Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,834 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,877 products)
- Chromatin/Epigenetics(2,613 products)
- Cytoskeletal Signaling(1,568 products)
- DNA Damage/DNA Repair(2,871 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,020 products)
- Immunology and Inflammation(3,905 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,257 products)
- Membrane Transporter/Ion Channel(3,155 products)
- Metabolism(10,133 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,473 products)
- Other Inhibitors(35,846 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,689 products)
- Stem Cell and Derivatives(732 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
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Found 66515 products of "Inhibitors"
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PptT-IN-2
PptT-IN-2 inhibits PptT enzyme crucial in tuberculosis, with 2.5 μM IC50, showing potential in TB research.Formula:C22H29N5O2Color and Shape:SolidMolecular weight:395.5Plagiochilin A
CAS:Plagiochilin A Inhibits Cytokinetic Abscission and Induces Cell DeathFormula:C15H14O7Color and Shape:SolidMolecular weight:306.27Monoamine Oxidase B inhibitor 2
MAO-B inhibitor 2: potent, reversible, oral, selective (IC50=1.33 nM), BBB-penetrant, with anti-oxidant and anti-inflammatory effects for Parkinson's study.Formula:C19H19FO3Color and Shape:SolidMolecular weight:314.35BMS-961955
CAS:BMS-961955 is an allosteric inhibitor of the hepatitis C virus NS5B polymerase.Formula:C37H43FN4O4SColor and Shape:SolidMolecular weight:658.83Ac-ATS010-KE
CAS:Ac-ATS010-KE is a novel Selective, irreversible, and Rapid Cell-Permeable Inhibitor of Human Caspase-3.Formula:C43H41F5N6O12SColor and Shape:SolidMolecular weight:960.88DMGF
CAS:DMGF, a biflavonoid from Taxus, induces apoptosis, autophagy, and inhibits B16F10 cell motility and MMP-2 expression, hindering melanoma metastasis.Formula:C32H22O10Color and Shape:SolidMolecular weight:566.51GNE-886
CAS:GNE-886 has a wide range of applications in life science related research.Formula:C28H30N6O3Purity:98%Color and Shape:SolidMolecular weight:498.59AL 6598
CAS:AL 6598, a prodrug of PGD2 agonist AL 6556, reduces IOP by 53% at 1μg twice daily in monkeys; binds DP receptors with Ki of 3.2μM.Formula:C23H39ClO5Color and Shape:SolidMolecular weight:431.01DNDI-8219
CAS:DNDI-8219 is an antitubercular agent. It has potent antileishmanial effects.Formula:C13H10F3N3O5Color and Shape:SolidMolecular weight:345.23Menin-MLL inhibitor 4
CAS:Menin-MLL inhibitor 4 has antitumor activity.Menin-MLL inhibitor 4 is an inhibitor of Menin- MLL (mixed-lineage leukemia protein) interaction .Formula:C32H38FN7O3Purity:98%Color and Shape:SolidMolecular weight:587.69FP0429
CAS:FP0429 is an agonist of mGlu4.Formula:C10H12N2O7Purity:98%Color and Shape:SolidMolecular weight:272.21DBCO-SS-PEG4-Biotin
DBCO-SS-PEG4-Biotin: cleavable ADC linker with 4-unit PEG, used in ADC synthesis.Formula:C45H62N6O9S3Purity:98%Color and Shape:SolidMolecular weight:927.2Mu opioid receptor antagonist 3
Potent, selective MOR antagonist (compound 26); crosses blood-brain barrier. Ki: 0.24 nM, EC50: 0.54 nM; for studying OUD.Formula:C25H28N2O4SColor and Shape:SolidMolecular weight:452.57GSK3527497 HCl
