Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,523 products)
- Apoptosis(5,792 products)
- Cell Cycle/Checkpoint(4,449 products)
- Chromatin/Epigenetics(2,238 products)
- Cytoskeletal Signaling(1,383 products)
- DNA Damage/DNA Repair(2,825 products)
- Endocrinology/Hormones(3,507 products)
- Enzyme(3,640 products)
- GPCR/G-Protein(8,333 products)
- Immunology and Inflammation(3,526 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(404 products)
- MAPK Signaling(1,202 products)
- Membrane Transporter/Ion Channel(2,790 products)
- Metabolism(9,448 products)
- Microbiology/Virology(6,981 products)
- Neuroscience(9,926 products)
- Other Inhibitors(37,926 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,400 products)
- Proteases/Proteasome(1,597 products)
- Stem Cell and Derivatives(831 products)
- Tyrosine Kinase/Adaptors(2,016 products)
- Ubiquitination(1,650 products)
Show 16 more subcategories
Found 66641 products of "Inhibitors"
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ORP-101
CAS:<p>ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.</p>Formula:C60H84N2O8Color and Shape:SolidMolecular weight:961.32GSD-11
<p>GSD-11: Potent, selective anti-austerity agent; blocks Akt/mTOR pathway, hinders PANC-1 cell migration & colony growth. Promising for pancreatic cancer study.</p>Formula:C20H28O2Color and Shape:SolidMolecular weight:300.44Fonadelpar
CAS:<p>Fonadelpar is an agonist of PPARδ. It also is used in the research of neuroparalytic keratopathy.</p>Formula:C25H23F3N2O4SPurity:98%Color and Shape:SolidMolecular weight:504.52Antibiotic MA 144M1
CAS:<p>Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.</p>Formula:C42H55NO15Color and Shape:SolidMolecular weight:813.88XO/COX/LOX-IN-1
<p>XO/COX/LOX-IN-1 targets XO/COX/LOX, used in research of inflammation, cancer, and metabolic disorders.</p>Formula:C24H20N4O2SColor and Shape:SolidMolecular weight:428.51Adafosbuvir
CAS:<p>Adafosbuvir has antiviral activity.</p>Formula:C22H29FN3O10PColor and Shape:SolidMolecular weight:545.457MCTR2
CAS:<p>MCTR2, synthesized from DHA in macrophages, aids in tissue repair and reduces inflammation by promoting eicosanoid PGD2 and PGF2α decrease.</p>Formula:C27H40N2O6SColor and Shape:SolidMolecular weight:520.68Isoleucyl tRNA synthetase-IN-1
CAS:<p>Isoleucyl tRNA synthetase-IN-1 is a selective and potent inhibitor (Ki: 88 nM) that targets isoleucyl tRNA synthetase (IleRS).</p>Formula:C23H35N5O7SColor and Shape:SolidMolecular weight:525.62BM635 hydrochloride
<p>BM635 hydrochloride, an MmpL3 inhibitor, strongly blocks Divergent bacteriophage H37Rv (MIC50: 0.08 μM), with doubled in vivo potency.</p>Formula:C25H30ClFN2OColor and Shape:SolidMolecular weight:428.97TBK1/IKKε-IN-1
CAS:<p>TBK1/IKKε-IN-1 is a dual inhibitor of TBK1 and IKKε (IC50s of <100 nM).</p>Formula:C28H26N4O5Purity:98%Color and Shape:SolidMolecular weight:498.53OP-2507
CAS:<p>OP-2507, a prostacyclin agonist, is used potentially for the treatment of hepatic insufficiency and hypertension.</p>Formula:C25H41NO4Purity:98%Color and Shape:SolidMolecular weight:419.6M1069
<p>M1069 is an oral A2A/A2B receptor antagonist, 100x more selective over A1/A3, with antitumor properties by blocking adenosine's immunosuppressive effects.</p>Formula:C25H30N4O8SColor and Shape:SolidMolecular weight:546.59ATM Inhibitor-4
<p>ATM Inhibitor -4: selective, potent (IC50: 0.32 nM), inhibits PI3K family, stable, stops mTOR at 1 μM.</p>Formula:C26H29FN6O3Color and Shape:SolidMolecular weight:492.55EGFR-IN-62
<p>EGFR-IN-62: IC50 of 10-242 nM for various EGFR mutations, blocks A549/H1975 cell cycle, induces apoptosis, and inhibits cell motility and proliferation.</p>Formula:C30H33N9O2Color and Shape:SolidMolecular weight:551.64Eravacycline
CAS:<p>Eravacycline (TP-434) is a potent and broad-spectrum antibacterial agent.</p>Formula:C27H31FN4O8Purity:97.46%Color and Shape:SolidMolecular weight:558.56DFBTA
<p>DFBTA inhibits ANO1 with IC50 of 24 nM, effectively treating inflammatory pain orally.</p>Formula:C18H10ClF2NO3SColor and Shape:SolidMolecular weight:393.79DC41SMe
CAS:<p>DC41SMe, a DC1 derivative and CC-1065 analogue, targets cancer with 18-25 pM IC50 against Ramos, Namalwa, HL60/s cells.</p>Formula:C38H36ClN5O4S2Purity:98%Color and Shape:SolidMolecular weight:726.31PI3K-IN-35
CAS:<p>PI3K-IN-35 (6l) selectively inhibits PI3K-α, β, δ (IC50: 13.98, 7.22, 10.94 μM), blocks G2/M phase, induces apoptosis, and is useful in leukemia research.</p>Formula:C25H23N7O2Color and Shape:SolidMolecular weight:453.5SARS-CoV-2-IN-8
<p>SARS-CoV-2-IN-8 is a major protease inhibitor of SARS-CoV-2 (IC50: 0.75 μM).</p>Formula:C35H38N6O3Color and Shape:SolidMolecular weight:590.71HOE-288
CAS:<p>HOE-288 is a converting enzyme (CE) inhibitor.</p>Formula:C27H38N2O5Color and Shape:SolidMolecular weight:470.60PAD2-IN-1 hydrochloride
<p>PAD2-IN-1 hydrochloride: potent, selective PAD2 inhibitor; 95x less on PAD4, 79x less on PAD3; benzimidazole derivative.</p>Formula:C25H30ClFN6O3Color and Shape:SolidMolecular weight:517HDAC-IN-33
