Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,833 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,612 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,015 products)
- Immunology and Inflammation(3,901 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,153 products)
- Metabolism(10,140 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,405 products)
- Other Inhibitors(35,850 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66518 products of "Inhibitors"
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KL8604166
CAS:KL8604166 (UCB-11056) is a potential puzzle compound.UCB-11056 amplifies the formation of inducible cyclic AMP in rat brain tissue.Formula:C12H21N5O2Purity:99.21%Color and Shape:SolidMolecular weight:267.33Ref: TM-T29038
1mg264.00€5mg650.00€10mg888.00€25mg1,369.00€50mg1,783.00€100mg2,250.00€1mL*10mM (DMSO)590.00€GAL-021 sulfate
CAS:GAL-021 sulfate is a BKCa channel blocker that inhibits the analgesic effects of opioids and is used in the study of respiratory control diseases.Formula:C11H24N6O5SPurity:99.92%Color and Shape:SolidMolecular weight:352.41BGT1-IN-9
CAS:BGT1-IN-9 is an M1 muscarinic agonist.Formula:C5H10ClN3O2Color and Shape:SolidMolecular weight:179.605Abivertinib HCl
CAS:Abivertinib (AC0010/Avitinib) is an EGFR/BTK inhibitor effective in AML, especially with FLT3-ITD mutations.Formula:C26H28Cl2FN7O2Color and Shape:SolidMolecular weight:560.4554Ridaifen-B
CAS:Ridaifen-B, a tamoxifen derivative, works by inducing independent autophagy of Bcl-2, without estrogen receptor involvement.Formula:C34H42N2O2Color and Shape:SolidMolecular weight:510.71SARS-CoV-2-IN-17
CAS:SARS-CoV-2-IN-17 inhibits NPro effectively, with EC50 of 2.18 μM and Kd of 7.82 μM, showing strong anti-viral properties.Formula:C19H19F3N2O3Color and Shape:SolidMolecular weight:380.36N,N-Dipropyldopamine (hydrobromide)
CAS:N,N-Dipropyldopamine is a dopamine agonist reducing DOPA and locomotion in rats and mice, reversible by spiroperidol.Formula:C14H24BrNO2Color and Shape:SolidMolecular weight:318.255CI 986
CAS:CI 986 is a novel nonulcerogenic anti-inflammatory agent.Formula:C21H35N3O2S2Color and Shape:SolidMolecular weight:425.65AZD7268
CAS:AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.Formula:C29H30N4O2SColor and Shape:SolidMolecular weight:498.64Diprafenone Free Base
CAS:Diprafenone Free Base is an antiarrhythmic beta adrenergic antagonist.Formula:C23H31NO3Color and Shape:SolidMolecular weight:369.5N-Fmoc-8-aminooctanoic acid
CAS:N-Fmoc-8-aminooctanoic acid: a PROTAC linker with deprotectable Fmoc-amine and reactive carboxylic end for stable amide bonds.Formula:C23H27NO4Color and Shape:SolidMolecular weight:381.46WX-081
CAS:WX-081 is an anti-TB drug effective against DS-TB (MIC: 0.083 μg/ml) and MDR-TB strains (MIC: 0.11 μg/ml) with hERG inhibition (IC50: 1.89 μM).Formula:C34H33ClN2O2Color and Shape:SolidMolecular weight:537.09LX-3
CAS:LX-3 activates p38 MAPK, enabling expression of genes normally silenced by DNA methylation.Formula:C20H13BrN4OSColor and Shape:SolidMolecular weight:437.31CDK4/6-IN-12
CAS:CDK4/6-IN-12 inhibits CDK4/6 with IC50s of 592.3 nM & 3090 nM, useful in cancer research.Formula:C12H10N6Color and Shape:SolidMolecular weight:238.25STING Agonist 12b
