Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,657 products)
- Apoptosis(6,058 products)
- Cell Cycle/Checkpoint(4,657 products)
- Chromatin/Epigenetics(2,354 products)
- Cytoskeletal Signaling(1,460 products)
- DNA Damage/DNA Repair(2,908 products)
- Endocrinology/Hormones(3,601 products)
- Enzyme(3,655 products)
- GPCR/G-Protein(8,703 products)
- Immunology and Inflammation(3,737 products)
- Influenza Virus(298 products)
- JAK/STAT signaling(403 products)
- MAPK Signaling(1,227 products)
- Membrane Transporter/Ion Channel(2,922 products)
- Metabolism(9,881 products)
- Microbiology/Virology(7,303 products)
- Neuroscience(10,209 products)
- Other Inhibitors(36,770 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,430 products)
- Proteases/Proteasome(1,669 products)
- Stem Cell and Derivatives(828 products)
- Tyrosine Kinase/Adaptors(2,042 products)
- Ubiquitination(1,681 products)
Show 16 more subcategories
Found 66609 products of "Inhibitors"
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CXCR2 antagonist 2
CAS:<p>CXCR2 antagonist 2 is a potent CXCR2 antagonist for cancer immunotherapy with an IC 50 value of 95 nM.</p>Formula:C17H17FN2O4SColor and Shape:SolidMolecular weight:364.39TM2 TEAD inhibitor
CAS:TM2 TEAD inhibitor, a robust and reversible inhibitor of the TEA domain transcription factor, presents dual inhibitory concentrations (IC50) of 38 nM for TEAD4Formula:C26H33N3O3Purity:99.91%Color and Shape:SolidMolecular weight:435.57L 659837
CAS:<p>L 659837 is an antagonist of ANC-2, lactam, and tackykinin.</p>Formula:C40H52N8O7SColor and Shape:SolidMolecular weight:788.96SAFit1
CAS:SAFit1 is an inhibitor of FK506 binding protein 51 (FKBP51)-specific (Ki: 4±0.3 nM).Formula:C42H53NO11Purity:98%Color and Shape:SolidMolecular weight:747.87(E)-LHF-535
CAS:(E)-LHF-535, an E-isomer antiviral, EC50 <1 μM vs Lassa/Machupo/Junin, 1-10 μM vs VSVg.Formula:C27H28N2O2Purity:98%Color and Shape:SolidMolecular weight:412.52L 694746
CAS:L 694746 is an inhibitor of HIV-1 protease.Formula:C35H42N2O8Purity:98%Color and Shape:SolidMolecular weight:618.72SAS-0132
CAS:<p>SAS-0132 is a modulator/antagonist of sigma2R/TMEM97 and has potential for treating TBIs, Alzheimer's disease, and neuropathic pain.</p>Formula:C24H29N3O2Color and Shape:SolidMolecular weight:391.51AMB639752
CAS:AMB639752 is a potent inhibitor of diacylglycerol kinase alpha (DGKα) that reinstates restimulation-induced cell death (RICD) in SAP-deficient lymphocytesFormula:C21H23N3O3Color and Shape:SolidMolecular weight:365.43SB-201076
CAS:<p>SB-201076 is a potent ATP citrate-lyase inhibitor. SB-204990 is the prodrug of SB-201076.</p>Formula:C18H24Cl2O6Color and Shape:SolidMolecular weight:407.29TNH
CAS:<p>TNH, a dimeric compound, possesses the ability to penetrate living cells and facilitate the recruitment of proteins into cellular structures [1].</p>Formula:C39H57ClN6O13Color and Shape:SolidMolecular weight:853.36WAY-325811
CAS:<p>WAY-325811 is an active pharmaceutical compound.</p>Formula:C18H18N2O2SColor and Shape:SolidMolecular weight:326.41Olgotrelvir
CAS:<p>Olgotrelvir is an antiviral agent [1].</p>Formula:C22H30N4O7SColor and Shape:SolidMolecular weight:494.56SAR502250
CAS:<p>SAR502250: potent, selective GSK3 inhibitor, IC50=12nM, oral, brain-penetrant, potential for AD research, antidepressant-like properties.</p>Formula:C19H18FN5O2Color and Shape:SolidMolecular weight:367.38HD-2a
CAS:<p>HA-2a inhibits the JAK2/STAT3 pathway by downregulating circDcbld2 expression in RAW264.7 cells [1].</p>Formula:C18H18O6Color and Shape:SolidMolecular weight:330.33Wieland-gumlich aldehyde
CAS:Wieland-Gumlich aldehyde is an indoline derived by chemical degradation from strychnine.Formula:C19H22N2O2Color and Shape:SolidMolecular weight:310.39Tiracizine HCl
CAS:<p>Tiracizine HCl, a new class I antiarrhythmic drug, was studied in patients with ischemic heart disease and shown to decrease myocardial contractile function.</p>Formula:C21H26ClN3O3Purity:98%Color and Shape:SolidMolecular weight:403.9OBBA
CAS:<p>OBBA is a phospholipase A2 antagonist.</p>Formula:C28H44O3Color and Shape:SolidMolecular weight:428.65Tuberculosis inhibitor 8
CAS:<p>Tuberculosis inhibitor 8 (compound 3b), a 3-methoxy-2-phenylimidazo[1,2-b]pyridazine derivative, exhibits potent activity against both Mycobacterium</p>Formula:C21H19FN4OColor and Shape:SolidMolecular weight:362.4STA-9584
CAS:<p>STA-9584, a vascular disrupting agent with a potent antitumor effect, targets tumor microvasculature and outperforms CA4P in certain cancer models.</p>Formula:C28H29N3O6Color and Shape:SolidMolecular weight:503.55Antitumor agent-66
CAS:<p>Antitumor agent-66 (Compound 4) is a derivative of (-)-cleistenolide, showcasing potential as a research tool for cancer diseases [1].</p>Formula:C18H17ClO8Color and Shape:SolidMolecular weight:396.78Sezolamide
CAS:<p>Sezolamide is a carbonic anhydrase inhibitor.</p>Formula:C11H18N2O4S3Color and Shape:SolidMolecular weight:338.47AR-L 100 BS
