Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,523 products)
- Apoptosis(5,792 products)
- Cell Cycle/Checkpoint(4,449 products)
- Chromatin/Epigenetics(2,238 products)
- Cytoskeletal Signaling(1,383 products)
- DNA Damage/DNA Repair(2,825 products)
- Endocrinology/Hormones(3,507 products)
- Enzyme(3,640 products)
- GPCR/G-Protein(8,333 products)
- Immunology and Inflammation(3,526 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(404 products)
- MAPK Signaling(1,202 products)
- Membrane Transporter/Ion Channel(2,790 products)
- Metabolism(9,448 products)
- Microbiology/Virology(6,981 products)
- Neuroscience(9,926 products)
- Other Inhibitors(37,926 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,400 products)
- Proteases/Proteasome(1,597 products)
- Stem Cell and Derivatives(831 products)
- Tyrosine Kinase/Adaptors(2,016 products)
- Ubiquitination(1,650 products)
Show 16 more subcategories
Found 66641 products of "Inhibitors"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
LGB-321 HCl
CAS:<p>LGB-321: potent, selective PIM kinase inhibitor, active against PIM2, halts diverse blood cancers' growth, orally effective in mice.</p>Formula:C23H23ClF3N5O2Color and Shape:SolidMolecular weight:493.91RS 2135
CAS:<p>RS 2135 is a novel class I antiarrhythmic agent to inhibit ischemia-induced ventricular arrhythmias.</p>Formula:C18H21ClN2O2Purity:98%Color and Shape:SolidMolecular weight:332.83Isoleucyl tRNA synthetase-IN-2
CAS:<p>Isoleucyl tRNA synthetase-IN-2 is a selective and potent inhibitor (Ki: 114 nM) that targets isoleucyl tRNA synthetase (IleRS).</p>Formula:C22H33N5O8SColor and Shape:SolidMolecular weight:527.59KRAS G12C inhibitor 44
<p>KRAS G12C inhibitor 44: potent, oral, anti-cancer; halts cell growth in MIA PaCA-2, H358; effective in vivo. IC50: MIA-0.016μM, H358-0.028μM.</p>Formula:C31H36ClFN6O2Color and Shape:SolidMolecular weight:579.11BMS-986339
CAS:<p>BMS-986339: oral, potent FXR agonist; binds to His298/ASN287; for PBC, PSC, NASH, anti-fibrosis research.</p>Formula:C35H41F4N3O4Color and Shape:SolidMolecular weight:643.71CK2 inhibitor 3
<p>CK2 inhibitor 3: potent CK2 blocker, IC50 of 280 nM, suppresses tumor cell growth, highly selective among 320 kinases.</p>Formula:C13H9BrN4O3SColor and Shape:SolidMolecular weight:381.2Ketomethylenebestatin
CAS:<p>Ketomethylenebestatin, a weaker carba-analog of aminopeptidase inhibitor bestatin, is 10x less potent.</p>Formula:C17H25NO4Purity:98%Color and Shape:SolidMolecular weight:307.38β-Glucuronidase/hCAII-IN-2
<p>β-Glucuronidase/hCAII-IN-2 is a potent inhibitor of β-glucuronidase and hCA II, and their IC50 values were 670.7 μM and 21.77 μM, respectively.</p>Formula:C31H23NO8Color and Shape:SolidMolecular weight:537.52BChE-IN-3
<p>BChE-IN-3: Selective, pseudo-irreversible BChE inhibitor (IC50: 56.9 nM); borderline reversible AChE inhibitor.</p>Formula:C26H41N3O2Color and Shape:SolidMolecular weight:427.62(R)-FL118
CAS:<p>FL118 inhibits human survivinion expression and activates tumor suppressor p53 as a MOA in p53 wild-type cancer cells.</p>Formula:C21H16N2O6Color and Shape:SolidMolecular weight:392.36HPK1-IN-3
<p>HPK1-IN-3: Selective HPK1 inhibitor, ATP-competitive, IC50=0.25nM; boosts IL-2 in PBMCs, EC50=108nM.</p>Formula:C23H22F4N6O2Color and Shape:SolidMolecular weight:490.45Anticancer agent 54
<p>Anticancer agent 54 blocks cell cycle in G0/G1, induces apoptosis, and fights cancer via DNA embedding and ROS.</p>Formula:C33H36N6Color and Shape:SolidMolecular weight:516.68NS2B/NS3-IN-3
CAS:<p>NS2B/NS3-IN-3 (Compd 66) is an inhibitor of Flavivirus NS2B-NS3 protease [1] .</p>Formula:C19H21N3O2Color and Shape:SolidMolecular weight:323.39rel-MDM2/4-p53-IN-3
<p>rel-MDM2/4-p53-IN-3 inhibits MDM2/4-p53 PPI, IC50: MDM2 18.5nM, MDM4 14.8nM, targets cancer research.</p>Formula:C25H24Cl2FN3O3Color and Shape:SolidMolecular weight:504.38TLR4/NF-κB/MAPK-IN-1
CAS:<p>TLR4/NF-κB/MAPK-IN-1 is a novel antineuroinflammatory agent that functions by inhibiting the TLR4/NF-κB/MAPK pathways.</p>Formula:C19H25BrO6Color and Shape:SolidMolecular weight:429.3Canosimibe
CAS:<p>Canosimibe is a cholesterol absorption inhibitor</p>Formula:C44H60FN3O10Color and Shape:SolidMolecular weight:809.96SHP2-IN-9
<p>SHP2-IN-9: Potent SHP2 inhibitor, IC50=1.174 μM, 85x SHP1 selectivity, crosses blood-brain barrier, hampers cancer growth.</p>Formula:C20H20FN3O2SColor and Shape:SolidMolecular weight:385.46MI-1481
CAS:<p>MI-1481: potent MML1 inhibitor, IC50 3.6 nM; disrupts menin-MLL1, active in MLL leukemia.</p>Formula:C29H30F3N7O2SPurity:98%Color and Shape:SolidMolecular weight:597.65NITD-688
CAS:<p>NITD-688 is a pan-serotype inhibitor targeting the dengue virus NS4B protein, effective through oral administration.</p>Formula:C25H32N4O3S2Color and Shape:SolidMolecular weight:500.68(-)-Mesembrine
CAS:<p>Mesembrine is a serotonin reuptake inhibitor and is also a weak inhibitor of the enzyme phosphodiesterase 4 (PDE4).</p>Formula:C17H23NO3Color and Shape:SolidMolecular weight:289.37BU09059
