Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,519 products)
- Apoptosis(5,787 products)
- Cell Cycle/Checkpoint(4,446 products)
- Chromatin/Epigenetics(2,235 products)
- Cytoskeletal Signaling(1,381 products)
- DNA Damage/DNA Repair(2,824 products)
- Endocrinology/Hormones(3,500 products)
- Enzyme(3,639 products)
- GPCR/G-Protein(8,317 products)
- Immunology and Inflammation(3,516 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(404 products)
- MAPK Signaling(1,200 products)
- Membrane Transporter/Ion Channel(2,787 products)
- Metabolism(9,416 products)
- Microbiology/Virology(6,968 products)
- Neuroscience(9,919 products)
- Other Inhibitors(37,928 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,400 products)
- Proteases/Proteasome(1,596 products)
- Stem Cell and Derivatives(831 products)
- Tyrosine Kinase/Adaptors(2,015 products)
- Ubiquitination(1,649 products)
Show 16 more subcategories
Found 66626 products of "Inhibitors"
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DNA crosslinker 4 dihydrochloride
CAS:<p>DNA Crosslinker 4 binds DNA's minor groove, inhibits NCI-H460, A2780, MCF-7 cancer cells, and is used in cancer research.</p>Formula:C16H24Cl2N8OColor and Shape:SolidMolecular weight:415.32CXCR2 antagonist 5
<p>CXCR2 antagonist 5 (compound 25) binds strongly (IC50=0.013μM) and mobilizes calcium (IC50=0.1μM).</p>Formula:C15H14F2N4O2SColor and Shape:SolidMolecular weight:352.36WEHI-9625
CAS:<p>WEHI-9625 is a tricyclic sulfone small molecule apoptosis inhibitor (EC50: 69 nM).</p>Formula:C34H27NO5S2Purity:98%Color and Shape:SolidMolecular weight:593.71FY-56
<p>FY-56: potent, selective LSD1/KDM1A inhibitor (IC50=42nM); differentiates MOLM-13/MV4-11 cells; promising for AML research.</p>Formula:C23H19FN2O3Color and Shape:SolidMolecular weight:390.41LolCDE-IN-2
CAS:<p>LolCDE-IN-2 is a potent Lol protein (LolCDE) inhibitor. LolCDE-IN-2 shows antibacterial activity with a MIC of 2 μg/ml against E. coli MG1655 [1].</p>Formula:C22H17N5OPurity:98%Color and Shape:SolidMolecular weight:367.40Dehydrocrenatidine
CAS:<p>Dehydrocrenatidine (Kumujian G) is an inhibitor of JAK and induces cell apoptosis.</p>Formula:C15H14N2O2Purity:98%Color and Shape:SolidMolecular weight:254.28Piperazinomycin
CAS:<p>Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.</p>Formula:C18H20N2O2Color and Shape:SolidMolecular weight:296.36Antifungal agent 19
<p>Antifungal agent 19 shows the potent antifungal activity ( EC 50 = 0.72 μM).</p>Formula:C19H18F4O2Color and Shape:SolidMolecular weight:354.34ERK2 IN-1
CAS:<p>ERK2 IN-1 is a selective ERK2 inhibitor with an IC50 of 7 nM.</p>Formula:C36H34FN7O2SPurity:98%Color and Shape:SolidMolecular weight:647.76Ornoprostil
CAS:<p>Ornoprostil, a prostaglandin E1 analogue, acts as a mucosal protectant.</p>Formula:C23H38O6Purity:98%Color and Shape:SolidMolecular weight:410.54UCN-02
CAS:<p>UCN-02 (7-epi-Hydroxystaurosporine) is a PKC inhibitor produced by Streptomyces N-126 strain, which inhibits PKA.</p>Formula:C28H26N4O4Purity:98%Color and Shape:SolidMolecular weight:482.53AChE/BuChE-IN-3
CAS:<p>AChE/BuChE-IN-3 inhibits AChE (IC50: 0.65 μM), BuChE (IC50: 5.77 μM), crosses BBB, and hinders Aβ1-42 aggregation for Alzheimer's research.</p>Formula:C30H30F3N3O6Color and Shape:SolidMolecular weight:585.57ZL-Pin13
CAS:<p>ZL-Pin13: potent Pin1 inhibitor (IC50: 67 nM), halts MDA-MB-231 cell growth, reduces Pin1 substrates.</p>Formula:C24H23ClN2O3SColor and Shape:SoildMolecular weight:454.97Burapitant
CAS:<p>Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity.</p>Formula:C31H35Cl2F6N3O3Purity:>99.99% - >99.99%Color and Shape:SolidMolecular weight:682.52PF-06380101
CAS:<p>PF-06380101, a potent auristatin analog and Dolastatin 10 derivative, shows strong anti-tumor activity and unique ADME attributes.</p>Formula:C39H62N6O6SPurity:98%Color and Shape:SolidMolecular weight:743.01Carboxylesterase-IN-3
CAS:<p>Carboxylesterase-IN-3 is a potent inhibitor of Carboxylesterase Notum (IC50 ≤ 10 nM).Carboxylesterase-IN-3 has the potential to study cancer diseases.</p>Formula:C11H6Cl2N4OSPurity:97.49% - 98.47%Color and Shape:SolidMolecular weight:313.16DN-F01
<p>DN-F01 exhibits a potent calcium-dependent inhibitory effect on cardiac myofibrillar ATPase activity, with an IC50 of 11 ± 4 nmol/L.</p>Formula:C22H16N2O2Color and Shape:SolidMolecular weight:340.37Fluperolone acetate
CAS:<p>Fluperolone acetate is a Glucocorticoid/Adrenal Cortex Hormone.</p>Formula:C24H31FO6Color and Shape:SolidMolecular weight:434.50PD-1/PD-L1-IN-15
<p>PD-1/PD-L1-IN-15 is a potent inhibitor of PD-1/PD-L1 (IC50: 60.1 nM) and has shown investigational potential for tumor immunotherapy.</p>Formula:C32H30N4O3Color and Shape:SolidMolecular weight:518.61Anticancer agent 45
<p>Anticancer agent 46, potent and selective, induces apoptosis, is cytotoxic to cancer cells, with low toxicity to human lymphocytes.</p>Formula:C22H14ClN3O6S2Color and Shape:SolidMolecular weight:515.95AKT-IN-3
