Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,834 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,613 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,015 products)
- Immunology and Inflammation(3,904 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,257 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,137 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,423 products)
- Other Inhibitors(35,848 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(732 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66516 products of "Inhibitors"
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Diethyl butylmalonate
CAS:Diethyl butylmalonate shows toxicity to T. pyriformis, with a log(IGC50 -1 ) of 0.557 [1].Formula:C11H20O4Color and Shape:SolidMolecular weight:216.27Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Formula:C19H26ClN3O2S2Color and Shape:SolidMolecular weight:428.01Dihydrogenistein
CAS:Dihydrogenistein, derived from Genistein, inhibits tyrosine kinases and EGF receptor autophosphorylation.Formula:C15H12O5Color and Shape:SolidMolecular weight:272.25Butyryl-L-carnitine (chloride)
CAS:Butyryl-L-carnitine, a butyrate ester, hinders carnitine/glycine transport in HRPE cells (IC50: 1.5 μM/4.6 mM).Formula:C11H22ClNO4Color and Shape:SolidMolecular weight:267.75Ceftibuten
CAS:Ceftibuten is a third-generation cephalosporin antibiotic.Formula:C15H14N4O6S2Purity:98%Color and Shape:SolidMolecular weight:410.42CPI-1612
CAS:CPI-1612: Oral EP300/CBP HAT inhibitor, IC50 8.1 nM, has anticancer properties.Formula:C27H26N6OColor and Shape:SolidMolecular weight:450.53Syntelin
CAS:Syntelin: a selective CENP-E inhibitor with an IC50 of 160 nM; distinct from GSK923295, effective on resistant mutants.Formula:C21H20N6O2S3Color and Shape:SolidMolecular weight:484.62Dinapsoline
CAS:Dinapsoline is a drug developed for the treatment of Parkinson's disease, that acts as a selective full agonist at the dopamine D1 receptor.Formula:C16H16BrNO2Color and Shape:SolidMolecular weight:334.21Nampt-IN-3
CAS:Nampt-IN-3 simultaneously inhibit nicotinamide phosphoribosyltransferase (NAMPT) and HDAC (IC50s of 31 nM and 55 nM, respectively).Formula:C29H25N7O2Purity:98%Color and Shape:SolidMolecular weight:503.55LEO 39652
CAS:LEO 39652: Dual-soft PDE4 inhibitor, IC50s: PDE4A/B: 1.2 nM, PDE4C: 3.0 nM, PDE4D: 3.8 nM; TNF-α IC50: 6.0 nM; for Atopic dermatitis research.Formula:C23H23N3O5Color and Shape:SolidMolecular weight:421.45CCR4 antagonist 3-1
CAS:CCR4 antagonist 3-1 is a weak inhibitor of [125I]TARC binding and CEM cell migration, with IC50 values of 1.7 μM and 6.4 μM, respectively.Formula:C14H12N2SPurity:99.87%Color and Shape:SolidMolecular weight:240.32Metallo-β-lactamase-IN-8
CAS:Metallo-β-lactamase-IN-8 (compound 17) is a potent, reversible and competitive broad-spectrum metallo-β-lactamases (MβLs) inhibitor with antibacterial activity.Formula:C13H11ClN2O4SColor and Shape:SolidMolecular weight:326.76Neuraminidase-IN-8
CAS:Neuraminidase-IN-8 (Compound 6d) is a powerful inhibitor of neuraminidase, exhibiting a low half-maximal inhibitory concentration (IC50) of 0.027 μM andFormula:C18H16FN3O3SColor and Shape:SolidMolecular weight:373.4LY 207702