CAS:<p>BU09059 is a potent, selective, short-acting antagonist of the κ-opioid receptor (KOR).</p>Formula:C28H37N3O5Purity:98%Color and Shape:SolidMolecular weight:495.61HIV-1 inhibitor-13
<p>HIV-1 inhibitor-13: oral NNRTI, IC50=0.14μM for HIV-1 RT, effective on resistant strains (EC50=2.85-18nM).</p>Formula:C30H32N6O3Color and Shape:SolidMolecular weight:524.61NVP-CFC218
CAS:<p>NVP-CFC218 is a novel potent and selective p53-HDM2 inhibitor.</p>Formula:C37H45ClN4O4Color and Shape:SolidMolecular weight:645.23Uprosertib hydrochloride
CAS:<p>Uprosertib hydrochloride is a potent and selective inhibitor of pan-Akt (IC50: 180/328/38 nM for Akt1/Akt2/Akt3, respectively).</p>Formula:C18H17Cl3F2N4O2Purity:98%Color and Shape:SolidMolecular weight:465.71MRS4458
CAS:<p>MRS4458 is an effective inhibitor of the P2Y14 Receptor.</p>Formula:C24H20F3N5O3SPurity:98%Color and Shape:SolidMolecular weight:515.51SARS-CoV-2-IN-8
<p>SARS-CoV-2-IN-8 is a major protease inhibitor of SARS-CoV-2 (IC50: 0.75 μM).</p>Formula:C35H38N6O3Color and Shape:SolidMolecular weight:590.71PrCP-7414
CAS:<p>PrCP-7414 is a potent PrCP inhibitor, CAS# 1252037-41-4, named after the CAS number's last four digits.</p>Formula:C31H33Cl2N5O2Color and Shape:SolidMolecular weight:578.53TAK-828F
CAS:<p>TAK-828F: potent, selective RORγt inverse agonist. Oral. IC50=1.9 nM; reporter gene IC50=6.1 nM.</p>Formula:C28H32FN3O5Purity:98%Color and Shape:SolidMolecular weight:509.57Artemisiane E
CAS:<p>Artemisiane E is a potent PI3K/AKT pathway inhibitor with an IC 50 of 8.9 μM .</p>Formula:C20H22O5Color and Shape:SolidMolecular weight:342.39ATM Inhibitor-2
<p>ATM Inhibitor -2 is a potent and selective inhibitor of ATM (IC50<1 nM).</p>Formula:C26H31N7O3Color and Shape:SolidMolecular weight:489.57STING agonist-7
<p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>Formula:C17H12N4O4Color and Shape:SolidMolecular weight:336.3AX15910
<p>AX15910 is a potent inhibitor of BRD4 and ERK5.</p>Formula:C32H38N6O3Color and Shape:SolidMolecular weight:554.7SCH-1473759
CAS:<p>SCH-1473759 is an inhibitor of the aurora (IC50s: 4 and 13 nM for Aurora A and B, respectively).</p>Formula:C20H26N8OSPurity:98%Color and Shape:SolidMolecular weight:426.54Methyl Streptonigrin
CAS:<p>Methyl Streptonigrin is an ABCG2 transporter function inhibitor.</p>Formula:C26H24N4O8Purity:98%Color and Shape:SolidMolecular weight:520.49PROTAC FKBP Degrader-3
CAS:<p>PROTAC FKBP Degrader-3, with FKBP and VHL binding groups linked, is a potent FKBP degrader.</p>Formula:C68H90N6O17SPurity:98%Color and Shape:SolidMolecular weight:1295.54ATP synthase inhibitor 2
CAS:<p>ATP synthase inhibitor 2 blocks P. aeruginosa ATP synthase; IC50=10 μg/mL, fully inhibits at 128 μg/mL.</p>Formula:C21H22N2O3SColor and Shape:SolidMolecular weight:382.48Fonsartan free acid
CAS:<p>Fonsartan: Angiotensin receptor blocker, halts angiotensin II effects on rat vascular cells.</p>Formula:C26H32N4O5S2Purity:98%Color and Shape:SolidMolecular weight:544.69CCW 28-3
CAS:<p>CCW 28-3 is a novel potent covalent BRD4 degrader, degrading BRD4 in a proteasome- and RNF4-dependent manner without inhibiting RNF4 autoubiquitination activity</p>Formula:C44H42Cl2N6O4SColor and Shape:SolidMolecular weight:821.81Anti-inflammatory agent 10
<p>Tilomisole-derived benzimidazole-thiazole, orally active, favors COX-2 inhibition over COX-1.</p>Formula:C17H13BrN4O3S2Color and Shape:SolidMolecular weight:465.34GRP78-IN-1
<p>GRP78-IN-1 binds to GRP78 protein, inhibits cell growth, and triggers apoptosis in breast cancer; has -8.07 kcal/mol binding energy.</p>Formula:C21H23FO3Color and Shape:SolidMolecular weight:342.4OSI-7904L free acid
CAS:<p>OSI-7904L is a folate-based thymidylate synthase inhibitor. It also has antimalarial and antitumor properties.</p>Formula:C27H24N4O6Purity:98%Color and Shape:SolidMolecular weight:500.5TRPC4/5-IN-1
<p>TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.</p>Formula:C21H21N3OColor and Shape:SolidMolecular weight:331.41DC1SMe
CAS:<p>DC1, a CC-1065-like ADC cytotoxin, is used in cancer-targeting antibody-drug conjugates. DC1Sme, a derivative, has IC50s: 22-250 pm in various cancer cells.</p>Formula:C35H30ClN5O4S2Purity:98%Color and Shape:SolidMolecular weight:684.23Teslexivir
CAS:<p>Teslexivir is a topical antiviral agent that is an effective and selective inhibitor of the interaction between two essential viral proteins, E1 and E2.</p>Formula:C35H36BrN3O4Purity:98%Color and Shape:SolidMolecular weight:642.586-trans-12-epi-Leukotriene B4
CAS:<p>6-trans-12-epi-Leukotriene B4, a metabolite of arachidonic acid, serves as a potent anti-inflammatory agent.</p>Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47CK2-IN-3
<p>CK2-IN-3: potent, selective CK2 inhibitor; Kd=12 nM, IC50: 1.51 μM (CK2α), 7.64 μM (CK2α'). For cancer research.</p>Formula:C22H26N4O7Color and Shape:SolidMolecular weight:458.46MtTMPK-IN-1
<p>MtTMPK-IN-1 inhibits MtTMPK with 2.5 μM IC50, shows moderate anti-tuberculosis activity, and is low in cytotoxicity.</p>Formula:C22H24N4O3Color and Shape:SolidMolecular weight:392.45PARP10/15-IN-3
