Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,824 products)
- Apoptosis(6,303 products)
- Cell Cycle/Checkpoint(4,862 products)
- Chromatin/Epigenetics(2,607 products)
- Cytoskeletal Signaling(1,553 products)
- DNA Damage/DNA Repair(2,875 products)
- Endocrinology/Hormones(3,752 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,998 products)
- Immunology and Inflammation(3,861 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(416 products)
- MAPK Signaling(1,253 products)
- Membrane Transporter/Ion Channel(3,155 products)
- Metabolism(10,145 products)
- Microbiology/Virology(7,618 products)
- Neuroscience(10,355 products)
- Other Inhibitors(35,866 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,426 products)
- Proteases/Proteasome(1,687 products)
- Stem Cell and Derivatives(737 products)
- Tyrosine Kinase/Adaptors(1,976 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66549 products of "Inhibitors"
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Closthioamide
CAS:Closthioamide is a potent inhibitor of bacterial DNA gyrase and highly active against MRSA, Ec, VRE, and Mv (MICs: 0.58 μM, 9.00 μM, 0.58 μM and 72.03 μM).Formula:C29H38N6O2S6Purity:98%Color and Shape:SolidMolecular weight:695.04GW-841819X
CAS:GW841819X: (+)-JQ1 analogue, BET bromodomain inhibitor, active in vivo against various cancers.Formula:C25H21N5O2Color and Shape:SolidMolecular weight:423.47Piribedil dihydrochloride
CAS:dopamine agonistFormula:C16H20Cl2N4O2Purity:98%Color and Shape:SolidMolecular weight:371.26AGLME
CAS:AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.Formula:C11H21N3O4Color and Shape:SolidMolecular weight:259.3SSR128129E free acid
CAS:SSR128129E free acid is an orally available and allosteric inhibitor of FGFR(IC50 of 1.9 μM for FGFR1).Formula:C18H16N2O4Purity:98%Color and Shape:SolidMolecular weight:324.33μ opioid receptor agonist 2
CAS:μ opioid receptor agonist 2 （Compound H-3）is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.Formula:C25H34N4OColor and Shape:SolidMolecular weight:406.56Osteoprotegerin
CAS:Osteoprotegerin, a secreted protein, blocks bone resorption by disrupting osteoclast signaling.Formula:C18H32O2Color and Shape:SolidMolecular weight:280.45IACS-8968
CAS:IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).Formula:C17H18F3N5O2Purity:98%Color and Shape:SolidMolecular weight:381.35LY 281217
CAS:LY 281217, an organic opioid agonist, can produce analgesic effects in mice.Formula:C32H42N4O6Purity:98%Color and Shape:SolidMolecular weight:578.7ZINC09659342
CAS:ZINC09659342 (compound 13) is an inhibitor of Lbc-RhoA interaction (IC50: 3.6 μM).Formula:C23H15F3N2O4Color and Shape:SolidMolecular weight:440.37L 364918
CAS:L 364918 is an oxytocin antagonist.Formula:C40H54N8O6Purity:98%Color and Shape:SolidMolecular weight:742.91Diethyl butylmalonate
CAS:Diethyl butylmalonate shows toxicity to T. pyriformis, with a log(IGC50 -1 ) of 0.557 [1].Formula:C11H20O4Color and Shape:SolidMolecular weight:216.27HDAC-IN-39
CAS:HDAC-IN-39 inhibits HDAC1-3 (IC50: 1.07-2.27 μM), arrests G2/M phase, hinders microtubule polymerization, and is effective against drug-resistant cancers.Formula:C27H26N4O4SColor and Shape:SolidMolecular weight:502.58Bisnafide mesylate