CAS:AR-L 100 BS is a bioactive chemical with cardiovascular effects and blood pressure.Formula:C16H17N3O3SColor and Shape:SolidMolecular weight:331.39Gliamilide
CAS:Gliamilide is a high-potency sulfamylurea hypoglycemic agent.Formula:C23H33N5O5SColor and Shape:SolidMolecular weight:491.6SARS-CoV-2 3CLpro-IN-10
<p>SARS-CoV-2 3CLpro-IN-10(5d) inhibits 3CL protease: 190 nM (SARS-CoV-2), 790 nM (SARS-CoV-1), 70 nM (MERS-CoV), and has broad-spectrum antiviral effects.</p>Formula:C24H33FN3NaO8SColor and Shape:SolidMolecular weight:565.59Fenquinotrione
CAS:Fenquinotrione, a 4-hydroxyphenylpyruvate dioxygenase (HPPD) inhibitor, exhibits IC50 values of 27.2 and 44.7 nM against HPPD from rice and Arabidopsis thalianaFormula:C22H17ClN2O5Color and Shape:SolidMolecular weight:424.83STING agonist-18
CAS:<p>STING Agonist-18 (Compound 1a) is a precursor for the synthesis of antibody-drug conjugates (ADCs), including Trastuzumab conjugates [1].</p>Formula:C38H45N13O6Color and Shape:SolidMolecular weight:779.85WAY-300569
CAS:<p>N-(3-Fluorophenyl)-3-(4-oxo-5-(thiophen-2-ylmethylene)-2-thioxothiazolidin-3-yl)propanamide is a chemical compound with biological activity.</p>Formula:C17H13FN2O2S3Color and Shape:SolidMolecular weight:392.49L 738167
CAS:<p>L 738167 is a potent antagonist of the long-acting fibrinogen receptor.</p>Formula:C25H34N6O6SColor and Shape:SolidMolecular weight:546.64RX-RA 85
CAS:<p>RX-RA 85 is a pyrimido-pyrimidine derivative that is an inhibitor of platelet and tumor phosphodiesterase.</p>Formula:C22H27N7OS2Color and Shape:SolidMolecular weight:469.63Dinophysistoxin 1
CAS:Dinophysistoxin 1 (DTX 1, 35-methylokadaic acid), a causative agent of diarrhetic shellfish poisoning, exhibits tumor-promoting activity and also acts as a skinFormula:C45H70O13Color and Shape:SolidMolecular weight:819.03KRAS inhibitor-11
<p>KRAS inhibitor-11 is a KRAS inhibitor .</p>Formula:C29H47N9O6Color and Shape:SolidMolecular weight:617.74HPK1-IN-9
CAS:HPK1-IN-9: Potent MAP4K family kinase inhibitor targeting hematopoietic progenitor cells; potential in HPK1 diseases. (Patent WO2021213317A1)Formula:C30H33N7O2Color and Shape:SolidMolecular weight:523.63Caroverine
CAS:Caroverine is a potential chemotherapeutical agent in HNSCC cell lines.Formula:C22H27N3O2Color and Shape:SolidMolecular weight:365.47Crobenetine hydrochloride
CAS:<p>Crobenetine hydrochloride, a sodium channel antagonist, is used potentially for the treatment of stroke.</p>Formula:C25H34ClNO2Color and Shape:SolidMolecular weight:416ICMT-IN-24
CAS:ICMT-IN-24 (compound 63) is an inhibitor of isoprenylcysteine carboxyl methyltransferase (ICMT), exhibiting potent activity with an IC50 value of 0.19 μM [1].Formula:C22H28ClNO2Color and Shape:SolidMolecular weight:373.92INX-SM-6
CAS:<p>INX-SM-6, a chemical compound, serves as a targeted delivery vehicle for anti-inflammatory agents and has shown efficacy in suppressing LPS-induced IL-1β</p>Formula:C32H36N2O6SColor and Shape:SolidMolecular weight:576.7CI-959 free acid
CAS:<p>CI-959 Free Acid is an orally effective inhibitor of cell activation in vitro and in animal models and also has anti-allergic/anti-inflammatory properties.</p>Formula:C14H15N5O3SColor and Shape:SolidMolecular weight:333.37ZINC08792355
CAS:ZINC08792355 is a novel inhibitor of SIRT1.Formula:C31H24N4O3Color and Shape:SolidMolecular weight:500.5515(S)-HEDE
CAS:<p>15(S)-HEDE is produced from 11Z,14Z-eicosadienoic acid by 15-LO. 15(S)-HEDE is an inhibitor of RBL-1 cell 5-LO with an IC50 value of 26 μM.</p>Formula:C20H36O3Color and Shape:SolidMolecular weight:324.5Biotin-hexanamide-(L-Thyroxine)
CAS:Biotin-hexanamide-(L-Thyroxine) is a biotinylated derivative of L-Thyroxine (Levothyroxine; T4), utilized as a synthetic hormone in hypothyroidism research [1].Formula:C31H36I4N4O7SColor and Shape:SolidMolecular weight:1116.32Tomicorat
CAS:<p>Tomicorat is an anti-inflammatory agent.</p>Formula:C32H30FNO5Color and Shape:SolidMolecular weight:527.58Anticancer agent 107
CAS:Compound 107 (Compd 11jc) exhibits potent antitumor activity and serves as an effective anticancer agent in the investigation of pulmonary metastatic melanoma [Formula:C24H19N3O4SColor and Shape:SolidMolecular weight:445.49Antibiofilm agent-2
CAS:<p>Antibiofilm Agent-2 (Compound 4T) serves as a potent biofilm inhibitor, exhibiting an IC50 of 3.6 μM, and impairs the quorum sensing system along with iron</p>Formula:C17H21NO5Color and Shape:SolidMolecular weight:319.35MK-8666
CAS:<p>MK-8666, a partial GPCR agonist targeting GPR40, may treat type 2 diabetes by enhancing insulin secretion and lowering glucose safely.</p>Formula:C29H31NO6SColor and Shape:SolidMolecular weight:521.62Org 43553
CAS:<p>Org 43553: oral LMW LH-R agonist; targets LH (EC50: 3.7nM) & FSH (EC50: 110nM); useful for endocrine research.</p>Formula:C24H30N6O3S2Color and Shape:SolidMolecular weight:514.6612R-LOX-IN-1
CAS:12R-LOX-IN-1 (Compound 4a), with an IC50 of 28.25 µM, is an inhibitor of 12R-LOX.Formula:C15H11NO2Color and Shape:SolidMolecular weight:237.255-Iodo-indirubin-3'-monoxime