<p>HDAC-IN-33 inhibits HDAC1/2/6 (IC50: 24/46/47 nM), exhibits potent antitumor activity in vitro and in vivo, and activates antitumor immunity.</p>Formula:C21H25N3O3Color and Shape:SolidMolecular weight:367.44PLAP-IN-1
CAS:<p>PLAP-IN-1: Potent, selective inhibitor of PLAP, IC50 of 32 nM; doesn't notably inhibit TNAP.</p>Formula:C25H21Cl2N3O5Color and Shape:SoildMolecular weight:514.36HbF inducer-1
<p>HbF inducer-1 is a fetal hemoglobin inducer which is orally bioavailable.</p>Formula:C18H19N3O3Color and Shape:SolidMolecular weight:325.36KRAS G12C inhibitor 15
CAS:<p>KRAS G12C inhibitor 15 is a potent KRAS G12C inhibitor .</p>Formula:C25H21ClF2N4O3Purity:98%Color and Shape:SolidMolecular weight:498.91ZD6021
CAS:<p>ZD6021 is an antagonist of neurokinin 1 receptor.</p>Formula:C35H35Cl2N3O2SPurity:98%Color and Shape:SolidMolecular weight:632.64Chitinase-IN-5
<p>Chitinase-IN-5 (8i) blocks OfChi-h (IC50: 0.051 μM), has insecticidal qualities, useful for eco-friendly pest control.</p>Formula:C20H21ClFN7Color and Shape:SolidMolecular weight:413.88Thioquinapiperifil dihydrochloride
CAS:<p>Thioquinapiperifil dihydrochloride is a potent, selective PDE-5 inhibitor (IC50: 0.074 nM) for research.</p>Formula:C24H29ClN6OSPurity:98.73%Color and Shape:SolidMolecular weight:485.05KOS-1584
CAS:<p>KOS-1584, a safer, more effective epothilone, inhibits cell division by stabilizing microtubules and evading P-gp.</p>Formula:C27H39NO5SColor and Shape:SolidMolecular weight:489.67AXKO-0046
<p>AXKO-0046 is an indole derivative and small-molecule LDHB selective inhibitor.</p>Formula:C25H33N3Color and Shape:SolidMolecular weight:375.55Arverapamil
CAS:<p>Arverapamil is a chiral metabolite of Verapamil.</p>Formula:C26H36N2O4Color and Shape:SolidMolecular weight:440.58Fabimycin
CAS:<p>Fabimycin, a FabI inhibitor, combats drug-resistant gram-negative bacterial infections effectively.</p>Formula:C23H25ClN4O3Color and Shape:SolidMolecular weight:440.924α-PDD
CAS:<p>4alpha-PDD activates transient receptor potential vanilloid 4 (TRPV4) channels and is inactive for signaling through PKC.</p>Formula:C40H64O8Color and Shape:SolidMolecular weight:672.93CXCR2 antagonist 7
<p>CXCR2 antagonist 7 is a powerful blocker with IC50s: 0.044 μM for binding, 0.66 μM for calcium mobilization.</p>Formula:C14H14F2N6OSColor and Shape:SolidMolecular weight:352.36N'-(2-Fluorophenyl)pyrazine-2-carbohydrazide
<p>N'-(2-Fluorophenyl)pyrazine-2-carbohydrazide is a Ole1p desaturase inhibitor as well as antifungal agent [1].</p>Formula:C11H9FN4OColor and Shape:SolidMolecular weight:232.21PNU-140457
CAS:<p>PNU-140457 is a bio-active chemical.</p>Formula:C14H14FN5O3Color and Shape:SolidMolecular weight:319.29Cicaprost
CAS:<p>Cicaprost (ZK 96480) is an IP agonist with artery relaxing effects; EC50 is 5.8 nM.</p>Formula:C22H30O5Color and Shape:SolidMolecular weight:374.47Seco-Duocarmycin SA
CAS:<p>Seco-Duocarmycin SA is a highly potent DNA alkylator used as an ADC cytotoxin.</p>Formula:C25H24ClN3O7Purity:98%Color and Shape:SolidMolecular weight:513.93Antiproliferative agent-8
<p>Compound 5a, an anticancer agent, enhances P53 and has antiproliferative effects.</p>Formula:C22H16ClN3O3Color and Shape:SolidMolecular weight:405.83p38 MAPK-IN-3
<p>Compound 2c is a potent p38α MAPK inhibitor with antitumor effects, enhancing apoptosis and ROS.</p>Formula:C22H17BrO2Color and Shape:SolidMolecular weight:393.27eIF4A3-IN-6
CAS:<p>eIF4A3-IN-6 is a potent eIF4A inhibitor, potentially used for treating eIF4A-related diseases like cancer. (US20170145026A1)</p>Formula:C26H25N3O5Color and Shape:SolidMolecular weight:459.49PI3K-IN-27
CAS:<p>PI3K-IN-27 is a potent PI3K inhibitor, relevant for cancer and immune disease research. See patent WO2021233227A1.</p>Formula:C30H26F2N6O2SColor and Shape:SolidMolecular weight:572.63AZD 4407
CAS:<p>AZD 4407 is a potent inhibitor of 5-lipoxygenase.</p>Formula:C19H21NO3S2Purity:98%Color and Shape:SolidMolecular weight:375.5Pol I-IN-1
<p>Pol I-IN-1 is a powerful inhibitor of RNA polymerase I (Pol I), specifically targeting the large catalytic subunit RPA194, demonstrating an inhibition</p>Formula:C23H22N4O2Color and Shape:SolidMolecular weight:386.45Colistin adjuvant-1
<p>Colistin adjuvant-1, inhibits NF-κB (IC50: 0.209 μM), boosts mucin against gram-negative bacteria.</p>Formula:C16H7F9N2OColor and Shape:SolidMolecular weight:414.23Dersimelagon phosphate
CAS:<p>Dersimelagon phosphate: MC1R agonist, boosts melanin, enhances light tolerance in EPP/XLP without sun.</p>Formula:C36H48F4N3O9PColor and Shape:SolidMolecular weight:773.75Antimalarial agent 2
<p>Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.</p>Formula:C27H25N3O5Color and Shape:SolidMolecular weight:471.5DC1SMe
CAS:<p>DC1, a CC-1065-like ADC cytotoxin, is used in cancer-targeting antibody-drug conjugates. DC1Sme, a derivative, has IC50s: 22-250 pm in various cancer cells.</p>Formula:C35H30ClN5O4S2Purity:98%Color and Shape:SolidMolecular weight:684.23(3S,4R)-Tofacitinib