CAS:LY 207702, a difluorinated purine nucleoside, exhibits antitumor activity in preclinical models.Formula:C10H12F2N6O3Purity:98%Color and Shape:SolidMolecular weight:302.24Adefovir diphosphate
CAS:Adefovir monophosphate: antiviral ANP active against HBV, herpes; ntRTI for hepatitis B, not HIV-1 effective.Formula:C8H13N5O7P2Color and Shape:SolidMolecular weight:353.17PF-03463275 2HCl
CAS:PF-03463275 is an orally available, CNS-penetrant inhibitor of SLC6A9, a GlyT1 glycine transporter.Formula:C19H24Cl3FN4OPurity:98%Color and Shape:SolidMolecular weight:449.78(3R,4R)-A2-32-01
CAS:(3R,4R)-A2-32-01 is the (R,R)-enantiomer of A2-32-01 and has potential antibacterial activity.Formula:C19H27NO2Purity:98.19%Color and Shape:SolidMolecular weight:301.42A 924
CAS:A 924 is an amino acid derivative with antineoplastic activity.Formula:C30H57N7O11Color and Shape:SolidMolecular weight:691.81Ici 186756
CAS:Ici 186756 is a novel, effective, and selective inhibitor of human neutrophil elastase.Formula:C33H49N5O9Purity:98%Color and Shape:SolidMolecular weight:659.77SCR1693
CAS:SCR1693 is a dual acetylcholinesterase inhibitor (AChEI) and a calcium channel blocker (CCB).Formula:C24H28ClN3O2Color and Shape:SolidMolecular weight:425.95DDPM-2571 HCl
CAS:DDPM-2571: Potent GABA transporter 1 inhibitor, anticonvulsant, anxiolytic, antidepressant, antinociceptive, prevents seizures, quick brain uptake.Formula:C21H21Cl3N2O3Color and Shape:SolidMolecular weight:455.76Rudolfomycin
CAS:Rudolfomycin is a class II anthracycline antitumor antibiotic that inhibit the synthesis of nucleolar RNA in intact tumor cells.Formula:C42H52N2O16Color and Shape:SolidMolecular weight:840.87Hexestrol dipropionate
CAS:Hexestrol dipropionate: synthetic ER agonist, halts microtubule growth, may cause cancer, disrupts cell division, and damages DNA.Formula:C24H30O4Color and Shape:SolidMolecular weight:382.49Diltiazem malate
CAS:Diltiazem malate is an ACE inhibitor and non-dihydropyridine calcium channel blocker used in the treatment of hypertension.Formula:C26H32N2O9SColor and Shape:SolidMolecular weight:548.60HPK1-IN-17
CAS:HPK1-IN-17 selectively inhibits HPK1, a MAP4Ks family kinase from blood progenitor cells; useful against HPK1-related diseases like cancer.Formula:C26H28N6OColor and Shape:SolidMolecular weight:440.54Tazolol HCl
CAS:Tazolol HCl is a selective beta1-agonist, coronartherapeutic agent, and cardiotonic agent.Formula:C9H17ClN2O2SColor and Shape:SolidMolecular weight:252.76mSIRK
CAS:mSIRK (G-Protein βγ Binding Peptide) is an ERK1 and ERK2 dual activator that promotes alpha-subunit dissociation.Formula:C93H150N20O25Purity:99.26%Color and Shape:SolidMolecular weight:1948.31Dipicrylamine Sodium Salt
CAS:Dipicrylamine sodium salt is an effective antagonist of the GABAA receptor.Formula:C12H5N7NaO12Color and Shape:SolidMolecular weight:462.199Diamthazole
CAS:Diamthazole (Dimazole) is an antifungal agent that can be used in the infection research[1].Formula:C15H23N3OSColor and Shape:SolidMolecular weight:293.43FQ
CAS:FQ is a novel reversible inhibitor of mixed-type tyrosinase.Formula:C14H9FN2OColor and Shape:SolidMolecular weight:240.23Epitizide
CAS:Epitizide, a benzothiadiazine, commonly found in combination Triamterene , is used to produce diuresis [1] .Formula:C10H11ClF3N3O4S3Color and Shape:SolidMolecular weight:425.86p,p'-DDMS