CAS:STING agonist 12b activates human/mouse STING, binds with Kd 26.4 μM, prompts interferon, and induces TNF-a, IL-6, IP-10, IL-1b in THP-1 cells.Formula:C16H15NO2Color and Shape:SolidMolecular weight:253.3Piperilate HCl
CAS:Piperilate HCl is an antispasmodic, antimuscarinic agent. It is a muscarinic cholinergic receptor antagonist.Formula:C21H26ClNO3Color and Shape:SolidMolecular weight:375.89M2WJ332
CAS:M2WJ332 is a novel M2-S31N inhibitor, showing antiviral activity against Influenza A virus.Formula:C18H22N2OSColor and Shape:SolidMolecular weight:314.45LH-708
CAS:LH-708 is an inhibitor of cystine stone formation for treatment of cystinuria.Formula:C16H36Cl4N6O2S2Color and Shape:SolidMolecular weight:550.42CK 2289
CAS:CK 2289 is an inhibitor of type III cyclic 3'5' -adenosine monophosphate phosphodiesterase with potential use in the treatment of congestive heart failure.Formula:C15H14N4O2Color and Shape:SolidMolecular weight:282.3SC 23133
CAS:SC 23133 is an antimineralocorticoid that is known to induce a marked but reversible inhibition of aldosterone biosynthesis.Formula:C23H30O3Color and Shape:SolidMolecular weight:354.48BRD9092
CAS:BRD9092 is a small molecule probe that elevates markers of oxidative stress without causing cell death.Formula:C24H18ClN3O3Purity:98.65%Color and Shape:SolidMolecular weight:431.87TX-1123
CAS:TX-1123: PTK/COX inhibitor, Src/eEF2-K/PKA/EGFR-K/PKC targeted, IC50 of 1.16μM(COX2), 15.7μM(COX1), low mitochondrial toxicity.Formula:C20H24O3Color and Shape:SolidMolecular weight:312.4AR524
CAS:AR524 surpasses kifunensine, strongly blocking human cancer cell-cluster formation at 10 μM.Formula:C26H30N2O3Color and Shape:SolidMolecular weight:418.53Androgen receptor antagonist 3
CAS:Androgen receptor antagonist 3 (Compound C18) has anticancer activities that is an antagonist of androgen receptor (AR) (IC 50 = 2.4 μM) [1].Formula:C22H18ClNColor and Shape:SolidMolecular weight:331.84EEDQ
CAS:EEDQ: irreversible dopamine antagonist; specifically reacts with carboxyl groups, couples acylamino acids without racemization.Formula:C14H17NO3Color and Shape:SolidMolecular weight:247.29Ro 47-1669
CAS:Ro 47-1669 is a bioactive chemical.Formula:C14H9NO7Color and Shape:SolidMolecular weight:303.22STAT3-IN-11
CAS:STAT3-IN-11 is a STAT3 inhibitor.STAT3-IN-11 promotes apoptosis in cancer cells and is a candidate compound for the treatment of cancer.Formula:C20H17NO4Purity:98.3%Color and Shape:SolidMolecular weight:335.35CAY10568
CAS:Most local anesthetics act by abolishing voltage gated sodium channel currents indiscriminately in all populations of neurons.Formula:C11H17IN2OColor and Shape:SolidMolecular weight:320.174Ronactolol
CAS:Ronactolol is an aminopropanol derivative with beta-adrenoreceptor blocking activity.Formula:C20H26N2O4Color and Shape:SolidMolecular weight:358.43Anti-hyperglycemic agent-1
CAS:Anti-hyperglycemic agent 1 is a potent inhibitor of alpha-glucosidase (IC50: 0.53 μM). anti-Hyperglycemic agent 1 can be used to study diabetes.Formula:C20H15BrN2O3Color and Shape:SolidMolecular weight:411.25Tolnidamine
CAS:Tolnidamine is an antineoplastic drug.Formula:C16H13ClN2O2Purity:98%Color and Shape:SolidMolecular weight:300.744,4'-Dicyanostilbene
CAS:4,4'-Dicyanostilbene: potent anti-Dd2 malaria, EC50=27nM; effective vs. MRSA.Formula:C16H10N2Color and Shape:SolidMolecular weight:230.26GX-585
