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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66641 products of "Inhibitors"

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  • (RS)-AMPA

    CAS:
    <p>(RS)-AMPA ((±)-AMPA) is a glutamate analog. (RS)-AMPA is an agonist of effective and selective excitatory neurotransmitter L-glutamic acid.</p>
    Formula:C7H10N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:186.17
  • Human enteropeptidase-IN-2


    <p>Human enteropeptidase-IN-2 is a potent inhibitor of enteropeptidase (enteropeptidase) and can be used in anti-obesity studies.</p>
    Formula:C20H19F3N4O7
    Color and Shape:Solid
    Molecular weight:484.38
  • SHR0687

    CAS:
    <p>SHR0687: potent KOR agonist, selective, favorable PK, effective in rat pain model, minimal BBB penetration, less CNS side effects.</p>
    Formula:C39H60N8O5
    Color and Shape:Solid
    Molecular weight:720.94
  • Antitumor agent-74


    <p>Antitumor agent-74, a quinazoline derivative, inhibits DNA, arrests cell cycle, and induces apoptosis with agent-75.</p>
    Formula:C26H23FN6
    Color and Shape:Solid
    Molecular weight:438.5
  • GABAA receptor agonist 2


    <p>Compound 4c, a potent GABAA agonist with anti-depressive effects in mouse FST/TST, shows promise in depression research.</p>
    Formula:C22H36O5
    Color and Shape:Solid
    Molecular weight:380.52
  • MMSET-IN-1

    CAS:
    <p>MMSET-IN-1 is an inhibitor of multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) .</p>
    Formula:C18H29N7O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:423.47
  • Cbl-b-IN-2

    CAS:
    <p>Cbl-b-IN-2 is an oral E3 enzyme inhibitor for immune-modulated diseases and cancer research.</p>
    Formula:C29H30F5N5O2
    Color and Shape:Solid
    Molecular weight:575.57
  • Ro 24-4383

    CAS:
    <p>Ro 24-4383 is a carbamate-linked dual-action antibacterial agent.</p>
    Formula:C32H31FN8O10S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:770.76
  • Niravoline

    CAS:
    <p>Niravoline is a kappa-opioid agonist.</p>
    Formula:C22H25N3O3
    Color and Shape:Solid
    Molecular weight:379.45
  • CD73-IN-7

    CAS:
    <p>CD73-IN-7: potent inhibitor of CD73, blocks adenosine production to treat tumors.</p>
    Formula:C13H11ClN4O2
    Color and Shape:Solid
    Molecular weight:290.7
  • α-Glucosidase-IN-15


    <p>α-Glucosidase-IN-15 (Compound 14B) exhibits potent inhibitory activity against α-glucosidase, with an IC50 value of 3.34 μM.</p>
    Formula:C24H24N2S
    Color and Shape:Solid
    Molecular weight:372.53
  • Antimalarial agent 9


    <p>Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.</p>
    Formula:C28H32BrN3O2
    Color and Shape:Solid
    Molecular weight:522.48
  • AGN-204396

    CAS:
    <p>AGN-204396 is an antagonist that selectively blocks the activity of prostamides (prostaglandin-ethanolamides).</p>
    Formula:C32H44FN3O4
    Color and Shape:Solid
    Molecular weight:553.71
  • Kaitocephalin

    CAS:
    <p>Kaitocephalin: naturally occurring, non-selective antagonist blocking glutamate receptors, made by Eupenicillium shearii fungus.</p>
    Formula:C18H21Cl2N3O9
    Color and Shape:Solid
    Molecular weight:494.28
  • PD-1/PD-L1-IN-23

    CAS:
    <p>PD-1/PD-L1-IN-23: potent, oral PD-1/PD-L1 inhibitor; L7's ester prodrug; exhibits strong antitumor effects.</p>
    Formula:C32H30BrCl2N3O6
    Color and Shape:Solid
    Molecular weight:703.41
  • BRD-7880

    CAS:
    <p>BRD-7880 is a potent and highly specific inhibitor of aurora kinases B and C.</p>
    Formula:C32H38N4O7
    Color and Shape:Solid
    Molecular weight:590.67
  • Cenicriviroc Sulfone