CAS:5-Iodo-indirubin-3'-monoxime is a potent GSK-3β, CDK5/P25 and CDK1/cyclin B inhibitor, competing with ATP for binding to the catalytic site of the kinase (IC50sFormula:C16H10IN3O2Color and Shape:SolidMolecular weight:403.17FGFR-IN-4
CAS:<p>FGFR-IN-4 is a potent inhibitor of FGFR. FGFR-IN-4 has potential for cancer disease studies.</p>Formula:C24H21N7O2Color and Shape:SolidMolecular weight:439.47Sunepitron HCl
CAS:<p>Sunepitron is a combined α2-adrenergic receptor antagonist and 5-HT1A receptor agonist.</p>Formula:C17H24ClN5O2Color and Shape:SolidMolecular weight:365.86Anticancer agent 112
CAS:<p>Anticancer agent 112[1], serves as a potent agent for cancer research.</p>Formula:C27H32ClN7OColor and Shape:SolidMolecular weight:506.04Duocarmycin analog-2
CAS:<p>Duocarmycin analog-2 is a potent DNA alkylating agent that exhibits antitumor effects and can be used in the synthesis of immunocouplers.</p>Formula:C29H23ClN4O3Color and Shape:SolidMolecular weight:510.97APJ receptor agonist 7
CAS:<p>APJ receptor agonist 7 (compound 37) is an orally active APJ (apelin receptor) agonist (Ki: 0.059 μM). arrestin (EC50: 0.063 μM).</p>Formula:C32H46N4O4Color and Shape:SolidMolecular weight:550.73Zabofloxacin
CAS:Zabofloxacin inhibits bacterial topoisomerases II/IV, effectively targeting gram-positive pathogens like S. aureus and S. pneumoniae.Formula:C19H20FN5O4Purity:98%Color and Shape:SolidMolecular weight:401.39ICMT-IN-2
CAS:ICMT-IN-2 (compound 45) serves as an ICMT inhibitor with an IC50 value of 0.168 μM [1].Formula:C21H26FNOColor and Shape:SolidMolecular weight:327.44(1s,4s)-Menin-MLL inhibitor-23
<p>(1s,4s)-Menin-MLL Inhibitor-23, an enantiomer of Menin-MLL Inhibitor-23 (Example 99A), functions as an inhibitor of the menin-MLL interaction [1].</p>Formula:C36H53FN6O4Color and Shape:SolidMolecular weight:652.84Artonin E
CAS:<p>Artonin E, a prenylated flavonoid, induces apoptosis and S-phase arrest, disrupting the mitochondrial pathway for cancer research.</p>Formula:C25H24O7Color and Shape:SolidMolecular weight:436.45TAC 363
CAS:<p>TAC 363 is a tachykinin NK-2-receptor antagonist.</p>Formula:C38H48N8O6Color and Shape:SolidMolecular weight:712.84L 163255
CAS:<p>L 163255 is a type of growth hormone secretagogue (GHS).</p>Formula:C28H38N4O4SColor and Shape:SolidMolecular weight:526.69LY 255262
CAS:<p>LY 255262 is an antibacterial agent in the class of pyrazolidinone.</p>Formula:C14H13N7O5SColor and Shape:SolidMolecular weight:391.36Flavokawain 1i
CAS:Flavokawain 1i, a derivative of chalcones flavokawain A, flavokawain B, and flavokawain C, exhibits anticancer and antiviral properties.Formula:C21H18O4Color and Shape:SolidMolecular weight:334.3715-PGDH-IN-1
CAS:15-PGDH-IN-1: potent oral 15-PGDH inhibitor, IC50=3nM, useful for tissue repair research.Formula:C24H22N4O2Color and Shape:SolidMolecular weight:398.46WAY-300570
CAS:N-(4-Chlorophenyl)-3-(4-oxo-5-(thiophen-2-ylmethylene)-2-thioxothiazolidin-3-yl)propanamide is an active chemical compound characterized by its complexFormula:C17H13ClN2O2S3Color and Shape:SolidMolecular weight:408.95SOS1-IN-7
CAS:SOS1-IN-7 (compound 18-p1) is a potent inhibitor of SOS1 and acts on SOS1-G12D (IC50: 20 nM) and SOS1-G12V (IC50: 67 nM).Formula:C23H25F3N4O3Color and Shape:SolidMolecular weight:462.467-Deaza-2',3'-dideoxyguanosine
CAS:<p>7-Deaza-2',3'-dideoxyguanosine (7-Deaza-ddG) is a 2′,3′-dideoxynucleoside 5′-triphosphate that inhibits HIV-1 reverse transcriptase with a Ki of 25 nM [1].</p>Formula:C11H14N4O3Color and Shape:SolidMolecular weight:250.25(Rac)-BRD0705
CAS:<p>(Rac)-BRD0705 is a less active racemate of BRD0705. BRD0705 is an effective and selective inhibitor of GSK3α.</p>Formula:C20H23N3OPurity:99.7%Color and Shape:SolidMolecular weight:321.42Disoxaril
CAS:<p>Disoxaril (BRN 3626820, WIN 51711), an anti-picornavirus, blocks enterovirus by targeting VP1; boosts poliovirus inhibition with Ambioxime, Bioxazole.</p>Formula:C20H26N2O3Color and Shape:SolidMolecular weight:342.43sEH/AChE-IN-3
CAS:sEH/AChE-IN-3 -15: potent dual sEH & AChE inhibitor; crosses BBB; IC50: hsEH 0.4nM, hAChE 1.94nM, hBChE 615nM, msEH 4.3nM, mAChE 2.61nM.Formula:C35H39ClF3N5O3Color and Shape:SolidMolecular weight:670.16PI3K/HDAC-IN-2
CAS:<p>PI3K/HDAC-IN-2: dual inhibitor with IC50s - PI3Kα: 226nM, β: 279nM, γ: 467nM, δ: 29nM; HDAC1: 1.3nM. Selective to PI3Kδ/class I/IIb HDAC, anticancer.</p>Formula:C23H23N7O4Color and Shape:SolidMolecular weight:461.47DXR Inhibitor 11a (free acid)
CAS:<p>DXR inhibitor 11a, with an IC50 of 0.11 µM, effectively inhibits P.</p>Formula:C10H12NO5PColor and Shape:SolidMolecular weight:257.20Vonifimod
CAS:<p>Vonifimod is an immunomodulator .</p>Formula:C17H34N4O2Color and Shape:SolidMolecular weight:326.48ICL-CCIC-0019
CAS:<p>ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.</p>Formula:C26H44Br2N4Purity:99.54%Color and Shape:SolidMolecular weight:572.46DGKζ-IN-4
CAS:DGKζ-IN-4 is a DGK-zeta inhibitor employed as an active ingredient in pharmaceutical formulations designed to treat cancers linked to immune cell activation orFormula:C23H25ClF3N3O6Color and Shape:SolidMolecular weight:531.91I-BET469
