Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,833 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,876 products)
- Chromatin/Epigenetics(2,613 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,015 products)
- Immunology and Inflammation(3,901 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,137 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,414 products)
- Other Inhibitors(35,849 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66517 products of "Inhibitors"
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HIV-1 inhibitor-34
CAS:HIV-1 inhibitor-34 (5q): potent, selective; EC50: 6.4 nM; MT-4 CC50: 16 μM; useful in AIDS research.Formula:C26H27N7OColor and Shape:SolidMolecular weight:453.54SCAL-255
CAS:SCAL-255 is a mitochondrial complex I (CI) inhibitor, exhibiting potent inhibition with an IC50 of 1.14 μM.Formula:C27H28F3N5O3Purity:98%Color and Shape:SolidMolecular weight:527.54I-138
CAS:I-138 is an orally active and reversible inhibitor of USP1-UAF1.I-138 induces mono-ubiquitination of FANCD2 and PCNA and inhibits USP1 auto-cleavage in cells.Formula:C26H23F3N6OPurity:99.41%Color and Shape:SolidMolecular weight:492.5Ref: TM-T73560
1mg170.00€5mg349.00€10mg492.00€25mg707.00€50mg982.00€100mg1,468.00€1mL*10mM (DMSO)384.00€Momelotinib Mesylate
CAS:Momelotinib Mesylate is an ATP-competitive JAK1/JAK2 inhibitor (IC50: 11 nM/18 nM). It has 10-fold selectivity versus JAK3.Formula:C24H26N6O5SPurity:98%Color and Shape:SolidMolecular weight:510.57SB 258585 hydrochloride
CAS:SB 258585 hydrochloride is a 5-HT6 receptor antagonist.Formula:C18H23ClIN3O3SPurity:98%Color and Shape:SolidMolecular weight:523.82QS11
CAS:QS11, a GTPase ARFGAP1, modulates ARF-GTP levels and synergizes with the Wnt/β-catenin signaling pathway to upregulate β-catenin nuclear translocation.Formula:C36H33N5O2Purity:98.59%Color and Shape:SolidMolecular weight:567.68Ref: TM-T4022
2mg34.00€5mg50.00€10mg80.00€25mg147.00€50mg215.00€100mg323.00€200mg442.00€1mL*10mM (DMSO)62.00€Tazanolast
CAS:Tazanolast is a selective mast-cell-stabilizing drug.Formula:C13H15N5O3Purity:98%Color and Shape:SolidMolecular weight:289.29Naprodoxime HCl
CAS:Naprodoxime HCl is an antidepressant. It also is an anti-aggressive agent.Formula:C13H15ClN2O2Purity:98%Color and Shape:SolidMolecular weight:266.72KD3010 tosylate
CAS:KD-3010 is a PPARδ agonist for possible diabetes and obesity treatment, reduces liver damage, and limits fibrosis more than GW501516 post-CCl₄ exposure.Formula:C30H33F3N2O8S2Color and Shape:SolidMolecular weight:670.7152Lercanidipine. (R)-
CAS:(R)-Lercanidipine enantiomer: antihypertensive, blocks L-type Ca2+ channels, dilates blood vessels.Formula:C36H41N3O6Color and Shape:SolidMolecular weight:611.73GSK2239633
CAS:GSK2239633: potent CCR4 antagonist, pIC50=7.9, promising for asthma due to T-helper 2 recruitment role.Formula:C21H19ClN4O5S2Color and Shape:SolidMolecular weight:506.98CB1R Allosteric modulator 2
CAS:Compound 18 is a potent CB1R allosteric modulator that acts as a negative modulator (NAM) for CB1R orthosteric ligands.Formula:C19H15ClFN3OColor and Shape:SolidMolecular weight:355.79CP 59430
CAS:CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.Formula:C21H22N8O3Color and Shape:SolidMolecular weight:434.45(4E)-SUN9221
CAS:(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity inFormula:C25H31FN4O3Purity:97.79%Color and Shape:SolidMolecular weight:454.54VU6010572