CAS:p,p'-DDMS is a water soluble and highly specific inhibitor of cytochrome P-450 omega-hydroxylase.Formula:C14H11Cl3Color and Shape:SolidMolecular weight:285.613-Hydroxystevane
CAS:13-Hydroxystevane shows an inhibitory action on oxidative phosphorylation.Formula:C20H34OPurity:98%Color and Shape:SolidMolecular weight:290.48Azalanstat HCl
CAS:Azalanstat: anti-obesity drug, inhibits cholesterol synthesis by blocking lanosterol 14α-demethylase, reduces LDL cholesterol in hamsters.Formula:C22H26Cl3N3O2SColor and Shape:SolidMolecular weight:502.879(Z)-4EGI-1
CAS:(Z)-4EGI-1, a Z-isomer, inhibits eIF4E/eIF4G; binds eIF4E (IC50=43.5 μM, Kd=8.74 μM); anticancer properties.Formula:C18H12Cl2N4O4SColor and Shape:SolidMolecular weight:451.28BRD4-BD1-IN-1
CAS:BRD4-BD1-IN-1 (Compound 9a) is a BRD4-BD1 inhibitor(IC50= 38.20 μM).Formula:C16H15BrN4O4Color and Shape:SolidMolecular weight:407.22U-89843A
CAS:U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].Formula:C16H24ClN5Purity:98%Color and Shape:SolidMolecular weight:321.85(R)-Viloxazine Hydrochloride
CAS:(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.Formula:C13H20ClNO3Purity:99.88% - 99.94%Color and Shape:SolidMolecular weight:273.76Ref: TM-T22413
1mg52.00€5mg111.00€10mg162.00€25mg235.00€50mg330.00€100mg452.00€200mg607.00€1mL*10mM (DMSO)101.00€Nimbocinone
CAS:Nimbocinone shows antidiabetogenic activity.Formula:C30H46O4Color and Shape:SolidMolecular weight:470.68GSK466317A
CAS:GSK466317A is a GRK2 inhibitor.Formula:C21H16ClF3N4O2Purity:98%Color and Shape:SolidMolecular weight:448.83UBP-282
CAS:AMPA and kainate receptor antagonistFormula:C15H15N3O6Purity:98%Color and Shape:SolidMolecular weight:333.3WJ35435
CAS:WJ35435 is a histone deacetylase and topoisomerase I dual inhibitor.Formula:C20H21N3O3Purity:98%Color and Shape:SolidMolecular weight:351.4OUP-186
CAS:OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.Formula:C19H30ClN3SColor and Shape:SolidMolecular weight:367.98TC-1698 dihydrochloride
CAS:TC-1698 dihydrochloride: selective α7 nicotinic agonist, with some β-receptor activity; neuroprotectant.Formula:C13H20Cl2N2Color and Shape:SolidMolecular weight:275.22Antitumor agent-90
CAS:Antitumor Agent-90 exhibits cytotoxic effects against PC 14 and MKN 45 cells, indicating its potential utility in cancer research.Formula:C10H4N4O2Color and Shape:SolidMolecular weight:212.16DNA-PK-IN-7
CAS:DNA-PK-IN-7 is a potent DNA-PK inhibitor (IC50= 1 nM) (WO2021104277A1, compound 5).Formula:C19H21N9O2Color and Shape:SolidMolecular weight:407.43ML309
CAS:ML309 inhibits R132H mutant IDH1, reduces 2-HG in U87 MG glioblastoma.Formula:C29H29FN4O2Color and Shape:SolidMolecular weight:484.56Dichlorodenafil
CAS:Dichlorodenafil is an inhibitor of phosphodiesterase type 5 enzyme (PDE-5).Formula:C19H20Cl2N4O2Color and Shape:SolidMolecular weight:407.29Caylin-2
CAS:Nutlin-3 activates p53 by blocking MDM2. Caylin-2, a nutlin-3 analog with trifluoromethyl instead of chlorine, is 10x less potent with an 8 μM IC50.Formula:C32H30F6N4O4Color and Shape:SolidMolecular weight:648.6Trichomonacid
CAS:Trichomonacid inhibits M. marinum MelF, halting M. marinum and M. tuberculosis growth.Formula:C27H43N4O15P3Color and Shape:SolidMolecular weight:756.57
