Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,746 products)
- Apoptosis(6,181 products)
- Cell Cycle/Checkpoint(4,806 products)
- Chromatin/Epigenetics(2,567 products)
- Cytoskeletal Signaling(1,498 products)
- DNA Damage/DNA Repair(2,897 products)
- Endocrinology/Hormones(3,701 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,960 products)
- Immunology and Inflammation(3,692 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,244 products)
- Membrane Transporter/Ion Channel(3,135 products)
- Metabolism(10,101 products)
- Microbiology/Virology(7,550 products)
- Neuroscience(10,300 products)
- Other Inhibitors(35,772 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,400 products)
- Proteases/Proteasome(1,670 products)
- Stem Cell and Derivatives(742 products)
- Tyrosine Kinase/Adaptors(1,922 products)
- Ubiquitination(1,715 products)
Show 16 more subcategories
Found 66578 products of "Inhibitors"
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Antileishmanial agent-13
CAS:Antileishmanial agent-13, a quinoline-isatin hybrid, targets L. Major with IC50s of 0.604 μM (promastigote) and 0.508 μM (amastigote).Formula:C17H10BrClN4OColor and Shape:SolidMolecular weight:401.64UL04
CAS:UL04 is an inhibitor of CREBBP bromodomain.Formula:C18H17NO5Color and Shape:SolidMolecular weight:327.33ARN726
CAS:ARN726, potent NAAA inhibitor, IC50 of 0.073 μM, reduces alcohol craving dose-dependently.Formula:C14H24N2O3Color and Shape:SolidMolecular weight:268.35Dizocilpine
CAS:MK-801 (Dizocilpine (MK-801)) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.Formula:C16H15NPurity:99.85% - 99.97%Color and Shape:SolidMolecular weight:221.3IDO1-IN-19
CAS:IDO1-IN-19 (Compound 17) is a potent inhibitor of IDO1 and has potential for cancer disease research.Formula:C25H22F4N2O3Color and Shape:SolidMolecular weight:474.45PF-5274857 mseylate (1373615-35-0 free base)
PF-5274857: oral hedgehog pathway inhibitor, IC50=5.8 nM, crosses blood-brain barrier, boosts survival in medulloblastoma mice.Formula:C21H29ClN4O6S2Purity:98%Color and Shape:SolidMolecular weight:533.06COX-2/sEH-IN-1
CAS:COX-2/sEH-IN-1, oral dual inhibitor: COX-2 (IC50=1.24 μM), sEH (IC50=0.40 μM); boosts anti-inflammatory action, cuts heart risk.Formula:C23H18F3N5O3SColor and Shape:SolidMolecular weight:501.48Autophagy inducer 4
CAS:Autophagy inducer 4, a Magnolol-based Mannich derivative, is an anticancer agent that blocks cancer cell migration & is 76x more toxic to T47D cells.Formula:C32H37NO6Color and Shape:SolidMolecular weight:531.64Ganstigmine
CAS:Ganstigmine is an acetylcholinesterase inhibitor for Alzheimer's disease.Formula:C22H27N3O3Color and Shape:SolidMolecular weight:381.47Flestolol sulfate
CAS:Flestolol sulfate is an anti-adrenergic beta-receptor.Formula:C15H24FN3O8SColor and Shape:SolidMolecular weight:425.43Gleditsioside A
CAS:Gleditsioside A is a useful organic compound for research related to life sciences. The catalog number is T125267 and the CAS number is 230302-68-8.Formula:C78H124O35Color and Shape:SolidMolecular weight:1621.82Oleyl Mesylate
CAS:Oleyl Mesylate is a derivative of oleyl alcohol that can be incorporated into various formulations.