<p>Compound 8a, a dual PARP10 & PARP15 inhibitor, has IC50s: PARP10 at 0.14μM & PARP15 at 0.40μM; it's cell-permeable & anti-apoptotic.</p>Formula:C12H12N2O3Color and Shape:SolidMolecular weight:232.24Pamiparib maleate
CAS:<p>Pamiparib (BGB-290) is a selective PARP inhibitor that blocks DNA repair and promotes apoptosis.</p>Formula:C44H42F2N8O14Purity:98%Color and Shape:SolidMolecular weight:944.859EZH2-IN-12
<p>EZH2-IN-12 (Compound 5) is a potent inhibitor of EZH2, which has potential for studies of CNS malignancies.</p>Formula:C23H23Cl2N3O3Color and Shape:SolidMolecular weight:460.35Sekdel sequence
CAS:<p>Sekdel sequence, as a signal, leads to retention of at least two proteins in the endoplasmic reticulum of animal cells.</p>Formula:C29H49N7O14Color and Shape:SolidMolecular weight:719.74Antifungal agent 43
<p>Antifungal agent 43 inhibits biofilms with low toxicity to human cancer cells.</p>Formula:C24H26N4Se2Color and Shape:SolidMolecular weight:528.41MK-6913
CAS:<p>MK-6913 is a potent and selective agonist of estrogen receptor β.</p>Formula:C25H27N3O2Purity:98%Color and Shape:SolidMolecular weight:401.5RAD51-IN-8
<p>RAD51-IN-8 inhibits RAD51-BRCA2 interaction and H4A4 with EC50 of 19 μM; a micromolar PPI inhibitor.</p>Formula:C16H14Cl2FN3O2Color and Shape:SolidMolecular weight:370.21Menin-MLL inhibitor 4
CAS:<p>Menin-MLL inhibitor 4 has antitumor activity.Menin-MLL inhibitor 4 is an inhibitor of Menin- MLL (mixed-lineage leukemia protein) interaction .</p>Formula:C32H38FN7O3Purity:98%Color and Shape:SolidMolecular weight:587.69ChE/Aβ1-42-IN-1
<p>ChE/Aβ1-42-IN-1 (compound 28) is a potent aggregation inhibitor of ChE and Aβ 1-42 with excellent BBB permeability.</p>Formula:C19H24N2O3Color and Shape:SolidMolecular weight:328.41MRGPRX1 agonist 3
<p>Compound 1f, a potent MRGPRX1 agonist, has an EC50 of 0.22 μM, useful for neuropathic pain studies.</p>Formula:C14H11FN2OSColor and Shape:SolidMolecular weight:274.31Udifitimod
CAS:<p>Udifitimod (BMS-986166) is a potent, selective, and orally active modulator of the S1P1R receptor, showing potential for research in autoimmune diseases.</p>Formula:C25H33NO2Color and Shape:SolidMolecular weight:379.54NDM-1 inhibitor-3
<p>NDM-1 inhibitor-3 is a New Delhi Metallo-β-lactamase-1 (NDM-1) inhibitor (Ki : 4 μM) widely found in nature and is associated with antibiotic resistance.</p>Formula:C16H12O4Purity:98.66%Color and Shape:SolidMolecular weight:268.26PD 135158
CAS:<p>PD 135158 is a CCK2 receptor antagonist.</p>Formula:C42H61N5O11Purity:98%Color and Shape:SolidMolecular weight:811.96ERK2 IN-1
CAS:<p>ERK2 IN-1 is a selective ERK2 inhibitor with an IC50 of 7 nM.</p>Formula:C36H34FN7O2SPurity:98%Color and Shape:SolidMolecular weight:647.76FTO-IN-6
CAS:<p>FTO-IN-6 is a selective inhibitor of fat mass and obesity associated protein (FTO).</p>Formula:C14H12N4O6Color and Shape:SolidMolecular weight:332.27DS89002333
<p>DS89002333: oral PRKACA inhibitor with 0.3 nM IC50, effective against FL-HCC with DNAJB1-PRKACA fusion in xenografts.</p>Formula:C22H20ClF2N3O3Color and Shape:SolidMolecular weight:447.86PIM1-IN-3
<p>PIM1-IN-3 (HL8) selectively blocks PIM1, induces Colo320 cell apoptosis, and may be researched for cancer.</p>Formula:C27H25BrN6OColor and Shape:SolidMolecular weight:529.43HDAC6-IN-13
<p>HDAC6-IN-13: potent, selective HDAC6 inhibitor; oral; IC50=0.019μM; targets HDAC1/2/3; crosses blood-brain barrier; anti-inflammatory.</p>Formula:C23H22N4OColor and Shape:SolidMolecular weight:370.45Antitubercular agent-29
<p>Compound 6xa inhibits drug-resistant tuberculosis with MICs 0.03 μg/mL for DS-Mtb and 0.03-0.06 for DR-Mtb, SI>40 for Vero cells.</p>Formula:C20H12ClN3O5Color and Shape:SolidMolecular weight:409.78M826
<p>M826, a non-peptide, potent, selective, and reversible caspase-3 inhibitor, exhibits an IC50 of 0.005 μM and demonstrates strong anti-apoptotic activity in</p>Formula:C28H45N7O6Purity:98%Color and Shape:SolidMolecular weight:575.7VHL Ligand 8
CAS:<p>VHL Ligand 8, a VHL ligand essential for synthesizing ARD-266, acts as a highly potent VHL E3 ligase-based androgen receptor (AR) PROTAC degrader.</p>Formula:C23H29N3O6Purity:98%Color and Shape:SolidMolecular weight:443.49Antitumor agent-37
<p>Antitumor agent-37: strong anti-growth, anti-spread, induces DNA damage, apoptosis via Bcl-2/Bax/caspase3, boosts immune response.</p>Formula:C16H18Cl2N2O4PtColor and Shape:SolidMolecular weight:568.32LSD1-IN-13 hydrochloride
CAS:<p>LSD1-IN-13 hydrochloride (7e) is an oral LSD1 inhibitor (IC50: 24.43 nM), promoting differentiation in AML cell lines.</p>Formula:C23H30ClN3O2SColor and Shape:SolidMolecular weight:448.02(S)-Seco-Duocarmycin SA
CAS:<p>(S)-Seco-Duocarmycin SA is a DNA alkylating agent and antibiotic with potent antitumor activity that can be used to synthesize ADC compounds.</p>Formula:C25H24ClN3O7Purity:98%Color and Shape:SolidMolecular weight:513.93ART615