CAS:<p>AKT-IN-3: potent oral Akt inhibitor with low hERG blockage. IC50: 1.4-1.7 nM for Akt1-3. Inhibits AGC kinases like PKA, PKC.</p>Formula:C23H23Cl2F2N5O3Purity:98%Color and Shape:SolidMolecular weight:526.36Monoamine Oxidase B inhibitor 1
<p>Potent, selective MAO-B inhibitor; reversible; oral; crosses BBB; IC50=0.02 nM; potential for Parkinson's research.</p>Formula:C18H15FO3Color and Shape:SolidMolecular weight:298.31U 80215
CAS:<p>U 80215 is an enzyme-competitive inhibitor.</p>Formula:C42H60N8O6SColor and Shape:SolidMolecular weight:805.04Salacinol
CAS:<p>Salacinol is a naturally occurring alpha-glucosidase inhibitor isolated from an Ayurvedic traditional medicine Salacia reticulata.</p>Formula:C9H18O9S2Color and Shape:SolidMolecular weight:334.37BGC-638
CAS:<p>BGC-638, an analogue of BGC-945, is a thymidylate synthase inhibitor specifically transported into α-folate receptor (α-FR)–overexpressing tumors.</p>Formula:C32H33N5O9Color and Shape:SolidMolecular weight:631.63CK156
CAS:<p>CK156 inhibits DAPK with high selectivity; IC50: 182 nM (DRAK1), 34 μM (CK2a1), 39 μM (CK2a2); key in autoimmune/inflammation research.</p>Formula:C21H25N5O3Color and Shape:SolidMolecular weight:395.45BRD-K98645985
CAS:<p>BRD-K98645985: BAF inhibitor, binds ARID1A, reverses HIV-1 latency, EC50 ~2.37μM, alters nucleosome placement.</p>Formula:C33H43N5O4Purity:98%Color and Shape:SolidMolecular weight:573.73Encephalitic alphavirus-IN-1
<p>Alphavirus-IN-1 blocks VEEV (EC50: 0.24 μM) & EEEV (EC50: 0.16 μM), non-toxic, stable in mice plasma.</p>Formula:C27H25FN6O2Color and Shape:SolidMolecular weight:484.52RGT-068A
CAS:<p>RGT-068A is a potent, selective and oral bioavailable MALT1 inhibitor .</p>Formula:C17H16ClN9O2Color and Shape:SolidMolecular weight:413.82CCR5 antagonist 1
CAS:<p>CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.</p>Formula:C39H46ClF2N5O3SPurity:98%Color and Shape:SolidMolecular weight:738.33Mifepristone methochloride
CAS:<p>Mifepristone methochloride is a glucocorticoid antagonist. This product will be sold for research use only.</p>Formula:C30H38ClNO2Color and Shape:SolidMolecular weight:480.08L 668411
CAS:<p>L 668411, the 2,3-ditritiated methyl ester of L 659699, inhibits HMG-CoA synthase.</p>Formula:C19H30O5Purity:98%Color and Shape:SolidMolecular weight:338.44α-Glucosidase-IN-13
<p>α-Glucosidase-IN-13 is an inhibitor of α-glucosidase (IC50: 5.69 μM).</p>Formula:C25H28N4O3S2Color and Shape:SolidMolecular weight:496.64FCE-27262
CAS:<p>FCE-27262 is a prostaglandin H2/thromboxane A2 receptor antagonist.</p>Formula:C23H31N3O3Color and Shape:SolidMolecular weight:397.51CCG258208
CAS:<p>GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).</p>Formula:C24H25FN4O4Purity:98%Color and Shape:SolidMolecular weight:452.48LY 190388
CAS:<p>LY 190388 is a penicillamine-containing enkephalin analog used as an mu receptor agonist with analgesia activity.</p>Formula:C30H41N5O7SPurity:98%Color and Shape:SolidMolecular weight:615.74AMG-25
CAS:<p>AMG-25 (c-Kit-IN-5-1) is a c-Kit inhibitor that inhibits c-Kit, KDR, p38, Lck, and Src, and can be used for the study of mast cell-associated fibrotic diseases.</p>Formula:C23H17N5O2Purity:98.16%Color and Shape:SolidMolecular weight:395.41Dinalbuphine sebacate
CAS:<p>Dinalbuphine sebacate: long-acting nalbuphine prodrug, μ-opioid partial agonist/antagonist, κ-opioid high-efficacy agonist.</p>Formula:C52H68N2O10Color and Shape:SolidMolecular weight:881.1T-Type calcium channel inhibitor 2
<p>Compound 6g inhibits T-type Ca channels (IC50: Cav3.1-31μM, Cav3.2-83μM), cytotoxic to A549 (IC50: 5μM) & HCT-116 cells (IC50: 6.4μM).</p>Formula:C36H39FN4OSColor and Shape:SolidMolecular weight:594.78SARS-CoV-2 nsp14-IN-2
<p>SARS-CoV-2 nsp14-IN-2: Strong Nsp14 methyltransferase inhibitor (IC50: 0.09 μM), potential for COVID-19 research.</p>Formula:C21H21N5O5SColor and Shape:SolidMolecular weight:455.49GLS1 Inhibitor-5
<p>GLS1 Inhibitor-5 (24y): Selective, oral glutaminase 1 inhibitor; IC50 68 nM; induces apoptosis; anti-tumor.</p>Color and Shape:SolidCemdomespib
CAS:<p>Cemdomespib (KU-596) is a potent Hsp90 modulator with neuroprotective effects and can improve diabetic neuropathy.</p>Formula:C24H30FNO6Color and Shape:SolidMolecular weight:447.5LSD1-IN-16
<p>LSD1-IN-16 (4b) inhibits LSD1, MAO-A/B; IC50: 0.015-0.366 μM. Halts prostate cancer cell growth; IC50: 15.2 μM.</p>Formula:C20H18N2OSColor and Shape:SolidMolecular weight:334.43Minnelide
CAS:<p>Minnelide is a prodrug of triptolide,and shows potent antitumor activity in a number of tumor types.</p>Formula:C21H25Na2O10PPurity:98.49% - 99.59%Color and Shape:SolidMolecular weight:514.37KRAS inhibitor-13
CAS:<p>KRAS inhibitor-13 blocks KRAS G12C (IC50: 0.883 μM) and p-ERK in some cancer cells; promising for pancreatic, colorectal, lung cancer research.</p>Formula:C25H19ClFN3O2SColor and Shape:SolidMolecular weight:479.95Anticancer agent 79
<p>Anticancer agent 79 (3d) has potent activity against breast cancer, with cytotoxic effects on T47-D, IC50=13.64±0.26μM.</p>Formula:C20H12F3NO5Color and Shape:SolidMolecular weight:403.31Acetoxycycloheximide
