Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,832 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,611 products)
- Cytoskeletal Signaling(1,563 products)
- DNA Damage/DNA Repair(2,873 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,900 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,141 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,369 products)
- Other Inhibitors(35,851 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,690 products)
- Stem Cell and Derivatives(735 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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(R)-KT109
CAS:(R)-KT109: potent DAGLβ inhibitor (IC50 = 0.79 nM), also blocks DAGLα and ABHD6 (IC50 = 2.51 nM), stronger than (S)-KT109.Formula:C27H26N4OColor and Shape:SolidMolecular weight:422.52DENV-IN-9
CAS:DENV-IN-9 is a DENV2 inhibitor with an EC 50 of 0.88 μM .Formula:C15H9BrO5Color and Shape:SolidMolecular weight:349.13MAC-5576
CAS:MAC-5576 a SARS-CoV-2 Protease inhibitor (IC50 = 81 nM).Formula:C10H6ClNO2SColor and Shape:SolidMolecular weight:239.68RTC14
CAS:RTC14 induces PTC readthrough, restoring dystrophin and aiding muscle function in Duchenne model mice.Formula:C17H18N2O3Color and Shape:SolidMolecular weight:298.34BMS 378806
CAS:BMS-378806 is an orally bioavailable HIV-1 inhibitor that interferes with gp120-CD4 interaction.Formula:C22H22N4O4Color and Shape:SolidMolecular weight:406.43Etintidine Free Base
CAS:Etintidine Free Base is a Histamine H2 Antagonist.Formula:C12H16N6SColor and Shape:SolidMolecular weight:276.36SC-III3
CAS:SC-III3, a scopoletin derivative, triggers autophagy in HepG2 cells via AMPK/mTOR and impairs cell/tumor growth, acting non-apoptotically.Formula:C19H14ClNO5Color and Shape:SolidMolecular weight:371.77JJO-1
CAS:JJO-1 is a bi-quinoline activating all AMPK αβγ isoforms except γ3; it requires low ATP and is unaffected by γ mutations or β deletions.Formula:C19H13N3Color and Shape:SolidMolecular weight:283.33MC4343
MC4343, a potent dual inhibitor targeting both EZH2 and histone deacetylase, presents promising potential for cancer research applications.Formula:C36H41N5O4Color and Shape:SolidMolecular weight:607.74SX-576
CAS:SX-576: potential pulmonary inflammation treatment, non-competitive boronic acid CXCR1/2 antagonist.Formula:C20H15BF4N2O4SColor and Shape:SolidMolecular weight:466.21F-050
CAS:F-050 inhibits platelet aggregation, potentially treating thrombosis in guinea pigs, rabbits, and rats.Formula:C21H20OColor and Shape:SolidMolecular weight:288.38F2276-0099
CAS:F2276-0099 is a PCAF/GCN5 BRD inhibitorFormula:C19H20N2O4Color and Shape:SolidMolecular weight:340.37Nrf2 activator-5
CAS:Nrf2 activator-5 combats oxidative stress and inflammation in microglia, with potent antioxidant effects.Formula:C25H30Cl2O6Color and Shape:SolidMolecular weight:497.41Looplure
CAS:Looplure is a chemosterilant, insect attractant and repellent.Formula:C14H26O2Color and Shape:SolidMolecular weight:226.35Tubulin polymerization-IN-18
CAS:Tubulin aggregation-IN-18 (compound 3) is a potent tubulin aggregation inhibitor with potential for breast cancer and drug-resistant colon cancer studies.Formula:C25H25NO6Color and Shape:SolidMolecular weight:435.47IKKß-IN-124
