Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,763 products)
- Apoptosis(6,205 products)
- Cell Cycle/Checkpoint(4,812 products)
- Chromatin/Epigenetics(2,553 products)
- Cytoskeletal Signaling(1,520 products)
- DNA Damage/DNA Repair(2,906 products)
- Endocrinology/Hormones(3,703 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,965 products)
- Immunology and Inflammation(3,749 products)
- Influenza Virus(297 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,244 products)
- Membrane Transporter/Ion Channel(3,118 products)
- Metabolism(10,123 products)
- Microbiology/Virology(7,569 products)
- Neuroscience(10,314 products)
- Other Inhibitors(35,804 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,411 products)
- Proteases/Proteasome(1,681 products)
- Stem Cell and Derivatives(752 products)
- Tyrosine Kinase/Adaptors(1,947 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66604 products of "Inhibitors"
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DN02
DN02: a potent, selective BRD8(1) bromodomain probe; Ki=32 nM; 30x more affine than BRD8(2).Formula:C22H24FN3O3Purity:98.22% - 99.74%Color and Shape:SolidMolecular weight:397.44Milademetan
CAS:Milademetan (DS-3032), an MDM2 inhibitor, exhibits antitumor activity, induces G1 cell cycle arrest and apoptosis, and can be used to study solid tumors.Formula:C30H34Cl2FN5O4Purity:>99.99%Color and Shape:SolidMolecular weight:618.53Ref: TM-T12040
1mg93.00€5mg167.00€10mg260.00€25mg492.00€50mg802.00€100mg1,378.00€1mL*10mM (DMSO)221.00€VX-984
CAS:VX-984 (M9831) is an oral DNA-PK inhibitor, crossing the blood-brain barrier, targeting GBM and NSC-LC.Formula:C23H21D2N7OPurity:97.65% - 99.98%Color and Shape:SolidMolecular weight:415.49Ref: TM-T11067
1mg117.00€5mg248.00€10mg369.00€25mg575.00€50mg863.00€100mg1,305.00€200mg1,755.00€1mL*10mM (DMSO)271.00€LLY-283
CAS:LLY-283, PRMT5 inhibitor, IC50 22 nM, Kd 6 nM, oral, selective, with antitumor effects.Formula:C17H18N4O4Purity:99.49%Color and Shape:SolidMolecular weight:342.35Picrotoxinin
CAS:Picrotoxinin blocks chloride channels, antagonizes GABAA noncompetitively (IC50: 1.15 μM, α1β2γ2L), and induces convulsions.Formula:C15H16O6Purity:98.07%Color and Shape:SolidMolecular weight:292.28BAY-3827
CAS:BAY-3827 is an AMPK inhibitor with antiproliferative activity and antitumor activity. BAY-3827 inhibits the phosphorylation of acetyl CoA carboxylase 1.Formula:C27H25FN6OPurity:99.90%Color and Shape:SolidMolecular weight:468.53Ref: TM-T73350
1mg56.00€5mg119.00€10mg187.00€25mg354.00€50mg590.00€100mg835.00€500mg1,663.00€1mL*10mM (DMSO)124.00€ELOVL1-IN-2
CAS:ELOVL1-IN-2 weakly inhibits ELOVL1 enzyme (IC50: 21 μM) and shows moderate potency in HEK293 cells (IC50: 6.7 μM).Formula:C18H15FN2OPurity:99.94%Color and Shape:SolidMolecular weight:294.32AZD-5672
CAS:AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.Formula:C32H38F2N2O5S2Purity:98.1%Color and Shape:SolidMolecular weight:632.78Ref: TM-T30260
1mg192.00€5mg434.00€10mg610.00€25mg888.00€50mg1,243.00€100mg1,693.00€1mL*10mM (DMSO)530.00€Cbl-b-IN-3
CAS:Cbl-b-IN-3 is a potent inhibitor of casitas b lineage lymphoma proto-oncogene-b (Cbl-b) (ic50 < 1 nM).Cost-effective and quality-assured.Formula:C30H34F3N5OPurity:97.63%Color and Shape:SolidMolecular weight:537.62Ref: TM-T63790
1mg70.00€5mg154.00€10mg202.00€25mg384.00€50mg590.00€100mg944.00€1mL*10mM (DMSO)175.00€NRX-103095
CAS:NRX-103095 increases β-catenin binding to SCFβ-TrCP E3 ligase; EC50 is 163 nM for pSer33/Ser37 affinity boost.Formula:C22H16Cl2F3N3O3SPurity:99.85% - 99.95%Color and Shape:SolidMolecular weight:530.35Ref: TM-T63730
1mg142.00€5mg344.00€10mg557.00€25mg1,108.00€50mg1,783.00€100mg2,673.00€1mL*10mM (DMSO)404.00€CCF0058981
CAS:CCF0058981: noncovalent inhibitor for SARS-CoV-2 & -1 proteases; IC50s: 68 nM (SC2) & 19 nM (SC1). Potential COVID-19 research use.