CAS:<p>Acetoxycycloheximide triggers TNF receptor 1, prompts apoptosis, and cytochrome c release by activating c-Jun N-terminal kinase.</p>Formula:C17H25NO6Color and Shape:SolidMolecular weight:339.38Belotecan
CAS:<p>Belotecan (CKD-602) inhibits DNA topoisomerase I, blocks cell cycle, induces apoptosis, and is a camptothecin-derived anticancer agent.</p>Formula:C25H27N3O4Color and Shape:SolidMolecular weight:433.5NA 382
CAS:<p>NA 382 is a staurosporine derivative that inhibits multidrug resistance.</p>Formula:C31H28N4O6Color and Shape:SolidMolecular weight:552.58A-9758
CAS:<p>A-9758: RORγt selective inverse agonist, IC50 5nM, inhibits IL-17A, Th17, and treats psoriasis.</p>Formula:C25H23Cl2F3N2O3Purity:98%Color and Shape:SolidMolecular weight:527.36Calcipotriol Impurity C
CAS:<p>Calcipotriol Impurity C is the impurity of Calcipotriol. Calcipotriol is a VDR-like receptors ligand.</p>Formula:C27H40O3Purity:98%Color and Shape:SolidMolecular weight:412.614Amdinocillin methylacetate
CAS:<p>Amdinocillin methylacetate is a Synthetic penicillin.</p>Formula:C18H27N3O4SColor and Shape:SolidMolecular weight:381.49Streptothricin F
CAS:<p>Streptothricin F is a biochemical.</p>Formula:C19H34N8O8Color and Shape:SolidMolecular weight:502.52EF1502 free base
CAS:<p>EF1502 is a potent and selective GABA transporter inhibitor.</p>Formula:C22H26N2O2S2Purity:98%Color and Shape:SolidMolecular weight:414.58hCAII-IN-5
CAS:<p>hCAII-IN-5 (compound 12h) is a potent, selective inhibitor of human carbonic anhydrase II (hCA II) with an inhibition constant (IC50) of 4.55 µM [1].</p>Formula:C29H18N2O7Color and Shape:SolidMolecular weight:506.46hDHODH-IN-10
<p>hDHODH-IN-10: selective oral inhibitor of hDHODH (IC50: 10.9 nM); blocks cancer cell growth, aids cancer research.</p>Formula:C21H15ClF4N2O4Color and Shape:SolidMolecular weight:470.8OXS007417
<p>OXS007417 induces AML cell differentiation at 48 nM EC50 and shows potent in vivo antitumor effects.</p>Formula:C20H14F3N3OColor and Shape:SolidMolecular weight:369.34CD73-IN-12
<p>CD73-IN-12, a compound from CN114437038A, shows strong anti-tumor activity by effectively inhibiting CD73 enzyme.</p>Formula:C17H14F2N4O2Color and Shape:SolidMolecular weight:344.32PX-316
CAS:<p>PX-316: AKT inhibitor, reduces Akt activity by 78% in HT-29 xenografts, effective against MCF-7 and HT-29 cancers, well-tolerated intravenously.</p>Formula:C28H57O10PColor and Shape:SolidMolecular weight:584.72(RS)-AMPA
CAS:<p>(RS)-AMPA ((±)-AMPA) is a glutamate analog. (RS)-AMPA is an agonist of effective and selective excitatory neurotransmitter L-glutamic acid.</p>Formula:C7H10N2O4Purity:98%Color and Shape:SolidMolecular weight:186.17ACT-281959
CAS:<p>ACT-281959, a prodrug of ACT-246475, is a potent P2Y12 antagonist, better than Clopidogrel, effective orally, and in human trials.</p>Formula:C38H55N6O14PColor and Shape:SolidMolecular weight:850.85GPR84 antagonist 1
<p>GPR84 antagonist 1 is a highly selective, high-affinity competitive antagonist of human GPR84.</p>Formula:C26H22N4O2Color and Shape:SolidMolecular weight:422.48WQ3810 TFA
<p>WQ3810 TFA is an orally available fluoroquinolone with antimicrobial activity against Mycobacterium tuberculosis and inhibits the DNA rotamase activity of</p>Formula:C24H23F6N5O5Purity:99.52%Color and Shape:SoildMolecular weight:575.46BMS-986120
CAS:BMS-986120: Oral, reversible PAR4 antagonist. IC50: 9.5 nM (human), 2.1 nM (monkey). Potent, selective antiplatelet.Formula:C23H23N5O5S2Color and Shape:SolidMolecular weight:513.59UK-432097
CAS:<p>UK 432097 is an adenosine A2A agonist.</p>Formula:C40H47N11O6Color and Shape:SolidMolecular weight:777.87QPX7728 methoxy acetoxy methy ester
CAS:<p>QPX7728 methoxy acetoxy methy ester is an inhibitor of boronic acid β-lactamase.</p>Formula:C14H14BFO7Purity:98%Color and Shape:SolidMolecular weight:324.07Befiradol hydrochloride
CAS:<p>Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 aggregation.</p>Formula:C20H23Cl2F2N3OPurity:99.1%Color and Shape:SolidMolecular weight:430.32L-I-OddU
CAS:<p>L-I-OddU: Selective anti-EBV, halts virus DNA/protein synthesis. EC50: 0.03 µM, low toxicity (CC50: 1000 nM).</p>Formula:C8H9IN2O5Color and Shape:SolidMolecular weight:340.07CY208-243 Mandelate
CAS:<p>CY208-243 is a D1 agonist boosting memory in T-maze, enhances adenylate cyclase (EC50=125nM), and alters monkey electroretinogram.</p>Formula:C27H26N2O3Color and Shape:SolidMolecular weight:426.52HBV-IN-20
<p>HBV-IN-20 is a potent, orally active HBV inhibitor (EC50: 0.46 μM). HBV-IN-20 is a classical type II CpAM (core protein assembly regulator).</p>Color and Shape:SolidSR 33805 oxalate
CAS:<p>Ca2+ channel antagonist</p>Formula:C34H42N2O9SPurity:98%Color and Shape:SolidMolecular weight:654.77Tandutinib (MLN518) HCl
<p>Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.</p>Formula:C31H43ClN6O4Purity:98%Color and Shape:SolidMolecular weight:599.16EGFR-IN-24
<p>EGFR-IN-24 is a potent inhibitor of EGFR and inhibits EGFR (del19/T790M/C797S) and EGFR (L858R/T790M/C797S).</p>Formula:C30H35FN6O3Color and Shape:SolidMolecular weight:546.64IRL 2500