CAS:IKKβ-IN-124 blocks NF-κB by inhibiting IκBα phosphorylation and securing IKKβ in inactive form.Formula:C17H26Cl2N2O3SColor and Shape:SolidMolecular weight:409.37hA2A/hCA XII modulator 1
CAS:Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.Formula:C24H19N7O4SColor and Shape:SolidMolecular weight:501.52Butixirate
CAS:Butixirate is a biochemical.Formula:C28H33NO2Color and Shape:SolidMolecular weight:415.577INU-101
CAS:INU-101: oral 11β-HSD1 inhibitor improves insulin sensitivity and reduces blood glucose, potential type 2 diabetes treatment.Formula:C21H28FN3O4SColor and Shape:SolidMolecular weight:437.53Vibsanin A
CAS:Vibsanin A, an activator of protein kinase C (PKC) and an inhibitor of HSP90, demonstrates anti-proliferative effects on human cancer cell lines.Formula:C25H38O4Color and Shape:SolidMolecular weight:402.57HDAC-IN-31
CAS:HDAC-IN-31: Oral HDAC inhibitor; targets HDAC1, 2, 3; weak on HDAC8; potential in fighting lymphoma.Formula:C25H24N4O2Color and Shape:SolidMolecular weight:412.48HDAC6-IN-14
HDAC6-IN-14, an inhibitor of HDAC6 (HDAC), exhibits high selectivity with an IC50 value of 42 nM, demonstrating over 100-fold selectivity compared to HDAC1,Formula:C24H30FN3O4Color and Shape:SolidMolecular weight:443.51L 738372
CAS:L 738372 is a non-nucleoside inhibitor of HIV-1 reverse transcriptase.Formula:C18H15N3OColor and Shape:SolidMolecular weight:289.33BML277 Acid
CAS:BML277 Acid is a metabolite of BML277 which is a selective checkpoint kinase 2 inhibitor.Formula:C20H13ClN2O3Color and Shape:SolidMolecular weight:364.78(+)-Cembrene A
CAS:(+)-Cembrene A, a nontoxic α-glucosidase inhibitor to human normal hepatocyte (LO2) cells, exhibits an IC50 value of 30.31 μM.Formula:C20H32Color and Shape:SolidMolecular weight:272.47IMB-10
CAS:IMB-10 is an alphaMbeta2 integrin modulator, inhibiting leukocyte migration and recruitment in vitro and in vivo.Formula:C19H15NOS2Color and Shape:SolidMolecular weight:337.46CGS 21595
CAS:CGS 21595 inhibits the formation of 5-hydroxyeicosatetraenoic acid and leukotriene B4; rapidly metabolized to CGS 19213.Formula:C21H25NO4Color and Shape:SolidMolecular weight:355.43SG2057
CAS:SG2057 (DRG16), a PBD dimer with pentyldioxy linkage, binds DNA minor groove, forms cross-links, and is a potent antitumor agent.Formula:C33H36N4O6Color and Shape:SolidMolecular weight:584.66Ametantrone Acetate
CAS:Ametantrone Acetate is a topoisomerase II inhibitor of anthrapyrazole family, which can lead to DNA covalent crosslinking.Formula:C24H32N4O6Color and Shape:SolidMolecular weight:472.542Naproxen ethyl ester
CAS:Naproxen ethyl ester, an NSAID similar to ibuprofen, reduces pain, fever, and inflammation. It's a non-selective COX inhibitor.Formula:C16H18O3Color and Shape:SolidMolecular weight:258.31CDK8-IN-6
CAS:CDK8-IN-6 (compound 9) is a potent inhibitor of cyclin-dependent kinase 8 (CDK8) (Kd: 13 nM), CDK8-IN-6 showed potential research value in AML cancers.Formula:C26H37ClN2Color and Shape:SolidMolecular weight:413.04LY191704
CAS:LY 191704 is a 5α-reductase type 1 inhibitor.Formula:C14H16ClNOColor and Shape:SolidMolecular weight:249.74PWT33597 mesylate
CAS:PWT33597 (VDC-597) is an oral PI3K alpha/mTOR dual inhibitor, potentially causing cancer cell death and growth inhibition.Formula:C27H34F2N8O7S2Color and Shape:SolidMolecular weight:684.7348VEGFR-2-IN-20