CAS:<p>(3S,4R)-Tofacitinib is an less active enantiomer of Tofacitinib. Tofacitinib is a JAK3 inhibitor(IC50 : 1 nM).</p>Formula:C16H20N6OPurity:98%Color and Shape:SolidMolecular weight:312.37Minnelide
CAS:<p>Minnelide is a prodrug of triptolide,and shows potent antitumor activity in a number of tumor types.</p>Formula:C21H25Na2O10PPurity:98.49% - 99.59%Color and Shape:SolidMolecular weight:514.37LSD1/2-IN-3
<p>LSD1/2-IN-3 selectively inhibits LSD1 (Ki 11 nM) over LSD2 (Ki 7 μM), and hinders tumor stem cell proliferation.</p>Formula:C9H8BrF2NColor and Shape:SolidMolecular weight:248.07Antibacterial agent 78
<p>Antibacterial agent 78 (compound 30) is an antibacterial agent with improved cytotoxicity profile[1].</p>Formula:C16H23N3S2Color and Shape:SolidMolecular weight:321.5CCR5 antagonist 1
CAS:<p>CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.</p>Formula:C39H46ClF2N5O3SPurity:98%Color and Shape:SolidMolecular weight:738.33Carbodine
CAS:<p>Carbodine is an antiviral targeting CTP synthetase, effective against influenza A0/PR-8/34 and A2/Aichi/2/68.</p>Formula:C10H15N3O4Purity:98%Color and Shape:SolidMolecular weight:241.24LAF-153
CAS:<p>LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.</p>Formula:C18H32N2O7Color and Shape:SolidMolecular weight:388.46STA 2
CAS:<p>STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.</p>Formula:C21H34O3SColor and Shape:SolidMolecular weight:366.56MA242
CAS:<p>MA242 is a nuclear factor of activated T cells 1 (NFAT1) for Pancreatic Cancer Therapy and dual inhibitor of murine double minute 2 (MDM2).</p>Formula:C26H21ClF3N3O5SPurity:98%Color and Shape:SolidMolecular weight:579.98HDAC-IN-34
<p>HDAC-IN-34 inhibits HDAC1 (IC50: 0.022 μM) & HDAC6 (IC50: 0.45 μM), binds DNA causing damage, and halts HCT-116 cell growth (IC50: 1.41 μM).</p>Formula:C24H26N6O3Color and Shape:SolidMolecular weight:446.5BTK inhibitor 18
<p>BTK inhibitor 18 is a selective, potent, covalent, orally active Btk inhibitor (IC50: 142 nM) that exhibits anti-inflammatory effects.</p>Formula:C29H25N5O4S2Color and Shape:SolidMolecular weight:571.67Calpain Inhibitor-2
CAS:<p>Calpain Inhibitor-2: Lipophilic, moderates growth of A-375, B-16F1, PC-3 cancers, and hinders 80% DU-145 cell invasion.</p>Formula:C26H33N3O5SColor and Shape:SolidMolecular weight:499.62DHU-Se1
<p>DHU-Se1: potent anti-inflammatory, releases reactive selenium from macrophages, inhibits iNOS/TNF-α, blocks M0 to M1 polarization.</p>Formula:C23H23N3OSSeColor and Shape:SolidMolecular weight:468.47RMS5
CAS:<p>RMS5: hambanine analogue, inhibits P-gp, anti-cancer with cytotoxic, anti-proliferative effects, reduces Bcl-2 proteins, cleaves PARP.</p>Formula:C35H38N2O5SColor and Shape:SolidMolecular weight:598.75SM-433 hydrochloride
<p>SM-433 hydrochloride, a Smac mimetic & IAP inhibitor, binds XIAP BIR3; potent IC50 <1 μM. (Patent WO2008128171A2)</p>Formula:C32H44ClN5O4Color and Shape:SolidMolecular weight:598.18EGFR-IN-17
<p>EGFR-IN-17: potent, selective EGFR inhibitor, IC50 of 0.2 nM, overcomes C797S drug resistance.</p>Formula:C27H31ClN7O3PColor and Shape:SolidMolecular weight:568.01Tovinontrine
CAS:<p>Tovinontrine (IMR-687) (IMR-687) is a potent and selective inhibitor of phosphodiesterase-9 (PDE9), designed to target sickle cell disease treatment.</p>Formula:C21H26N6O2Purity:98.14%Color and Shape:SolidMolecular weight:394.47G12Si-1
<p>G12Si-1 selectively binds and inhibits K-Ras(G12S) to block oncogenic signaling and nucleotide exchange.</p>Formula:C29H32ClN5O3Color and Shape:SolidMolecular weight:534.05MALT1-IN-5
CAS:<p>MALT1-IN-5 is a potent inhibitor of the MALT1 protease and can be used in cancer research.</p>Formula:C17H17ClF2N6O3Color and Shape:SolidMolecular weight:426.80BMS-248360
CAS:<p>BMS-248360: Oral dual hAT1/hETA antagonist with Kis of 10nM & 1.9nM, respectively; treats hypertension.</p>Formula:C36H45N5O5SPurity:98%Color and Shape:SolidMolecular weight:659.84SP inhibitor 1
<p>SP inhibitor 1 blocks SARS-CoV-2 replication in vitro (0.3250<5.98 μM) and targets SP protein (IC50: 3.26 μM) with antiviral effects.</p>Formula:C36H38N2O2Color and Shape:SolidMolecular weight:530.7FGFR3-IN-4
CAS:<p>FGFR3-IN-4 is a selective inhibitor targeting FGFR3, demonstrating an IC50 value of under 50 nM.</p>Formula:C26H24ClN7OColor and Shape:SolidMolecular weight:485.97A25822B
CAS:<p>A25822B is an antifungal agent.</p>Formula:C28H45NOPurity:98%Color and Shape:SolidMolecular weight:411.66CVN636
CAS:<p>CVN636, a potent and selective allosteric agonist for the mGluR7 receptor, exhibits oral activity and CNS permeability [1], with an EC50 of 7 nM for human</p>Formula:C19H20FNO4SColor and Shape:SolidMolecular weight:377.43AP5
CAS:<p>AP5: GPR40 agonist, positive allosteric modulator; rat hIP1 EC50: 0.49 nM.</p>Formula:C28H28FNO4Purity:98%Color and Shape:SolidMolecular weight:461.52PTP1B-IN-18
