Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,833 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,612 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,015 products)
- Immunology and Inflammation(3,901 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,153 products)
- Metabolism(10,139 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,391 products)
- Other Inhibitors(35,852 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66520 products of "Inhibitors"
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Dacopafant
CAS:Dacopafant is an antagonist of platlet activationg factor receptor.Formula:C12H11N3OSColor and Shape:SolidMolecular weight:245.3UNC5452
CAS:UNC5452 is a Nek1 inhibitor.Formula:C17H20N4O2SColor and Shape:SolidMolecular weight:344.43Primapterin
CAS:Primapterin, 7-Substituted pterins, is a new type of mammalian pteridines.Formula:C9H11N5O3Color and Shape:SolidMolecular weight:237.22ML-148
CAS:ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM).Formula:C20H21N3OPurity:99.88%Color and Shape:SolidMolecular weight:319.4Ref: TM-T38163
1mg60.00€5mg165.00€10mg254.00€25mg459.00€50mg658.00€100mg935.00€200mg1,283.00€1mL*10mM (DMSO)188.00€Methanesulfonic acid, compd. with α-(ethylthio)-4-(octyloxy)-m-toluidine (7CI)
CAS:Methanesulfonic acid, compd. with alpha-(ethylthio)-4-(octyloxy)-m-toluidine (7CI) is a bioactive chemical.Formula:C18H33NO4S2Color and Shape:SolidMolecular weight:391.59ATSP-7041
CAS:ATSP-7041 is a novel potent and selective dual inhibitor of mdm2 (ki = 0.9 nm) and mdmx (ki = 7 nm)Formula:C87H125N17O21Color and Shape:SolidMolecular weight:1745.02Chlorozotocin
CAS:Chlorozotocin is a nitrosourea. It is used for cancer therapy.Formula:C9H16ClN3O7Color and Shape:SolidMolecular weight:313.69Pacrinolol
CAS:Pacrinolol is a beta adrenergic receptor antagonist.Formula:C23H28N2O4Color and Shape:SolidMolecular weight:396.48Cafaminol
CAS:Cafaminol (methylcoffanolamine) is a vasoconstrictor and anticatarrhal of the methylxanthine family related to caffeine which is used as a nasal decongestant.Formula:C11H17N5O3Color and Shape:SolidMolecular weight:267.28LFS-829
CAS:LFS-829: small molecule, inhibits exportin-1, low nanomolar activity, orally reverses colitis in mice, low toxicity, promising for clinical trials.Formula:C13H9F6NOS2Color and Shape:SolidMolecular weight:373.34β-Lactamase-IN-7
CAS:β-Lactamase-IN-7 (compound 14) effectively inhibit Klebsiella pneumoniae that is a potent inhibitor of VIM-Type metallo-β-lactamase with Ki values of 1.26 μMFormula:C16H15N3S2Color and Shape:SolidMolecular weight:313.44Amthamine dihydrobromide
CAS:H2 agonistFormula:C6H13Br2N3SPurity:98%Color and Shape:SolidMolecular weight:319.06HMR-1566
CAS:HMR-1566 is a potent and selective Iks channel blocker.Formula:C18H26F3NO5SColor and Shape:SolidMolecular weight:425.46AGI-41998
CAS:AGI-41998: a potent MAT2A inhibitor that crosses the blood-brain barrier, targeting SAM enzymes for cancer therapy and CNS research.Formula:C22H16BrF3N4O2Color and Shape:SolidMolecular weight:505.29PF-06279794
CAS:PF-06279794 is a potent, selective and ATP-competitive TNIK inhibitor.Formula:C22H20N4OColor and Shape:SolidMolecular weight:356.42AHR-5645B free base