Formula:C19H38O3SPurity:99.64%Color and Shape:SolidMolecular weight:346.57Sarcolysine hydrochloride
CAS:Sarcolysine hydrochloride, also known as Melphalan HCl, is a nitrogen mustard and alkylating agent that has been studied for use in multiple myeloma therapy.Formula:C13H19Cl3N2O2Color and Shape:SolidMolecular weight:341.66YH-306
CAS:YH-306 (TRV055 acetate ) is a modulator of the FAK signaling pathway that acts by suppressing colorectal tumor growth and metastasis.Formula:C19H18N2O2Purity:98.06%Color and Shape:SolidMolecular weight:306.36CDK9/CycT1-IN-93
CAS:CDK9/CycT1-IN-93 is a highly specific, ATP-competitive inhibitor of CDK9/CycT1 with antiviral activity.Formula:C27H28N3O3PColor and Shape:SolidMolecular weight:473.54-CPI
CAS:4-CPI inhibits non-active site mutants of cytochrome P450 2B4.Formula:C9H7ClN2Purity:98%Color and Shape:SolidMolecular weight:178.62OX11
CAS:OX11 is a selective inhibitor of S. pneumoniae, P. aeruginosa and E. coli bacteria.Formula:C17H10Cl2N4O3S2Color and Shape:SolidMolecular weight:453.32Novembichin
CAS:Novembichin is a nitrogen mustard agent that crosslinks with DNA, causing inhibition of DNA synthesis.Formula:C7H15Cl4NColor and Shape:SolidMolecular weight:255THK-5117
CAS:THK-5117, a tau PET probe, has a high tau fibril affinity (Ki 10.5 nM) and binds well to AD brain aggregates.Formula:C19H19FN2O2Color and Shape:SolidMolecular weight:326.36Fuberidazole
CAS:Fuberidazole is an antifungal agent.Formula:C11H8N2OPurity:98.95%Molecular weight:184.19BMH-9
CAS:BMH-9 is an RNA polymerase I inhibitor that acts by causing nucleolar stress and showing potent anticancer activity across many tumor types.Formula:C19H27N3O2Color and Shape:SolidMolecular weight:329.44Sulforemate
CAS:Sulforemate is a phase II enzyme inducer for chemopreventive activities.Formula:C7H15NOS3Color and Shape:SolidMolecular weight:225.4DA 4626
CAS:DA 4626 is an H2-receptor antagonist with KB values akin to those in standard assays.Formula:C14H18N4Purity:98%Color and Shape:SolidMolecular weight:242.32LEI-101
CAS:LEI-101: potent CB2 agonist, pEC50=8, bioavailable, >100x selective over CB1, potential for inflammatory diseases.Formula:C23H25FN4O4SPurity:98%Color and Shape:SolidMolecular weight:472.53HUHS2002
CAS:HUHS2002 is a free fatty acid derivative that works as a potentiator of GluA1 AMPA receptor responses and α7 ACh receptor responses.Formula:C17H24O3Purity:98%Color and Shape:SolidMolecular weight:276.37SARS-CoV-2 3CLpro-IN-1
CAS:SARS-CoV-2 3CLpro-IN-1 is a potent inhibitor of the key enzyme 3CL pro in coronaviruses, promising for antiviral drug R&D.Formula:C27H30ClN3O3SColor and Shape:SolidMolecular weight:512.06AL 8697
CAS:AL 8697 is a selective p38α MAPK inhibitor (IC50 = 6 nM) with 14-fold selectivity over p38β (IC50 = 82 nM) and 300-fold selectivity over a panel of 91 kinases.