<p>PTP1B-IN-18 is an orally active, fully mixed protein tyrosine phosphatase 1B (PTP1B) inhibitor (Ki: 35.2 μM).PTP1B-IN-18 can be used to study type 2 diabetes.</p>Formula:C26H19N3O4SColor and Shape:SolidMolecular weight:469.51SR 140333
CAS:<p>SR 140333 is a NK1 receptor antagonist.</p>Formula:C37H45Cl3N2O2Purity:98%Color and Shape:SolidMolecular weight:656.12IDX-320
CAS:<p>IDX-320 is an HCV protease inhibitor.</p>Formula:C37H43F3N6O7S2Color and Shape:SolidMolecular weight:804.9Hypoglycemic agent 1
CAS:<p>Hypoglycemic agent 1 has an action for lowering blood sugar. It acts as a therapeutic and/or prophylactic agent for diabetes.</p>Formula:C25H24FN5O4Purity:98%Color and Shape:SolidMolecular weight:477.49SGE-516
CAS:<p>SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.</p>Formula:C23H35N3O2Purity:98%Color and Shape:SolidMolecular weight:385.54MSX-3 free acid
CAS:<p>MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.</p>Formula:C21H23N4O7PColor and Shape:SolidMolecular weight:474.40GPX4-IN-3
CAS:<p>GPX4-IN-3 (26a) is a potent GPX4 inhibitor, inducing selective ferroptosis with 71.7% inhibition at 1 μM.</p>Formula:C29H24ClN3O3SColor and Shape:SolidMolecular weight:530.04Antibacterial agent 88
<p>Antibacterial agent 88 is an effective antibacterial agent against B. subtilis (MIC: 4 μg/ml) with MIC values of ≤0.0156 μg/mL for MRSA, MRSE and S. aureus.</p>Formula:C31H44N2O6SColor and Shape:SolidMolecular weight:572.76Cap-dependent endonuclease-IN-25
CAS:<p>Cap-dependent endonuclease-IN-25 is a potent inhibitor of CEN, useful in studying Orthomyxoviridae viruses. (See WO2020075080A1, compound 4.)</p>Formula:C25H25N3O3Color and Shape:SolidMolecular weight:415.48MraY-IN-2
<p>MraY-IN-2 (compound 6) is an effective inhibitor of bacterial transposase MraY (IC50=4.5 μ M), and can be used for antibacterial research.</p>Formula:C16H23N3O9Color and Shape:SolidMolecular weight:401.37IRAK4-IN-11
<p>IRAK4-IN-11 (compound 6) is a potent inhibitor of IRAK4 with an IC 50 of 0.008 μM. IRAK4-IN-11 exhibits cell pIRAK4 potencies with an IC 50 of 0.19 μM [1].</p>Formula:C16H19N7OColor and Shape:SolidMolecular weight:325.37β-Secretase Inhibitor III
<p>β-Secretase Inhibitor III is a highly selective inhibitor of BACE1 with a Ki value of 0.13 nM.</p>Formula:C20H20F2N4O3SColor and Shape:SolidMolecular weight:434.46L-Afegostat
CAS:<p>L-Afegostat (5-epi-Isofagomine), an iminosugar, inhibits glycosidase and β-Glucosidase (K i 30 μM), aids in carbohydrate synthesis.</p>Formula:C6H13NO3Color and Shape:SolidMolecular weight:147.17Anticancer agent 64
CAS:<p>Anticancer agent 64 (5m) induces apoptosis, has IC50 2.4μM in CCRF-CEM, activates caspases, cleaves PARP, affects mitochondria.</p>Formula:C31H46N2O2SColor and Shape:SolidMolecular weight:510.77(2S,4S)-Sacubitril
CAS:<p>(2S,4S)-Sacubitril (Sacubitril Impurity C) is a stereoisomer derived from Sacubitril which is a potent NEP inhibitor.</p>Formula:C24H29NO5Purity:98%Color and Shape:SolidMolecular weight:411.49LY3130481
CAS:<p>LY3130481: TARP γ-8 dependent AMPA receptor blocker; selectively targets AMPA/TARP γ-8 with 65 nM IC50.</p>Formula:C19H18N4O3SColor and Shape:SolidMolecular weight:382.44Tofogliflozin
CAS:<p>Tofogliflozin specifically inhibits SGLT2; IC50s are 2.9 nM (human), 14.9 nM (rat), 6.4 nM (mouse).</p>Formula:C22H26O6Purity:98%Color and Shape:SolidMolecular weight:386.44GR 122222X
CAS:<p>GR 122222X is an inhibitor of topoisomerase II.</p>Formula:C26H35N5O11SPurity:98%Color and Shape:SolidMolecular weight:625.65CaMKIIα-IN-1
<p>CaMKIIα-IN-1 (Compound 4d) is an orally active inhibitor of Ca 2+ /calmodulin-dependent protein kinase II α (CaMKIIα) with a Kd of 219 nM for CaMKIIα WT hub.</p>Formula:C14H11ClO4Color and Shape:SolidMolecular weight:278.69NVP-CGM097 sulfate
CAS:<p>NVP-CGM097 sulfate is a potent and selective inhibitor of MDM2 (hMDM2, IC50 of 1.7±0.1 nM).</p>Formula:C38H49ClN4O8SPurity:98%Color and Shape:SolidMolecular weight:757.34Gimatecan
CAS:<p>Gimatecan (STI481) is a potent topoisomerase I inhibitor. Gimatecan is an orally bioavailable camptothecin analogue with antitumor activity.</p>Formula:C25H25N3O5Purity:98.47%Color and Shape:SolidMolecular weight:447.48SLN124
<p>SLN124, a GalNAc-siRNA targeting TMPRSS6, may normalize iron balance by restoring ferroregulation.</p>Color and Shape:SolidCP-481715
CAS:<p>CP 481715 is an effective selective CCR1 antagonist with potential therapeutic significance for inflammatory diseases.</p>Formula:C26H31FN4O4Color and Shape:SolidMolecular weight:482.55AChE-IN-5
<p>AChE-IN-5: oral, crosses blood-brain barrier, targets AChE/5-HT1A/SERT, potent with 2.29 nM IC50.</p>Formula:C38H45N5OColor and Shape:SolidMolecular weight:587.85-HT6/5-HT2AR antagonist-1
<p>Potent 5-HT6/5-HT2A receptors dual antagonist with K i of 11 nM & 39 nM.</p>Formula:C21H26N6SColor and Shape:SolidMolecular weight:394.54S-1033
CAS:<p>S-1033 is an FP receptor agonist.</p>Formula:C20H33NaO4Color and Shape:SolidMolecular weight:360.4698hCA IX-IN-1