CAS:Bisnafide, a naphthalimide analogue, inhibits DNA/topo II and has antiangiogenic properties to enhance cytotoxic drug delivery to tumors.Formula:C34H36N6O14S2Color and Shape:SolidMolecular weight:816.81Linagliptin mixture with metformin
CAS:Linagliptin mixture with metformin is used for the treatment of type 2 diabetes.Formula:C29H39N13O2Color and Shape:SolidMolecular weight:601.71Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Formula:C19H26ClN3O2S2Color and Shape:SolidMolecular weight:428.01GPI-15427
CAS:GPI-15427: a potent PARP-1 inhibitor, crosses the blood-brain barrier, boosts TMZ's effects on CNS tumors, and sensitizes cancer to radiotherapy.Formula:C20H20N4O2Color and Shape:SolidMolecular weight:348.4Piperphentonamine HCl
CAS:Piperphentonamine HCL is a potential calcium sensitizer for the treatment of heart failure.Formula:C21H24ClNO4Color and Shape:SolidMolecular weight:389.88Trimopam
CAS:Trimopam is a dopamine receptor agonist of the benzazepine group.Formula:C19H23NO2Color and Shape:SolidMolecular weight:297.39CAY10680
CAS:CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.Formula:C18H16N2O2SColor and Shape:SolidMolecular weight:324.4MSU38225
CAS:MSU38225, an Nrf-2 inhibitor, elevates reactive oxygen species (ROS) levels and suppresses the proliferation of human lung cancer cells.Formula:C21H19N3Color and Shape:SolidMolecular weight:313.4Hexamide
CAS:Hexamide is a protein inhibitor.Formula:C13H17NOColor and Shape:SolidMolecular weight:203.28STA-2842
CAS:STA-2842 is an inhibitor of heat shock protein 90 (HSP90).Formula:C29H38N6O5Color and Shape:SolidMolecular weight:550.65BMY-27709
CAS:BMY-27709 inhibits influenza growth (IC50: 3-8 μM, A/WSN/33), targets H1/H2 subtypes via hemagglutinin, ineffective against H3/B Lee/40.Formula:C17H24ClN3O2Purity:97.83% - 98.37%Color and Shape:SolidMolecular weight:337.84Pirifibrate
CAS:Pirifibrate (EL-466) can be used in the hyperlipoproteinemias research that is a hypolipemic substance [1].
Formula:C17H18ClNO4Color and Shape:SolidMolecular weight:335.78P 34081
CAS:P 34081 rapidly blocks parasite cysteine proteinase activity in vivo.Formula:C25H30FN3O4Color and Shape:SolidMolecular weight:455.53Dexetimide HCl
CAS:Dexetimide HCl is a muscarinic antagonist that has been used to treat neuroleptic-induced parkinsonism. Benzetimide is the (-)-enantimorph of dexetimide.Formula:C23H27ClN2O2Color and Shape:SolidMolecular weight:398.93S 332
CAS:S332 is a beta3-agonist, better at enhancing bladder storage than clenbuterol but weaker in reducing bladder contraction during micturition.Formula:C16H17N3O3SColor and Shape:SolidMolecular weight:331.39YS-121
CAS:YS121 inhibits mPGES-1 (IC50=3.4μM) & 5-LOX (IC50=6.5μM), and lowers PGE2 in A549 cells (EC50=12μM).Formula:C20H26ClN3O2SColor and Shape:SolidMolecular weight:407.96SLK/STK10-IN-1
CAS:SLK/STK10-IN-1 is a selective and potent inhibitor of SLK and STK10 with potential antitumor activity.Formula:C17H13ClN2O3Purity:99.34%Color and Shape:SolidMolecular weight:328.75Cyclazocine
CAS:Cyclazocine is an analgesic with mixed narcotic agonist-antagonist properties.Formula:C18H25NOColor and Shape:SolidMolecular weight:271.4PF-184298
CAS:PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.Formula:C15H20Cl2N2OPurity:98.67%Color and Shape:SolidMolecular weight:315.24Boc-7-Aminoheptanoic acid