CAS:I-BET469 is a Bromodomain and Extraterminal Inhibitor with a Low Predicted Human Dose.Formula:C23H30N4O4Color and Shape:SolidMolecular weight:426.51H-201-70
CAS:<p>H-201-70 is a partial beta1 agonist with adrenoreceptor stimulatory effects.</p>Formula:C23H39N3O6Color and Shape:SolidMolecular weight:453.57ICMT-IN-14
CAS:ICMT-IN-14 (compound 50) serves as an inhibitor of isoprenylcysteine carboxyl methyltransferase (ICMT), exhibiting potent activity with an IC50 of 0.025 μM [1].Formula:C21H25ClFNOColor and Shape:SolidMolecular weight:361.88RO-5328673
CAS:<p>RO-5328673 is a high-affinity, insurmountable dual NK2/NK3 antagonist with fast kinetics, affecting dopaminergic activity and reversing locomotion in gerbils.</p>Formula:C29H32Cl2FN3O4Color and Shape:SolidMolecular weight:576.49Kuwanon T
CAS:<p>Kuwanon T, an isoprenylated flavonoid extracted from the root bark of Morus alba, exhibits protective effects against t-BHP-induced oxidative stress, presenting</p>Formula:C25H26O6Color and Shape:SolidMolecular weight:422.47Indacaterol xinafoate
CAS:<p>Indacaterol xinafoate is an ultra-long-acting beta-adrenoceptor agonist.</p>Formula:C35H36N2O6Color and Shape:SolidMolecular weight:580.67Himbacine
CAS:<p>Himbacine is a muscarine receptor antagonist.</p>Formula:C22H35NO2Color and Shape:SolidMolecular weight:345.52NT113
CAS:NT113: ERBB inhibitor, penetrates brain, hinders GBM growth (high EGFR/EGFRvIII), targets ERBB/Akt phosphorylation in vivo/in vitro.Formula:C27H25ClFN5O2Color and Shape:SolidMolecular weight:505.97GSK2647544
CAS:<p>GSK2647544 inhibits Lp-PLA2, a pro-inflammatory enzyme from macrophages, orally active, calcium-independent.</p>Formula:C24H18ClF3N4O3Color and Shape:SolidMolecular weight:502.87FAP Ligand 1
CAS:FAP Ligand 1 (FL), a high-affinity small molecule targeting fibroblast activation protein (FAP), facilitates the delivery of conjugated therapeutics to FAP-Formula:C15H17F2N5O2Color and Shape:SolidMolecular weight:337.32Plomestane
CAS:<p>Plomestane is a selective inhibitor of aromatization in human breast tissue and may provide a mechanism for controlling estrogen responsive processes.</p>Formula:C21H26O2Color and Shape:SolidMolecular weight:310.43L-697661
CAS:L-697661, a reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.Formula:C16H15Cl2N3O2Color and Shape:SolidMolecular weight:352.22SM-1295
CAS:SM-1295: IAP antagonist, Kd 3077 nM XIAP-BIR3, 3.2 nM c-IAP1-BIR3, 9.5 nM c-IAP2-BIR3.Formula:C29H36BrN5O4Color and Shape:SolidMolecular weight:598.53ATM-IN-1
CAS:<p>ATM-IN-1 is a potent inhibitor of ATM. ATM-IN-1 has shown research potential in cancer and neurological diseases.</p>Formula:C30H36N6O3Color and Shape:SolidMolecular weight:528.65GYKI-46903 HCl
CAS:GYKI-46903 is a noncompetitive 5-HT3 receptor antagonist.Formula:C17H21ClFNO2Color and Shape:SolidMolecular weight:325.81AZD 4017
CAS:AZD 4017 is an inhibitor of 11β-Hydroxysteroid Dehydrogenase Type 1(11β-HSD1) (IC50: 7 nM).Formula:C22H33N3O3SPurity:99.61%Color and Shape:SolidMolecular weight:419.58LMP7-IN-2
CAS:<p>LMP7-IN-2 is an inhibitor of LMP7 and may be utilized in the treatment of associated inflammatory diseases and disorders [1].</p>Formula:C28H27N3O3SColor and Shape:SolidMolecular weight:485.6PTC725
CAS:PTC725 is a selective HCV 1b replicons inhibitor. It has been shown to target the nonstructural protein 4B.Formula:C23H18F4N6O2SPurity:98%Color and Shape:SolidMolecular weight:518.49JNK3 inhibitor-1
CAS:JNK3 inhibitor-1: potent, selective, IC50 of 0.005 μM, orally bioavailable, brain-penetrant.Formula:C21H17ClFN5O2SColor and Shape:SolidMolecular weight:457.91JNJ-19567470
CAS:JNJ-19567470 is a selective, non-peptide CRF receptor 1 antagonist.Formula:C22H27BrN4OColor and Shape:SolidMolecular weight:443.38Keap1-Nrf2-IN-16
CAS:<p>Keap1-Nrf2-IN-16 is a biologically active peptide with KEAP1 binding activity.</p>Formula:C73H114N16O26Color and Shape:SolidMolecular weight:1631.78SR11237
CAS:<p>SR11237 is a Pan retinoid X receptor (RXR) agonist.</p>Formula:C24H28O4Purity:98.79%Color and Shape:SolidMolecular weight:380.48WAY-648936
CAS:WAY-648936 is an active compound.Formula:C17H21N3O4Color and Shape:SolidMolecular weight:331.37Immuno modulator-1
CAS:Immuno modulator-1 (compound 22) effectively suppresses the secretion of TNFα and IL-2 in human peripheral blood mononuclear cells (hPBMC) with IC50 values of 4Formula:C32H31FN6O4Color and Shape:SolidMolecular weight:582.62TOP1362
CAS:<p>TOP1362: a kinase inhibitor for dry eye and ocular inflammation; targets p38α, Syk, Src, Lck; reduces cytokines and cell infiltration.</p>Formula:C43H51N7O8SColor and Shape:SolidMolecular weight:825.97WAY-324572
CAS:WAY-324572 is an active compound.Formula:C20H21FN2OColor and Shape:SolidMolecular weight:324.397'-Hydroxy ABA
CAS:<p>7'-Hydroxy ABA (7'-OH ABA), a metabolite of Abscisic acid (ABA), arises from the hydroxylation at the 7'-carbon of ABA.</p>Formula:C15H20O5Color and Shape:SolidMolecular weight:280.32BMS-496