CAS:AHR-5645B free base is a substituted benzamide which has been shown to inhibit 3H-spiperone binding to bovine anterior pituitary membranes.Formula:C18H27N3OColor and Shape:SolidMolecular weight:301.43Oxypertine
CAS:Oxypertine, an indole-derived antipsychotic, treats psychoses like mania, schizophrenia, and severe anxiety, akin to chlorpromazine.Formula:C23H29N3O2Color and Shape:SolidMolecular weight:379.5CYD-2-11
CAS:CYD-2-11 is an effective and selective Bax agonist. It acts by targeting the structural pocket proximal to S184 in the C-terminal region of Bax.Formula:C22H18N2O3Color and Shape:SolidMolecular weight:358.39Methsuximide
CAS:Methsuximide is an anticonvulsant agent which appeared to be effective in petit mal, psychomotor and focal motor attacks [1].Formula:C12H13NO2Color and Shape:Crystals From Dilute Alcohol SolidMolecular weight:203.24RA-2
CAS:RA-2 is a pan-negative-gating modulator of KCa2/3 channels that acts by inhibiting EDH-type relaxation in coronary arteries.Formula:C22H16F2O6Color and Shape:SolidMolecular weight:414.36S7958
CAS:S7958 is a is a TAS2R8 antagonist. It was found to be non-mutagenic in vitro.Formula:C21H23N5O4Color and Shape:SolidMolecular weight:409.44TRPC6-IN-3
CAS:TRPC6-IN-3 is an oral TRPC6 ion channel inhibitor, regulating calcium levels and membrane potential.Formula:C22H22FN5O3Color and Shape:SolidMolecular weight:423.44Tubulin inhibitor 18
CAS:"Tubulin inhibitor 18 (5j), a potent chalcone, uniquely structured for cancer research."Formula:C22H26O5Color and Shape:SolidMolecular weight:370.44Synstab A
CAS:Synstab A is a microtubule stabilizer.Formula:C15H13BrCl3N3O3SColor and Shape:SolidMolecular weight:501.61PI3-Kinase α Inhibitor 2
CAS:Phosphatidylinositol 3-kinase (PI3K) catalyzes the phosphorylation of the 3' hydroxyl position of PIs to produce the second messengers PtdIns-(3,4)-P2 andFormula:C16H15N3O2SColor and Shape:SolidMolecular weight:313.37Dichloro-all-trans-retinone
CAS:Dichloro-all-trans-retinone is a selective inhibitor for retinaldehyde dehydrogenase enzymes, thereby irreversibly inhibiting RALDH1, 2, and 3.Formula:C21H28Cl2OColor and Shape:SolidMolecular weight:367.35Antiviral agent 23
CAS:Antiviral agent 23 targets EV71 with 94 nM EC50 and suppresses METTL3/14, useful in infection research.Formula:C18H21N5O4Color and Shape:SolidMolecular weight:371.39A-971432
CAS:A-971432: selective S1P5 agonist, IC50 = 0.006 µM. Enhances blood-brain barrier, reduces Huntington’s symptoms in mice at 0.1 mg/kg.Formula:C18H17Cl2NO3Color and Shape:SolidMolecular weight:366.24A-366833
CAS:A-366833: Abbott's nicotinic receptor ligand, Ki=3.1 nM at agonist site, selective for alpha4beta2 NACHR.Formula:C11H12N4Color and Shape:SolidMolecular weight:200.24BzDANP
CAS:BzDANP is a modulator of pre-miR-29a maturation by Dicer.Formula:C18H24N6Color and Shape:SolidMolecular weight:324.42Isodispar B
CAS:Isodispar B: an anticancer drug, halts many cancer types' growth, triggers cell death.Formula:C20H18O5Color and Shape:SolidMolecular weight:338.35Mipicoledine
CAS:DM-CHOC-PEN is a DNA alkylation agent that may be used to treat brain cancer.Formula:C35H48Cl5NO4Color and Shape:SolidMolecular weight:724.02Tyrphostin A46
CAS:Tyrphostin A46 is an antagonist of the epidermal growth factor-urogastrone receptor.Formula:C10H8N2O3Purity:98%Color and Shape:Off-White SolidMolecular weight:204.18α-Glucosidase-IN-8