<p>ART615 is a related isomer of ART558. ART615 inhibits Polθ by <10% at 12 μM and is able to act as a control for ART558 (IC50:7.9 nM).</p>Formula:C21H21F3N4O2Color and Shape:SolidMolecular weight:418.41AZ-PFKFB3-67 quarterhydrate
<p>AZ-PFKFB3-67 quarterhydrate inhibits PFKFB3 (IC50: 11 nM), PFKFB2 (159 nM), and PFKFB1 (1130 nM).</p>Formula:C26H27N5O4Color and Shape:SolidMolecular weight:460.01MT-134
<p>MT-134 is a SkMII -specific inhibitor and has excellent exposure in muscles.</p>Formula:C19H16N4O3Color and Shape:SolidMolecular weight:348.36Efrapeptin F
CAS:<p>Efrapeptin F, from Tolypocladium fungi, inhibits mitochondrial complex V and targets nutrient-deprived tumor cells.</p>Formula:C82H141N18O16Color and Shape:SolidMolecular weight:1635.11Samuraciclib
CAS:<p>Samuraciclib (CT7001) is an oral CDK7 inhibitor with 41 nM IC50, notable for its high selectivity and potency against breast cancer cells.</p>Formula:C22H30N6OColor and Shape:SolidMolecular weight:394.51RET-IN-14
CAS:<p>RET-IN-14 inhibits RET (IC50: <0.51-9.3 nM) & BTK (C481S) (IC50: 9.2-15 nM), promising for tumor research.</p>Formula:C24H23FN8O4Color and Shape:SolidMolecular weight:506.49Metesind Glucuronate
CAS:<p>Metesind Glucuronate is an antineoplastic. It also is a specific thymidylate synthase inhibitor.</p>Formula:C29H34N4O10SColor and Shape:SolidMolecular weight:630.67MA242
CAS:<p>MA242 is a nuclear factor of activated T cells 1 (NFAT1) for Pancreatic Cancer Therapy and dual inhibitor of murine double minute 2 (MDM2).</p>Formula:C26H21ClF3N3O5SPurity:98%Color and Shape:SolidMolecular weight:579.98D-473
CAS:<p>D-473 is a novel orally active triple reuptake inhibitor targeting dopamine, serotonin and norepinephrine transporters.</p>Formula:C26H27F2NO3Color and Shape:SolidMolecular weight:439.49VU6005806
CAS:<p>VU6005806 is a potent M4 PAM with EC50s: 94 nM (human), 28 nM (rat), 87 nM (dog), 68 nM (cyno); studied for neuropsychiatric disorders.</p>Formula:C17H16F3N7O2SPurity:98%Color and Shape:SolidMolecular weight:439.4114α-Demethylase/DNA Gyrase-IN-1
<p>14α-Demethylase/DNA Gyrase-IN-1 (Compound 7c) is a potent inhibitor of 14α-Demethylase/DNA Gyrase with antibacterial activity.</p>Formula:C26H22N4O4Color and Shape:SolidMolecular weight:454.48Topoisomerase I inhibitor 8
CAS:<p>Topoisomerase I inhibitor 8, a hexacyclic analogue of camptothecin, is also a potent inhibitor of topoisomerase I and is toxic to tumour cells.</p>Formula:C24H21FN2O4Color and Shape:SolidMolecular weight:420.43Nikkomycin Z
CAS:<p>Nikkomycin Z (Nikkomycin Z from Streptomyces tendae) is a competitive chitin synthase inhibitor.It inhibitor of the growth of filamentous fungi, insects,</p>Formula:C20H25N5O10Purity:98%Color and Shape:SolidMolecular weight:495.44LP-284
CAS:<p>LP-284 is a DNA alkylating agent effective against solid tumors and hematologic cancers like MCL.</p>Formula:C16H20N2O4Color and Shape:SolidMolecular weight:304.34Sinulatumolin E
CAS:<p>Sinulatumolin E, a terpenoid, inhibits TNF-α (IC 50: 3.6 μM); has anti-inflammatory properties.</p>Formula:C15H22O2Color and Shape:SolidMolecular weight:234.33Antitubercular agent-22
<p>Antitubercular agent-22 combats Candida albicans (MIC: 2.34 μg/ml) and M. tuberculosis (MIC: 2 μg/ml).</p>Formula:C24H28FN5O8Color and Shape:SolidMolecular weight:533.51Napsagatran hydrate
CAS:<p>Napsagatran hydrate is a novel and specific inhibitor of thrombin.</p>Formula:C26H36N6O7SPurity:98%Color and Shape:SolidMolecular weight:576.66YKL-05-093
CAS:<p>YKL-05-093 is a alt inducible kinase (SIK) inhibitor. YKL-05-093 increases bone formation and bone mass.</p>Formula:C35H40N6O4Color and Shape:SolidMolecular weight:608.73AChE-IN-10
<p>AChE-IN-10 (24r) inhibits AChE (IC50=2.4 nM), reducing amyloid buildup, tau phosphorylation, and promotes neuron health.</p>Formula:C23H27F2NO4SColor and Shape:SolidMolecular weight:451.53Aeruginosin 98-B
CAS:<p>Aeruginosin 98-B, a protease inhibitor, effectively inhibits trypsin, plasmin, and thrombin with IC50 values of 0.6, 7.0, and 10.0 μg/mL, respectively.</p>Formula:C29H46N6O9SColor and Shape:SolidMolecular weight:654.78T-Type calcium channel inhibitor 2
<p>Compound 6g inhibits T-type Ca channels (IC50: Cav3.1-31μM, Cav3.2-83μM), cytotoxic to A549 (IC50: 5μM) & HCT-116 cells (IC50: 6.4μM).</p>Formula:C36H39FN4OSColor and Shape:SolidMolecular weight:594.78Mal-PEG4-VA-PBD
CAS:<p>Mal-PEG4-VA-PBD is a drug-linker conjugate for Antibody-Drug Conjugates (ADCs), comprising the antitumor antibiotic Pyrrolobenzodiazepine (PBD), connected</p>Formula:C68H79N9O17Purity:98%Color and Shape:SolidMolecular weight:1294.41(25S)-δ7-Dafachronic acid
CAS:<p>(25S)-delta7-Dafachronic acid, an orphan nuclear receptor DAF-12 ligand, inhibits the dauer-promoting activity of DAF-12.</p>Formula:C27H42O3Purity:98%Color and Shape:SolidMolecular weight:414.62Tacrolimus anhydrous 8-epimer
CAS:<p>Tacrolimus anhydrous 8-epimer, an immunosuppressive l-pipecolic acid macrolide, blocks T cell growth by hindering IL-2.</p>Formula:C44H69NO12Color and Shape:SolidMolecular weight:804.02VEGFR2-IN-1