CAS:<p>BMS-496 is a dual DGKα/ζ lipid kinase inhibitor exhibiting IC50 values of 0.09 μM (DGKα) and 0.006 μM (DGKζ) [1].</p>Formula:C26H22BrF2N5O3Color and Shape:SolidMolecular weight:570.39Khellinol
CAS:Khellinol, a vasodilator, has bronchodilatory action.Formula:C13H10O5Color and Shape:SolidMolecular weight:246.22Nepaprazole
CAS:Nepaprazole (TY-11345) is a potent proton pump inhibitor; IC50: 5.8µM at pH 6.0, 9.9µM at pH 7.4. Better inhibition in weak acid.Formula:C18H19N3O2SPurity:98%Color and Shape:SolidMolecular weight:341.43YM49598
CAS:YM49598 is a tachykinin receptor antagonist with high affinity for NK(1) and NK(2). It inhibits rat bladder contraction induced by NK(1) agonists.Formula:C36H45Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:608.66mTOR inhibitor 9a
CAS:<p>mTOR inhibitor 9a inhibited the growth of human LNCap cells with an ic50 of 80 nm.</p>Formula:C20H21N5O2SPurity:99.78%Color and Shape:SoildMolecular weight:395.48ICMT-IN-26
CAS:<p>ICMT-IN-26 (compound 38) acts as an ICMT inhibitor with an IC50 value of 0.36 μM [1].</p>Formula:C21H26ClNOColor and Shape:SolidMolecular weight:343.89SUCNR1-IN-2
CAS:SUCNR1-IN-2 (Statement 35) serves as an inhibitor of both succinate and succinate receptor 1, utilized in research pertaining to neurodegenerative disorders,Formula:C17H13F3N2O6Color and Shape:SolidMolecular weight:398.29Phototrexate
CAS:Phototrexate, a photochromic Methotrexate analog, is a UVA-activated, reversible DHFR inhibitor with antifolate properties (IC50: 6 nM cis vs. 34 μM trans).Formula:C20H19N7O5Color and Shape:SolidMolecular weight:437.41mp-dLAE-PABC-MMAE
CAS:<p>mp-dLAE-PABC-MMAE is an agent-linker conjugate for antibody-drug conjugates (ADCs) that incorporates the potent tubulin inhibitor Monomethyl auristatin E (MMAE</p>Formula:C68H102N10O17Color and Shape:SolidMolecular weight:1331.59Lys(MMT)-PAB-oxydiacetamide-PEG8-N3
CAS:<p>Lys(MMT)-PAB-oxydiacetamide-PEG8-N3 is a cleavable linker for antibody-drug conjugate (ADC) synthesis that facilitates the attachment of therapeutic agents to</p>Formula:C55H77N7O14Color and Shape:SolidMolecular weight:1060.24SW106
CAS:SW106 blocks PTHR1 cAMP signaling, not affecting mutant PTHR1-T410P/H223R.Formula:C16H14F5NO2Color and Shape:SolidMolecular weight:347.28cis-Clopidogrel-MP derivative
CAS:cis-Clopidogrel-MP derivative, also Clopidogrel-MP-AM, is a 3'-methoxyacetophenone Clopidogrel metabolite and oral P2Y12 receptor platelet inhibitor.Formula:C25H26ClNO6SColor and Shape:SolidMolecular weight:503.99WAY-323756
CAS:WAY-323756 is a research-active molecule utilized in the study of amyloid diseases and synucleinopathies.Formula:C16H18N2O2SColor and Shape:SolidMolecular weight:302.397Ethanol-10NH2-11F-Camptothecin
CAS:7Ethanol-10NH2-11F-Camptothecin, an antibody drug conjugate (ADC), demonstrates inhibitory effects on tumor growth and is utilized in cancer research [1].Formula:C21H18FN3O5Color and Shape:SolidMolecular weight:411.38Verzistobart
CAS:<p>Verzistobart, an IgG1κ antibody, specifically targets the hepatitis A virus cellular receptor, HAVCR2.</p>Color and Shape:LiquidR-130823
CAS:R-130823 inhibits MAP kinase p38alpha (IC50=22 nM) and blocks cytokine release, reducing rat arthritis swelling and pain better than methotrexate.Formula:C28H26FN3Color and Shape:SolidMolecular weight:423.52MDK-0757
CAS:MDK-0757 is a novel inhibitor of heat shock protein 90 (Hsp90).Formula:C20H18FN5OPurity:98%Color and Shape:SolidMolecular weight:363.39Orexin receptor antagonist 4
CAS:Orexin antagonist 4: potent, selective for OX2R (IC50=4.27 nM); less for OX1R (IC50=295 nM).Formula:C22H24FN5O2Color and Shape:SolidMolecular weight:409.46Teropavimab
CAS:<p>Teropavimab (3BNC117-LS), an antibody, is utilized in the research of HIV infection [1].</p>Color and Shape:LiquidL-749329
CAS:L-749329 is a ligand of ET(A) and ET(B) endothelin receptor.Formula:C28H29NO8SPurity:98%Color and Shape:SolidMolecular weight:539.6ML115
CAS:ML115 is a potent and selective activator of transcription 3 (STAT3), with abn EC50 of 2.0 nM, and is inactive against the related STAT1 and NFκB anti-targets.Formula:C15H15ClN2O4Purity:99.97%Color and Shape:SolidMolecular weight:322.742-Deoxy-D-galactose
CAS:<p>2-Deoxy-D-galactose is a glucose analog and glucose antagonist that inhibits the maintenance of hippocampal LTP.</p>Formula:C6H12O5Purity:99.41% - 99.91%Color and Shape:SolidMolecular weight:164.16Anticancer agent 101
CAS:Anticancer Agent 101, a tetracaine derivative, exhibits anti-cancer activity [1].Formula:C19H20F3N3OColor and Shape:SolidMolecular weight:363.38WAY-311474
CAS:<p>WAY-311474 is an investigational compound targeting amyloid-related diseases and synucleinopathies.</p>Formula:C15H19Cl2NO2Color and Shape:SolidMolecular weight:316.22Solitomab
CAS:Solitomab (AMG 110) is a bispecific antibody targeting CD3 and EpCAM, used in uterine/ovarian carcinosarcoma research.Purity:95%Color and Shape:Liquidβ-catenin-IN-6
