX2, triggers apoptosis, halts EMT, and stifles cancer cell growth and migration.</p>Color and Shape:SoildJTE 151A
CAS:<p>JTE-151 is a novel RORγ inverse agonist.</p>Formula:C26H30ClN3O5Color and Shape:SolidMolecular weight:499.99Anticancer agent 36
<p>Compound 11: Sulfonylurea derivative, antimicrobial, anticancer; MIC 0.039-0.156 mg/mL; A549 IC50: 19.7 μg/mL, PC3 IC50: 11.9 μg/mL.</p>Formula:C21H17N3O3S2Color and Shape:SolidMolecular weight:423.51COX-2/PI3K-IN-1
<p>COX-2/PI3K-IN-1 (compound 5d) is a potent inhibitor of PI3K (IC50: 1.14 nM). COX-2/PI3K-IN-1 is a selective inhibitor of COX-2 (Ki: 3.24 nM).</p>Formula:C19H14ClN5S2Color and Shape:SolidMolecular weight:411.93DSM705 hydrochloride
<p>DSM705 hydrochloride: potent antimalarial, pyrrole-based DHODH inhibitor effective against Plasmodium, non-toxic to mammalian DHODH.</p>Formula:C19H20ClF3N6OColor and Shape:SolidMolecular weight:440.85T-3764518
CAS:<p>T-3764518 is a novel and potent inhibitor of stearoyl coenzyme A desaturase (SCD)(IC50 of 4.7 nM).</p>Formula:C20H17F6N5O2Purity:98%Color and Shape:SolidMolecular weight:473.37DWN-12088 HCl
CAS:<p>DWN-12088 HCl is the salt form of DWN-12088 Free Base, an orally administered small molecule prolyl-tRNA synthetase (PRS) inhibitor</p>Formula:C15H21Cl4N3OColor and Shape:SolidMolecular weight:401.15Oxythiamine diphosphate ammonium
<p>Oxythiamin diphosphate ammonium is a potent inhibitor of transketolase (TK).</p>Color and Shape:SolidPM-060184
CAS:<p>PM-060184, a tubulin polymerisation inhibitor, is used potentially for the treatment of solid tumours and breast cancer.</p>Formula:C31H45N3O7Purity:98%Color and Shape:SolidMolecular weight:571.7(R)-FL118
CAS:<p>FL118 inhibits human survivinion expression and activates tumor suppressor p53 as a MOA in p53 wild-type cancer cells.</p>Formula:C21H16N2O6Color and Shape:SolidMolecular weight:392.36Flurandrenolone Acetate
CAS:<p>Flurandrenolone Acetate, a synthetic glucocorticoid derived from Flurandrenolide, is used to study skin issues like eczema and psoriasis.</p>Formula:C26H35FO7Color and Shape:SolidMolecular weight:478.55PF-06462894
CAS:<p>PF-06462894: morpholinopyrimidone, mGlu5 antagonist (Ki=6nM), no immune activation in mouse model.</p>Formula:C18H23N3O3Purity:98%Color and Shape:SolidMolecular weight:329.39NB-533
CAS:<p>NB-533 is a macrocyclic peptidic BACE-1 inhibitor.</p>Formula:C33H55N3O4Color and Shape:SolidMolecular weight:557.81PAT-347
CAS:<p>PAT-347 is a potent inhibitor of Autotaxin, an enzyme linked to cell survival and diseases like cancer and fibrosis.</p>Formula:C28H21ClF2N2O3SColor and Shape:SolidMolecular weight:538.99RORγt Inverse agonist 2
CAS:<p>RORγt Inverse agonist 2 is a selective, orally active inverse agonist of RORγt(EC50 of 119 nM).</p>Formula:C27H25F8NO5SPurity:98%Color and Shape:SolidMolecular weight:627.54HDAC6-IN-12