<p>hCA IX-IN-1 inhibits human carbonic anhydrases I, II, IX, and XII with Ki values of 331.4, 28.4, 9.4, 17.8 nM and exhibits anticancer properties.</p>Formula:C19H18N2O3SColor and Shape:SolidMolecular weight:354.42LAS195319
CAS:<p>LAS195319 is a potent and selective inhaled PI3Kδ Inhibitor (IC50 = 0.5 nM) for the Treatment of Respiratory Diseases.</p>Formula:C29H26N10O3SColor and Shape:SolidMolecular weight:594.65PKG1α activator 3
<p>PKG1α activator 3 is a PKG1α activator (EC50basal/partial=13/0.52 μM).</p>Formula:C27H26Cl2N2O6Color and Shape:SolidMolecular weight:545.41EGFR/HER2-IN-8
<p>EGFR/HER2-IN-8 inhibits EGFR, HER2, DHFR (IC50: 0.45, 0.244, 5.669 μM); useful in cancer research, safe and selective.</p>Formula:C16H16N4O2SColor and Shape:SolidMolecular weight:328.39Antitumor agent-51
<p>Antitumor agent-51 targets osteosarcoma with 21.9 nM IC50, high selectivity, and low toxicity.</p>Formula:C23H25N5O2SColor and Shape:SolidMolecular weight:435.54DNA crosslinker 1 dihydrochloride
CAS:<p>DNA Crosslinker 1 binds DNA minor groove with 1.1°C affinity increase; used in cancer research.</p>Formula:C15H22Cl2N8OColor and Shape:SolidMolecular weight:401.29GSK864
CAS:<p>GSK864 is an inhibitor of isocitrate dehydrogenase 1 (IDH1) mutant. GSK864 inhibits IDH1 mutants R132C, R132H, and R132G (IC50: 8.8, 15.2, and 16.6 nM).</p>Formula:C30H31FN6O4Purity:97.07%Color and Shape:SolidMolecular weight:558.6EBI-907
CAS:<p>EBI-907 is a potent, oral B-RafV600E inhibitor with an IC50 of 4.9 nM, over 10x stronger than Vemurafenib, and effective against key cancer kinases.</p>Formula:C23H21ClF2N4O3SColor and Shape:SolidMolecular weight:506.95PF-06463922 acetate
CAS:<p>PF-06463922 acetate: ALK/ROS1 inhibitor, brain- penetrable, active vs crizotinib-resistant mutants, in NSCLC trials.</p>Formula:C23H23FN6O4Color and Shape:SolidMolecular weight:466.46eIF4A3-IN-4
<p>eIF4A3-IN-4 is a novel inhibitor of eIF4A (IC50: 8.6 μM).</p>Formula:C24H20N2O5Color and Shape:SolidMolecular weight:416.43Prohibitin ligand 1
<p>Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.</p>Formula:C20H22N2OColor and Shape:SolidMolecular weight:306.4Lasonolide A
CAS:<p>Lasonolide A, an anticancer compound from Forcepia sponge, shows nanomolar growth inhibition and unique cytotoxicity in the NCI 60-cell-line screen.</p>Formula:C41H60O9Color and Shape:SolidMolecular weight:696.91Omesdafexor
CAS:<p>Omesdafexor is an FXR agonist that can be used to study diseases caused by liver disease or metabolic inflammation.</p>Formula:C34H43N3O3Color and Shape:SolidMolecular weight:541.72Anti-inflammatory agent 13
<p>Pentacyclic triterpene, Anti-inflammatory 13 inhibits DAMP/PAMP inflammation models.</p>Formula:C30H48O4Color and Shape:SolidMolecular weight:472.7Hexedine
CAS:<p>Hexedine is a biochemical.</p>Formula:C22H45N3Color and Shape:SolidMolecular weight:351.61Flutimide
CAS:<p>Flutimide: Endonuclease inhibitor, IC50 = 3μM, for research on acute respiratory diseases like influenza.</p>Formula:C12H18N2O3Color and Shape:SolidMolecular weight:238.28GZN39838
CAS:<p>GZN39838, a natural Kv1.2 blocker, induces C-type inactivation without blocking the outer pore.</p>Formula:C22H30O6Color and Shape:SolidMolecular weight:390.47D18
CAS:<p>D18: Dual agonist for TLR7/8, boosts PD-L1, aids tumor sensitivity to PD-1/PD-L1 inhibitors, and is a cytotoxin for ADC HE-S2.</p>Formula:C21H28N6Color and Shape:SolidMolecular weight:364.49CRV431
CAS:<p>CRV431 is a novel Pan-Cyclophilin Inhibitor, potently inhibiting all cyclophilin isoforms tested - A, B, D, and G (IC50 values ranged from 1-7 nM).</p>Formula:C67H122N12O13Color and Shape:SolidMolecular weight:1303.76Turoctocog alfa
CAS:<p>Turoctocog alfa: recombinant FVIII from CHO cells for hemophilia A study.</p>Color and Shape:SolidHIV-1 protease-IN-6
<p>HIV-1 protease-IN-6 (17d) strongly inhibits HIV-1 protease (IC50: 21 pM, Ki: 4.7 pM) and effectively targets DRV-resistant mutants.</p>Formula:C27H31FN2O6SColor and Shape:SolidMolecular weight:530.61Leu-AMS R enantiomer
CAS:<p>Leu-AMS R enantiomer is the R enatiomer of Leu-AMS. Leu-AMS is a potent leucyl-tRNA synthetase (LRS) inhibitor that inhibits the bacteria growth.</p>Formula:C16H25N7O7SPurity:98%Color and Shape:SolidMolecular weight:459.48Niravoline
CAS:<p>Niravoline is a kappa-opioid agonist.</p>Formula:C22H25N3O3Color and Shape:SolidMolecular weight:379.45GABAA receptor agonist 2
<p>Compound 4c, a potent GABAA agonist with anti-depressive effects in mouse FST/TST, shows promise in depression research.</p>Formula:C22H36O5Color and Shape:SolidMolecular weight:380.5217β-HSD1-IN-1
<p>17β-HSD1-IN-1 (Compound 1) can be used in the non-small cell lung cancer (NSCLC) research.</p>Formula:C21H21NO3Color and Shape:SolidMolecular weight:335.4Antitumor agent-74
<p>Antitumor agent-74, a quinazoline derivative, inhibits DNA, arrests cell cycle, and induces apoptosis with agent-75.</p>Formula:C26H23FN6Color and Shape:SolidMolecular weight:438.5ent-8-iso-15(S)-Prostaglandin F2α