CAS:<p>IRL 2500 is an antagonist of Endothelin receptor with IC50s of 1.3 and 94 nM for Endothelin A receptor and Endothelin B receptor.</p>Formula:C36H35N3O4Purity:99.36%Color and Shape:White Crystalline SolidMolecular weight:573.68Topoisomerase I inhibitor 8
CAS:<p>Topoisomerase I inhibitor 8, a hexacyclic analogue of camptothecin, is also a potent inhibitor of topoisomerase I and is toxic to tumour cells.</p>Formula:C24H21FN2O4Color and Shape:SolidMolecular weight:420.43Carbodine
CAS:<p>Carbodine is an antiviral targeting CTP synthetase, effective against influenza A0/PR-8/34 and A2/Aichi/2/68.</p>Formula:C10H15N3O4Purity:98%Color and Shape:SolidMolecular weight:241.24Multi-kinase-IN-1
CAS:<p>Multi-kinase-IN-1, a powerful kinase inhibitor, exhibits antitumor properties by inducing cell apoptosis.</p>Formula:C35H36F2N6O6SColor and Shape:SolidMolecular weight:706.76Homodestcardin
CAS:<p>Homodestcardin: cyclic depsipeptide from T. roseum with immunosuppressant properties; inhibits mouse T cell proliferation.</p>Formula:C32H55N5O7Color and Shape:SolidMolecular weight:621.81Arverapamil
CAS:<p>Arverapamil is a chiral metabolite of Verapamil.</p>Formula:C26H36N2O4Color and Shape:SolidMolecular weight:440.58Gusperimus
CAS:<p>Gusperimus was synthesized by chemical modification of spergualin and in combination with cyclosporine A to prevent diabetes in susceptible NOD mice.</p>Formula:C17H37N7O3Color and Shape:SolidMolecular weight:387.52FMK-MEA
CAS:<p>FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.</p>Formula:C21H26FN5O2Purity:98%Color and Shape:SolidMolecular weight:399.46BM635 hydrochloride (1493762-74-5 free base)
<p>BM635 hydrochloride is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).</p>Formula:C25H30ClFN2OPurity:98%Color and Shape:SolidMolecular weight:428.97SCH-1473759
CAS:<p>SCH-1473759 is an inhibitor of the aurora (IC50s: 4 and 13 nM for Aurora A and B, respectively).</p>Formula:C20H26N8OSPurity:98%Color and Shape:SolidMolecular weight:426.54Adecypenol
CAS:<p>Adecypenol is a unique adenosine deaminase inhibitor. It shows effective inhibitory activity against calf intestinal adenosine deaminase.</p>Formula:C12H16N4O4Purity:98%Color and Shape:SolidMolecular weight:280.28HCV-IN-7
CAS:<p>HCV-IN-7: potent oral HCV NS5A inhibitor, pan-genotypic, IC50s 3-47 pM, good pharmacokinetics, favorable liver uptake.</p>Formula:C40H48N8O6SPurity:98%Color and Shape:SolidMolecular weight:768.92ROPA
CAS:<p>ROPA, a potent PKCalpha and PKCgamma activator, promotes tumor growth through PKC-activation.</p>Formula:C28H32O6Purity:98%Color and Shape:SolidMolecular weight:464.55U91356
CAS:<p>U91356 is an agonist of the dopamine receptors.</p>Formula:C13H17N3OPurity:98%Color and Shape:SolidMolecular weight:231.29Iralukast (CGP 45715A)
CAS:<p>Iralukast is a cysteinyl-leukotriene antagonist (CysLT) with a pKi of 7.8 for CysLT1.</p>Formula:C38H37F3O8SColor and Shape:SolidMolecular weight:710.76Esorubicin
CAS:<p>Esorubicin, a doxorubicin derivative, intercalates DNA, inhibits topoisomerase II, has less cardiotoxicity, but more myelosuppression.</p>Formula:C27H29NO10Color and Shape:SolidMolecular weight:527.52L-739750
CAS:<p>L-739,750 is an inhibitor (FTI) of peptidomimetic farnesyltransferase.</p>Formula:C23H39N3O6S2Purity:98%Color and Shape:SolidMolecular weight:517.7FtsZ-IN-4
<p>FtsZ-IN-4 is an oral FtsZ inhibitor with strong antibacterial effects and good drug traits, low toxicity (CC50 >20μg/mL).</p>Formula:C21H16ClF2NO2Color and Shape:SolidMolecular weight:387.81CD73-IN-2
<p>CD73-IN-2 is a potent inhibitor of CD73 (IC50: 0.09 nM).</p>Formula:C17H25ClN5O7PColor and Shape:SolidMolecular weight:477.84Elocalcitol
CAS:<p>Elocalcitol is a calcitriol analog for inhibition of prostate cell growth.</p>Formula:C29H43FO2Color and Shape:SolidMolecular weight:442.65LSD1-IN-13 hydrochloride
CAS:<p>LSD1-IN-13 hydrochloride (7e) is an oral LSD1 inhibitor (IC50: 24.43 nM), promoting differentiation in AML cell lines.</p>Formula:C23H30ClN3O2SColor and Shape:SolidMolecular weight:448.02PD 113271
CAS:<p>PD 113,271 is an analog of the fermentation products fostriecin with antitumor activity in vitro and in vivo.</p>Formula:C19H27O10PPurity:98%Color and Shape:SolidMolecular weight:446.39MDL-100173
CAS:<p>MDL-100173 is a dual angiotensin-converting enzyme (ACE)/neutral endopeptidase (NEP) inhibitor.</p>Formula:C24H26N2O4SColor and Shape:SolidMolecular weight:438.54Vimirogant
CAS:<p>Vimirogant is a RORγ inhibitor (Ki: <100 nM).</p>Formula:C27H35F3N4O3SPurity:98%Color and Shape:SolidMolecular weight:552.65ETX0282
CAS:<p>ETX0282, oral class A/C β-lactamase inhibitor, developed by Entasis with cefpodoxime for bacterial infections.</p>Formula:C13H18FN3O5Color and Shape:SolidMolecular weight:315.30ONO-DI-004
CAS:<p>ONO-DI-004 is a selective EP1 Prostanoid receptor agonist.</p>Formula:C24H38O6Color and Shape:SolidMolecular weight:422.55Antifungal agent 11
<p>Antifungal agent 11 has a good antifungal effect.</p>Formula:C21H19F2N7O3S2Color and Shape:SolidMolecular weight:519.55Antitumor agent-48