    CAS:
    <p>Cenicriviroc Sulfone, a Cenicriviroc derivative, inhibits CCR2/CCR5 to block HIV entry into cells.</p>
    Formula:C41H52N4O5S
    Color and Shape:Solid
    Molecular weight:712.94
  • Nomelidine

    CAS:
    <p>Nomelidine, the active N-demethylated metabolite of zimelidine, has been used as an antidepressant and analgesic.</p>
    Formula:C15H15BrN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:303.20
  • PI3K-IN-35

    CAS:
    <p>PI3K-IN-35 (6l) selectively inhibits PI3K-α, β, δ (IC50: 13.98, 7.22, 10.94 μM), blocks G2/M phase, induces apoptosis, and is useful in leukemia research.</p>
    Formula:C25H23N7O2
    Color and Shape:Solid
    Molecular weight:453.5
  • VEGFR-2-IN-10


    <p>VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.</p>
    Formula:C20H21N3O2
    Color and Shape:Solid
    Molecular weight:335.4
  • Bulgecin A

    CAS:
    <p>Bulgecin A is an inhibitor of binuclear metallo-beta-lactamases and Lytic transglycosolase.</p>
    Formula:C16H29N3O14S2
    Color and Shape:Solid
    Molecular weight:551.54
  • LSD1-IN-22


    <p>LSD1-IN-22: potent LSD1 inhibitor, K_i 98 nM, curbs cancer cell growth.</p>
    Formula:C9H8BrF2N
    Color and Shape:Solid
    Molecular weight:248.07
  • AL-GDa62


    <p>AL-GDa62, a gastric cancer treatment lead, has EC50 of 3.2 μM (MCF10A-WT) and 2 μM (MCF10A-CDH1 -/-).</p>
    Formula:C24H28FN3O
    Color and Shape:Solid
    Molecular weight:393.5
  • HDAC8-IN-2


    <p>HDAC8-IN-2 (5o) inhibits both smHDAC8 and hHDAC8 with IC50s of 0.27 μM, 0.32 μM, kills schistosome larvae, and lowers egg laying.</p>
    Formula:C21H16N2O5
    Color and Shape:Solid
    Molecular weight:376.36
  • RS 61756-007

    CAS:
    <p>RS 61756-007 is a selective thromboxane receptor (TP) agonist.</p>
    Formula:C23H28O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:384.47
  • AK-295

    CAS:
    <p>AK 295, also known as CX 295, is a dipeptide inhibitor of alpha-ketoamide calpain.</p>
    Formula:C26H40N4O6
    Color and Shape:Solid
    Molecular weight:504.62
  • LY 292728

    CAS:
    <p>LY 292728 is a highly potent antagonist of leukotriene B4 receptor.</p>
    Formula:C34H29FO9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:600.59
  • L 156903

    CAS:
    <p>L 156903 is a bioactive chemical. It also inhibits the binding of neurotensin to brain tissue.</p>
    Formula:C35H41N7O5S
    Color and Shape:Solid
    Molecular weight:671.81
  • L-threo-Sphingosine C-18

    CAS:
    <p>L-threo-Sphingosine C-18 is a protein kinase C inhibitor.</p>
    Formula:C18H37NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.49
  • Porphobilinogen

    CAS:
    <p>Porphobilinogen act as a phytotoxin, a metabotoxin, and a neurotoxin.</p>
    Formula:C10H14N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:226.23
  • (2R,3S)-Azelaprag

    CAS:
    <p>(2R,3S)-N-(4-(2,6-dimethoxyphenyl)-5-(5-methylpyridin-3-yl)-4H-1,2,4-triazol-3-yl)-3-(5-methylpyrimidin-2-yl)butane-2-sulfonamide is an Apelin receptor agonist</p>
    Formula:C25H29N7O4S
    Purity:97.47% - >99.99%
    Color and Shape:Soild
    Molecular weight:523.61
  • MAFP

    CAS:
    <p>MAFP (Methyl Arachidonyl Fluorophosphonate) is an effective irreversible inhibitor of anandamide amidase.</p>
    Formula:C21H36FO2P
    Color and Shape:Solid
    Molecular weight:370.48
  • GSK5852


    <p>GSK5852, an HCV NS5B inhibitor, has IC50 of 50 nM; potently fights HCV with EC50 of 3.0 nM for GT1a and 1.7 nM for GT1b.</p>
    Formula:C27H27BF2N2O6S
    Color and Shape:Solid
    Molecular weight:556.39
  • AZD 4407

