Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,804 products)
- Apoptosis(6,264 products)
- Cell Cycle/Checkpoint(4,847 products)
- Chromatin/Epigenetics(2,597 products)
- Cytoskeletal Signaling(1,538 products)
- DNA Damage/DNA Repair(2,878 products)
- Endocrinology/Hormones(3,748 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,990 products)
- Immunology and Inflammation(3,807 products)
- Influenza Virus(299 products)
- JAK/STAT signaling(416 products)
- MAPK Signaling(1,252 products)
- Membrane Transporter/Ion Channel(3,149 products)
- Metabolism(10,141 products)
- Microbiology/Virology(7,596 products)
- Neuroscience(10,350 products)
- Other Inhibitors(35,822 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,420 products)
- Proteases/Proteasome(1,684 products)
- Stem Cell and Derivatives(742 products)
- Tyrosine Kinase/Adaptors(1,959 products)
- Ubiquitination(1,725 products)
Show 16 more subcategories
Found 66559 products of "Inhibitors"
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Exp 631
CAS:Exp 631 is a centrally-acting non-opioid analgesic; exhibits serotonin and norepinephrine reuptake inhibiting activities.Formula:C30H46N2O6S2Color and Shape:SolidMolecular weight:594.83ML263
CAS:ML263 inhibits NF-kB activation induced by B-cell specific antigen receptor.Formula:C15H18N2O3Color and Shape:SolidMolecular weight:274.32ALRT 1550
CAS:ALRT 1550, a retinoic acid agent (RAR) agonist, is used potentially for the treatment of cervical carcinoma.Formula:C23H32O2Color and Shape:SolidMolecular weight:340.5BMY 22089
CAS:BMY 22089 is a bioactive chemical.Formula:C23H20F2N4O3Color and Shape:SolidMolecular weight:438.43AM-211 sodium
CAS:AM-211 sodium: potent DP2 receptor antagonist, active against allergic inflammation, selective, and orally bioavailable in rats and dogs.Formula:C27H26F3N2NaO4Color and Shape:SolidMolecular weight:522.5RU 58642
CAS:RU 58642 is an effective systemic antiandrogen for androgen-dependent disorders.Formula:C15H11F3N4O2Purity:98%Color and Shape:SolidMolecular weight:336.27TWS-119
CAS:TWS-119 blocks GSK-3β, prompting neuronal formation in mouse stem cells.Formula:C22H16F6N4O6Color and Shape:SolidMolecular weight:546.38Fluorocarazolol
CAS:Fluorocarazolol is a high-affinity beta-adrenergic receptor antagonist .Formula:C18H21FN2O2Color and Shape:SolidMolecular weight:315.37Selenolanthionine
CAS:Selenolanthionine is the major water-soluble selenium compound in the selenium tolerant plant Cardamine violifolia.Formula:C6H12N2O4SeColor and Shape:SolidMolecular weight:255.13SHP2-IN-8
CAS:SHP2-IN-8: reversible, selective SHP2 inhibitor; IC50=23 nM; induces AKT dephosphorylation and Hela cell apoptosis.Formula:C17H21Cl2N5SColor and Shape:SolidMolecular weight:398.35Eclanamine maleate
CAS:Eclanamine found to be mildly mutagenic in AS52 test, evaluated in various short-term genetic assays.Formula:C20H26Cl2N2O5Color and Shape:SolidMolecular weight:445.34GPR120-IN-1
CAS:GPR120-IN-1 is a novel GPR120 inhibitor, showing ~90% inhibitory effects on cell growth with micromolar affinities against SW480.Formula:C31H28N2O2SColor and Shape:SolidMolecular weight:492.63Oleyl Anilide
CAS:"Oleyl analide (OA) inhibits ACAT (IC50 26 μM), linked to toxic oil syndrome (TOS) with eosinophilia, T-cell activation, and high IL-4, IL-2R, IL-5."Formula:C24H39NOColor and Shape:SolidMolecular weight:357.57VEGFR-2-IN-19