CAS:<p>VEGFR2-IN-1 is a VEGFR2 inhibitor with antitumor activity used in the study of breast cancer.</p>Formula:C22H18N6SPurity:98.15%Color and Shape:SolidMolecular weight:398.48Tubulin polymerization-IN-4
CAS:<p>Tubulin polymerization-IN-4: inhibits tubulin (IC50=4.6 μM), blocks G2/M phase, induces apoptosis, hinders cell cloning/migration, damages vasculature.</p>Formula:C21H21ClN2O4Color and Shape:SolidMolecular weight:400.86PI3kδ inhibitor 1
CAS:<p>PI3kδ inhibitor 1 is a selective inhibitor of PI3Kδ (IC50 of 3.8 nM).</p>Formula:C28H33FN6O2Purity:98%Color and Shape:SolidMolecular weight:504.60Salacinol
CAS:<p>Salacinol is a naturally occurring alpha-glucosidase inhibitor isolated from an Ayurvedic traditional medicine Salacia reticulata.</p>Formula:C9H18O9S2Color and Shape:SolidMolecular weight:334.37Antibacterial agent 118
<p>Antibacterial agent 118, potent against various mycobacteria, has MIC values ranging from 10.2 to 163.0 μM. Useful in TB research.</p>Formula:C19H21N5O2SColor and Shape:SolidMolecular weight:383.47LIT-001 free base
CAS:<p>LIT-001, a nonpeptide OT-R agonist, enhances mouse autism-like behavior, with EC50=55 nM and Ki=226 nM.</p>Formula:C28H33N7O2SPurity:98%Color and Shape:SolidMolecular weight:531.67Dual AChE-MAO B-IN-1
<p>Dual AChE-MAO B-IN-1: orally active CNS-permeable, safe, stable neuroprotective agent; AChE IC50=550 nM, MAO-B IC50=8.2 nM.</p>Formula:C23H25F2NO4Color and Shape:SolidMolecular weight:417.45Epiderstatin
CAS:<p>Epiderstatin is isolated from Streptomyces pulveraceus subsp. epiderstagenes; inhibits mitogenic activity of epidermal growth factor.</p>Formula:C15H20N2O4Color and Shape:SolidMolecular weight:292.33URAT1 inhibitor 2
<p>URAT1 inhibitor 2: oral URAT1/CYP blocker, IC50 of 1.36μM (URAT1), 16.97μM (CYP1A2), 5.22μM (CYP2C9); potential gout treatment.</p>Formula:C21H18BrN3O2SColor and Shape:SolidMolecular weight:456.36LSD1-IN-22
<p>LSD1-IN-22: potent LSD1 inhibitor, K_i 98 nM, curbs cancer cell growth.</p>Formula:C9H8BrF2NColor and Shape:SolidMolecular weight:248.07XIAP/cIAP1 antagonist-1
<p>Potent oral XIAP/cIAP1 inhibitor with EC50s: XIAP 5.1 nM, cIAP1 0.32 nM; curbs tumor growth in vivo.</p>Color and Shape:SolidGSK866
CAS:<p>GSK866 is a selective glucocorticoid receptor agonist (SEGRA).</p>Formula:C23H21Cl2F4N5O3Color and Shape:SolidMolecular weight:562.34Aurora B inhibitor 1
CAS:<p>Aurora B inhibitor 1 is an Aurora B (Aurora-1) inhibitor (Ki <0.010 uM) with potential anticancer activity for cancer research.</p>Formula:C25H26ClF2N7O2Purity:98.37%Color and Shape:SolidMolecular weight:529.97Iroxanadine hydrobromide
CAS:<p>Iroxanadine hydrobromide is a MAPK p38 inhibitor potentially for the treatment of atherosclerosis.</p>Formula:C14H21BrN4OColor and Shape:SolidMolecular weight:341.25Dyrk1A-IN-1
<p>Dyrk1A-IN-1 is a triple inhibitor of Dyrk1A kinase activity, aggregation of tau and α-syn oligomers, with an IC50 value of 119 nM for Dyrk1A kinase.</p>Formula:C23H20N4O3SColor and Shape:SolidMolecular weight:432.49Alpibectir
CAS:<p>Alpibectir has antibacterial activity [1].</p>Formula:C12H14F6N2O2Color and Shape:SolidMolecular weight:332.24KDM1/CDK1-IN-1
<p>KDM1/CDK1-IN-1 inhibits KDM1 (IC50: 0.096 μM) & CDK1 (IC50: 0.078 μM), blocks HOP-92 G2/M phase, induces apoptosis, toxic to cancer cells.</p>Formula:C22H17N5O3SColor and Shape:SolidMolecular weight:431.47(-)-15-Deoxyspergualin
CAS:<p>(-)-15-Deoxyspergualin is a potent antitumor agent that demonstrates significant inhibition against mouse leukemia L-1210.</p>Formula:C17H37N7O3Color and Shape:SolidMolecular weight:387.52COX-2-IN-10
<p>COX-2-IN-10 is a potent COX-2 inhibitor, reducing IL-6, TNF-α, IL-1β, PGE2 (IC50=2.54 μM), and iNOS expression.</p>Formula:C31H32FN5O2SColor and Shape:SolidMolecular weight:557.68SAR-114137
CAS:<p>SAR-114137 is a histone sphingomyelin kinase inhibitor used in the study of molluscum arteriosum and peripheral neuropathic pain.</p>Formula:C25H34N4O7SPurity:99.09% - 99.91%Color and Shape:SolidMolecular weight:534.63Cav 3.2 inhibitor 1
<p>Cav 3.2 inhibitor 1 targets T-type calcium channels, weakly binds D2 receptors, and aids physical and visceral pain research.</p>Formula:C32H39N3OColor and Shape:SolidMolecular weight:481.67UCN-02
CAS:<p>UCN-02 (7-epi-Hydroxystaurosporine) is a PKC inhibitor produced by Streptomyces N-126 strain, which inhibits PKA.</p>Formula:C28H26N4O4Purity:98%Color and Shape:SolidMolecular weight:482.53Fosmanogepix
CAS:<p>Fosmanogepix (APX001) is a broad-spectrum oral antifungal that targets Gwt1 enzyme, transforming into active APX001A in the body.</p>Formula:C22H21N4O6PPurity:98%Color and Shape:SolidMolecular weight:468.40AFP464 free base
CAS:<p>AFP464 (NSC710464) free base is an active HIF-1α inhibitor (IC50: 0.25 μM) and a potent aryl hydrocarbon receptor (AhR) activator.</p>Formula:C22H23F3N4O3Purity:98%Color and Shape:SolidMolecular weight:448.44GSK945237
CAS:<p>GSK945237 is a type IIA topoisomerase inhibitor, effective on Gram-positive and negative bacteria, with favorable pharmacokinetics and in vivo efficacy.</p>Formula:C24H26FN5O3Color and Shape:SolidMolecular weight:451.49L 731735