    CAS:
    <p>AZD 4407 is a potent inhibitor of 5-lipoxygenase.</p>
    Formula:C19H21NO3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:375.5
  • Azotomycin

    CAS:
    <p>Azotomycin is an antagonist of L-glutamine and may be used as an immunosuppressant.</p>
    Formula:C17H23N7O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:453.41
  • Diospyrin

    CAS:
    <p>Diospyrin is a plant product that has significant inhibitory effect on the growth of Leishmania donovani promastigotes.</p>
    Formula:C22H14O6
    Color and Shape:Solid
    Molecular weight:374.34
  • 2R,4S-Sacubitril

    CAS:
    <p>2R,4S-Sacubitril (Sacubitril Enantiomer) is the impurity of Sacubitril which is a neprilysin inhibitor.</p>
    Formula:C24H28NO51Ca
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.49
  • KY-02327 acetate


    <p>KY-02327 acetate inhibits Dvl-CXXC5, stabilizes Wnt/β-catenin signaling, and enhances osteoblast differentiation.</p>
    Formula:C22H31N3O6
    Color and Shape:Solid
    Molecular weight:433.5
  • PDE4-IN-6


    <p>PDE4-IN-6: Potent PDE4 inhibitor, IC50 - 0.125μM (B), 0.43μM (D), anti-inflammatory, for arthritis research.</p>
    Formula:C25H20FNO5S
    Color and Shape:Solid
    Molecular weight:465.49
  • Chitinase-IN-5


    <p>Chitinase-IN-5 (8i) blocks OfChi-h (IC50: 0.051 μM), has insecticidal qualities, useful for eco-friendly pest control.</p>
    Formula:C20H21ClFN7
    Color and Shape:Solid
    Molecular weight:413.88
  • OP-5244 sodium


    <p>OP-5244 sodium: potent oral CD73 inhibitor (IC50: 0.25 nM), potential in cancer research by hindering adenosine, reversing immunosuppression.</p>
    Formula:C19H28ClN5NaO9P
    Color and Shape:Solid
    Molecular weight:559.87
  • L 671776

    CAS:
    <p>L 671776 is an inositol monophosphatase inhibitor.</p>
    Formula:C23H32O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:388.5
  • LSD1-IN-17


    <p>LSD1-IN-17, a potent LSD1/CoREST/MAO inhibitor, IC50: 0.005/0.028/0.820 μM; hinders LNCaP prostate cancer cell growth, IC50: 17.2 μM.</p>
    Formula:C20H18N2OS
    Color and Shape:Solid
    Molecular weight:334.43
  • Antifungal agent 39

    CAS:
    <p>Antifungal agent 39 (Compound 9h) is a broad-spectrum antifungal agent.</p>
    Formula:C23H22ClN3O5
    Color and Shape:Solid
    Molecular weight:455.89
  • Beloxepin

    CAS:
    <p>Beloxepin is an oral dual selective inhibitor of serotonin and norepinephrine uptake.</p>
    Formula:C19H21NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:295.38
  • LXR agonist 2


    <p>LXR agonist 2 is a potent agonist of the LXR (liver X receptor). LXR agonist 2 stabilises NCOA1 (coactivator), which in turn agonises the LXR.</p>
    Formula:C35H40ClN3O3
    Color and Shape:Solid
    Molecular weight:586.16
  • PD-L1-IN-1


    <p>PD-L1-IN-1, potent PD-L1 inhibitor with 115 nM IC50, suppresses tumors, boosts immune response, and spares healthy cells.</p>
    Formula:C21H23N5O2
    Color and Shape:Solid
    Molecular weight:377.44
  • GNE-203

    CAS:
    <p>GNE-203 is a Met inhibitor.</p>
    Formula:C30H29Cl2F3N8O3
    Color and Shape:Solid
    Molecular weight:677.50
  • NBD-10007

    CAS:
    NBD-10007 is an inhibitor of HIV-1 entry.
    Formula:C20H25ClN4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.96
  • Homopteroic Acid

    CAS:
    <p>Homopteroic Acid, a precursor to Homofolic Acid, inhibits L1210 mouse leukemia growth by targeting folate uptake.</p>
    Formula:C15H14N6O3
    Color and Shape:Solid
    Molecular weight:326.31
  • Antitubercular agent-23