CAS:VEGFR-2-IN-19 (15b) effectively inhibits VEGFR2, induces apoptosis, and increases oxidative stress, showing potential as an anticancer drug.Formula:C21H19N3O2Color and Shape:SolidMolecular weight:345.39Peficitinib hydrochloride
CAS:Peficitinib HCl (ASP015K) is an oral JAK inhibitor with IC50s: JAK1 (3.9 nM), JAK2 (5.0 nM), JAK3 (0.7 nM), Tyk2 (4.8 nM).Formula:C18H23ClN4O2Color and Shape:SolidMolecular weight:362.86Etibendazole
CAS:Etibendazole is a microtubule inhibitor.Formula:C18H16FN3O4Color and Shape:SolidMolecular weight:357.34Z 124-73
CAS:Z 124-73 is an agent of antiviral.Formula:C27H28N4O2SPurity:98%Color and Shape:SolidMolecular weight:472.6Clofibride
CAS:Clofibrin is a kind of hypolipidemic drug, which can reduce Hypertriglyceride and hypercholesterolemia.Formula:C16H22ClNO4Color and Shape:SolidMolecular weight:327.8SC-58272
CAS:SC-58272 is an inhibitor of N-myristoyltransferase (Nmt), a target for anti-fungal and anti-viral therapy.Formula:C33H52N6O4Purity:98%Color and Shape:SolidMolecular weight:596.8NLX-219
CAS:NLX-219 is a selective 5-HT1A receptor-biased agonists.Formula:C21H23ClF2N2O2Color and Shape:SolidMolecular weight:408.87Methylsilanol ascorbate
CAS:Methylsilanol ascorbate is a silanol analogue and inhibitor of angiotensin-converting enzyme.Formula:C7H12O8SiColor and Shape:SolidMolecular weight:252.25FK409
CAS:FK409 is a cell permeable NO donor which produces vasorelaxation.Formula:C8H13N3O4Color and Shape:SolidMolecular weight:215.21S.pombe lumazine synthase-IN-1
CAS:S.pombe lumazine synthase-IN-1 inhibits lumazine synthases: Ki of 243μM for S.pombe, 9.6μM for M.tuberculosis.Formula:C14H13N3O6Color and Shape:SolidMolecular weight:319.275-Hydroxylansoprazole sulfone
CAS:5-hydroxylansoprazole is an in vitro metabolism-dependent CYP2C19 inhibitor.Formula:C16H14F3N3O4SColor and Shape:SolidMolecular weight:401.36hCAXII-IN-3
CAS:hCAXII-IN-3 (Compound 6o) is a selective inhibitor of human carbonic anhydrase XII (hCAXII) (Ki: 10.0 nM).Formula:C26H20BrN5O3SColor and Shape:SolidMolecular weight:562.44HIV-1 inhibitor-19
CAS:HIV-1 inhibitor-19 is a potent NNRTI targeting L100I, K103N, V106A/F227L mutants; EC50s: 7.3, 9.2, 21.0 nM respectively.Formula:C24H22BClN2O5SColor and Shape:SolidMolecular weight:496.77Antitumor agent-55
CAS:Antitumor agent-55 (5q) inhibits PC3 (IC50: 0.91 μM), blocks G1/S phase, induces apoptosis, and halts migration.Formula:C32H34N6O4SColor and Shape:SolidMolecular weight:598.72CID-1304264
CAS:CID-1304264 is an HIV-1 Rev pre-integration inhibitor.Formula:C23H21ClN4O3SColor and Shape:SolidMolecular weight:468.96Flupirtine HCl
CAS:Flupirtine HCl, non-opioid central analgesic sold as Katadolon/others since 1984, opens potassium channels, modulates NMDA/GABAA receptors.Formula:C15H18ClFN4O2Color and Shape:SolidMolecular weight:340.78Kadsurenone
CAS:Kadsurenone, from haifenteng, blocks PAF/PTAFR pathway, promising for breast cancer bone metastases treatment.Formula:C21H24O5Color and Shape:SolidMolecular weight:356.41hGGPPS-IN-2
CAS:hGGPPS-IN-2, a C2-ThP-BP analogue, inhibits hGGPPS, targets MM cells, induces apoptosis, and has anti-myeloma effects.Formula:C20H18FN5O7P2SColor and Shape:SolidMolecular weight:553.43-Fucosyllactose
CAS:3-Fucosyllactose, a key fucosylated oligosaccharide in human milk, offers prebiotic and immune benefits.Formula:C18H32O15Color and Shape:SolidMolecular weight:488.44Neratinib dimethylamine N-oxide