CAS:GSK3527497: potent TRPV4 inhibitor, IC50=12 nM, targets heart/respiratory issues, for oral/IV use, low-dose effective.Formula:C17H17Cl2FN4O4SColor and Shape:SolidMolecular weight:463.3054FGFR4-IN-4
CAS:FGFR4-IN-4 is a FGFR4 inhibitor with anti-tumor activity.Formula:C28H32Cl2N6O5Purity:98%Color and Shape:SolidMolecular weight:603.5Homomoschatoline
CAS:Homomoschatoline is an antibacterial isolated from Artabotrys crassifolius.Formula:C19H15NO4Purity:98%Color and Shape:SolidMolecular weight:321.33GSK864
CAS:GSK864 is an inhibitor of isocitrate dehydrogenase 1 (IDH1) mutant. GSK864 inhibits IDH1 mutants R132C, R132H, and R132G (IC50: 8.8, 15.2, and 16.6 nM).Formula:C30H31FN6O4Purity:97.07%Color and Shape:SolidMolecular weight:558.6GSK1820795A
CAS:GSK1820795A: Telmisartan analog, selective hGPR132a antagonist, blocks yeast activation by N-acylamides, angiotensin II antagonist, partial PPARγ agonist.Formula:C35H34N8Color and Shape:SolidMolecular weight:566.7GPX4-IN-3
CAS:GPX4-IN-3 (26a) is a potent GPX4 inhibitor, inducing selective ferroptosis with 71.7% inhibition at 1 μM.Formula:C29H24ClN3O3SColor and Shape:SolidMolecular weight:530.04SSR-182289A (Free)
CAS:SSR-182289A (Free) is a thrombin inhibitor.Formula:C30H33F2N5O4SPurity:98%Color and Shape:SolidMolecular weight:597.68LSD1-IN-13 hydrochloride
CAS:LSD1-IN-13 hydrochloride (7e) is an oral LSD1 inhibitor (IC50: 24.43 nM), promoting differentiation in AML cell lines.Formula:C23H30ClN3O2SColor and Shape:SolidMolecular weight:448.02SS-RJW100
SS-RJW100 is an enantiomer of RJW100 targeting LRH-1, SF-1, enhances Tif2 interaction, and disrupts LRH-1 networks with lowered stability.Formula:C28H34OColor and Shape:SolidMolecular weight:386.57DS89002333
DS89002333: oral PRKACA inhibitor with 0.3 nM IC50, effective against FL-HCC with DNAJB1-PRKACA fusion in xenografts.Formula:C22H20ClF2N3O3Color and Shape:SolidMolecular weight:447.86Antibacterial agent 68
Antibacterial agent 68 targets drug-resistant E. coli at 0.007 mM with low cytotoxicity.Formula:C26H25BrN4O7Color and Shape:SolidMolecular weight:585.4CAII-IN-2
CAII-IN-2 (3g): potent, selective CA-II inhibitor; IC50-12.1 μM for bovine CA-II; valuable in CA-related disorder research.Formula:C18H19BrN4SColor and Shape:SolidMolecular weight:403.34LY2934747
CAS:LY2934747 is a novel, potent, and systemically bioavailable mGlu2/3 receptor agonist, exhibiting both antipsychotic and analgesic properties in vivo.Formula:C10H13NO4Color and Shape:SolidMolecular weight:211.21DNA gyrase B-IN-1
DNA gyrase B-IN-1, a potent inhibitor of P. aeruginosa DNA gyrase B, has IC50 of 2.2 μM with high affinity and stability.Formula:C23H18ClF3N6O4SColor and Shape:SolidMolecular weight:566.94Kahweol linoleate
CAS:Kahweol linoleate, a semi-synthetic from coffee, blocks osteoclast creation, fights cancerous cells, prevents DNA damage, and reduces oxidative stress.Formula:C38H56O4Color and Shape:SolidMolecular weight:576.85GNE-203
CAS:GNE-203 is a Met inhibitor.Formula:C30H29Cl2F3N8O3Color and Shape:SolidMolecular weight:677.50Anti-inflammatory agent 13
Pentacyclic triterpene, Anti-inflammatory 13 inhibits DAMP/PAMP inflammation models.Formula:C30H48O4Color and Shape:SolidMolecular weight:472.7SF0166
CAS:SF0166: potent αvβ3 antagonist, IC50: 0.6 nM. Blocks cell adhesion, IC50: 7.6 pM-76 nM. Reduces neovascularization in mice.Formula:C23H27F2N5O4Color and Shape:SolidMolecular weight:475.49Antibacterial agent 88