CAS:<p>Isoprostanes are produced by the non-enzymatic, free radical peroxidation of phospholipid-esterified arachidonic acid.</p>Formula:C20H34O5Color and Shape:SolidMolecular weight:354.48Anti-inflammatory agent 9
<p>Benzimidazothiazole-derived Compound 28 from tilomisole targets COX-2, has potent anti-inflammatory effects & is orally bioavailable.</p>Formula:C18H15N5O2SColor and Shape:SolidMolecular weight:365.41EBOV-GP-IN-1
<p>EBOV-GP-IN-1 (Compound 28) is a potent inhibitor of Ebola entry, acting on the Ebola virus envelope glycoprotein (EBOV-GP) (IC50: 0.05 μM).</p>Formula:C25H40ClN3O2Color and Shape:SolidMolecular weight:450.06Ivaltinostat formic
<p>Ivaltinostat (CG-200745) is an oral panHDAC inhibitor, inducing apoptosis and enhancing cancer drug sensitivity.</p>Formula:C25H35N3O6Color and Shape:SolidMolecular weight:473.56Carazostatin
CAS:<p>Carazostatin is an antioxidant, free radical scavenger, and potent lipid peroxidation inhibitor.</p>Formula:C20H25NOPurity:98%Color and Shape:Pale Yellow SolidMolecular weight:295.42Coleon-U-quinone
CAS:<p>Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.</p>Formula:C20H24O5Color and Shape:SolidMolecular weight:344.4Epolactaene
CAS:<p>Epolactaene: neuritogenic, inhibits mammalian DNA polymerases & human DNA topoisomerase II.</p>Formula:C21H27NO6Color and Shape:SolidMolecular weight:389.44Antileishmanial agent-4
<p>Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].</p>Formula:C17H18N4O4Color and Shape:SolidMolecular weight:342.35BTK-IN-15
<p>BTK-IN-15: Oral BTK inhibitor, IC50 0.7 nM, induces cancer cell apoptosis, selective with anti-tumor effects.</p>Formula:C28H24FN5O2Color and Shape:SolidMolecular weight:481.52Hydrolyzed Fumonisin B2
CAS:<p>Hydrolyzed Fumonisin B2 (HFB2) is a hydrolysis product of fumonisins (HF), which retains biological activity. It exhibits phytotoxicity.</p>Formula:C22H47NO4Purity:98%Color and Shape:SolidMolecular weight:389.61Topoisomerase I/II inhibitor 4
<p>Topoisomerase I/II inhibitor 4 halts cell growth and spread, induces apoptosis, and is used in liver cancer research.</p>Formula:C27H21N5O6Color and Shape:SolidMolecular weight:511.49LXR antagonist 2
<p>LXR antagonist 2 inhibits adipogenesis, downregulates LXR genes, and reduces lipids in hyperlipidemic mice (LXRβ IC50: 0.36μM, LXRα IC50: 2.25μM).</p>Formula:C34H40N2O5SColor and Shape:SolidMolecular weight:588.76NTPDase-IN-3
CAS:<p>NTPDase-IN-3 inhibits NTPDase1/2/3/8 (IC50: 0.21/1.07/0.38/0.05 μM), useful for cancer and thrombosis research.</p>Formula:C22H24ClN3OS2Color and Shape:SolidMolecular weight:446.03Terguride
CAS:<p>Terguride: treats hyperprolactinemia, blocks 5-HT2A/B, activates dopamine receptors, studied for PAH.</p>Formula:C20H28N4OColor and Shape:SolidMolecular weight:340.46Dictyostatin
CAS:<p>Dictyostatin: potent microtubule stabilizer & anticancer agent with antiproliferative effects; researched for tauopathies.</p>Formula:C32H52O6Color and Shape:SolidMolecular weight:532.75Antibacterial agent 110
<p>Compound 4e, an antibacterial against P. aeruginosa, disrupts cell membranes (MIC: 1 μg/ml).</p>Formula:C22H21N5O4SColor and Shape:SolidMolecular weight:451.5MAO-B-IN-5
CAS:<p>MAO-B-IN-5: potent, selective oral MAO-B inhibitor, IC50=0.204μM, potential for Parkinson's research.</p>Formula:C19H21FN2O2Purity:97.68%Color and Shape:SolidMolecular weight:328.38PF-06751979
CAS:<p>PF-06751979 is an inhibitor of β-site amyloid precursor protein cleaving enzyme 1 (BACE1) (IC50 of 7.3 nM in BACE1 binding assay).</p>Formula:C18H19F2N5O3S2Purity:98%Color and Shape:SolidMolecular weight:455.5CB2 receptor antagonist 1
CAS:<p>Compound 29 is a potent, CB2-selective antagonist/reverse agonist. Derivatives 23 & 24 offer antinociception; 24 activates cannabinoid/TRPV1 receptors.</p>Formula:C28H47NO3Color and Shape:SolidMolecular weight:445.68Antibacterial agent 66
<p>Compound 6q, a trifluoromethylpyridine oxadiazole, targets Xanthomonas oryzae with EC50 of 7.2 μg/mL.</p>Formula:C17H10ClF6N3O2SColor and Shape:SolidMolecular weight:469.79SML-10-70-1
CAS:<p>SML-10-70-1 is a Novel Active Site Inhibitor of Oncogenic K-Ras G12C.</p>Formula:C25H42ClN7O13P2Color and Shape:SolidMolecular weight:746.04DI-404
CAS:<p>DI-404: Potent DCN1-UBC12 inhibitor, selectivity blocks cullin 3 neddylation, Kd=6.9 nM.</p>Formula:C35H45ClN6O6SPurity:98%Color and Shape:SolidMolecular weight:713.29Flurdihydroergotamine
CAS:<p>Flurdihydroergotamine, a serotonin 5HT1 receptor agonist, is used as an antimigraine drug.</p>Formula:C34H36F3N5O5Purity:98%Color and Shape:SolidMolecular weight:651.68FTO-IN-1 TFA
<p>FTO-IN-1 TFA: FTO enzyme inhibitor, anti-obesity, IC50 < 1μM, potential cancer research tool.</p>Formula:C20H17Cl2F3N4O4Color and Shape:SolidMolecular weight:505.27K252d
CAS:<p>K252d: indolocarbazole alkaloid in Nocardiopsis; inhibits PKC in rat brain and bovine heart phosphodiesterase.</p>Formula:C26H23N3O5Color and Shape:SolidMolecular weight:457.48MIV-150