CAS:Neratinib dimethylamine N-oxide is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity.Formula:C30H29ClN6O4Color and Shape:SolidMolecular weight:573.04CAY10416
CAS:CAY10416: dual COX-2/5-LO inhibitor, IC50: COX-2 (50 nM), 5-LO (3 nM); >200x selectivity for COX-2; anti-inflammatory, prostate cancer agent.Formula:C29H29FN2O5SColor and Shape:SolidMolecular weight:536.61AK 275
CAS:AK 275 is a calpain inhibitor that prevents degradation of cytoskeletal and myelin proteins in spinal cord in vitro.Formula:C20H31N3O4Color and Shape:SolidMolecular weight:377.48Inz-4
CAS:Inz-4 is a fungal-selective inhibitor of mitochondrial cytochrome bc1.Formula:C18H14F4N2O2Color and Shape:SolidMolecular weight:366.31Pifexole
CAS:Pifexole, a 1,2,4-oxadiazole derivative, shows muscle-relaxant effects in animals and is 7x more potent than chlorzoxazone in rats.Formula:C13H8ClN3OColor and Shape:SolidMolecular weight:257.68SYNTi
SYNTi, a PDZ inhibitor, disrupts syndecan/syntenin interaction with an IC50 of 400 nM, LE of 0.24, for breast cancer study.Formula:C28H24BrFN2O5Color and Shape:SolidMolecular weight:567.4Dot1L-IN-7
CAS:Dot1L-IN-7 (compound 25), a potent DOT1L inhibitor with an IC50 of 1.0 μM, selectively kills MLL-AF9, sparing E2A-HLF cells.Formula:C23H27N9O2Color and Shape:SolidMolecular weight:461.52TBK1/IKKε-IN-4
CAS:TBK1/IKKε-IN-4, a 6-aminopyrazolopyrimidine derivative, serves as a potent, selective inhibitor for TBK1 and IKKε, demonstrating IC50 values of 13 nM and 59 nMFormula:C28H35N7O4Color and Shape:SolidMolecular weight:533.62Lauroylglycyrrhetinic acid
CAS:Lauroylglycyrrhetinic acid, an analog of carbenoxolone, can be used in the treatment of stomach ulcer.Formula:C42H68O5Color and Shape:SolidMolecular weight:652.99Erioflorin
CAS:Erioflorin is an ATP-competitive selective c-Jun N-terminal kinase (JNK) inhibitor.Formula:C19H24O6Color and Shape:SolidMolecular weight:348.39Topoisomerase II inhibitor 4
CAS:Compound E17, a topoisomerase II inhibitor, halts cell cycle at G2/M, possesses anticancer properties and cytotoxic effects.Formula:C25H25N5O4Color and Shape:SolidMolecular weight:459.5BIR2
CAS:BIR2 triggers hESC self-organization into 3D balloon structures during differentiation.Formula:C9H10N2S2Color and Shape:SolidMolecular weight:210.32SJP-L-5
CAS:SJP-L-5 is a inhibitor of HIV-1 infection by blocking viral DNA nuclear entry.Formula:C18H19NO5Color and Shape:SolidMolecular weight:329.35NSC145366
CAS:NSC145366 inhibits Hsp90, targeting its C-terminal for allosteric client downregulation (IC50=119μM), without competing with ATP.Formula:C37H63ClN2O4Color and Shape:SolidMolecular weight:635.36FL3
CAS:FL3 is a novel potent eIF4F inhibitor, it induces the death of cancer cells by an original mechanism that involves the apoptosis-inducing factor and caspase 12.Formula:C25H23BrO5Color and Shape:SolidMolecular weight:483.35TbPTR1 inhibitor 1
CAS:TbPTR1 inhibitor 1 effectively targets kinetochore PTR1 with IC50 <0.1 nM, EC50 0.66 μM against Trypanosoma brucei.Formula:C22H21N7OColor and Shape:SolidMolecular weight:399.45DC-034
CAS:DC-034, a strong MYC transcription suppressor in cancer via G4 mechanism, targets MYC more than other G4 genes.Formula:C24H25F3N2O3Color and Shape:SolidMolecular weight:446.46RDEA-806 free acid
CAS:RDEA-806, a reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.Formula:C24H18BrClN4O3SColor and Shape:SolidMolecular weight:557.85