Antibacterial agent 88 is an effective antibacterial agent against B. subtilis (MIC: 4 μg/ml) with MIC values of ≤0.0156 μg/mL for MRSA, MRSE and S. aureus.Formula:C31H44N2O6SColor and Shape:SolidMolecular weight:572.76Antimalarial agent 9
Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.Formula:C28H32BrN3O2Color and Shape:SolidMolecular weight:522.48BILA 1906 BS
CAS:BILA 1906 BS is an inhibitor of substrate analog protease.Formula:C41H52N6O4SPurity:98%Color and Shape:SolidMolecular weight:724.95P7170
CAS:P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.Formula:C21H16F3N9Color and Shape:SolidMolecular weight:451.42SIK1 activator 1
CAS:SIK1 activator 1 boosts SIK1 phosphorylation, reduces type 2 diabetes hyperglycemia, and inhibits liver gluconeogenesis.Formula:C23H32O6Color and Shape:SolidMolecular weight:404.508(S),15(S)-DiHETE
CAS:8(S),15(S)-DiHETE, from 15(S)-HETE's oxidation by 15-LO, triggers eosinophil movement at 1.5 μM; it counteracts pain and LTB4 effects.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47Acetylpepstatin
CAS:Acetylpepstatin is an inhibitor of HIV-1 protease, HIV-2 protease, aspartyl protease.Formula:C33H61N5O11Purity:98%Color and Shape:SolidMolecular weight:703.875NS2B/NS3-IN-5
Compound 25b inhibits DENV2/ZIKV NS2B/NS3 proteases; IC50: ZIKV 0.67μM, DENV2 4.38μM.Formula:C14H9IN2O3SColor and Shape:SolidMolecular weight:412.2AL-6556
CAS:AL-6556 is a prostaglandin DP receptor agonist.Formula:C20H33ClO5Color and Shape:SolidMolecular weight:388.93Tezampanel hydrate
CAS:Tezampanel is used for the treatment of migraine, neuropathic pain.Formula:C13H23N5O3Color and Shape:SolidMolecular weight:297.35A-9758
CAS:A-9758: RORγt selective inverse agonist, IC50 5nM, inhibits IL-17A, Th17, and treats psoriasis.Formula:C25H23Cl2F3N2O3Purity:98%Color and Shape:SolidMolecular weight:527.36GW311616 hydrochloride
CAS:GW-311616 hydrochloride is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).Formula:C19H32ClN3O4SPurity:98%Color and Shape:SolidMolecular weight:433.99Afeletecan HCl
CAS:Afeletecan (BAY 56-3722) is a water-soluble, anti-cancer camptothecin conjugated to a carbohydrate, inhibiting DNA replication and inducing apoptosis.Formula:C45H50ClN7O11SColor and Shape:SolidMolecular weight:932.44KRAS G12C inhibitor 37
CAS:KRAS G12C inhibitor 37 targets a key signaling protein, showing promise for cancer research involving KRAS G12C.Formula:C35H39F3N8O2Color and Shape:SolidMolecular weight:660.73BXL0124
CAS:BXL0124 is a gemini vitamin D analog which targets CD44-STAT3 signaling and inhibits breast cancer invasion.Formula:C32H44F6O4Color and Shape:SolidMolecular weight:606.68KRAS G12D inhibitor 16
CAS:KRAS G12D inhibitor 16 targets KRAS G12D with IC50 of 0.7 nM and mutant form at 0.35 μM, useful in various cancer studies.Formula:C32H39IN6O3Color and Shape:SolidMolecular weight:682.59Rosiptor acetate
CAS:Rosiptor (AQX-1125) activates SHIP1, inhibits Akt, and reduces inflammation and allergy in rodents.Formula:C22H39NO4Purity:98%Color and Shape:Solid PowderMolecular weight:381.55PCSK9-IN-17
CAS:PCSK9-IN-17 is a PCSK9 inhibitor utilized in the research of cholesterol metabolism.Formula:C16H19N5OSColor and Shape:SolidMolecular weight:329.42NVP-CFC218
