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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66687 products of "Inhibitors"

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  • PDHK-IN-4


    PDHK-IN-4 inhibits PDHK2 (IC50: 0.0051 μM) & PDHK4 (IC50: 0.0122 μM), with potential for cancer research.
    Formula:C24H25N5O3
    Color and Shape:Solid
    Molecular weight:431.49
  • MDK-3298

    CAS:
    MDK-3298 is a reversible covalent inhibitor of Mcl-1, a target of protein-protein interaction (PPI).
    Formula:C35H32BN3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:617.46
  • Mifepristone methochloride

    CAS:
    Mifepristone methochloride is a glucocorticoid antagonist. This product will be sold for research use only.
    Formula:C30H38ClNO2
    Color and Shape:Solid
    Molecular weight:480.08
  • WAY-855

    CAS:
    WAY-855 is an EAAT2-preferring, nonsubstrate inhibitor of high-affinity glutamate uptake.
    Formula:C9H11NO4
    Color and Shape:Solid
    Molecular weight:197.19
  • E6201

    CAS:
    E6201, a dual kinase inhibitor, blocks MEK1/FLT3 and has anti-tumor/psoriasis effects with low IC50s: ERK2 (5.2 nM), JNK (91 nM), p38 MAPK (19 nM).
    Formula:C21H27NO6
    Color and Shape:Solid
    Molecular weight:389.44
  • EGFR-IN-17


    EGFR-IN-17: potent, selective EGFR inhibitor, IC50 of 0.2 nM, overcomes C797S drug resistance.
    Formula:C27H31ClN7O3P
    Color and Shape:Solid
    Molecular weight:568.01
  • Antitumor agent-58


    Antitumor agent-58 suppresses tumor growth, colony formation, cell migration, and induces mitochondrial dysfunction in MGC-803 cells.
    Formula:C27H28F3N9S
    Color and Shape:Solid
    Molecular weight:567.63
  • CDK1-IN-5


    CDK1-IN-5 is a selective inhibitor for CDK1 (IC50: 42.19 nM), CDK2, CDK5, halting cancer cell growth.
    Formula:C27H26ClN5OS
    Color and Shape:Solid
    Molecular weight:504.05
  • Antileishmanial agent-4


    Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].
    Formula:C17H18N4O4
    Color and Shape:Solid
    Molecular weight:342.35
  • PPARγ agonist 1


    PPARγ agonist 1 is a potent agonist of PPARγ that efficiently activates hPPARγ without causing full agonism, thereby avoiding adverse effects.
    Formula:C34H39NO3
    Color and Shape:Solid
    Molecular weight:509.68
  • M-525

    CAS:
    M-525, a potent first-in-class menin-MLL inhibitor, binds at 3 nM IC50 and curbs MLL leukemia cell growth & gene expression.
    Formula:C39H51FN6O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:734.92
  • Rpi 856 C

    CAS:
    Rpi 856 C is a retrovirus protease inhibitor from Streptomyces that is effective against HIV-1 and HTLV-1 proteases.
    Formula:C39H56N6O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:768.90
  • LJ-4517


    LJ-4517 is an effective A2AAR antagonist (Ki=18.3 nM). LJ-4517 can effectively replace the binding of [3H] ZM241385 at WT A2AAR.
    Formula:C19H21N5O3S
    Color and Shape:Solid
    Molecular weight:399.47
  • BDZ-h

    CAS:
    BDZ-h inhibits both closed/open states of all 4 homomeric & 2 GluA2R-complex AMPA receptors.
    Formula:C21H21N5O3S
    Color and Shape:Solid
    Molecular weight:423.49
  • UCN-01

    CAS:
    inhibitor of Akt, protein kinase C, PDK1 and cyclin-dependent kinases
    Formula:C28H26N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:482.53
  • G12Si-1


    G12Si-1 selectively binds and inhibits K-Ras(G12S) to block oncogenic signaling and nucleotide exchange.
    Formula:C29H32ClN5O3
    Color and Shape:Solid
    Molecular weight:534.05
  • TD-0212

    CAS:
    TD-0212: Oral dual antagonist for AT1 (pKi 8.9) & NEP inhibitor (pIC50 9.2).
    Formula:C28H34FN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:527.65
  • CCT369260

    CAS:
    CCT369260 (compound 1), an orally active inhibitor targeting B-cell lymphoma 6 (BCL6), demonstrates anti-tumor efficacy with an IC50 value of 520 nM [1].
    Formula:C24H31ClF2N6O2
    Color and Shape:Solid
    Molecular weight:508.99
  • DYRKs-IN-1 hydrochloride

    CAS:
    DYRKs-IN-1 HCl inhibits DYRK1A (5 nM IC50) & DYRK1B (8 nM IC50) with antitumor properties.
    Formula:C30H31Cl2N7O4
    Color and Shape:Solid
    Molecular weight:624.52
  • Befiradol hydrochloride

    CAS:
    <p>Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 aggregation.</p>
    Formula:C20H23Cl2F2N3O
    Purity:99.1%
    Color and Shape:Solid
    Molecular weight:430.32