CAS:VU6010572: potent, selective mGlu3 modulator, IC50 245 nM, high CNS penetration.Formula:C20H18FNO3Color and Shape:SolidMolecular weight:339.36Dimetacrine
CAS:Dimetacrine is a useful antidepressant.Formula:C20H26N2Purity:98%Color and Shape:SolidMolecular weight:294.43INO-1001 methanesulfonate
CAS:INO-1001 methanesulfonate is a strong PARP inhibitor with chemosensitization and radiosensitization effects.Formula:C24H29N3O7S2Color and Shape:SolidMolecular weight:535.63Imatinib hydrochloride
CAS:Imatinib: treats CML/GISTs, inhibits v-Abl/c-Kit/PDGFR (IC50: 0.6/0.1/0.1 μM).Formula:C29H32ClN7OPurity:98%Color and Shape:SolidMolecular weight:530.06(R)-Bambuterol
CAS:Bambuterol is a β2-agonist prodrug for asthma and COPD, taken daily, with a good safety profile and reduces plasma LDL-C and cholesterol.Formula:C18H29N3O5Color and Shape:SolidMolecular weight:367.44FGFR3-IN-5
CAS:FGFR3-IN-5: potent, selective FGFR3 inhibitor. IC50: 3 nM FGFR3, 44 nM FGFR2, 289 nM FGFR1. For cancer research.Formula:C24H24FN7O3Color and Shape:SolidMolecular weight:477.49Furamidine
CAS:Furamidine is a PRMT1-selective, cell-permeable inhibitor (IC50: 9.4μM), also targeting TDP-1, and is an antiparasitic bisbenzamidine derivative.Formula:C18H16N4OPurity:98%Color and Shape:SolidMolecular weight:304.35CAY10641
CAS:cPLA2α breaks down arachidonic acid, starting prostaglandin and leukotriene synthesis. CAY10641, its inactive alcohol form, is a potent anti-inflammatory.Formula:C28H27NO6Color and Shape:SolidMolecular weight:473.52BLT-3
CAS:BLT-3 is a novel scavenger receptor BI (SR-BI) inhibitor.Formula:C19H13NOPurity:98%Color and Shape:SolidMolecular weight:271.31ETMTC
CAS:ETMTC is a inhibitor of inflammatory cell adhesion molecules (cams)Formula:C14H18O4SColor and Shape:SolidMolecular weight:282.36OUN10989
CAS:OUN10989, an analog of LP-261, is a potent antimitotic inhibiting G2/M phase, first reported in J. Med. Chem 2011; no formal name yet.Formula:C19H15N3OColor and Shape:SolidMolecular weight:301.34PF-739
CAS:PF-739 is an AMPK agonist that has been shown to activate AMPK in hepatocytes and skeletal muscle.Formula:C23H23ClN2O5Purity:98%Color and Shape:SolidMolecular weight:442.89α-Lipoic Acid Choline Ester
CAS:Alpha-Lipoic Acid Choline Ester is used potentially to treat presbyopia.Formula:C13H26ClNO2S2Purity:98%Color and Shape:SolidMolecular weight:327.93COR167
CAS:COR167 is a CB2 agonist with immunomodulatory effects, protective brain properties, and antinociception.Formula:C28H38N2O2Color and Shape:SolidMolecular weight:434.61Btm 1042
CAS:Btm 1042 is an antispasmodic drug. It has been found to depress twitch responses in the ileum of guinea pigs.Formula:C21H26ClN3OSColor and Shape:SolidMolecular weight:403.97Tubulin polymerization-IN-7
CAS:Tubulin aggregation-IN-7 is a potent tubulin aggregation inhibitor that has shown research potential for cancer diseases.Formula:C28H24N4O6SColor and Shape:SolidMolecular weight:544.58Butabindide
CAS:Butabindide (UCL-1397) selectively inhibits TPP II, protecting CCK-8, with Ki of 10 μM (TPP I) and 7 nM (TPP II).Formula:C17H25N3O2Color and Shape:SolidMolecular weight:303.4MR 2266
CAS:MR 2266 is a narcotic antagonist.Formula:C21H27NO2Color and Shape:SolidMolecular weight:325.44Acolbifene