CAS:<p>β-Catenin-IN-6 is an inhibitor of the canonical Wnt/β-catenin signaling pathway, effectively impeding the proliferation of human colorectal cancer cells and</p>Formula:C22H19ClN6OColor and Shape:SolidMolecular weight:418.88Yonkenafil HCl
CAS:Yonkenafil HCl, a PDE5 inhibitor, is used potentially for the treatment of erectile dysfunction.Formula:C24H34ClN5O4SColor and Shape:SolidMolecular weight:524.08BePI
CAS:BePI can be a specific intercalator of both double and triple-helical DNA.Formula:C20H22N4OColor and Shape:SolidMolecular weight:334.41Osemozotan Free Base
CAS:Osemozotan Free Base is a 5-HT(1A) receptor agonist.Formula:C19H21NO5Color and Shape:SolidMolecular weight:343.37Sontigidomide
CAS:Sontigidomide (Compound 5) is an antineoplastic agent that demonstrates over 80% inhibition of MOLM-13 cell proliferation at a concentration of 1 μM after 3Formula:C26H22F3N3O5Color and Shape:SolidMolecular weight:513.47CycLuc1
CAS:<p>CycLuc1 is a brain penetrant luciferase substrate.</p>Formula:C13H11N3O2S2Purity:98.38%Color and Shape:SolidMolecular weight:305.38EHT 5372
CAS:<p>EHT 5372 inhibits DYRK kinases; IC50: 0.22-221 nM for DYRK1A/B, DYRK2/3, CLK1/2/4, GSK-3α/β.</p>Formula:C17H11Cl2N5OSColor and Shape:SolidMolecular weight:404.27GPR3 agonist-2
CAS:GPR3 agonist-2 (compound 32) is a potent full agonist of the G protein-coupled receptor 3 (GPR3), exhibiting an IC50 value of 260 nM [1].Formula:C14H7F6IO4SColor and Shape:SolidMolecular weight:512.16URAT1 inhibitor 8
CAS:URAT1 Inhibitor 8 (example 247) serves as a highly potent inhibitor of URAT1, demonstrating an IC50 value of 0.001 μM.Formula:C19H13ClFN3O4SColor and Shape:SolidMolecular weight:433.84MDL-74156
CAS:MDL-74156 is an active metabolite of dolasetron and a 5-hydroxy-tryptamine3 (5-HT3) antagonist.Formula:C19H22N2O3Color and Shape:SolidMolecular weight:326.39WAY-354436
CAS:<p>WAY-354436 is an active molecule.</p>Formula:C19H22FN3SColor and Shape:SolidMolecular weight:343.46Anti-inflammatory agent 43
CAS:Compound 43, also known as compound 3, is a 6-methoxyflavonol glycoside exhibiting anti-inflammatory activity.Formula:C34H42O22Color and Shape:SolidMolecular weight:802.68WAY-634964
CAS:WAY-634964 is an active molecule.Formula:C9H7N3O2Color and Shape:SolidMolecular weight:189.17Phosphazide
CAS:Phosphazide is a zidovudine prodrug.Formula:C10H14N5O6PColor and Shape:SolidMolecular weight:331.22NMS-P515
CAS:<p>NMS-P515 is an effective, orally active, and stereospecific PARP-1 inhibitor (Kd: 16 nM and an IC50: 27 nM (in Hela cells)). It has anti-tumor activity.</p>Formula:C21H29N3O2Purity:98%Color and Shape:SolidMolecular weight:355.47AMPA receptor modulator-6
CAS:<p>AMPA receptor modulator-6, an AMPA receptor positive allosteric modulator (PAM), is utilized in the research of neurological diseases [1].</p>Formula:C24H36N2O4S2Purity:98%Color and Shape:SolidMolecular weight:480.68THK-5105
CAS:<p>THK-5105, a tau-binding arylquinoline, could be an 18F-PET imaging probe for Alzheimer's disease.</p>Formula:C20H21FN2O2Color and Shape:SolidMolecular weight:340.39ARN 11391
CAS:<p>ARN 11391 enhances the function of the IP3-gated calcium channel ITPR1 (Inositol 1,4,5-trisphosphate (IP3) receptor type 1), boosting intracellular calcium ion</p>Formula:C22H29N3O3Color and Shape:SolidMolecular weight:383.49ARTD3/PARP3-IN-1
CAS:ARTD3/PARP3-IN-1 is a non-selective inhibitor targeting diphtheria toxin-like ADP-ribosyltransferase 3 (ARTD3)/PARP3 [1].Formula:C17H16N4O2Color and Shape:SolidMolecular weight:308.33PNU109291
CAS:PNU109291, a potent and selective agonist of the 5-HT1D receptor, effectively mitigates dural plasma extravasation induced by trigeminal ganglion stimulation.Formula:C24H31N3O3Purity:98%Color and Shape:SolidMolecular weight:409.52WAY-119918
CAS:WAY-119918 is an active molecule.Formula:C14H20N2OColor and Shape:SolidMolecular weight:232.32MF266-1
CAS:MF266-1, a selective E prostanoid receptor 4 antagonist, relieves joint inflammation and pain in rodent models of osteoarthritis and rheumatoid.Formula:C24H17ClF3NO3SColor and Shape:SolidMolecular weight:491.91YM-543 choline
CAS:YM-543/ASP-543: Potent, selective SGLT2 inhibitor, reduces blood sugar and improves glucose tolerance in diabetic mice.Formula:C28H37NO7Color and Shape:SolidMolecular weight:499.6BMS-332
CAS:BMS-332 is a dual inhibitor of the lipid kinases DGKα and DGKζ, demonstrating half-maximal inhibitory concentrations (IC50) of 0.005 μM for DGKα and 0.001 μMFormula:C29H27F2N5OColor and Shape:SolidMolecular weight:499.55HDM-201 succinate
CAS:<p>HDM-201 succinate is an orally bioavailable human double minute 2 homolog (HDM2) inhibitor with potential antineoplastic activity.</p>Formula:C30H30Cl2N6O8Color and Shape:SolidMolecular weight:673.5PI5P4K-β-IN-1
CAS:<p>PI5P4K-β-IN-1 (compound vs1) is a potent PI5P4K-β inhibitor with an IC50 of 0.80 μM [1].</p>Formula:C23H17Cl2N3O2Color and Shape:SolidMolecular weight:438.31Giminabant
CAS:Giminabant is an antagonist of cannabinoid receptor antagonist (veterinary use).Formula:C26H22Cl2N4Color and Shape:SolidMolecular weight:461.39MN-05