    <p>Antitubercular agent-23 combats Candida albicans (MIC: 1.1 μg/ml) and M. tuberculosis (MIC: 1 μg/ml).</p>
    Formula:C20H22FN5O8S
    Color and Shape:Solid
    Molecular weight:511.48
  • KOS-1584

    CAS:
    <p>KOS-1584, a safer, more effective epothilone, inhibits cell division by stabilizing microtubules and evading P-gp.</p>
    Formula:C27H39NO5S
    Color and Shape:Solid
    Molecular weight:489.67
  • SID 26681509 quarterhydrate


    <p>SID 26681509 is a selective inhibitor of cathepsin L (IC50: 56 nM) and blocks Plasmodium falciparum (IC50: 15.4 μM) and Leishmania major (IC50: 12.5 μM).</p>
    Formula:C27H35N5O6S
    Color and Shape:Solid
    Molecular weight:544.16
  • BRD7539

    CAS:
    <p>BRD7539B: PfDHODH inhibitor, IC50 0.033μM; selective vs HsDHODH, IC50 &gt;50μM.</p>
    Formula:C23H22FN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:391.44
  • Silvestrol

    CAS:
    <p>Silvestrol is a eukaryotic translation initiation factor 4A inhibitor. Silvestrol causes autophagy and caspase-mediated apoptosis.</p>
    Formula:C34H38O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:654.66
  • CXCR7 modulator 2

    CAS:
    <p>CXCR7 modulator 2 is a 7-type C-X-C chemokine receptor (CXCR7) modulator with a Ki of 13 nM.</p>
    Formula:C29H42N6O3
    Color and Shape:Solid
    Molecular weight:522.68
  • GNE684

    CAS:
    <p>GNE684 inhibits RIP1; Ki app: 21 nM (human), 189 nM (mouse), 691 nM (rat).</p>
    Formula:C23H24N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.48
  • LY3130481

    CAS:
    <p>LY3130481: TARP γ-8 dependent AMPA receptor blocker; selectively targets AMPA/TARP γ-8 with 65 nM IC50.</p>
    Formula:C19H18N4O3S
    Color and Shape:Solid
    Molecular weight:382.44
  • Refametinib R enantiomer

    CAS:
    <p>Refametinib R enantiomer (RDEA119 R enantiomer) is an MEK inhibitor with an EC50 of 2.0-15 nM.Refametinib (R enantiomer) has anticancer activity and can be used</p>
    Formula:C19H20F3IN2O5S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:572.34
  • CA IX-IN-1


    <p>CA IX-IN-1 (compound 12g) is a potent and highly selective hCA IX inhibitor (IC50: 7 nM) that exhibits antitumour effects.</p>
    Formula:C16H22N4O8S
    Color and Shape:Solid
    Molecular weight:430.43
  • BXL0124

    CAS:
    <p>BXL0124 is a gemini vitamin D analog which targets CD44-STAT3 signaling and inhibits breast cancer invasion.</p>
    Formula:C32H44F6O4
    Color and Shape:Solid
    Molecular weight:606.68
  • DS01080522


    <p>DS01080522: PRKACA inhibitor, IC50: kinase 0.8 nM, CREB 66 nM; potential for cancer research.</p>
    Formula:C23H20Cl2N4O3
    Color and Shape:Solid
    Molecular weight:471.34
  • A25822B

    CAS:
    <p>A25822B is an antifungal agent.</p>
    Formula:C28H45NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.66
  • AP5

    CAS:
    <p>AP5: GPR40 agonist, positive allosteric modulator; rat hIP1 EC50: 0.49 nM.</p>
    Formula:C28H28FNO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:461.52
  • Cgs 25155

    CAS:
    <p>Cgs 25155 is an orally active inhibitor of NEP 24.11.</p>
    Formula:C25H34N2O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:490.61
  • ODN 21158

    CAS:
    <p>ODN 21158 is a potent, non-cytotoxic inhibitor of G-modified TLR3 and TLR9. ODN 21158 dose-dependently inhibits IFN-α secretion.</p>
    Color and Shape:Solid
  • ONL-1204

    CAS:
    <p>ONL-1204 is a small molecule, CD95 antigen inhibitor (Fas inhibitor) being developed by ONL Therapeutics for the treatment of retinal detachment.</p>
    Formula:C71H100N18O16
    Color and Shape:Solid
    Molecular weight:1461.66
  • E-3030 free acid