CAS:Acolbifene (SCH 57068) is a selective antagonist of estrogen receptors with IC50s of 2 nM and 0.4 nM for estradiol-induced transcriptional activity of ERα andFormula:C29H31NO4Purity:98.17%Color and Shape:SolidMolecular weight:457.56AKCI
CAS:AKCI is a PPI inhibitor that acts by targeting the AURKC-IκBα interaction.Formula:C19H27N7OPurity:98%Color and Shape:SolidMolecular weight:369.46CVT-2759
CAS:CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.Formula:C17H24N6O6Color and Shape:SolidMolecular weight:408.41NKP-1339
CAS:NKP-1339 (IT-139) induces G2/M cell cycle arrest, blockage of DNA synthesis, and induction of apoptosis via the mitochondrial pathway.Formula:C14H12Cl4N4NaRuPurity:98%Color and Shape:SolidMolecular weight:502.14EGFR-IN-26
CAS:EGFR-IN-26 is an EGFR inhibitor that can be used in cancer research.Formula:C29H34N6O3Color and Shape:SolidMolecular weight:514.62Blancoxanthone
CAS:Blancoxanthone, a plant-derived molecule, may inhibit COVID-19, influenza, SARS, and MERS-CoV.Formula:C23H22O5Color and Shape:SolidMolecular weight:378.42Zaldaride maleate
CAS:Zaldaride maleate blocks Ca2+, Na+, K+ currents, and nAChR; inhibits CaM cAMP PDE (IC50: 3.3 nM) and estrogen signaling.Formula:C30H32N4O6Purity:98%Color and Shape:SolidMolecular weight:544.6Tilmacoxib
CAS:Tilmacoxib is a highly selective, time-dependent, and irreversible inhibitor of human COX-2 ( IC50: 85 nM in an enzyme assay).Formula:C16H19FN2O3SPurity:98%Color and Shape:SolidMolecular weight:338.4RU 24926
CAS:RU 24926 is a di-(phenethyl)-amine derivative that used as a dopamine-D2 receptor agonist.Formula:C19H25NO2Color and Shape:SolidMolecular weight:299.41BisQ
CAS:BisQ is an agonist of photochromic. It used for the muscle-type nAChR.Formula:C20H30IN4Purity:98%Color and Shape:SolidMolecular weight:453.392Profadol hydrochloride
CAS:Profadol hydrochloride acts as a mixed agonist-antagonist of the μ-opioid receptor with analgesic activity.Formula:C14H22ClNOPurity:98%Color and Shape:SolidMolecular weight:255.78Aronixil
CAS:Aronixil is a biochemical.Formula:C14H15ClN4O2Color and Shape:SolidMolecular weight:306.75Cl-Necrostatin-1
CAS:Cl-Necrostatin-1 is an inhibitor of receptor-interacting protein kinase. It inhibits RIPK1 activity.Formula:C13H12ClN3OSColor and Shape:SolidMolecular weight:293.77THK-5470
CAS:THK-5470, a selective MAO-B probe, binds strongly (IC50=4.2 nM) and aids in studying neurological diseases.Formula:C18H17FN2O2Color and Shape:SolidMolecular weight:312.34ICI 195739
CAS:ICI 195739 is a newer antifungal agent. It inhibits neutrophil random migration, chemotaxis, and hexose monophosphate shunt activity.Formula:C24H20F6N6O2Purity:98%Color and Shape:SolidMolecular weight:538.45Neuraminidase-IN-13
CAS:Neuraminidase-IN-13 (Compound 10), a neuraminidase inhibitor exhibiting antiviral activity, demonstrates significant inhibition of NDV infection in Vero cellsFormula:C13H13F7N4O7Purity:98%Color and Shape:SolidMolecular weight:470.25SDH-IN-5
CAS:SDH-IN-5 (compound 7d), a potent inhibitor of succinate dehydrogenase (SDH) with an IC50 of 3.293 μM, additionally demonstrates antifungal efficacy, exhibitingFormula:C16H19F2N3O2Color and Shape:SolidMolecular weight:323.34MFZ 10-7 hydrochloride
CAS:MFZ 10-7 hydrochloride is a highly potent and selective negative allosteric modulator of mGluR5 NAMFormula:C15H10ClFN2Purity:98%Color and Shape:SolidMolecular weight:272.71