CAS:NVP-CFC218 is a novel potent and selective p53-HDM2 inhibitor.Formula:C37H45ClN4O4Color and Shape:SolidMolecular weight:645.23ABL-001-Amide-PEG3-acid
ABL-001-Amide-PEG3-acid, an analogue to ABL-001, primarily serves as a labeled chemical or fluorescent probe.Formula:C29H33ClF2N6O9Purity:98%Color and Shape:SolidMolecular weight:683.06ent-8-iso-15(S)-Prostaglandin F2α
CAS:Isoprostanes are produced by the non-enzymatic, free radical peroxidation of phospholipid-esterified arachidonic acid.Formula:C20H34O5Color and Shape:SolidMolecular weight:354.48β-N-Acetyl-D-hexosaminidase-IN-1
β-N-Acetyl-D-hexosaminidase-IN-1 is a newly discovered chemical compound that acts as an inhibitor for β-N-acetyl-D-hexosaminidase.Formula:C18H13F2NO2SColor and Shape:SolidMolecular weight:345.36ONO-8809
CAS:ONO-8809: Thromboxane A2 antagonist, reduces airway hyperresponse, macrophage accumulation, and MMP-9 in SHRSP brains.Formula:C30H46BrNO4SPurity:98%Color and Shape:SolidMolecular weight:596.66DRX-065
CAS:DRX-065, a deuterated R-enantiomer of pioglitazone, treats NASH without PPARγ weight gain issues.Formula:C19H20N2O3SColor and Shape:SolidMolecular weight:357.45LPA5 antagonist 1
LPA5 antagonist 1: selective, potent (IC50=32 nM), high brain permeability, studies inflammatory/neuropathic pain.Formula:C28H26N2O4SColor and Shape:SolidMolecular weight:486.58A 70450
CAS:A 70450, an inhibitor of aspartyl proteinase, can be used as an antifungal agent and may have a role in HIV protease inhibition therapy.Formula:C42H71ClN6O5Purity:98%Color and Shape:SolidMolecular weight:775.50(-)-Mesembrine
CAS:Mesembrine is a serotonin reuptake inhibitor and is also a weak inhibitor of the enzyme phosphodiesterase 4 (PDE4).Formula:C17H23NO3Color and Shape:SolidMolecular weight:289.37Domitroban
CAS:Domitroban, also known as S-145, is a thromboxane (Tx) A2-receptor antagonist with partial agonistic activity in vascular smooth muscle.Formula:C20H27NO4SColor and Shape:SolidMolecular weight:377.5Fabimycin
CAS:Fabimycin, a FabI inhibitor, combats drug-resistant gram-negative bacterial infections effectively.Formula:C23H25ClN4O3Color and Shape:SolidMolecular weight:440.92HPK1-IN-14
CAS:HPK1-IN-14 is a potent inhibitor of HPK1. HPK1-IN-14 has potential for the study of HPK1-related diseases.Formula:C24H23FN6O2Color and Shape:SolidMolecular weight:446.48Teslexivir hydrochloride
CAS:Teslexivir (BTA074) HCl inhibits HPV 6/11 by blocking E1-E2 protein interaction, vital for DNA replication. Used in condyloma research.Formula:C35H37BrClN3O4Color and Shape:SolidMolecular weight:679.04Antioxidant agent-3
Antioxidant agent-3 shows strong DPPH and ABTS+ radical scavenging (IC50: 26.58, 30.31 μM). Boosts ROS, SOD, GSH; lowers LDH in H2O2-exposed HepG2 cells.Formula:C18H14O8Color and Shape:SolidMolecular weight:358.3MIF2-IN-1
MIF2-IN-1, potent inhibitor of MIF2 (IC50: 1μM), halts non-small cell lung cancer growth via MAPK pathway.Formula:C26H19F3N2O2SColor and Shape:SolidMolecular weight:480.5KT5926
CAS:KT5926 selectively inhibits myosin light chain kinase and NGF-dependent neurite growth; it's a K-252a analogue.Formula:C30H27N3O6Purity:98%Color and Shape:SolidMolecular weight:525.55PS-519
CAS:PS-519 is a human tissue plasminogen activator and proteasome inhibitor.Formula:C12H19NO4Color and Shape:SolidMolecular weight:241.28Lunacalcipol