<p>Antitumor agent-48, a 2,3-dehydrosilybin derivative, exhibits cytotoxicity on MCF-7, NCI-H1299, HepG2, HT29 cells; IC50 ranging 8.06-16.51 µM.</p>Formula:C35H34N2O14Color and Shape:SolidMolecular weight:706.65Lumirubin
CAS:<p>Lumirubin is a water-soluble photoproduct of bilirubin formed in vivo during phototherapy.</p>Formula:C33H36N4O6Color and Shape:SolidMolecular weight:584.66GABAA receptor agonist 1
<p>Compound 3e, a potent GABAA agonist, targets GABA sites and has potential anti-depressive effects in mice.</p>Formula:C20H30O3Color and Shape:SolidMolecular weight:318.45Pareptide monohydrochloride
CAS:<p>Pareptide monohydrochloride is a metabolically stable analog of melatonin inhibitor (MIF).</p>Formula:C14H27ClN4O3Purity:98%Color and Shape:SolidMolecular weight:334.84Akt/NF-κB/JNK-IN-1
<p>Akt/NF-κB/JNK-IN-1 (Compound 2i) is an inhibitor of Akt, NF-κB and JNK signalling pathways.Akt/NF-κB/JNK-IN-1 exhibits an inhibitory effect on nitric oxide</p>Formula:C22H22N2O6Color and Shape:SolidMolecular weight:410.42FTI-2148
CAS:<p>FTI-2148 blocks RAS-related FT-1 & GGT-1; IC50: 1.4 nM & 1.7 μM.</p>Formula:C24H28N4O3SPurity:98%Color and Shape:SolidMolecular weight:452.57CHK1-IN-4
CAS:<p>CHK1-IN-4 is a potent inhibitor of checkpoint kinase 1 (chk1) and potently inhibits chk1 phosphorylation in the tumor cells with anti-tumor activity.</p>Formula:C18H18BrN7O2Purity:98%Color and Shape:SolidMolecular weight:444.29Ambuic acid
CAS:<p>Ambuic acid: cyclohexanone with antifungal, quorum-inhibiting, antibacterial properties, blocks cyclic peptides; reduces MRSA abscesses in mice.</p>Formula:C19H26O6Color and Shape:SolidMolecular weight:350.41(R)-FL118
CAS:<p>FL118 inhibits human survivinion expression and activates tumor suppressor p53 as a MOA in p53 wild-type cancer cells.</p>Formula:C21H16N2O6Color and Shape:SolidMolecular weight:392.36HDAC-IN-35
<p>HDAC-IN-35 (Compound 14) is an effective and selective inhibitor of VEGFR-2 and HDAC, with IC50 values of 13.2 and 0.166 μM for VEGFR-2 and HDAC6, respectively.</p>Formula:C17H13ClF3N3O3Color and Shape:SolidMolecular weight:399.75C.I. Pigment Red 60
CAS:<p>C.I. Pigment Red 60 is a bright, scarlet, semi-transparent red pigment.</p>Formula:C17H9N2Na3O9S2Purity:98%Color and Shape:SolidMolecular weight:518.35GPX100 HCl
CAS:<p>GPX-100, a non-cardiotoxic doxorubicin analog, intercalates DNA and inhibits replication, repair, and protein synthesis.</p>Formula:C27H32ClNO10Color and Shape:SolidMolecular weight:566MraY-IN-3
<p>MraY-IN-3 (12a) is a potent inhibitor of the bacterial translocase MraY (IC50: 140 μM). 46 μg/ml).</p>Formula:C35H45N3O5Color and Shape:SolidMolecular weight:587.75A1AR antagonist 1
<p>Compound 18g, a potent A1AR blocker with Ki: 2.08 nM (hA1), 6.91 nM (hA2A), 31.2 nM (hA2B).</p>Formula:C18H14N4OColor and Shape:SolidMolecular weight:302.332R,4R-Sacubitril
CAS:<p>2R,4R-Sacubitril is the impurity of Sacubitril. Sacubitril is used in combination with valsartan for the treatment of patients with heart failure.</p>Formula:C24H29NO5Purity:98%Color and Shape:SolidMolecular weight:411.49ADH-6
CAS:<p>ADH-6, a tripyridylamide, disrupts mutant p53 aggregates in cancer cells, reviving its function and inducing apoptosis.</p>Formula:C29H36N8O9Color and Shape:SolidMolecular weight:640.64PF-06648671
CAS:<p>PF-06648671 is a γ-secretase modulator for the treatment of neurodegenerative and/or neurological disorders.</p>Formula:C25H23ClF4N4O3Purity:98%Color and Shape:SolidMolecular weight:538.92Kaitocephalin
CAS:<p>Kaitocephalin: naturally occurring, non-selective antagonist blocking glutamate receptors, made by Eupenicillium shearii fungus.</p>Formula:C18H21Cl2N3O9Color and Shape:SolidMolecular weight:494.28KRAS G12D inhibitor 1
CAS:<p>KRAS G12D inhibitor 1 (example 243) is an inhibitor of KRAS G12D with an IC 50 of 0.8 nM for KRAS G12D-mediated ERK phosphorylation [1].</p>Formula:C33H32F2N6O2Color and Shape:SolidMolecular weight:582.64Ketomethylenebestatin
CAS:<p>Ketomethylenebestatin, a weaker carba-analog of aminopeptidase inhibitor bestatin, is 10x less potent.</p>Formula:C17H25NO4Purity:98%Color and Shape:SolidMolecular weight:307.38Monlunabant
CAS:<p>Monlunabant ((S)-MRI-1891), a solid dispersion compound, functions as an inhibitor of the cannabinoid CB1 receptor [1].</p>Formula:C26H22ClF3N6O3SPurity:98%Color and Shape:SolidMolecular weight:591.00Prohibitin ligand 1
<p>Compound 22i, a prohibitin ligand, protects the heart at nanomolar levels by inducing STAT3 phosphorylation.</p>Formula:C20H22N2OColor and Shape:SolidMolecular weight:306.4VEGFR-2-IN-18
<p>VEGFR-2-IN-18 is a potent VEGFR-2 inhibitor with a 60 nM IC50, promoting cell apoptosis and anticancer effects.</p>Formula:C20H13ClN4O2Color and Shape:SolidMolecular weight:376.8MALT1-IN-11
CAS:<p>MALT1-IN-11: MALT1 inhibitor, IC50 <10-100 nM, reduces IL10, for cancer/autoimmune research.</p>Formula:C20H16F4N8OColor and Shape:SolidMolecular weight:460.39PD-1/PD-L1-IN-23
CAS:<p>PD-1/PD-L1-IN-23: potent, oral PD-1/PD-L1 inhibitor; L7's ester prodrug; exhibits strong antitumor effects.</p>Formula:C32H30BrCl2N3O6Color and Shape:SolidMolecular weight:703.41LTD4 antagonist 1