Formula:C21H21F3N4OPurity:99.55% - 99.89%Color and Shape:SolidMolecular weight:402.41Saikosaponin B4
CAS:Saikosaponin B4 is isolated from the MeOH extract of the roots of Bupleurum falcatum L.Formula:C43H72O14Purity:99.03%Color and Shape:SolidMolecular weight:813.02JNJ-10191584
CAS:JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammationFormula:C13H15ClN4OColor and Shape:SolidMolecular weight:278.74Aminochlorthenoxazin
CAS:Aminochlorthenoxazin is an antipyretic and analgesic agent.Formula:C10H11ClN2O2Purity:98%Color and Shape:SolidMolecular weight:226.66Ibulocydine
CAS:Ibulocydine: potent CDK inhibitor, targets Cdk7/9, more effective than others on HCC cells, minimal impact on normal hepatocytes, induces apoptosis.Formula:C16H20BrN5O6Color and Shape:SolidMolecular weight:458.262-PAT
CAS:2-PAT: reversible MAO-A inhib., IC50=0.721 µM; MAO-B inactivator, IC50=14.6 µM; potential in Parkinson's/depression study.Formula:C13H15NColor and Shape:SolidMolecular weight:185.26Estrogen receptor antagonist 2
CAS:ER antagonist 2 selectively suppresses ERα, a key breast cancer driver, with research potential in the disease.Formula:C26H31F4N5Color and Shape:SolidMolecular weight:489.55AKT-IN-5
CAS:AKT-IN-5, an Akt inhibitor, targets Akt1/Akt2 with IC50s: 450/400 nM.Formula:C23H20N4O2Color and Shape:SolidMolecular weight:384.43SKF-83566 hydrobromide
CAS:D1-like dopamine receptor antagonistFormula:C17H19BrClNOPurity:98%Color and Shape:SolidMolecular weight:368.7L162441
CAS:L162441 is an antagonist of Angiotensin type 1 receptor.Formula:C34H43N5O5SPurity:98%Color and Shape:SolidMolecular weight:633.8LabMol-301
CAS:LabMol-301 blocks NS5 RdRp/NS2B-NS3pro (IC50: 0.8/7.4µM), protects cells from ZIKV death.Formula:C18H16N6Color and Shape:SolidMolecular weight:316.36Carboxyamidotriazole
CAS:Carboxyamidotriazole is a cytostatic inhibitor of non-voltage-operated calcium channels and calcium channel-mediated signaling pathways.Formula:C17H12Cl3N5O2Purity:98%Color and Shape:SolidMolecular weight:424.67LY-104119
CAS:LY-104119: weight loss agent, lowers noradrenaline in brown fat, heart, liver.Formula:C19H25ClN2O2Color and Shape:SolidMolecular weight:348.87EF-7412
CAS:EF-7412 is a ligand that is characterized as an antagonist in vivo in pre- and postsynaptic 5-HT(1A)R sites.Formula:C22H33N5O4SColor and Shape:SolidMolecular weight:463.59ANAPP3
CAS:ANAPP3 is a P2x-purinoceptor antagonist. It affects contractions in various muscle groups and tissues.Formula:C19H23N10O16P3Color and Shape:SolidMolecular weight:740.37Remeglurant
CAS:Remeglurant is used as a selective antagonist of the mGlu5 receptor.Formula:C17H15BrN4OColor and Shape:SolidMolecular weight:371.23Suclofenide
CAS:Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.Formula:C16H13ClN2O4SPurity:98%Color and Shape:SolidMolecular weight:364.8Keap1-Nrf2-IN-14
CAS:Keap1-Nrf2-IN-14, a KEAP1-NRF2 inhibitor (IC50: 75 nM, Kd: 24 nM), boosts NRF2 gene expression, antioxidative and anti-inflammatory response.Formula:C30H29NO8SColor and Shape:SolidMolecular weight:563.62EGFR/HER2-IN-3
CAS:EGFR/HER2-IN-3 (Compound ZINC21942954) is a dual EGFR and HER2 inhibitor.Formula:C26H23N5O3Color and Shape:SolidMolecular weight:453.49SN00799639
CAS:SN00799639 (SN639) inhibits Haemonchus contortus larvae; IC50: 8.4 μM (motility), 0.29 μM (development).Formula:C17H18N4OSColor and Shape:SolidMolecular weight:326.42ICRF-196
CAS:ICRF-196 is a Topoisomerase II Inhibitor and antineoplastic agent.Formula:C12H18N4O4Color and Shape:SolidMolecular weight:282.3Rolafagrel
CAS:Rolafagrel is a novel inhibitor of thromboxane synthase.Formula:C14H12N2O2Color and Shape:SolidMolecular weight:240.26HAT-IN-1
CAS:HAT-IN-1 is an inhibitor of HAT used in the research of cancer.Formula:C23H18BrF4N3O4Purity:98%Color and Shape:SolidMolecular weight:556.3VMY-1-101
CAS:VMY-1-101: synthetic fluorescent CDK inhibitor with strong activity, increases G2/M arrest, and induces more apoptosis than purvalanol B.Formula:C33H40ClN9O4SColor and Shape:SolidMolecular weight:694.25