CAS:<p>L 731735 is a farnesyltransferase inhibitor.</p>Formula:C19H40N4O4SPurity:98%Color and Shape:SolidMolecular weight:420.61J-104871
CAS:<p>J-104871 (UNII-6137X5QNJF) is an FTase inhibitor that inhibits tumor growth in nude mice transplanted with activated H-ras-transformed NIH3T3 cells.</p>Formula:C38H32N2O12Purity:98%Color and Shape:SolidMolecular weight:708.67A 76889
CAS:<p>A 76889 is an inhibitor of HIV-1 protease.</p>Formula:C44H58N8O6Purity:98%Color and Shape:SolidMolecular weight:794.98Netupitant metabolite Monohydroxy Netupitant
CAS:<p>Monohydroxy Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.</p>Formula:C30H32F6N4O2Purity:98%Color and Shape:SolidMolecular weight:594.59Mesulergine hydrochloride
CAS:<p>5-HT2A and 2C receptor antagonist</p>Formula:C18H27ClN4O2SPurity:98%Color and Shape:SolidMolecular weight:398.95BMS-986163
CAS:<p>BMS-986163, a prodrug, quickly becomes BMS-986169, a GluN2B inhibitor (Ki=4 nM, IC50=24 nM).</p>Formula:C23H28FN2O5PPurity:98%Color and Shape:SolidMolecular weight:462.45Antifungal agent 39
CAS:<p>Antifungal agent 39 (Compound 9h) is a broad-spectrum antifungal agent.</p>Formula:C23H22ClN3O5Color and Shape:SolidMolecular weight:455.89PROTAC CDK12/13 Degrader-1
<p>PROTAC CDK12/13 Degrader-1 (7f) selectively degrades CDK12/13 at nanomolar potency, targeting breast cancer.</p>Color and Shape:SolidMAO-B-IN-5
CAS:<p>MAO-B-IN-5: potent, selective oral MAO-B inhibitor, IC50=0.204μM, potential for Parkinson's research.</p>Formula:C19H21FN2O2Purity:97.68%Color and Shape:SolidMolecular weight:328.38Lu 26-046
CAS:<p>Lu 26-046 is a muscarinic receptor agonist.</p>Formula:C10H12N2OSColor and Shape:SolidMolecular weight:208.28hCAIX/XII-IN-5
<p>Coumarin 9a: Selective inhibitor of hCA IX/XII (Ki 93.3/85.7 nM), blocks cancer cell growth, and induces apoptosis.</p>Formula:C18H13NO3Color and Shape:SolidMolecular weight:291.3AM-6494
CAS:<p>AM-6494 is a potent and orally active BACE1 inhibitor (IC50: 0.4 nM) with in vivo selectivity over BACE2 (IC50: 18.6 nM).</p>Formula:C22H21F2N5O3SPurity:98%Color and Shape:SolidMolecular weight:473.5CS-0777
CAS:<p>CS-0777 is a potent, selective, and orally active S1P1 agonist (sphingosine 1-phosphate receptor modulator).</p>Formula:C21H31N2O5PColor and Shape:SolidMolecular weight:422.45CDK5-IN-2
CAS:<p>CDK5-IN-2 (compound 15) is a highly selective CDK5 inhibitor that acts on CDK5/p25 (IC50: 0.2 nM) and CDK2/CycA (IC50: 23 nM).</p>Formula:C29H28FN5OColor and Shape:SolidMolecular weight:481.56GSD-11
<p>GSD-11: Potent, selective anti-austerity agent; blocks Akt/mTOR pathway, hinders PANC-1 cell migration & colony growth. Promising for pancreatic cancer study.</p>Formula:C20H28O2Color and Shape:SolidMolecular weight:300.44SARS-CoV-2 nsp14-IN-1
<p>SARS-CoV-2 nsp14-IN-1 inhibits Nsp14 Mtase with an IC50 of 0.061 μM, affecting multiple substrates.</p>Formula:C20H20N6O5SColor and Shape:SolidMolecular weight:456.48Bim-IN-1
<p>Bim-IN-1 is a potent inhibitor of Bim expression with low toxicity, Bim-IN-1 reduces Bim expression levels with little inhibition of protein kinase A.</p>Formula:C19H20Cl2FNO2SColor and Shape:SolidMolecular weight:416.34SB 224289
CAS:<p>SB 224289: selective 5-HT1B antagonist, pKi 8.2, 60x selectivity, effective orally.</p>Formula:C32H32N4O3Purity:98%Color and Shape:SolidMolecular weight:520.62Antibiotic MA 144M1
CAS:<p>Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.</p>Formula:C42H55NO15Color and Shape:SolidMolecular weight:813.88Adafosbuvir
CAS:<p>Adafosbuvir has antiviral activity.</p>Formula:C22H29FN3O10PColor and Shape:SolidMolecular weight:545.457BM635 hydrochloride
<p>BM635 hydrochloride, an MmpL3 inhibitor, strongly blocks Divergent bacteriophage H37Rv (MIC50: 0.08 μM), with doubled in vivo potency.</p>Formula:C25H30ClFN2OColor and Shape:SolidMolecular weight:428.97GDC-0927 Racemate
CAS:<p>GDC-0927 Racemate is a degrader of estrogen receptor, is used in the research of ER-related diseases, potently inhibits ER-α activity, with an IC50 of 0.2 nM.</p>Formula:C28H28FNO4Purity:98%Color and Shape:SolidMolecular weight:461.52C.I. Pigment Red 60
CAS:<p>C.I. Pigment Red 60 is a bright, scarlet, semi-transparent red pigment.</p>Formula:C17H9N2Na3O9S2Purity:98%Color and Shape:SolidMolecular weight:518.35Flutimide
CAS:<p>Flutimide: Endonuclease inhibitor, IC50 = 3μM, for research on acute respiratory diseases like influenza.</p>Formula:C12H18N2O3Color and Shape:SolidMolecular weight:238.28Vanin-1-IN-3
<p>Vanin-1-IN-3 (OMP-7) is a vanin-1 inhibitor with an IC 50 of 0.038 μM [1].</p>Formula:C17H22F3NO5Color and Shape:SolidMolecular weight:377.36SB 243213 hydrochloride
CAS:<p>SB 243213 hydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8).It</p>Formula:C22H20ClF3N4O2Purity:98%Color and Shape:SolidMolecular weight:464.87Cap-dependent endonuclease-IN-6
CAS:<p>Cap-dependent endonuclease-IN-6 (compound 13) is a Cap-dependent endonuclease (CEN) inhibitor that inhibits influenza virus.</p>Formula:C23H21N3O3SColor and Shape:SolidMolecular weight:419.5Rostratin B