CAS:<p>LTD4 antagonist 1 is a potent and orally active antagonist of leukotriene D4 (LTD4; Ki: 0.57 nM).</p>Formula:C31H32F3N3O5SPurity:98%Color and Shape:SolidMolecular weight:615.66Valopicitabine
CAS:<p>Valopicitabine is an effective prodrug of the effective anti-HCV drug 2'-C-methylcytidine and can be used as a promising antiviral drug for the study of chronic</p>Formula:C15H24N4O6Purity:98%Color and Shape:SolidMolecular weight:356.37LY367385 hydrochloride
CAS:<p>LY367385 hydrochloride: selective mGluR1a antagonist, IC50 = 8.8 μM, neuroprotective, anticonvulsant, antiepileptic.</p>Formula:C10H12ClNO4Color and Shape:SolidMolecular weight:245.66MDL-43291
CAS:<p>MDL-43291 is a leukotriene receptor antagonist.</p>Formula:C25H42O4SColor and Shape:SolidMolecular weight:438.66EGFR-IN-62
<p>EGFR-IN-62: IC50 of 10-242 nM for various EGFR mutations, blocks A549/H1975 cell cycle, induces apoptosis, and inhibits cell motility and proliferation.</p>Formula:C30H33N9O2Color and Shape:SolidMolecular weight:551.64GSK5852
<p>GSK5852, an HCV NS5B inhibitor, has IC50 of 50 nM; potently fights HCV with EC50 of 3.0 nM for GT1a and 1.7 nM for GT1b.</p>Formula:C27H27BF2N2O6SColor and Shape:SolidMolecular weight:556.39Antioxidant agent-3
<p>Antioxidant agent-3 shows strong DPPH and ABTS+ radical scavenging (IC50: 26.58, 30.31 μM). Boosts ROS, SOD, GSH; lowers LDH in H2O2-exposed HepG2 cells.</p>Formula:C18H14O8Color and Shape:SolidMolecular weight:358.3Enpp-1-IN-7
<p>Enpp-1-IN-7: potent enpp-1 inhibitor, broad specificity, potential in cancer/infectious disease research. (WO2021203772A1)</p>Formula:C18H19N7O4SColor and Shape:SolidMolecular weight:429.45MsbA-IN-2
<p>MsbA-IN-2 is a potent inhibitor of the lipopolysaccharide transporter MsbA and is able to act on E. coli MsbA (IC50: 2 nM).</p>Formula:C23H19Cl2NO3Color and Shape:SolidMolecular weight:428.31Pulvomycin
CAS:<p>Pulvomycin is a protein biosynthesis inhibitor preventing ternary complex formation between elongation factor Tu, GTP, and aminoacyl-tRNA.</p>Formula:C47H66O13Purity:98%Color and Shape:SolidMolecular weight:839.032FGFR4-IN-9
<p>FGFR4-IN-9 is a selective inhibitor of FGFR4 (IC50: 75.3 nM) that effectively inhibits the growth and angiogenesis of hepatocellular carcinoma cells.</p>Formula:C24H22ClF3N4O4Color and Shape:SolidMolecular weight:522.9Ro 31-8472
CAS:<p>Ro 31-8472 is an angiotensin-converting enzyme (ACE) inhibitor and an analog of cilazaprilat.</p>Formula:C20H27N3O6Purity:98%Color and Shape:SolidMolecular weight:405.44MMAF sodium
CAS:<p>MMAF sodium, a potent tubulin inhibitor in ADCs like Vorsetuzumab mafodotin and SGN-CD19A, acts as an antitumor agent.</p>Formula:C39H64N5NaO8Purity:98%Color and Shape:SolidMolecular weight:753.94Antibacterial agent 76
<p>Antibacterial agent 76 (compound 9) is a potent antibacterial agent.</p>Formula:C23H27N3O2SColor and Shape:SolidMolecular weight:409.54Bleomycin Free Base
CAS:<p>Bleomycin Free Base, a glycopeptide antibiotic, halts DNA function and treats solid tumors.</p>Formula:C55H84N17O21S3Color and Shape:SolidMolecular weight:1415.55AZD-3409
CAS:<p>AZD-3409 is a more potent prenyl transferase inhibitor than lonafarnib with varied IC(50) in cells, acting on gefitinib-resistant breast cancer.</p>Formula:C34H41FN4O4S2Color and Shape:SolidMolecular weight:652.84Furametpyr
CAS:<p>Furametpyr is a kind of low toxicity pesticides used to control plant diseases caused by various pathogenic microorganisms.</p>Formula:C17H20ClN3O2Purity:98%Color and Shape:SolidMolecular weight:333.81LAS195319
CAS:<p>LAS195319 is a potent and selective inhaled PI3Kδ Inhibitor (IC50 = 0.5 nM) for the Treatment of Respiratory Diseases.</p>Formula:C29H26N10O3SColor and Shape:SolidMolecular weight:594.65LY 245769
CAS:<p>LY 245769 is an inhibitor of leukotriene E4 (LTE4).</p>Formula:C25H33F3N8OSPurity:98%Color and Shape:SolidMolecular weight:550.64Anti-TSWV agent 1
<p>Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV).</p>Formula:C22H27ClN4OS3Color and Shape:SolidMolecular weight:495.12MK-8825
CAS:<p>MK-8825 is a CGRP receptor antagonist.</p>Formula:C31H30F2N6O3Color and Shape:SolidMolecular weight:572.61Apoptosis inducer 5
<p>Apoptosis Inducer 5, a lignan enantiomer extracted from Crataegus pinnatifida, demonstrates cytotoxic properties through inducing apoptosis and autophagy in</p>Formula:C23H26O7Color and Shape:SolidMolecular weight:414.45BMS-066
CAS:<p>BMS-066 is an IKKβ/Tyk2 pseudokinase inhibitor. With IC50s of 9 nM and 72 nM, respectively.</p>Formula:C19H21N7O2Purity:98%Color and Shape:SolidMolecular weight:379.42Ph-Ph+
<p>Ph-Ph+ is a dimerized phenanthroline derivative with antitumor, antibacterial, and antifungal effects.</p>Formula:C24H17N4Color and Shape:SolidMolecular weight:361.4212(S)-HETE
CAS:<p>Enpatoran hydrochloride (M5049 hydrochloride) is a TLR7/8 inhibitor with antiviral activity that is used in the study of autoimmune diseases.</p>Formula:C20H32O3Color and Shape:SolidMolecular weight:320.47HDAC8-IN-2
<p>HDAC8-IN-2 (5o) inhibits both smHDAC8 and hHDAC8 with IC50s of 0.27 μM, 0.32 μM, kills schistosome larvae, and lowers egg laying.</p>Formula:C21H16N2O5Color and Shape:SolidMolecular weight:376.36KRAS G12C inhibitor 46