    CAS:
    <p>E-3030 free acid, a PPAR agonist, lowers blood glucose, triglycerides, and insulin; boosts adiponectin; reduces apo C-III; and raises lipoprotein lipase.</p>
    Formula:C22H23ClFNO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:435.87
  • BAY-7598

    CAS:
    <p>BAY-7598 is a potent, selective, and orally bioavailable MMP12 inhibitor (IC50s: 0.085, 0.67, and 1.1 nM for human/murine/rat MMP12).</p>
    Formula:C28H31N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:505.56
  • Plumbemycin B

    CAS:
    <p>Plumbemycin B is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>
    Formula:C12H21N4O8P
    Color and Shape:Solid
    Molecular weight:380.29
  • Naltrindole

    CAS:
    <p>Naltrindole is a delta opioid receptor antagonist.</p>
    Formula:C26H26N2O3
    Color and Shape:Solid
    Molecular weight:414.5
  • Turoctocog alfa

    CAS:
    <p>Turoctocog alfa: recombinant FVIII from CHO cells for hemophilia A study.</p>
    Color and Shape:Solid
  • Arverapamil

    CAS:
    <p>Arverapamil is a chiral metabolite of Verapamil.</p>
    Formula:C26H36N2O4
    Color and Shape:Solid
    Molecular weight:440.58
  • ZK824859 hydrochloride


    <p>ZK824859 hydrochloride: oral uPA inhibitor with IC50 of 79 nM (uPA), 1580 nM (tPA), 1330 nM (fibrin).</p>
    Formula:C23H23ClF2N2O4
    Color and Shape:Solid
    Molecular weight:464.89
  • β-Glucuronidase/hCAII-IN-1

    CAS:
    <p>β-Glucuronidase/hCAII-IN-2 (Compound 12e) is a compound that effectively inhibits both β-glucuronidase and human Carbonic Anhydrase II (hCA II), exhibiting IC50</p>
    Formula:C30H21NO9
    Color and Shape:Solid
    Molecular weight:539.49
  • OP-5244

    CAS:
    <p>OP-5244 has comparable potency to bisphosphonic acid series and targets CD73.</p>
    Formula:C19H29ClN5O9P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:537.89
  • CRV431

    CAS:
    <p>CRV431 is a novel Pan-Cyclophilin Inhibitor, potently inhibiting all cyclophilin isoforms tested - A, B, D, and G (IC50 values ranged from 1-7 nM).</p>
    Formula:C67H122N12O13
    Color and Shape:Solid
    Molecular weight:1303.76
  • Pomaglumetad methionil

    CAS:
    <p>Pomaglumetad methionil is an oral methionine prodrug of the potent specific agonist of mGlu2/3 receptor LY404039.</p>
    Formula:C12H20N2O8S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:384.43
  • c-Met-IN-2

    CAS:
    <p>c-Met-IN-2 is a selective and orally available c-Met inhibitor (IC50: 0.6 nM) with antitumor activity.</p>
    Formula:C24H21FN10O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:484.49
  • Imidocarb dihydrochloride monohydrate


    <p>Imidocarb dihydrochloride monohydrate is an effective antiprotozoal agent against the parasite B. bovis (IC50: 87 μg/ml).</p>
    Formula:C19H24Cl2N6O2
    Color and Shape:Solid
    Molecular weight:439.34
  • CDK7-IN-17

    CAS:
    <p>CDK7-IN-17, a pyrimidine-based CDK7 inhibitor, shows promise for various cancers, especially with abnormal transcription.</p>
    Formula:C24H26F3N6OP
    Color and Shape:Solid
    Molecular weight:502.47
  • COTC

    CAS:
    <p>COTC is an anticancer bacterial metabolite; inhibits glyoxalase with GSH, halts HeLa cell growth, and fights tumor in Ehrlich murine model.</p>
    Formula:C11H14O6
    Color and Shape:Solid
    Molecular weight:242.23
  • CEase-IN-1


    <p>CEase-IN-1 (A1H3), potent CEase inhibitor, IC50 0.36μM, for hypercholesterolemia study.</p>
    Formula:C13H15F3N2O2
    Color and Shape:Solid
    Molecular weight:288.27
  • DLK-IN-1