CAS:MN-05 is a neuroprotective and vasodilator for neurodegenerative diseases.Formula:C13H22N2O3Color and Shape:SolidMolecular weight:254.33BO-1158
CAS:BO-1158 is an antibacteria agent.Formula:C13H16FN5O8S2Purity:98%Color and Shape:SolidMolecular weight:453.42STING agonist-10
CAS:<p>STING agonist-10 is a potent activator of the STING small molecule cyclic urea class (EC50: 2600 nM).STING activation is a highly promising immunotherapy.</p>Formula:C25H20ClF4N3O2Color and Shape:SolidMolecular weight:505.89Cathepsin K inhibitor 3
CAS:Cathepsin K inhibitor 3: Selective, IC50 of 0.5 nM, good pharmacokinetics, potential for OA research.Formula:C30H31FN4O4SColor and Shape:SolidMolecular weight:562.65Fulvestrant (S enantiomer)
CAS:Fulvestrant S enantiomer is the less active S enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.Formula:C32H47F5O3SPurity:98%Color and Shape:SolidMolecular weight:606.7720-HETE inhibitor-1
CAS:20-HETE Inhibitor-1 (Comp 83) serves as an inhibitor of 20-HETE formation [1].Formula:C19H24N4OColor and Shape:SolidMolecular weight:324.42GTPγS tetralithium
CAS:<p>GTPγS tetralithium (Guanosine 5'-[γ-thio]triphosphate tetralithium) is a G-protein activator and a non-hydrolyzable GTP analog.</p>Formula:C10H12Li4N5O13P3SPurity:75%Color and Shape:SolidMolecular weight:562.985-Methyldihydrofolate
CAS:5-Methyldihydrofolate is the primary biologically active form of folate used for DNA reproduction, the cysteine cycle, and the regulation of homocysteine.Formula:C20H23N7O6Color and Shape:SolidMolecular weight:457.44Deoxyharringtonine
CAS:<p>Deoxyharringtonine, an alkaloid extracted from the Cephalotaxus genus, exhibits significant anti-leukemic properties [1].</p>Formula:C28H37NO8Color and Shape:SolidMolecular weight:515.6TMC-649128
CAS:TMC-649128, a RNA polymerase NS5B inhibitor, is used for the treatment of HCV infection.Formula:C18H26N6O6Color and Shape:SolidMolecular weight:422.44TAMRA-probe 1
TAMRA-probe 1 is a fluorescent probe for labeling.Formula:C46H62N8O10Purity:98%Color and Shape:SolidMolecular weight:887.03TRV-1387
CAS:<p>TRV-1387, a benzofurazan derivative, inhibits the aggregation of tau and amyloid-β [1].</p>Formula:C23H25F3N4O2Color and Shape:SolidMolecular weight:446.47[D-Ala6]-LH-RH
CAS:[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].Formula:C56H77N17O13Color and Shape:SolidMolecular weight:1196.32SREBP/SCAP-IN-2
CAS:SREBP/SCAP-IN-2 (compound 13) acts as a selective inhibitor of SREBP/SCAP [1].Formula:C27H37ClF2N4OColor and Shape:SolidMolecular weight:507.06Brevicompanine B
CAS:<p>Brevicompanine B: fungal metabolite, regulates plant growth/circadian rhythm, inhibits Arabidopsis roots, affects gene transcription, anti-P. falciparum.</p>Formula:C22H29N3O2Color and Shape:SolidMolecular weight:367.48Macimorelin acetate
CAS:Macimorelin acetate (EP-1572) is an oral GHSR agonist for AGHD and CACS research.Formula:C28H34N6O5Color and Shape:SolidMolecular weight:534.61p-fin4
CAS:p-fin4, a peptide, inhibits STEP-GluA2 interaction, Ki 0.4 μM; may enhance cognition, has anxiolytic and antidepressant effects.Formula:C39H53N8O18PColor and Shape:SolidMolecular weight:952.85Rosuvastatin zinc salt
CAS:Rosuvastatin zinc salt (Rosuvastatin zinc), a zinc-infused variant of Rosuvastatin, functions as an HMG-CoA reductase inhibitor, utilized primarily inFormula:C44H54F2N6O12S2ZnColor and Shape:SolidMolecular weight:1026.47CDK9-IN-23
CAS:<p>CDK9-IN-23 (Example 4) is a potent inhibitor of CDK9, exhibiting an IC50 value of less than 20 nM [1].</p>Formula:C22H25ClN4O3Purity:98%Color and Shape:SolidMolecular weight:428.91Antitumor agent-120
CAS:<p>Antitumor agent-120 (compound 1), a flavonoid derived from Kudzu root, exhibits negligible inhibitory effects on LNCaP and PC3 cancer cells, with IC50 values</p>Formula:C17H16N2O3Color and Shape:SolidMolecular weight:296.3214,15-Epoxyeicosatrienoic acid
CAS:<p>14,15-Epoxyeicosatrienoic acid (14,15-EET), derived from Arachidonic acid metabolism, significantly inhibits platelet aggregation in vivo and enhances</p>Formula:C20H32O3Color and Shape:SolidMolecular weight:320.47ASB-16165
CAS:<p>ASB-16165, a PDE7A inhibitor, may treat psoriasis by slowing keratinocyte growth.</p>Formula:C23H29N5O2SColor and Shape:SolidMolecular weight:439.57CBP/p300-IN-5
CAS:P300/CBP-IN-5 is a potent inhibitor of p300/CBP histone acetyltransferase (IC50 of 18.8 nM).Formula:C29H27F5N6O4Purity:98%Color and Shape:SolidMolecular weight:618.55Mal-PEG8-Phe-Lys-PAB-Exatecan
CAS:Compound 15, Mal-PEG8-Phe-Lys-PAB-Exatecan, is an antibody-drug conjugate (ADC) comprised of the degradable linker Mal-PEG8-Phe-Lys-PAB and the cytotoxic agentFormula:C73H92FN9O20Color and Shape:SolidMolecular weight:1434.56Bio-AMS
CAS:<p>Bio-AMS is a potent inhibitor of bacterial biotin protein ligase, exhibiting selective activity against Mycobacterium tuberculosis (Mtb) and disrupting fatty</p>Formula:C20H29N9O7S2Color and Shape:SolidMolecular weight:571.63Prostaglandin B2
CAS:<p>Prostaglandin B2 is a dehydration product of PGE2/PGA2 with weak TP receptor activity, raising rabbit pulmonary pressure at >5 ug/kg.</p>Formula:C20H30O4Color and Shape:SolidMolecular weight:334.45DU-125530