CAS:Boc-7-Aminoheptanoic acid is a PROTAC linker with a Boc-protected amine and terminal carboxylic acid for stable amide formation.Formula:C12H23NO4Color and Shape:SolidMolecular weight:245.32Glucosylceramide synthase-IN-1
CAS:Potent oral GCS inhibitor T-036, crosses BBB, targets human (IC50: 31 nM) and mouse GCS (IC50: 51 nM), for Gaucher disease research.Formula:C24H20F4N2O3Color and Shape:SolidMolecular weight:460.42Telomerase-IN-4
CAS:Telomerase-IN-4 is a potent inhibitor of telomerase with antiproliferative properties and induces apoptosis [1].Formula:C21H18N4OS2Purity:98%Color and Shape:SolidMolecular weight:406.52Lefucoxib
CAS:Lefucoxib is a cyclooxygenase-2 (COX-2) inhibitor.Formula:C19H17F3N2O2SColor and Shape:SolidMolecular weight:394.41Hemustine
CAS:Hemustine is an inhibitor of human glutathione reductase and widely used as an anti-tumor agent.Formula:C5H10ClN3O3Color and Shape:SolidMolecular weight:195.6GSK-598809 L-tartrate sesquihydrate
CAS:GSK-598809 L-tartrate sesquihydrate is an acute D3 antagonist.Formula:C26H29F4N5O7SH2OColor and Shape:SolidMolecular weight:658.62Bizine dihydrochloride
CAS:Bizine dihydrochloride is a potent LSD1 inhibitor in vitro, being selective versus monoamine oxidases A/B and the LSD1 homologue, LSD2.Formula:C18H25Cl2N3OColor and Shape:SolidMolecular weight:370.32L-771688
CAS:L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benignFormula:C28H33F2N5O5Purity:94.15%Color and Shape:SolidMolecular weight:557.59Leucine thiorphan
CAS:Leucine thiorphan is an inhibitor of enkephalinase.Formula:C16H23NO3SPurity:98%Color and Shape:SolidMolecular weight:309.42GSK5750
CAS:GSK5750 is the ribonuclease H activity inhibitor.Formula:C16H12N4O2SColor and Shape:SolidMolecular weight:324.36D13
CAS:D13 acylhydrazone antifungal; MIC80: 0.06 μg/ml vs. C. neoformans; boosts mouse survival against fungal infections at 20 mg/kg/day orally.Formula:C14H9Br3N2O2Color and Shape:SolidMolecular weight:476.95Bromotetrandrine
CAS:Bromotetrandrine enhances chemo by inhibiting P-glycoprotein, countering efflux pumps.Formula:C38H41BrN2O6Color and Shape:SolidMolecular weight:701.65NSC-639829
CAS:NSC-639829 is an anti-tumor compound that requires a solubilizing agent for dissolution.Formula:C21H20BrN5O3Purity:99.53% - 99.77%Color and Shape:SolidMolecular weight:470.32P-CAB agent 2
CAS:Potent P-CAB agent 2 blocks gastric acid secretion; H+/K+-ATPase IC50 <100 nM, hERG IC50 18.69 μM; non-toxic.Formula:C22H25FN2O4SColor and Shape:SolidMolecular weight:432.51FR-198248
CAS:FR-198248, a new anti-influenza agent, shows antiinfluenza virus activity in Madin-Darby canine kidney (MDCK) cells in vitro.Formula:C9H10O5Color and Shape:SolidMolecular weight:198.17JNJ525
JNJ525, a TNFα inhibitor, blocks protein function by hindering TNFα/TNFR1 and TNFα/TNFR2 complexes; IC50s: 1.2 μM (TNFR1), 1.1 μM (TNFR2).Formula:C31H30N8Color and Shape:SolidMolecular weight:514.64Methapyrilene
CAS:Methapyrilene is a histamine H1 antagonist with sedative action.Formula:C14H19N3SColor and Shape:Liquid Physical Description Clear Colorless Liquid (Ntp 1992)Molecular weight:261.39SHP244
CAS:SHP244 is an allosteric inhibitor of SHP2 with modest thermal stabilization of the enzyme.Formula:C23H17ClN4O3Color and Shape:SolidMolecular weight:432.86