CAS:α-Glucosidase-IN-8 (Compound 4k) is a potent, competitive inhibitor of α-glucosidase. It displays an impressive IC50 value of 0.18 μg/mL [1].Formula:C19H20FN3O2Color and Shape:SolidMolecular weight:341.38GK-136901
CAS:GK-136901 is a first-in-class, potent, and orally bioavailable NADPH oxidase isoform 4 (Nox4) inhibitor.Formula:C20H18N4O2Color and Shape:SolidMolecular weight:346.384,4'-Dicyanostilbene
CAS:4,4'-Dicyanostilbene: potent anti-Dd2 malaria, EC50=27nM; effective vs. MRSA.Formula:C16H10N2Color and Shape:SolidMolecular weight:230.26BI-1622
CAS:BI-1622, an oral HER2 inhibitor, IC50: 7 nM, >25x selectivity over EGFR, shows effective in vivo antitumor activity.Formula:C26H24N10O2Color and Shape:SolidMolecular weight:508.53Vilazodone carboxylic acid
CAS:Vilazodone carboxylic acid is a vilazodone metabolite observed in both urine and plasma.Formula:C26H26N4O3Purity:98%Color and Shape:SolidMolecular weight:442.51S-methyl DM1
CAS:S-methyl DM1 is a thiomethyl derivative of Maytansine. S-methyl DM1 binds to tubulin(Kd of 0.93 μM) and inhibts microtubule polymerization.Formula:C36H50ClN3O10SPurity:98%Color and Shape:SolidMolecular weight:752.31CAY10506
CAS:CAY10506, a hybrid lipoic acid-TZD, activates PPARγ to control glucose and lipid levels with an EC50 of 10 μM.Formula:C20H26N2O4S3Color and Shape:SolidMolecular weight:454.63Anti-inflammatory agent 15
CAS:Compound 29, anti-inflammatory and antimycobacterial, halts Mtb H37Rv and M299 growth; MIC50 at 2.3 and 7.8 μM. Blocks iNOS, TNF-α, IL-1β.Formula:C17H20N2SColor and Shape:SolidMolecular weight:284.42A23887
CAS:A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formula:C22H24ClNPurity:98%Color and Shape:SolidMolecular weight:337.89Ro 22-0654
CAS:Ro 22-0654, a novel lipid synthesis inhibitor, has antiobesity effects.Formula:C8H11NO2SPurity:98%Color and Shape:SolidMolecular weight:185.24SC 42619
CAS:SC 42619 is a tripeptide analogue that inhibits aggregation of, and secretion from, human platelets.Formula:C15H28N2O3Color and Shape:SolidMolecular weight:284.39KRAS inhibitor-15
CAS:KRAS inhibitor-15 blocks KRAS G12C and p-ERK in cancer cells; potent against pancreatic and lung cancers. IC50: 0.954 μM (KRAS), 2.03/>33.3 μM (p-ERK).Formula:C20H17Cl2FN4OSColor and Shape:SolidMolecular weight:451.34Darexaban glucuronide
CAS:Darexaban glucuronide is the major component in plasma after oral administration of darexaban to humans. Darexaban (YM150) is a direct inhibitor of factor Xa.Formula:C33H38N4O10Color and Shape:SolidMolecular weight:650.68Lexibulin dihydrochloride
CAS:Lexibulin 2HCl inhibits tubulin polymerization (IC50: 10-100 nM) and shows potent anti-cancer cytotoxicity and vascular disruption in vitro/vivo.Formula:C24H32Cl2N6O2Purity:98%Color and Shape:SolidMolecular weight:507.46Chlorambucyl-proline
CAS:Chlorambucyl-proline is a chlorambucil derivative of L-proline. It is an inhibitor of bovine lung angiotensin I-converting enzyme.Formula:C19H26Cl2N2O3Purity:98%Color and Shape:SolidMolecular weight:401.33OXA-06 Dihydrochloride
CAS:OXA-06 Dihydrochloride is a PANC-1 cell migration and MYPT1 phosphorylation inhibitor.Formula:C21H18FN3Purity:98%Color and Shape:SolidMolecular weight:331.39IND8
CAS:IND8 is a selective and potent α7-nAChR agonist.Formula:C17H19N5Color and Shape:SolidMolecular weight:293.37