<p>HDAC6-IN-12 is a potent inhibitor of HDAC6 that binds in the DNA chain, causing DNA damage and exhibiting anticancer effects that can be used in cancer research</p>Formula:C24H39F2N3O5Color and Shape:SolidMolecular weight:487.58Antiangiogenic agent 3
<p>Antiangiogenic agent 3 blocks HUVEC cell migration, chemotaxis, and lowers Src, cdc42, MAPK gene expression.</p>Formula:C19H20O7Color and Shape:SolidMolecular weight:360.36MtTMPK-IN-9
<p>MtTMPK-IN-9 moderately inhibits MtbTMPK (IC50: 48 μM), has submicromolar Mycobacterium activity, and is non-toxic, aiding tuberculosis research.</p>Formula:C25H26N6O7Color and Shape:SolidMolecular weight:522.51ddCTP trisodium
<p>ddCTP trisodium, an HIV reverse transcriptase target, aids AIDS research and DNA sequencing as a ddNTP.</p>Formula:C9H13N3Na3O12P3Color and Shape:SolidMolecular weight:517.1VEGFR-2-IN-14
<p>VEGFR-2-IN-14 (Compound 5) is a potent inhibitor of VEGFR-2, which inhibits the growth of HepG2 cells in the Pre-G1 phase and induces apoptosis.</p>Formula:C24H23N3O3SColor and Shape:SolidMolecular weight:433.52KMH-233
CAS:<p>KMH-233 effectively blocks LAT1, inhibiting L-leucine uptake and cell growth, boosting betastatin and cisplatin efficacy at 25 μM.</p>Formula:C32H25N7O5Color and Shape:SolidMolecular weight:587.58Ganoderic acid R
CAS:<p>Ganoderic acid R: potent anticancer, induces apoptosis, cytotoxic to MDR and sensitive tumor cells.</p>Formula:C34H50O6Color and Shape:SolidMolecular weight:554.76BPN-15606 besylate
<p>BPN-15606 besylate is a potent oral γ-secretase regulator reducing Aβ42 and Aβ40 with good pharmacokinetics. IC50: 7 nM (Aβ42), 17 nM (Aβ40).</p>Formula:C29H29FN6O4SColor and Shape:SolidMolecular weight:576.64Resolvin E2
CAS:<p>RvE2, a bioactive lipid from the SPM family, is made from EPA and reduces inflammatory neutrophil infiltration and helps treat NAFLD and other diseases.</p>Formula:C20H30O4Color and Shape:SolidMolecular weight:334.45AR-13324 M1 metabolite
CAS:<p>AR-13324 M1 metabolite is a hydrolysis metabolite of AR-13324 mesylate.</p>Formula:C19H19N3O2Purity:98%Color and Shape:SolidMolecular weight:321.37HDAC2-IN-1
<p>HDAC2-IN-1 is an oral HDAC2 inhibitor (IC50: 0.5 μM), crosses the blood-brain barrier, and inhibits HDAC1 and HDAC8.</p>Formula:C22H23ClN4OSColor and Shape:SolidMolecular weight:426.96RWJ-56110
CAS:<p>protease-activated receptor-1 (PAR1) antagonist</p>Formula:C41H43Cl2F2N7O3Purity:98%Color and Shape:SolidMolecular weight:790.73EGFR-IN-62
<p>EGFR-IN-62: IC50 of 10-242 nM for various EGFR mutations, blocks A549/H1975 cell cycle, induces apoptosis, and inhibits cell motility and proliferation.</p>Formula:C30H33N9O2Color and Shape:SolidMolecular weight:551.64PTP1B-IN-16
<p>PTP1B-IN-16: selective benzimidazole inhibitor of PTP1B, Ki: 12.6 μM, potential for type 2 diabetes research.</p>Formula:C26H18ClN3O4SColor and Shape:SolidMolecular weight:503.96Nepaprazole sodium