CAS:Lunacalcipol is used for the treatment of Secondary Hyperparathyroidism.Formula:C28H42O4SColor and Shape:SolidMolecular weight:474.7KRAS inhibitor-13
CAS:KRAS inhibitor-13 blocks KRAS G12C (IC50: 0.883 μM) and p-ERK in some cancer cells; promising for pancreatic, colorectal, lung cancer research.Formula:C25H19ClFN3O2SColor and Shape:SolidMolecular weight:479.95MAO-B-IN-6
MAO-B-IN-6 is a selective, potent, orally active MAO-B inhibitor (IC50: 0.019 μM). MAO-B-IN-6 is superior to Safinamide both in vitro and in vivo.Color and Shape:SolidJAK3-IN-7
CAS:JAK3-IN-7 is a potent and selective JAK3 inhibitor (IC50<0.01 μM) for the treatment of rejection in organ transplantation, graft-versus-host reaction afterFormula:C17H20N6OPurity:98.81%Color and Shape:SolidMolecular weight:324.38LpxC-IN-10
CAS:LpxC-IN-10 is a selective LpxC inhibitor with an MIC of 0.5 μg/mL against E. coli and K. pneumoniae and is capable of being used to study bacterial infections.Formula:C30H31N5O3Color and Shape:SolidMolecular weight:509.6Nonsteroidal aromatase inhibitor 1
Compound 13h, a nonsteroidal aromatase inhibitor, has a potent IC50 of 0.09 nM against CYP19A1, showing promise for breast cancer research.Formula:C22H16N4O2Color and Shape:SolidMolecular weight:368.39GSK2578999A
CAS:GSK2578999A is a betulin derivative with antitumor activity.Formula:C46H62ClNO7Purity:98%Color and Shape:SolidMolecular weight:776.44L 731735
CAS:L 731735 is a farnesyltransferase inhibitor.Formula:C19H40N4O4SPurity:98%Color and Shape:SolidMolecular weight:420.61NITD-688
CAS:NITD-688 is a pan-serotype inhibitor targeting the dengue virus NS4B protein, effective through oral administration.Formula:C25H32N4O3S2Color and Shape:SolidMolecular weight:500.68PI4KIIIbeta-IN-11
CAS:PI4KIIIbeta-IN-11 is a PI4KIIIβ inhibitor (mean pIC50=9.1) that can be used to study diseases caused by RNA viruses and Plasmodium falciparum.Formula:C33H39N7O3Color and Shape:SolidMolecular weight:581.71Thioquinapiperifil dihydrochloride
CAS:Thioquinapiperifil dihydrochloride is a potent, selective PDE-5 inhibitor (IC50: 0.074 nM) for research.Formula:C24H29ClN6OSPurity:99.81%Color and Shape:SolidMolecular weight:485.05Ref: TM-T9773
1mg58.00€5mg130.00€1mL*10mM (DMSO)148.00€10mg187.00€25mg304.00€50mg393.00€100mg552.00€200mg725.00€rel-MDM2/4-p53-IN-2
Potent dual MDM2/MDM4 inhibitor & p53 activator; IC50: 70.7 nM (MDM2), 81.4 nM (MDM4); regulates cell cycle, triggers apoptosis, anti-cancer.Formula:C25H17Cl3FN3O3Color and Shape:SolidMolecular weight:532.78KRAS G12D inhibitor 3
CAS:KRAS G12D Inhibitor 3, a compound targeting the KRAS G12D mutation, demonstrates potent antitumor efficacy with an inhibitory concentration (IC50) of less thanFormula:C34H31ClF3N5O2Color and Shape:SolidMolecular weight:634.09VEGFR-2-IN-14
VEGFR-2-IN-14 (Compound 5) is a potent inhibitor of VEGFR-2, which inhibits the growth of HepG2 cells in the Pre-G1 phase and induces apoptosis.Formula:C24H23N3O3SColor and Shape:SolidMolecular weight:433.52MtTMPK-IN-1
MtTMPK-IN-1 inhibits MtTMPK with 2.5 μM IC50, shows moderate anti-tuberculosis activity, and is low in cytotoxicity.Formula:C22H24N4O3Color and Shape:SolidMolecular weight:392.45NF-κB-IN-4
NF-κB-IN-4 (compound 17) is a potent inhibitor of NF-κB pathway which can cross blood brain barrier (BBB).Formula:C18H15FN4OColor and Shape:SolidMolecular weight:322.34IDO1-IN-13