CAS:<p>MIV-150 is a nonnucleoside inhibitor of reverse transcriptase (NNRT). MIV-150 also blocking HIV-1 and HIV-2 infections (EC50<1 nM against HIV-1/HIV-2MN).</p>Formula:C19H17FN4O3Purity:98%Color and Shape:SolidMolecular weight:368.36FXIa-IN-10
<p>FXIa-IN-10 is a potent, orally bioavailable inhibitor of Activator XI (FXIa) (Ki: 0.17 nM).</p>Formula:C23H18Cl2F3N9O2Color and Shape:SolidMolecular weight:580.35THR-β agonist 5
CAS:<p>THR-β agonist 5 (compound 54) is a potent THR-β agonist, with an EC 50 of <50 nM [1].</p>Formula:C22H23N5O2Color and Shape:SolidMolecular weight:389.45PptT-IN-2
<p>PptT-IN-2 inhibits PptT enzyme crucial in tuberculosis, with 2.5 μM IC50, showing potential in TB research.</p>Formula:C22H29N5O2Color and Shape:SolidMolecular weight:395.5sEH inhibitor-4
<p>Compound B15: potent sEH inhibitor (0.03 nm), reduces inflammation & pain.</p>Formula:C27H28Cl2N4O3Color and Shape:SolidMolecular weight:527.44HS-731
CAS:<p>HS-731 is a μ-Opioid Receptor Agonist.</p>Formula:C20H26N2O5Color and Shape:SolidMolecular weight:374.43VU6005806
CAS:<p>VU6005806 is a potent M4 PAM with EC50s: 94 nM (human), 28 nM (rat), 87 nM (dog), 68 nM (cyno); studied for neuropsychiatric disorders.</p>Formula:C17H16F3N7O2SPurity:98%Color and Shape:SolidMolecular weight:439.41Symplostatin 1
CAS:<p>Symplostatin 1 is a dolastatin 10 analog from the marine cyanobacterium Symploca hydnoides.</p>Formula:C43H70N6O6SColor and Shape:SolidMolecular weight:799.12RORγt inhibitor 2
CAS:<p>RORγt Inhibitor 2, a potent inhibitor of RORγt, exhibits an IC50 of 9.2 nM and is utilized in the study of cancer, inflammation, or autoimmune diseases that are</p>Formula:C31H33F5N2O7SColor and Shape:SolidMolecular weight:672.66PI3K-IN-23
<p>PI3K-IN-23 is a (E)-9-oxooctadec-10-en-12-ynoic acid analogue that promotes glucose uptake (EC50: 7.00 μM).</p>Formula:C24H33NO4SColor and Shape:SolidMolecular weight:431.59Antifungal agent 40
<p>Antifungal agent 40 blocks C. albicans CYP51 in pocket II, hindering lanosterol demethylase and biofilm growth.</p>Formula:C22H20Cl2N4SeColor and Shape:SolidMolecular weight:490.29Anticancer agent 142
CAS:<p>Compound 142 (also known as Compound 235) is a PTPN inhibitor with potential applications in cancer research [1].</p>Formula:C13H14BrF2N2O7PS2Purity:98%Color and Shape:SolidMolecular weight:523.26Hetrombopag olamine
CAS:<p>Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity.</p>Formula:C29H36N6O7Purity:98%Color and Shape:SolidMolecular weight:580.63HDAC6-IN-12
<p>HDAC6-IN-12 is a potent inhibitor of HDAC6 that binds in the DNA chain, causing DNA damage and exhibiting anticancer effects that can be used in cancer research</p>Formula:C24H39F2N3O5Color and Shape:SolidMolecular weight:487.58PEN-866
CAS:<p>PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.</p>Formula:C49H49N7O9Color and Shape:SolidMolecular weight:879.95Cdc7-IN-8
CAS:<p>Cdc7-IN-8, inhibits Cdc7 kinase, key in DNA replication, and is promising for cancer research. (WO2021032170A1)</p>Formula:C19H21N5O2Color and Shape:SolidMolecular weight:351.40ABL-L
CAS:<p>ABL-L is able to induce apoptosis in human laryngeal cancer cells using a p53-dependent pathway.</p>Formula:C29H46O6Color and Shape:SolidMolecular weight:490.67BW 443C
CAS:<p>BW 443C is a selective agonist of mu-opioid receptor.</p>Formula:C33H46N10O10Color and Shape:SolidMolecular weight:742.791Pisiferic acid
CAS:<p>Pisiferic acid is a novel PP2C activator and an an antimicrobial diterpenoid</p>Formula:C20H28O3Color and Shape:SolidMolecular weight:316.43UTPγS trisodium salt
CAS:<p>P2Y2 and P2Y4 receptor agonist</p>Formula:C9H12N2Na3O14P3SPurity:98%Color and Shape:SolidMolecular weight:566.15Fradafiban
CAS:<p>Fradafiban binds to the human platelet GP IIb/IIIa complex with a Kd value of 148 nM. Fradafiban is a non-polypeptide platelet glycoprotein IIb/IIIa antagonist.</p>Formula:C20H21N3O4Purity:98%Color and Shape:SolidMolecular weight:367.40AZD 2066 hydrate
<p>AZD 2066 hydrate is a selective, orally active, and brain-penetrant antagonist of mGluR5. It exhibits antinociceptive effects [1].</p>Formula:C19H18ClN5O3Color and Shape:SolidMolecular weight:386.33WDR5-IN-5
CAS:<p>WDR5-IN-5: Selective oral inhibitor for WDR5's WIN site with high affinity (Ki<0.02 nM) and anti-cancer properties. Good pharmacokinetics.</p>Formula:C29H29F3N6OColor and Shape:SolidMolecular weight:534.58PPI-2458
CAS:<p>PPI-2458, a fumagillin derivative, irreversibly blocks MetAP2, hindering abnormal cell growth and angiogenesis with improved toxicity.</p>Formula:C22H36N2O6Color and Shape:SolidMolecular weight:424.53A 74273
CAS:<p>A 74273, a nonpeptidic and renin inhibitor, may be used to treat cardiovascular diseases due to renin inhibition.</p>Formula:C44H74N4O8Purity:98%Color and Shape:SolidMolecular weight:787.08Bometolol Hydrochloride