CAS:<p>KRAS G12C inhibitor 46 is a potent inhibitor of KRAS G12C.</p>Formula:C32H33F2N7O2Color and Shape:SolidMolecular weight:585.658(S),15(S)-DiHETE
CAS:<p>8(S),15(S)-DiHETE, from 15(S)-HETE's oxidation by 15-LO, triggers eosinophil movement at 1.5 μM; it counteracts pain and LTB4 effects.</p>Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47RET-IN-7
CAS:<p>RET-IN-7 exhibits strong inhibitory effects against RET kinase in vitro and shows significant efficacy in treating RET-driven tumor xenografts in mice through</p>Formula:C22H24ClFN6O2Color and Shape:SolidMolecular weight:458.92NBD-10007
CAS:NBD-10007 is an inhibitor of HIV-1 entry.Formula:C20H25ClN4O3SPurity:98%Color and Shape:SolidMolecular weight:436.96RdRP-IN-5
CAS:<p>RdRP-IN-5 (compound 20), a potent inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), has potential application in influenza research [1].</p>Formula:C23H21N3O5Purity:98%Color and Shape:SolidMolecular weight:419.43Moflomycin
CAS:<p>Moflomycin is an anthracycline derivative. It exhibits a higher antileukemic activity compared to other anthracyclines.</p>Formula:C25H25IO10Purity:98%Color and Shape:SolidMolecular weight:612.36ORIC-101
CAS:<p>ORIC-101 is a highly effective and selective glucocorticoid receptor antagonist (EC50: 5.6 nM). It also has anti-cancer activity.</p>Formula:C34H47NO2Purity:98%Color and Shape:SolidMolecular weight:501.74UK 356618
CAS:<p>UK 356618 is a potent and selective inhibitor of matrix metalloprotease-3 (IC50: 5.9 nM).</p>Formula:C34H43N3O4Purity:98%Color and Shape:SolidMolecular weight:557.72Anticancer agent 143
CAS:<p>Anticancer Agent 143 (Compound 369), a potent dual inhibitor targeting PTPN2 and PTP1B, exhibits IC50 values below 2.5 nM.</p>Formula:C19H15BrF2N3O6PS2Purity:98%Color and Shape:SolidMolecular weight:594.34Sekikaic Acid
CAS:<p>Sekikaic acid, a phenolic lichen metabolite in H. obscurata, has antioxidant and antiviral properties, inhibiting MLL1-CBP.</p>Formula:C22H26O8Color and Shape:SolidMolecular weight:418.44Dopamine D3 receptor antagonist-1
<p>Dopamine D3 receptor antagonist-1 is a dopamine D3 receptor selective or multi-targeting ligand with a Ki value of 1.58 nM that has demonstrated therapeutic</p>Formula:C31H35Cl2N3O3Color and Shape:SolidMolecular weight:568.53(S)-ZG197
<p>(S)-ZG197 is a compound that acts as a highly selective activator of the Staphylococcus aureus Caseinolytic Protease P (Sa ClpP), demonstrating efficacy at a</p>Formula:C28H35F3N4O3Color and Shape:SolidMolecular weight:532.6T01-1
CAS:<p>T01-1, a derivative of camptothecin, is an anticancer agent demonstrating significant anti-proliferative activity.</p>Formula:C26H29N3O6SColor and Shape:SolidMolecular weight:511.59UK-370106
CAS:<p>UK-370106 is a potent and highly selective inhibitor of MMP-3 with IC50 of 23 nM and MMP-12 with IC50 of 42 nM, and potently inhibits cleavage of [3H]-</p>Formula:C35H44N2O5Purity:98%Color and Shape:SolidMolecular weight:572.73JBJ-02-112-05
CAS:<p>JBJ-02-112-05 is a potent, mutant-selective, allosteric and orally active inhibitor of EGFR with an IC 50 of 15 nM for EGFR L858R/T790M [1].</p>Formula:C27H20N4O2SPurity:98%Color and Shape:SolidMolecular weight:464.54Glycotriosyl glutamine
CAS:<p>Glycotriosyl glutamine is a nephritogenoside analog.</p>Formula:C23H40N2O18Color and Shape:SolidMolecular weight:632.57PHGDH-IN-2
<p>PHGDH-IN-2: potent PHGDH inhibitor, IC50=5.2μM; hinders PHGDH cancer cell growth & serine synthesis in MDA-MB-468.</p>Formula:C22H20N4O3SColor and Shape:SolidMolecular weight:420.48Marizomib
CAS:<p>Marizomib is a novel irreversible brain-permeable proteasome inhibitor that inhibits CT-L, CT-T-laspase-like, and trypsin-like 20S proteasomes.Cost-effective and quality-assured.</p>Formula:C15H20ClNO4Purity:98.03% - 99.41%Color and Shape:SolidMolecular weight:313.78Antibacterial agent 88
<p>Antibacterial agent 88 is an effective antibacterial agent against B. subtilis (MIC: 4 μg/ml) with MIC values of ≤0.0156 μg/mL for MRSA, MRSE and S. aureus.</p>Formula:C31H44N2O6SColor and Shape:SolidMolecular weight:572.76Implitapide
CAS:<p>Implitapide is an inhibitor of microsomal triglyceride transfer protein (MTP).</p>Formula:C35H37N3O2Purity:98%Color and Shape:SolidMolecular weight:531.69GNE-431
CAS:<p>GNE-431: potent, selective noncovalent Btk inhibitor, IC50=3.2 nM; effective against C481R, T474I, T474M mutants, may counter ibrutinib resistance.</p>Formula:C30H32N10O2Color and Shape:SolidMolecular weight:564.64G-4120
CAS:<p>G-4120 is a biochemical that has been shown to have a dose-dependent complete inhibition of arterial and venous thrombosis.</p>Formula:C26H36N8O11SColor and Shape:SolidMolecular weight:668.68PF-06795071
CAS:<p>PF-06795071 is an effective and selective covalent inhibitor of MAGL (IC50: 3 nM).</p>Formula:C18H17F4N3O3Purity:98%Color and Shape:SolidMolecular weight:399.34MraY-IN-1
<p>MraY-IN-1 inhibits MraY (IC50: 140μM), fights E. coli K12, B. subtilis W23, P. fluorescens (MIC50: 7-46μg/ml), for antimicrobial research.</p>Formula:C35H46N3O5Color and Shape:SolidMolecular weight:588.76SLC4101431