    CAS:
    DLK-IN-1: Oral DLK (MAP3K12) inhibitor, Ki=3nM, effective in Alzheimer's model, CNS permeable, well-tolerated with sustained brain levels.
    Formula:C20H24F3N5O2
    Color and Shape:Solid
    Molecular weight:423.43
  • Top/HDAC-IN-2


    <p>Top/HDAC-IN-2 (45b) is a dual inhibitor of Top and HDAC that induces apoptosis and exhibits significant anti-tumour effects.</p>
    Formula:C30H32N8O4
    Color and Shape:Solid
    Molecular weight:568.63
  • XIAP/cIAP1 antagonist-1


    <p>Potent oral XIAP/cIAP1 inhibitor with EC50s: XIAP 5.1 nM, cIAP1 0.32 nM; curbs tumor growth in vivo.</p>
    Color and Shape:Solid
  • EGFR-IN-24


    <p>EGFR-IN-24 is a potent inhibitor of EGFR and inhibits EGFR (del19/T790M/C797S) and EGFR (L858R/T790M/C797S).</p>
    Formula:C30H35FN6O3
    Color and Shape:Solid
    Molecular weight:546.64
  • DC41SMe

    CAS:
    <p>DC41SMe, a DC1 derivative and CC-1065 analogue, targets cancer with 18-25 pM IC50 against Ramos, Namalwa, HL60/s cells.</p>
    Formula:C38H36ClN5O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:726.31
  • SP-471


    <p>SP-471 is a potent inhibitor of dengue virus (DENV) protease (IC50: 18 μM) and inhibits the inter- and intramolecular protease processes of DENV.</p>
    Formula:C33H26BrN5
    Color and Shape:Solid
    Molecular weight:572.5
  • Lometrexol disodium

    CAS:
    <p>Lometrexol disodium: Inhibits hSHMT1/2 and GARFT, anticancer by blocking purine synthesis, induces apoptosis and cell cycle arrest.</p>
    Formula:C21H23N5Na2O6
    Color and Shape:Solid
    Molecular weight:487.424
  • Leu-AMS R enantiomer

    CAS:
    <p>Leu-AMS R enantiomer is the R enatiomer of Leu-AMS. Leu-AMS is a potent leucyl-tRNA synthetase (LRS) inhibitor that inhibits the bacteria growth.</p>
    Formula:C16H25N7O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.48
  • Exicorilant

    CAS:
    <p>Exicorilant is a selective oral GR antagonist (Ki: 7 nM) that may reduce obesity, glucose intolerance, &amp; dyslipidemia.</p>
    Formula:C26H23F4N7O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:589.56
  • SR121566A

    CAS:
    <p>SR121566A is a novel non-peptide antagonist of Glycoprotein IIb/IIIa (GP IIb-IIIa).</p>
    Formula:C20H25N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.51
  • Indinavir monohydrate

    CAS:
    <p>Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.</p>
    Formula:C36H49N5O5
    Color and Shape:Solid
    Molecular weight:631.82
  • J-104132

    CAS:
    <p>J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.</p>
    Formula:C31H33NO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.60
  • ICA-105665

    CAS:
    <p>ICA-105665 is an orally active Kv7.2/7.3/7.5 channel opener, CNS-penetrant with antiseizure effects, and low hepatocyte cytotoxicity.</p>
    Formula:C19H15F2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:355.34
  • SGLT inhibitor-1

    CAS:
    <p>SGLT inhibitor-1 is a potentsodium glucose co-transporter proteins (SGLTs) dual inhibitor(hSGLT1 and hSGLT2 with IC50s of 43 nM and 9 nM, respectively).</p>
    Formula:C24H27FO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:462.46
  • GZN39838

    CAS:
    <p>GZN39838, a natural Kv1.2 blocker, induces C-type inactivation without blocking the outer pore.</p>
    Formula:C22H30O6
    Color and Shape:Solid
    Molecular weight:390.47
  • CE-2072

    CAS:
    <p>CE-2072 is a synthetic host serine proteases inhibitor.</p>
    Formula:C33H41N5O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:603.71
  • ACT 178882

    CAS:
    <p>ACT 178882 is a new Renin inhibitor (IC50: 1.4 nM).</p>
    Formula:C33H38Cl3N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:647.03