CAS:<p>Rostratin B, a cytotoxic disulfide, demonstrates in vitro cytotoxicity against human colon carcinoma (HCT-116), exhibiting an IC50 value of 1.9 μg/mL.</p>Formula:C18H20N2O6S2Color and Shape:SolidMolecular weight:424.49Mesulergine
CAS:<p>Mesulergine is metabolized into dopaminergic agonists.</p>Formula:C18H26N4O2SColor and Shape:SolidMolecular weight:362.49α-Glucosidase-IN-13
<p>α-Glucosidase-IN-13 is an inhibitor of α-glucosidase (IC50: 5.69 μM).</p>Formula:C25H28N4O3S2Color and Shape:SolidMolecular weight:496.64Glutaminyl Cyclase Inhibitor 3
CAS:<p>Designed anti-Alzheimer’s compound; potent Glutaminyl Cyclase inhibitor; IC50 at 4.5 nM; reduces brain Aβ; improves cognition.</p>Formula:C24H32N6O2SPurity:98%Color and Shape:SolidMolecular weight:468.61KUSC-5037
<p>KUSC-5037 inhibits HIF-1 (IC50 = 1.2 μM) and mitochondrial complex V/FoF1ATP synthase.</p>Formula:C18H17F3N6O2Color and Shape:SolidMolecular weight:406.13651SSR 146977
CAS:<p>NK3 receptor antagonist</p>Formula:C35H42Cl2N4O2Purity:98%Color and Shape:SolidMolecular weight:621.64SDM25N hydrochloride
CAS:<p>δ receptor antagonist</p>Formula:C26H27ClN2O3Purity:98%Color and Shape:SolidMolecular weight:450.96B-3852
CAS:<p>B-3852 is a Bradykinin inhibitor.</p>Formula:C55H74F3N15O11Color and Shape:SolidMolecular weight:1178.27IRAK4-IN-15
CAS:<p>IRAK4-IN-15: selective IRAK4 inhibitor, IC50 0.002 μM, good PK, low clearance, synergizes with Acalabrutinib in MyD88/CD79 mutant ABC-DLBCL.</p>Formula:C25H29FN10Color and Shape:SolidMolecular weight:488.56Complex III-IN-2
<p>Complex III-IN-2 inhibits complex III, with antifungal EC50: 29.31 mg/L vs R. solani, 29.98 mg/L vs S. sclerotiorum.</p>Formula:C15H21ClN2O2SColor and Shape:SolidMolecular weight:328.86FT001
CAS:<p>FT001: Oral BET Bromodomain inhibitor, IC50=0.46μM, suppresses MYC, anti-cancer, effective in vitro/vivo.</p>Formula:C25H29N3O4SPurity:99.9%Color and Shape:SolidMolecular weight:467.58p38-α MAPK-IN-5
CAS:<p>p38-α MAPK-IN-5: potent p38α inhibitor, IC50s: 0.1 nM (α), 0.2 nM (β), 944 nM (γ), 4100 nM (δ); anti-inflammatory, promising for asthma/COPD research.</p>Formula:C37H49N11O2Color and Shape:SolidMolecular weight:679.86EGFR-IN-48
<p>EGFR-IN-48: potent EGFR inhibitor, oral, IC50: 0.193-66.7 nM, blocks EGFR mutants & BaF3/PC-9 cell proliferation.</p>Color and Shape:SolidHeme Oxygenase-2-IN-1
<p>Heme Oxygenase-2-IN-1 is a selective HO-2 inhibitor with IC50s: 14.9 μM (HO-1), 0.9 μM (HO-2).</p>Formula:C19H17N3O2Color and Shape:SolidMolecular weight:319.36Naldemedine tosylate
CAS:<p>Naldemedine (S-297995) tosylate, a PAMORA, targets μ-, δ-, κ-opioid receptors, aiding OIC research, may bind to SARS-CoV2's 3CL pro.</p>Formula:C39H42N4O9SColor and Shape:SolidMolecular weight:742.84Topoisomerase II inhibitor 6
<p>Topoisomerase II inhibitor 6, a potent tryptanthrin derivative, blocks G2 phase in CCRF-CEM cells, induces DNA breaks, and may be used for cancer research.</p>Formula:C19H18N4O2Color and Shape:SolidMolecular weight:334.37KPH2f
CAS:<p>KPH2f: dual URAT1/GLUT9 inhibitor, orally active, IC50: 0.24μM (URAT1), 9.37μM (GLUT9), minimal OAT1/ABCG2 impact.</p>Formula:C24H16N3NaO2SColor and Shape:SolidMolecular weight:433.46CAII-IN-2
<p>CAII-IN-2 (3g): potent, selective CA-II inhibitor; IC50-12.1 μM for bovine CA-II; valuable in CA-related disorder research.</p>Formula:C18H19BrN4SColor and Shape:SolidMolecular weight:403.34(Rac)-PT2399
CAS:<p>(Rac)-PT2399 is a potent and specific inhibitor of hypoxia-inducible factor 2a (HIF-2α)(IC50 of 0.01 μM).</p>Formula:C17H10F5NO4SColor and Shape:SolidMolecular weight:419.32SS-RJW100
<p>SS-RJW100 is an enantiomer of RJW100 targeting LRH-1, SF-1, enhances Tif2 interaction, and disrupts LRH-1 networks with lowered stability.</p>Formula:C28H34OColor and Shape:SolidMolecular weight:386.57LY3325656
CAS:<p>LY3325656, a GPR142 agonist with anti-diabetic properties, progresses to phase 1 trials for Type 2 diabetes.</p>Formula:C21H23F3N6O2Color and Shape:SolidMolecular weight:448.447(Z),11(Z)-Nonacosadiene
CAS:<p>7(Z),11(Z)-Nonacosadiene, a female fly pheromone, spurs male courtship; it's a C29 diene made by a female-specific elongase.</p>Formula:C29H56Color and Shape:SolidMolecular weight:404.75MK-8825
CAS:<p>MK-8825 is a CGRP receptor antagonist.</p>Formula:C31H30F2N6O3Color and Shape:SolidMolecular weight:572.61Anti-MRSA agent 6
<p>Anti-MRSA agent 6 (compound 3q6) is a potent anti-methicillin-resistant Staphylococcus aureus (anti-MRSA) agent with low cytoxicity for MCF-7, A549 cells [1].</p>Formula:C16H11F2N3Color and Shape:SolidMolecular weight:283.28ERRγ agonist-1
<p>ERRγ agonist-1 can be used in neuropsychological disorders research.</p>Formula:C17H21N5OColor and Shape:SolidMolecular weight:311.38KU-32
CAS:<p>KU-32 is a novel and novobiocin-based Hsp90 inhibitor. It can protect against neuronal cell death.</p>Formula:C20H25NO8Purity:98%Color and Shape:SolidMolecular weight:407.41EB-0156