CAS:<p>Nepaprazole Na (TY-11345), a proton pump inhibitor, may treat gastric ulcers; it reduces H+/K(+)-ATPase activity, with IC50 of 5.8-9.9 microM.</p>Formula:C18H18N3NaO2SColor and Shape:SolidMolecular weight:363.41Aplaviroc
CAS:<p>Aplaviroc (AK 602), a SDP derivative, is a CCR5 antagonist. With IC50s of 0.1-0.4 nM for HIV-1Ba-L, HIV-1JRFL and HIV-1MOKW.</p>Formula:C33H43N3O6Purity:97.98% - 98.26%Color and Shape:SolidMolecular weight:577.71G-744
CAS:<p>G-744 is a selective and orally active inhibitor of Btk (IC50: 2 nM).</p>Formula:C29H29N5O3SPurity:98%Color and Shape:SolidMolecular weight:527.64trans-Doxercalciferol
CAS:<p>trans-Doxercalciferol is an isomer of Doxercalciferol. Doxercalciferol is an activator of the Vitamin D receptor and prevents renal disease.</p>Formula:C28H44O2Purity:98%Color and Shape:SolidMolecular weight:412.65SLC4011540
<p>SLC4011540 is a potent and selective SphK1/2 dual inhibitor with Ki value of 120 nM and 90 nM respectively.</p>Formula:C24H23ClF3N7OSColor and Shape:SolidMolecular weight:550Azonafide-PEABA
CAS:<p>Azonafide-PEABA is a drug moiety with cytotoxic [1].</p>Formula:C32H33N5O4Purity:98%Color and Shape:SolidMolecular weight:551.64STAT3-IN-9
<p>STAT3-IN-9 hinders STAT3 at Tyr705, doesn't affect STAT1 Tyr701, induces apoptosis, and arrests cells in G2/M phase.</p>Formula:C22H21N3O4Color and Shape:SolidMolecular weight:391.42Anticancer agent 16
<p>Anticancer agent 16 showed good cytotoxic effects on HCT-116 cell line (IC50: 8.55 μM), NCI-H460 cell line (IC50: 5.41 μM) and SKOV3 cell line (IC50: 6.4 μM).</p>Formula:C27H33N5O6Color and Shape:SolidMolecular weight:523.58QPX7728 methoxy acetoxy methy ester
CAS:<p>QPX7728 methoxy acetoxy methy ester is an inhibitor of boronic acid β-lactamase.</p>Formula:C14H14BFO7Purity:98%Color and Shape:SolidMolecular weight:324.07YW3-56 (hydrochloride) (technical grade)
CAS:<p>YW3-56: PAD2 & PAD4 inhibitor (IC50 = 0.5-5 μM), halts U2OS cell growth (IC50 ~2.5 μM), reduces S-180 & MDA-MB-231 tumor growth in mice.</p>Formula:C27H33Cl2N5O2Color and Shape:SolidMolecular weight:530.493'-Hydroxy Repaglinide
CAS:<p>'3'-Hydroxy Repaglinide, a CYP2C8 metabolite of Repaglinide, treats type II diabetes.</p>Formula:C27H36N2O5Purity:98%Color and Shape:SolidMolecular weight:468.59HER2-IN-11
<p>HER2-IN-11 is a psoralen derivative that induces apoptosis. HER2-IN-11 shows light-activated cytotoxicity and also exhibits anti-breast cancer activity [1].</p>Formula:C17H11NO6Color and Shape:SolidMolecular weight:325.27ND-654
CAS:<p>ND-654 is an acetyl CoA carboxylase inhibitor.</p>Formula:C29H33N3O8SColor and Shape:SolidMolecular weight:583.6516,16-Dimethyl prostaglandin E2
CAS:<p>16,16-Dimethyl prostaglandin E2 regulates hematopoietic stem cells via EP2/EP4 and Wnt, taken orally.</p>Formula:C22H36O5Purity:98%Color and Shape:SolidMolecular weight:380.52CBP/p300-IN-16