Formula:C24H19ClN6OPurity:98.94%Color and Shape:SoildMolecular weight:442.9Ref: TM-T60095
1mg46.00€2mg60.00€5mg92.00€10mg160.00€25mg324.00€50mg449.00€100mg562.00€500mgTo inquireAldometanib
CAS:Aldometanib (LXY-05-029) is an oral aldolase inhibitor that maintains metabolic balance by blocking FBP and activating lysosomal AMPK.Formula:C27H43Cl2IN2Purity:99.32% - 99.55%Color and Shape:SolidMolecular weight:593.46BAY-8400
BAY-8400 is an orally active, potent and selective DNA-dependent protein kinase ( DNA-PK ) inhibitor ( IC 50 =81 nM) which shows synergistic efficacy inFormula:C21H17F2N5OPurity:99.53%Color and Shape:SolidMolecular weight:393.39Ref: TM-T9498
1mg80.00€5mg147.00€10mg215.00€25mg439.00€50mg750.00€100mg1,009.00€1mL*10mM (DMSO)161.00€Rineterkib
CAS:Rineterkib (ERK-IN-1) is an inhibitor of RAF and ERK1/2 activating mutations in the MAPK pathway.Formula:C26H27BrF3N5O2Purity:99.73%Color and Shape:SolidMolecular weight:578.42Ref: TM-T11224
1mg87.00€5mg170.00€10mg318.00€25mg538.00€50mg765.00€100mg1,035.00€1mL*10mM (DMSO)224.00€XMD-17-51 Trifluoroacetate
CAS:XMD-17-51 Trifluoroacetate is a pyrimido-diazepinone compound that regulates protein kinases.Formula:C23H25F3N8O3Purity:99.65%Color and Shape:SolidMolecular weight:518.49FGI-106 tetrahydrochloride
CAS:FGI-106 tetrahydrochloride demonstrates potent inhibitory activity across a broad spectrum of viruses, including those causing hemorrhagic fevers such as EbolaFormula:C28H42Cl4N6Purity:99.68%Color and Shape:SolidMolecular weight:604.48Ref: TM-T11281L
1mg82.00€5mg161.00€10mg245.00€25mg406.00€50mg572.00€100mg772.00€200mg1,035.00€1mL*10mM (DMSO)207.00€TGFβRI-IN-3
CAS:TGFβRI-IN-3 inhibits TGFβR1 with an IC 50 of 0.79 nM with 2000-fold selectivity against MAP4K4.Formula:C28H23N3O2SPurity:99.85%Color and Shape:SoildMolecular weight:465.57Ref: TM-T9523
1mg84.00€5mg177.00€10mg281.00€25mg552.00€50mg859.00€100mg1,234.00€500mg2,457.00€1mL*10mM (DMSO)177.00€Gemcitabine elaidate hydrochloride
CAS:CP-4126, a lipophilic pro-drug of Gemcitabine, converts to active form by esterases, allowing oral administration with dose-dependent effects.
Formula:C27H44ClF2N3O5Purity:98.50% - 99.6%Color and Shape:SolidMolecular weight:564.11Rolapitant hydrochloride
CAS:Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.Formula:C25H27ClF6N2O2Purity:98.35% - 99.79%Color and Shape:SolidMolecular weight:536.94Ref: TM-T3724
1mg153.00€5mg365.00€10mg520.00€25mg780.00€50mg1,054.00€100mg1,425.00€200mg1,882.00€1mL*10mM (DMSO)439.00€BRD0639
CAS:BRD0639 is a first-in-class PRMT5-substrate interaction inhibitor for PBM-dependent PRMT5 activity studies.Formula:C21H22ClN5O4SPurity:99.85%Color and Shape:SolidMolecular weight:475.95