CAS:<p>Bometolol Hydrochloride is a beta-adrenergic blocking compound used for the treatment of cardiovascular disease.</p>Formula:C25H33ClN2O7Purity:98%Color and Shape:SolidMolecular weight:508.99FAK inhibitor 6
CAS:<p>Compound 26F: potent enzyme inhibitor (IC50=28.2nM), low cytotoxicity (IC50=3.32μM), induces dose-dependent apoptosis in MDA-MB-231, blocks G0/G1 phase.</p>Formula:C25H24FN5O2SColor and Shape:SolidMolecular weight:477.55HDAC/Top-IN-1
CAS:<p>HDAC/Top-IN-1, an oral HDAC/Top inhibitor, targets HDAC1-3,6,8 with low IC50s; blocks S-phase & induces apoptosis in HEL cells.</p>Formula:C29H25FN4O4Color and Shape:SolidMolecular weight:512.53CDK8-IN-11 hydrochloride
<p>CDK8-IN-11 HCl: potent, selective CDK8 inhibitor (IC50: 46 nM), blocks WNT/β-catenin pathway, used in colon cancer research.</p>Formula:C19H16ClF3N4O2Color and Shape:SolidMolecular weight:424.8SIK1 activator 1
CAS:<p>SIK1 activator 1 boosts SIK1 phosphorylation, reduces type 2 diabetes hyperglycemia, and inhibits liver gluconeogenesis.</p>Formula:C23H32O6Color and Shape:SolidMolecular weight:404.50Ro 31-8472
CAS:<p>Ro 31-8472 is an angiotensin-converting enzyme (ACE) inhibitor and an analog of cilazaprilat.</p>Formula:C20H27N3O6Purity:98%Color and Shape:SolidMolecular weight:405.44Steroid sulfatase/17β-HSD1-IN-1
<p>Steroid sulfatase/17β-HSD1-IN-1 is a highly effective inhibitor of both steroid sulfatase and 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1) activities,</p>Formula:C19H18N2O5SColor and Shape:SolidMolecular weight:386.42Oral antiplatelet agent 1
CAS:<p>Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.</p>Formula:C23H24N4O5SPurity:98%Color and Shape:SolidMolecular weight:468.53MIF2-IN-1
<p>MIF2-IN-1, potent inhibitor of MIF2 (IC50: 1μM), halts non-small cell lung cancer growth via MAPK pathway.</p>Formula:C26H19F3N2O2SColor and Shape:SolidMolecular weight:480.5P2X7 receptor antagonist-1
<p>P2X7 receptor antagonist-1 is a purinergic P2X7 receptor antagonist with anti-neuroinflammatory effects.</p>Formula:C22H20F4N2O3Color and Shape:SolidMolecular weight:436.4TLR7/8 antagonist 2
<p>TLR7/8 antagonist 2: potent, orally active, IC50: 4.9 nM (TLR7), 0.6 nM (TLR8); potential for lupus therapy research.</p>Formula:C22H26FN5Color and Shape:SolidMolecular weight:379.47Carbonic anhydrase inhibitor 8
<p>R-13, a carbonic anhydrase inhibitor, has Ki of 60.7 nM (hCA I), 320.7 nM (hCA II), and 2298 nM (hCA IV).</p>Formula:C20H25N3O4SColor and Shape:SolidMolecular weight:403.5AGN-795
CAS:<p>AGN-795 is a biochemical.</p>Formula:C14H20N2Color and Shape:SolidMolecular weight:216.328(±)-ANAP hydrochloride (1185251-08-4 free base)
<p>(±)-ANAP hydrochloride is the amino acid analog of prodan. It can be used as a fluorescent probes and enhance environmental sensitivity.</p>Formula:C15H17ClN2O3Purity:98%Color and Shape:SolidMolecular weight:308.76Lp-PLA2-IN-10
<p>Lp-PLA2-IN-10, a potent Lp-PLA2 inhibitor, may research neurodegenerative and cardiovascular diseases.</p>Formula:C21H15F5N4O4Color and Shape:SolidMolecular weight:482.36Tacrolimus anhydrous 8-epimer
CAS:<p>Tacrolimus anhydrous 8-epimer, an immunosuppressive l-pipecolic acid macrolide, blocks T cell growth by hindering IL-2.</p>Formula:C44H69NO12Color and Shape:SolidMolecular weight:804.02TP003
CAS:<p>TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for α1β2gam2, α2β3gam2, α3β3gam2, α5β2gam2, EC50 of 20.3, 10.6, 3.24, 5.</p>Formula:C23H16F3N3OPurity:99.17%Color and Shape:SolidMolecular weight:407.39SAR-114137
CAS:<p>SAR-114137 is a histone sphingomyelin kinase inhibitor used in the study of molluscum arteriosum and peripheral neuropathic pain.</p>Formula:C25H34N4O7SPurity:99.09% - 99.91%Color and Shape:SolidMolecular weight:534.63Sulprostone
CAS:<p>EP3 and EP1 receptor agonist</p>Formula:C23H31NO7SPurity:98%Color and Shape:White To Off-White SolidMolecular weight:465.56γ-Secretase modulator 11 hydrochloride
CAS:<p>γ-Secretase modulator 11 hydrochloride is a potent, orally active γ-secretase modulator (IC50: 0.029 μM).</p>Formula:C28H23ClF2N4O2Color and Shape:SolidMolecular weight:520.96VEGFR-2-IN-14
<p>VEGFR-2-IN-14 (Compound 5) is a potent inhibitor of VEGFR-2, which inhibits the growth of HepG2 cells in the Pre-G1 phase and induces apoptosis.</p>Formula:C24H23N3O3SColor and Shape:SolidMolecular weight:433.52MEK1/2-IN-2
<p>MEK1/2-IN-2 is a potent, ATP-competitive MEK1/2 inhibitor that exhibits equal inhibitory effects on wild-type MEK1/2 and a group of MEK1/2 mutant cells.</p>Formula:C28H22ClFN6OColor and Shape:SolidMolecular weight:512.97AMPK Activator SC4
CAS:<p>SC4 is a potent, direct AMPK activator. SC4 preferentially activates α2 complexes and stimulates skeletal muscle glucose uptake.</p>Formula:C26H18ClN3O4Color and Shape:SolidMolecular weight:471.89Novokinin
CAS:<p>Angiotensin AT2 receptor agonist</p>Formula:C39H61N11O7Purity:98%Color and Shape:SolidMolecular weight:795.97U 80215
CAS:<p>U 80215 is an enzyme-competitive inhibitor.</p>Formula:C42H60N8O6SColor and Shape:SolidMolecular weight:805.04