<p>CBP/p300-IN-16 (compound 1) is a potent inhibitor of EP300/CBP HAT, acting on HAT EP300 (IC50: 0.61 μM) and LK2 H3K27 (IC50: 2.24 μM).</p>Formula:C26H31N3O4Color and Shape:SolidMolecular weight:449.54ODN 21158
CAS:<p>ODN 21158 is a potent, non-cytotoxic inhibitor of G-modified TLR3 and TLR9. ODN 21158 dose-dependently inhibits IFN-α secretion.</p>Color and Shape:SolidONL-1204
CAS:<p>ONL-1204 is a small molecule, CD95 antigen inhibitor (Fas inhibitor) being developed by ONL Therapeutics for the treatment of retinal detachment.</p>Formula:C71H100N18O16Color and Shape:SolidMolecular weight:1461.66Latrunculins A
CAS:<p>Latrunculins A is a novel marine toxin, disrupts microfilament organization in cultured cells.</p>Formula:C22H31NO6SColor and Shape:SolidMolecular weight:437.55C.I. Pigment Red 60
CAS:<p>C.I. Pigment Red 60 is a bright, scarlet, semi-transparent red pigment.</p>Formula:C17H9N2Na3O9S2Purity:98%Color and Shape:SolidMolecular weight:518.35MCTR3
CAS:<p>MCTR3, derived from DHA via maresin 1 in macrophages, hastens tissue healing and reduces inflammation and eicosanoids post-E. coli infection in mice.</p>Formula:C25H37NO5SColor and Shape:SolidMolecular weight:463.63CYP2C1/CYP2C19-IN-2
<p>CYP2C1/CYP2C19-IN-2 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>Formula:C27H28N2O6SColor and Shape:SolidMolecular weight:508.59O-Desmethyl Midostaurin
CAS:<p>O-Desmethyl Midostaurin is the active Midostaurin metabolite via cytochrome P450 liver enzyme metabolism.</p>Formula:C34H28N4O4Purity:98%Color and Shape:SolidMolecular weight:556.61α-Glucosidase-IN-13
<p>α-Glucosidase-IN-13 is an inhibitor of α-glucosidase (IC50: 5.69 μM).</p>Formula:C25H28N4O3S2Color and Shape:SolidMolecular weight:496.64CB2 receptor antagonist 1
CAS:<p>Compound 29 is a potent, CB2-selective antagonist/reverse agonist. Derivatives 23 & 24 offer antinociception; 24 activates cannabinoid/TRPV1 receptors.</p>Formula:C28H47NO3Color and Shape:SolidMolecular weight:445.68P-gp inhibitor 2
CAS:<p>Potent P-gp inhibitor 2 reverses Doxorubicin resistance in colorectal carcinoma cells with IC50 of 0.22 µM.</p>Formula:C29H26N2O6Color and Shape:SolidMolecular weight:498.53Purine phosphoribosyltransferase-IN-1
<p>Compound (S,R)-48 inhibits Pf, Pv, & Tbr PRT with Ki of 50, 20, 2 nM.</p>Formula:C11H15N5Na4O10P2Color and Shape:SolidMolecular weight:531.17Detoxin D1
CAS:<p>Detoxin D1 is a selective blasticidin S antagonist.</p>Formula:C28H41N3O8Purity:98%Color and Shape:SolidMolecular weight:547.64SML-10-70-1
CAS:<p>SML-10-70-1 is a Novel Active Site Inhibitor of Oncogenic K-Ras G12C.</p>Formula:C25H42ClN7O13P2Color and Shape:SolidMolecular weight:746.04B-3852
CAS:<p>B-3852 is a Bradykinin inhibitor.</p>Formula:C55H74F3N15O11Color and Shape:SolidMolecular weight:1178.27IRAK4-IN-15
CAS:<p>IRAK4-IN-15: selective IRAK4 inhibitor, IC50 0.002 μM, good PK, low clearance, synergizes with Acalabrutinib in MyD88/CD79 mutant ABC-DLBCL.</p>Formula:C25H29FN10Color and Shape:SolidMolecular weight:488.56