<p>EB-0156: potent ER α-glucosidase inhibitor, IC50 of 0.0479/ <0.001 μM, N-substituted valerian, broad-spectrum antiviral potential.</p>Formula:C21H32N6O7Color and Shape:SolidMolecular weight:480.51CBP/p300-IN-2
CAS:<p>CBP/EP300-IN-2 is an inhibitor of CBP/EP300 (IC50s: 1.07 nM and 5.96 nM for CBP/HTRF and Myc).</p>Formula:C27H29F2N7O2Purity:98%Color and Shape:SolidMolecular weight:521.56MRS2500
CAS:<p>MRS2500 is a highly potent and selective platelet P2Y1 receptor antagonist.</p>Formula:C13H18IN5O8P2Purity:98%Color and Shape:SolidMolecular weight:561.16L 767679
CAS:<p>L 767679 is an antagonist of the fibrinogen receptors.</p>Formula:C20H24N4O4Purity:98%Color and Shape:SolidMolecular weight:384.43Detajmium
CAS:<p>Detajmium is an anti-arrhythmia compound. It is an Na(+)-channel-blocking drug with an extremely long recovery from use-dependent sodium channel block.</p>Formula:C27H42N3O3Purity:98%Color and Shape:SolidMolecular weight:456.64ETX0282
CAS:<p>ETX0282, oral class A/C β-lactamase inhibitor, developed by Entasis with cefpodoxime for bacterial infections.</p>Formula:C13H18FN3O5Color and Shape:SolidMolecular weight:315.30Antibacterial agent 112
<p>Compound 112: Powerful antibacterial, MIC 1250 μM against B. subtilis, E. coli, E. faecalis, S. typhimurium, S. aureus; also an HIV-1 antibody.</p>Formula:C35H23N5O5Color and Shape:SolidMolecular weight:593.59FtsZ-IN-4
<p>FtsZ-IN-4 is an oral FtsZ inhibitor with strong antibacterial effects and good drug traits, low toxicity (CC50 >20μg/mL).</p>Formula:C21H16ClF2NO2Color and Shape:SolidMolecular weight:387.81IACS-8779
CAS:<p>IACS-8779 is a potent STING agonist that efficiently stimulates interferon gene activity and exhibits strong systemic antitumor effects.</p>Formula:C21H25N9O10P2S2Purity:98%Color and Shape:SolidMolecular weight:689.55HBV-IN-20
<p>HBV-IN-20 is a potent, orally active HBV inhibitor (EC50: 0.46 μM). HBV-IN-20 is a classical type II CpAM (core protein assembly regulator).</p>Color and Shape:SolidPTP1B-IN-3 diammonium
<p>PTP1B-IN-3 diammonium, an oral enzyme inhibitor, has potent antidiabetic and anticancer effects, with a 120 nM IC50.</p>Formula:C12H13BrF2N3O3PColor and Shape:SolidMolecular weight:396.12L 668411
CAS:<p>L 668411, the 2,3-ditritiated methyl ester of L 659699, inhibits HMG-CoA synthase.</p>Formula:C19H30O5Purity:98%Color and Shape:SolidMolecular weight:338.44WIN 66306
CAS:<p>WIN 66306: Cyclic heptapeptide, blocks NK1/NK2 receptors, inhibits substance P-triggered contractions in guinea pig ileum.</p>Formula:C41H52N8O9Color and Shape:SolidMolecular weight:800.9VU0463271 quarterhydrate
<p>VU0463271 quarterhydrate is a potent KCC2 antagonist, with an IC 50 of 61 nM [1].</p>Formula:C19H20N4O2S2Color and Shape:SolidMolecular weight:387MurB-IN-1
<p>MurB-IN-1 (compound 44) inhibits key bacterial enzyme MurB with 3.57 μM affinity, offering treatment potential against P. aeruginosa.</p>Formula:C12H7Cl2F3N2O2Color and Shape:SolidMolecular weight:339.1Fipravirimat
CAS:<p>Fipravirimat is a potent inhibitor of HIV-1 with potential applications in HIV and AIDS research.</p>Formula:C43H67FN2O4SColor and Shape:SolidMolecular weight:727.07Kahweol Acetate
CAS:<p>Kahweol Acetate, a semi-synthetic coffee bean derivative, inhibits osteoclasts, cancer cells, DNA damage, and oxidative stress.</p>Formula:C22H28O4Color and Shape:SolidMolecular weight:356.46U91356
CAS:<p>U91356 is an agonist of the dopamine receptors.</p>Formula:C13H17N3OPurity:98%Color and Shape:SolidMolecular weight:231.29(R)-CSN5i-3
CAS:<p>(R)-CSN5i-3 is CSN5i-3 of the R configuration.</p>Formula:C28H29F2N5O2Purity:99.76% - 99.97%Color and Shape:SolidMolecular weight:505.56Riminkefon
CAS:<p>Riminkefon is a kappa opioid receptor agonist .</p>Formula:C38H57N7O6Color and Shape:SolidMolecular weight:707.9BRD4 D1-IN-1
<p>BRD4 D1-IN-1 selectively inhibits BRD4 D1 (IC50 <0.092 μM, Kd 18 nM) with >500-fold specificity versus D2.</p>Formula:C32H37F3N6OColor and Shape:SolidMolecular weight:578.67Antibiotic MA 144M2
CAS:<p>Antibiotic MA 144M2, an anthracycline glycoside, targets gram-positive bacteria and tumors, derived from Streptomyces and aclacinomycin A conversion.</p>Formula:C42H55NO16Color and Shape:SolidMolecular weight:829.88CHK1-IN-2
CAS:<p>CHK1-IN-2 is an inhibitor of checkpoint kinase 1 (CHK1; IC50: 6 nM).</p>Formula:C20H22N4OSPurity:98%Color and Shape:SolidMolecular weight:366.48AFP-07 free acid
CAS:<p>AFP 07 free acid is a 7,7-difluoroprostacyclin derivative. It also acts as a selective and highly potent agonist for the IP receptor.</p>Formula:C22H30F2O5Purity:98%Color and Shape:SolidMolecular weight:412.47PI3Kα-IN-8
<p>PI3Kα-IN-8 is a selective inhibitor of PI3Kα (IC50: 0.012 μM).</p>Formula:C26H27BrN4O2Color and Shape:SolidMolecular weight:507.42Lentiginosine
CAS:<p>Lentiginosine is a selective amyloglucosidase inhibitor.</p>Formula:C8H15NO2Color and Shape:SolidMolecular weight:157.21Heparastatin
CAS:<p>Heparastatin is an inhibitor of heparanase.</p>Formula:C8H11F3N2O5Purity:98%Color and Shape:SolidMolecular weight:272.18