CAS:DU-125530 is a 5-HT1A receptor antagonist.Formula:C23H26ClN3O5SColor and Shape:SolidMolecular weight:491.99Sjc 13
CAS:Sjc 13 is an azaindolidine derivative that is a cell adhesion molecule inhibitor.Formula:C17H18N3NaO4Color and Shape:SolidMolecular weight:351.3378Clocortolone pivalate
CAS:Clocortolone pivalate, a synthetic steroid, treats dermatitis and psoriasis.Formula:C27H36ClFO5Color and Shape:SolidMolecular weight:495.02Deleobuvir sodium
CAS:Deleobuvir sodium (BI207127), a hepatitis C NS5B inhibitor, showed promise in some trials but was discontinued in 2013 due to insufficient efficacy.Formula:C34H32BrN6NaO3Color and Shape:SolidMolecular weight:675.56RET-IN-25
CAS:<p>RET-IN-25 (compound 6b) is an anticancer RET kinase inhibitor that demonstrates efficacy against medullary thyroid carcinoma (MTC), exhibiting half-maximal</p>Formula:C22H17N3O5SColor and Shape:SolidMolecular weight:435.45(R)-BDP9066
CAS:(R)-BDP9066 blocks MRCK to curb cancer cell spread, aiding research on diseases like cancer.Formula:C20H24N6Color and Shape:SolidMolecular weight:348.44PD-1/PD-L1-IN-27
CAS:PD-1/PD-L1-IN-27: potent anti-cancer, IC50 134nM, minimal T cell harm, boosts CD8+ T cells, reduces fatigue.Formula:C44H35NO6Purity:98%Color and Shape:SolidMolecular weight:673.75VU 0546110
CAS:<p>VU 0546110, a selective inhibitor of the sperm-specific potassium channel SLO3 (IC50= 64 μM), demonstrates 40-fold selectivity over SLO1.</p>Formula:C24H31NO4S2Color and Shape:SolidMolecular weight:461.64DQP-26
CAS:<p>DQP-26, a potent negative allosteric modulator of NMDA receptors (NMDARs), exhibits IC50 values of 0.77 μM for GluN2C and 0.44 μM for GluN2D subunits,</p>Formula:C28H21Cl2N3O4Purity:98%Color and Shape:SolidMolecular weight:534.39UNC3474
CAS:UNC3474, a small molecule ligand, selectively interacts with the aromatic methyl-lysine binding cage of the tumor protein 53BP1 Tudor domain (TT), exhibiting aFormula:C17H28N2OColor and Shape:SolidMolecular weight:276.42Heclin
CAS:<p>Heclin is an inhibitor of HECT E3 ubiquitin ligase that acts by inhibiting Smurf2, Nedd4, and WWP1 with IC50 values of 6.8, 6.3, and 6.9 μM, respectively.</p>Formula:C17H17NO3Purity:95.79%Color and Shape:SolidMolecular weight:283.32GSK 2833503A
CAS:GSK 2833503A: potent TRPC6/3 antagonist; IC50: 3-16/21-100 nM; >63x selective; inhibits cardiac hypertrophy signaling.Formula:C18H21ClFN3OSColor and Shape:SolidMolecular weight:381.9CBP/p300-IN-15
CAS:CBP/p300-IN-15 inhibits p300 (IC50: 2.5 nM) & CBP (28 nM), affects OVCAR-3 (EC50: 0.865 μM) & A2780 cells (2.71 μM) for ovarian cancer research.Formula:C26H28N4O5Color and Shape:SolidMolecular weight:476.52SHR5133
CAS:SHR5133 is a potent, orally active regulator of HBV capsid assembly that reduces HBV DNA (EC50: 26.6 nM).Formula:C19H18F4N6O2Color and Shape:SolidMolecular weight:438.38Anticancer agent 170
CAS:<p>Compound 3a, an anticancer agent and ketone derivative, exhibits potent activity against the A549 cancer cell line, demonstrating an inhibitory concentration (</p>Formula:C16H16O5Color and Shape:SolidMolecular weight:288.3NaPi2b Inhibitor 15
CAS:<p>NaPi2b, key in phosphate balance, is in intestines, lungs, testes. Blocking it may treat hyperphosphatemia by lowering serum phosphate.</p>Formula:C44H58ClF3N4O11SColor and Shape:SolidMolecular weight:943.46AMPK-IN-1
CAS:AMPK-IN-1 is an activator of the AMP-activated protein kinase (AMPK) enzyme, specifically targeting the α2β2γ1 isoform with an EC50 of 551 nM.Formula:C24H18ClN3O3Color and Shape:SolidMolecular weight:431.87N8-Acetylspermidine dihydrochloride
CAS:<p>N8-Acetylspermidine dihydrochloride is a polyamine that regulates ischemic cardiac apoptosis and resultant cardiac dysfunction.</p>Formula:C9H23Cl2N3OPurity:98% - 99.98%Color and Shape:SolidMolecular weight:260.2VKGILS-NH2 TFA
CAS:<p>VKGILS-NH2 TFA, a non-impacting control peptide for PAR2 agonist SLIGKV-NH2, doesn't affect DNA synthesis.</p>Formula:C30H55F3N8O9Color and Shape:SolidMolecular weight:728.8BAY-7081
BAY-7081 is a cyanopyridone-based compound that functions as a potent, selective, and orally active PDE9A inhibitor, demonstrating an inhibition concentration (Formula:C19H27ClN4OColor and Shape:SolidMolecular weight:362.9Butylate
CAS:<p>Butylate is a herbicide of thiocarbamate.</p>Formula:C11H23NOSColor and Shape:Less Liquid Which Darkens Upon Exposure To Light Air And Moisture Colorless Liquid Which Darkens Upon Exposure To Light Air And MoistureMolecular weight:217.37GLP-1R agonist 9
CAS:GLP-1R agonist 9 acts as a GLP-1R agonist, demonstrating efficacy with EC50 values of 1.1 nM and 11 nM against CHO GLP-1R Clone H6 and Clone C6, respectively.Formula:C32H30ClF2N3O5Color and Shape:SolidMolecular weight:610.05PYR01
CAS:PYR01 is a potent nonnucleoside reverse transcriptase inhibitor of HIV-1 and concurrently acts as a targeted activator to eliminate cells expressing HIV-1 [1].Formula:C21H13F7N4O3Color and Shape:SolidMolecular weight:502.34