IDO1-IN-13 is a potent IDO1 inhibitor (IC50: 61.6 nM, EC50: 30 nM in HeLa) that reduces kyn/trp ratio by 51% in SK-OV-3 tumors.Formula:C20H16BrN5O2SColor and Shape:SolidMolecular weight:470.34BTK-IN-10
CAS:BTK-IN-10 is a potent inhibitor of BTK, acting on wild-type BTK (IC50<5 nM) or mutant BTK (C481S) (IC50<5 nM).Formula:C25H24F2N4O2Color and Shape:SolidMolecular weight:450.48Laulimalide
CAS:Microtubule stabilizer; halts cancer cell growth (IC50: 3-30 nM); arrests cells in prometaphase; prevents bipolar spindle formation.Formula:C30H42O7Color and Shape:SolidMolecular weight:514.65PEN-866
CAS:PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.Formula:C49H49N7O9Color and Shape:SolidMolecular weight:879.95BI-207524
CAS:BI-207524 is a novel NS5B Thumb Pocket 1 Inhibitor with Improved Potency for the Potential Treatment of Chronic Hepatitis C Virus Infection.Formula:C35H36ClN5O5Color and Shape:SolidMolecular weight:642.14CDK9-IN-11
CAS:CDK9-IN-11 is a potent CDK9 inhibitor that is the ligand for the PROTAC CDK9 Degrader-1 [1].Formula:C20H25N3O4Purity:98%Color and Shape:SolidMolecular weight:371.43ACSS2-IN-1
CAS:ACSS2-IN-1, a potent ACSS2 inhibitor, has IC50 0.01-<1 nM; useful in cancer research.Formula:C27H25ClN6O2Color and Shape:SolidMolecular weight:500.98AD013
AD013 is a selective ACE inhibitor and NEP inhibitor with potential anti-hypertensive and cardioprotective benefits.Formula:C24H28N2O5Color and Shape:SolidMolecular weight:424.49SCH 563705
CAS:SCH 563705 is a CXCR2 and CXCR1 antagonist used in the study of acute respiratory syndrome, chronic obstructive pulmonary disease, and inflammation.Formula:C23H27N3O5Purity:98.03%Color and Shape:SolidMolecular weight:425.48(1R,3S)-THCCA-Asn
(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.Formula:C24H24N4O6Color and Shape:SolidMolecular weight:464.47Diacylglycerol acyltransferase inhibitor-1
CAS:Diacylglycerol Acyltransferase Inhibitor-1, a diacylglycerol acyltransferase (DGAT1) inhibitor, effectively suppresses the activity of DGAT1.Formula:C21H23N5O2Purity:98%Color and Shape:SolidMolecular weight:377.44TRβ agonist 1
CAS:TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.Formula:C29H25FN2O8Color and Shape:SolidMolecular weight:548.52AY 17,605
CAS:AY 17,605 is an inhibitor of bovine heart and rat brain nucleoside-3',5'- monophosphate phosphodiesterase.Formula:C25H36O5Color and Shape:SolidMolecular weight:416.55sEH inhibitor-2
SEH inhibitor-2 is an orally active sEH blocker (IC50=0.9 nM) with predicted 71.2-88.4% absorption, potentially aiding cardiovascular health.Formula:C23H18N4O3Color and Shape:SolidMolecular weight:398.41P-gp modulator 3
P-gp modulator 3 (Compound 37) is a potent, competitive, metabotropic P-glycoprotein (P-gp) modulator.Formula:C31H37N3O5Color and Shape:SolidMolecular weight:531.64BRD7929
CAS:BRD7929 is a multistage antimalarial inhibitor for single-dose treatment of malaria in mouse models.Formula:C33H38N4O2Color and Shape:SolidMolecular weight:522.68DI-404
CAS:DI-404: Potent DCN1-UBC12 inhibitor, selectivity blocks cullin 3 neddylation, Kd=6.9 nM.Formula:C35H45ClN6O6SPurity:98%Color and Shape:SolidMolecular weight:713.29TCMDC-135051 TFA (2413716-15-9 free base)
TCMDC-135051 TFA is a highly selective and potent inhibitor of protein kinase PfCLK3.Formula:C31H34F3N3O5Purity:98%Color and Shape:SolidMolecular weight:585.61