CAS:GX-585 is a novel potent inhibitor of NaV1.7 and highly selective against NaV1.5, having limited selectivity against NaV1.1 and NaV1.2.Formula:C24H25Cl2FN4O3SPurity:99.02% - 99.03%Color and Shape:SolidMolecular weight:539.45Sibopirdine
CAS:Sibopirdine is a new type of cognitive enhancer and intelligence booster that has been studied as a cognitive enhancer for the treatment of Alzheimer's disease.Formula:C23H18N4Color and Shape:SolidMolecular weight:350.42F-17
CAS:F-17 inhibits biofilm, elastase, pyocyanin, and motility, binds to LasR/PqsR, and is non-cytotoxic.Formula:C17H15BrO4Color and Shape:SolidMolecular weight:363.2Quinoprazine
CAS:Quinoprazine: inhibits Vaccinia virus (IC50=10μM), antimalarial vs Plasmodium berghei, reduces PrPSc, antiprion.Formula:C25H26N4Color and Shape:SolidMolecular weight:382.5OSU-53
CAS:OSU-53 is an AMPK activator, inhibiting mTOR signaling and autophagy stimulation. OSU-53 also activates mutations in RAS or BRAF.Formula:C25H24F3N3O6S2Color and Shape:SolidMolecular weight:583.6AY-16804
CAS:AY-16804 is an inhibitor of platelet aggregation.Formula:C12H18O3Color and Shape:SolidMolecular weight:210.27UCK2 Inhibitor-1
CAS:UCK2 Inhibitor-1 is a non-competitive UCK2 inhibitor with an IC 50 of 4.7 µM .Formula:C27H21N3O4SColor and Shape:SolidMolecular weight:483.54(rel)-Oxaliplatin
CAS:(rel)-Oxaliplatin, a DNA inhibitor, induces crosslinks, hinders replication/transcription, and triggers apoptosis; used in cancer studies.Formula:C8H14N2O4PtColor and Shape:SolidMolecular weight:397.29THK-523
CAS:THK-523 selectively binds to tau in Alzheimer's, potent in vitro/vivo. 18F-THK523 excels in tau imaging.Formula:C17H15FN2OColor and Shape:SolidMolecular weight:282.31SANT-2
CAS:SANT-2 is a potent inhibitor of Shh signaling pathway.Formula:C23H20ClN3O4Color and Shape:SolidMolecular weight:437.88Diallyl G
CAS:Diallyl G is a delta-opioid receptor antagonist agent.Formula:C38H53N5O8Color and Shape:SolidMolecular weight:707.86α-Glucosidase-IN-5
CAS:α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.Formula:C15H13NO3Color and Shape:SolidMolecular weight:255.27α-Glucosidase-IN-16
CAS:α-Glucosidase-IN-16 is a highly effective and orally bioavailable inhibitor of α-glucosidase, displaying a remarkable IC50 value of 3.28 μM.Formula:C22H18FNSColor and Shape:SolidMolecular weight:347.45BN80933
CAS:BN80933 is a dual inhibitor of lipid peroxidation and neuronal nitric oxide synthase; Neuroprotectant.Formula:C29H34N4O3SColor and Shape:SolidMolecular weight:518.67Binifibrate
CAS:Binifibrate is a hyperlipemiant drug used for the treatment of hyperlipidemia.Formula:C25H23ClN2O7Color and Shape:SolidMolecular weight:498.91EMI56
CAS:EMI56, a derivative of EMI1, exhibits enhanced potency against mutant EGFR compared to EMI1. Additionally, EMI56 effectively inhibits EGFR triple mutants[1].Formula:C21H20N2O3Color and Shape:SolidMolecular weight:348.4Bexin-1
CAS:Bexin-1 blocks Munc13-4 from binding to membranes, targeting its C2 domain and stopping ANF-EGFP release induced by ionomycin.Formula:C20H26ClN5OSColor and Shape:SolidMolecular weight:419.97KDM5B-IN-3
CAS:KDM5B-IN-3 inhibits KDM5B/JARID1B with IC50 of 9.32 μM, useful in gastric cancer studies.Formula:C19H25ClN4O2Color and Shape:SolidMolecular weight:376.88