CAS:VEGFR-2-IN-20 (Compound 7) is a highly effective VEGFR inhibitor with significant potential for cancer research [1].Formula:C20H20N4O3SColor and Shape:SolidMolecular weight:396.46BAY-846
CAS:BAY-846: allosteric MEK inhibitor, long-lasting, highly bioavailable, low brain entry, effective in K-Ras A549 model.Formula:C19H13F4IN4O4SColor and Shape:SolidMolecular weight:596.29TRK-IN-16
CAS:TRK-IN-16 (X-21) is a potent TRK inhibitor for research in diseases related to protein kinases.Formula:C19H20FN5OColor and Shape:SolidMolecular weight:353.39Sulfamethomidine
CAS:Sulfamethomidine has antibacterial activity [1].Formula:C12H14N4O3SColor and Shape:SolidMolecular weight:294.33Antitumor agent-44
CAS:Antitumor agent-44 (Compound 5n) elicits potent antitumor effects by inducing disruption of mitochondrial homeostasis, cell cycle arrest, and apoptosis in humanFormula:C24H15N3O3Color and Shape:SolidMolecular weight:393.39SAR296968
CAS:SAR296968 is a novel selective NCX inhibitor, improving cardiac function and restoring sympathovagal balance in heart failure.Formula:C22H22N2O4SColor and Shape:SolidMolecular weight:410.49Antitubercular agent-31
CAS:Antitubercular agent-31 is an antitubercular agent that inhibits M. tuberculosisH37Rv (MIC: 0.03 μM) and also inhibits DprE1 (IC50: 1.1 μM).Formula:C20H24F2N4O5S2Color and Shape:SolidMolecular weight:502.56Germination-IN-1
CAS:Germination-IN-1 (compound 11) is a potent germination inhibitor (IC50: 4 μM) with anti-germination effects (germination rate = 14%).Formula:C30H45NO3Color and Shape:SolidMolecular weight:467.68UCSF924NC
CAS:UCSF924NC, a DRD4 antagonist, has 1/2500th affinity of its counterpart, UCSF924.Formula:C19H21N3OColor and Shape:SolidMolecular weight:307.39α-Synuclein inhibitor 3
CAS:α-Synuclein inhibitor 3 (Compound 7g) is a potent inhibitor of α-synuclein (α -Syn) aggregation.Formula:C20H23N5O2Color and Shape:SolidMolecular weight:365.432-(1-hydroxypentyl)benzoic Acid
CAS:Potassium-Hydroxypentyl Benzoate is a drug potentially for the treatment of acute ischemic stroke (AIS)Formula:C12H16O3Color and Shape:SolidMolecular weight:208.25Tubulin polymerization-IN-27
CAS:Compound 5j inhibits tubulin polymerization, arrests cell cycle at G2/M phase, and induces apoptosis.Formula:C22H20N2O2Color and Shape:SolidMolecular weight:344.41Exp 063
CAS:Exp 063 is a hybrid compound that possesses both the angiotensin II antagonist activity and the β-blocking activity. EXP 063 also acts as a partial β-agonist.Formula:C37H41N9O5Color and Shape:SolidMolecular weight:691.78BW 373U86
CAS:BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [Formula:C27H37N3O2Color and Shape:SolidMolecular weight:435.6Ap44mSe
CAS:Ap44mSe: potent, selective antitumor. Lowers cellular iron, alters iron protein levels, boosts metastasis suppressor NDRG1.Formula:C10H14N4SeColor and Shape:SolidMolecular weight:269.2NAGKi
CAS:NAGKi is an inhibitor of N-acetylmannosamine kinase (NAMK) and N-acetylglucosamine kinase (NAGK).Formula:C9H17NO6Purity:98%Color and Shape:SolidMolecular weight:235.23UK-356202
CAS:UK-356,202: potent, selective inhibitor of urokinase-type plasminogen activator (Ki=37 nM), target for breast/ovarian/pancreatic cancer therapy.Formula:C17H13ClN4O2Color and Shape:SolidMolecular weight:340.76