<p>SLC4101431 is a potent SphK2 inhibitor with Ki value of 90 nM.</p>Formula:C29H28ClN7OSColor and Shape:SolidMolecular weight:558.1Teslexivir hydrochloride
CAS:<p>Teslexivir (BTA074) HCl inhibits HPV 6/11 by blocking E1-E2 protein interaction, vital for DNA replication. Used in condyloma research.</p>Formula:C35H37BrClN3O4Color and Shape:SolidMolecular weight:679.04MRS2500
CAS:<p>MRS2500 is a highly potent and selective platelet P2Y1 receptor antagonist.</p>Formula:C13H18IN5O8P2Purity:98%Color and Shape:SolidMolecular weight:561.16hMAO-B/MB-COMT-IN-2
<p>Dual inhibitor hMAO-B/MB-COMT-IN-2 targets hMAO-B (IC50: 4.27μM) & MB-COMT (IC50: 2.69μM), aids in neurodegenerative research.</p>Formula:C17H18N2O3Color and Shape:SolidMolecular weight:298.34AZD2353
CAS:<p>AZD2353 is a potent inhibitor of diacylglycerol acetyl transferase 1 (DGAT1).</p>Formula:C22H19ClFN3O3Color and Shape:SolidMolecular weight:427.86HIV-1 protease-IN-6
<p>HIV-1 protease-IN-6 (17d) strongly inhibits HIV-1 protease (IC50: 21 pM, Ki: 4.7 pM) and effectively targets DRV-resistant mutants.</p>Formula:C27H31FN2O6SColor and Shape:SolidMolecular weight:530.61Rafutrombopag
CAS:<p>Rafutrombopag is a thrombopoietin (TPO) agonist.</p>Formula:C25H22N4O5Color and Shape:SolidMolecular weight:458.47LRRK2-IN-4
CAS:<p>LRRK2-IN-4: Potent, selective LRRK2 inhibitor, oral, BBB-penetrating, IC50=2.6 nM, potential for Parkinson's.</p>Formula:C25H29ClF2N6O2Color and Shape:SolidMolecular weight:518.99GSK8814
CAS:<p>GSK8814 is a selective and ATAD2/2B bromodomain chemical probe and inhibitor (binding constant pKd=8.1 and a pKi=8.9 in BROMOscan).</p>Formula:C28H35F2N5O3Purity:98%Color and Shape:SolidMolecular weight:527.6120S Proteasome-IN-4
CAS:<p>20S Proteasome-IN-4: brain-penetrant, parasite-specific, oral, inhibits T.b. brucei proteasome (IC50: 6.3nM), for HAT research.</p>Formula:C20H18ClF2N3O3Color and Shape:SolidMolecular weight:421.83CGC 11144
CAS:<p>CGC 11144 is a Polyamine analogue inhibit tumor growth in vitro and in vivo.</p>Formula:C40H100Cl10N10Color and Shape:SolidMolecular weight:1075.82SHR0687
CAS:<p>SHR0687: potent KOR agonist, selective, favorable PK, effective in rat pain model, minimal BBB penetration, less CNS side effects.</p>Formula:C39H60N8O5Color and Shape:SolidMolecular weight:720.94Anti-inflammatory agent 23
<p>Anti-inflammatory agent 23 blocks LPS-induced NO (IC50: 0.449 μM) and binds p65 well.</p>Formula:C34H49NO6Color and Shape:SolidMolecular weight:567.76C108297
CAS:<p>C108297: glucocorticoid modulator, combats diet obesity/inflammation, reduces appetite/lipid storage, boosts fat burn.</p>Formula:C30H36FN3O4SPurity:98%Color and Shape:SolidMolecular weight:553.69Anti-MRSA agent 6
<p>Anti-MRSA agent 6 (compound 3q6) is a potent anti-methicillin-resistant Staphylococcus aureus (anti-MRSA) agent with low cytoxicity for MCF-7, A549 cells [1].</p>Formula:C16H11F2N3Color and Shape:SolidMolecular weight:283.28Human enteropeptidase-IN-2
<p>Human enteropeptidase-IN-2 is a potent inhibitor of enteropeptidase (enteropeptidase) and can be used in anti-obesity studies.</p>Formula:C20H19F3N4O7Color and Shape:SolidMolecular weight:484.38Hit 1
<p>Hit 1 is an activator of insulin-degrading enzymes (IDE) (EC50: 5.5 μM) and reduces glucose-stimulated insulin secretion.</p>Formula:C22H24N4O3S2Color and Shape:SolidMolecular weight:456.58LPA5 antagonist 2
<p>LPA5 antagonist 2, compound 65, water-soluble, reduces nociception, for inflammatory/neuropathic pain study.</p>Formula:C26H25FN2O4SColor and Shape:SolidMolecular weight:480.55Ivaltinostat formic
<p>Ivaltinostat (CG-200745) is an oral panHDAC inhibitor, inducing apoptosis and enhancing cancer drug sensitivity.</p>Formula:C25H35N3O6Color and Shape:SolidMolecular weight:473.56PARP10/15-IN-3
<p>Compound 8a, a dual PARP10 & PARP15 inhibitor, has IC50s: PARP10 at 0.14μM & PARP15 at 0.40μM; it's cell-permeable & anti-apoptotic.</p>Formula:C12H12N2O3Color and Shape:SolidMolecular weight:232.24VEGFR-2-IN-17
<p>VEGFR-2-IN-17 (15a) is a potent VEGFR-2 inhibitor with an IC50 of 67.25 nM, showing significant antitumor effects.</p>Formula:C21H14ClN3O2Color and Shape:SolidMolecular weight:375.81SB 243213 hydrochloride
CAS:<p>SB 243213 hydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8).It</p>Formula:C22H20ClF3N4O2Purity:98%Color and Shape:SolidMolecular weight:464.87Metesind Glucuronate
CAS:<p>Metesind Glucuronate is an antineoplastic. It also is a specific thymidylate synthase inhibitor.</p>Formula:C29H34N4O10SColor and Shape:SolidMolecular weight:630.67HDAC6-IN-3
<p>HDAC6-IN-3 (Compound 14) is an oral anti-prostate cancer agent, inhibiting HDACs and MAO-A, with IC50 of 0.02-1.54 μM.</p>Formula:C19H27N3O3Color and Shape:SolidMolecular weight:345.44Heme Oxygenase-1-IN-2
<p>Heme Oxygenase-1-IN-2 is a novel inhibitor of heme oxygenase-1 (HO-1), displaying potent antiproliferative activity in vitro, with an IC50 value of 0.95 μM.</p>Formula:C19H18ClN3OColor and Shape:SolidMolecular weight:339.82
