Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,782 products)
- Apoptosis(6,263 products)
- Cell Cycle/Checkpoint(4,792 products)
- Chromatin/Epigenetics(2,441 products)
- Cytoskeletal Signaling(1,528 products)
- DNA Damage/DNA Repair(2,965 products)
- Endocrinology/Hormones(3,707 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,009 products)
- Immunology and Inflammation(3,875 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,248 products)
- Membrane Transporter/Ion Channel(3,033 products)
- Metabolism(10,209 products)
- Microbiology/Virology(7,592 products)
- Neuroscience(10,381 products)
- Other Inhibitors(36,040 products)
- Oxidation-Reduction(42 products)
- PI3K/Akt/mTOR Signaling(1,442 products)
- Proteases/Proteasome(1,724 products)
- Stem Cell and Derivatives(826 products)
- Tyrosine Kinase/Adaptors(2,035 products)
- Ubiquitination(1,717 products)
Show 16 more subcategories
Found 66683 products of "Inhibitors"
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TTA-Q6
CAS:TTA-Q6 is a T-type Ca2+ channel antagonist that inhibits the uptake of extracellular calcium ions by tumour cells for the treatment of neurological diseases.Formula:C20H15ClF3N3OPurity:99.97%Color and Shape:SolidMolecular weight:405.8MG 1
CAS:MG 1 is a potent alpha-1 adrenergic receptor antagonist.Formula:C17H25N3O2Purity:98.98% - >99.99%Color and Shape:SolidMolecular weight:303.4Desethylreboxetine
CAS:Desethylreboxetine is an desethylated metabolite of Reboxetine (R142000), a selective noradrenaline reuptake inhibitor and an antidepressant.Formula:C17H19NO3Color and Shape:SolidMolecular weight:285.34Formylmethionyl-alanyl-leucine
CAS:Formylmethionyl-alanyl-leucine is formed by E coli ribosomal protein L10 gene.Formula:C15H27N3O5SColor and Shape:SolidMolecular weight:361.46KDM2B-IN-3
CAS:KDM2B-IN-3, from patent WO2016112284A1 as compound 183c, potently inhibits histone demethylase KDM2B, with cancer research potential.Formula:C25H30N2O2Color and Shape:SolidMolecular weight:390.52AI-3
CAS:Nrf2/Keap1 and Keap1/Cul3 interaction inhibitorFormula:C11H13ClO3S2Purity:98%Color and Shape:SolidMolecular weight:292.8HIV-1 inhibitor-24
CAS:HIV-1 inhibitor-24 (S-12a) blocks HIV reverse transcription effectively (IC50: 9.5 nM), low toxicity, well-tolerated in mice, good heart safety.Formula:C26H19N5O2Color and Shape:SolidMolecular weight:433.46Emlenoflast sodium
CAS:Emlenoflast sodium (MCC7840 sodium), a sulfonylurea, is a selective NLRP3 inflammasome inhibitor with an IC50 value of less than 100 nM for NLRP3 inflammasome,Formula:C19H24N4NaO3SColor and Shape:SolidMolecular weight:411.47AF40431
CAS:AF40431 is the first reported small-molecule ligand of sortilin (IC50: 4.4 μM; Kd: 0.7 μM). AF40431 is bound in the neurotensin-binding site of sortilin.Formula:C17H21NO5Color and Shape:SolidMolecular weight:319.35Ro-15-2041
CAS:Ro 15-2041 is a selective inhibitor of platelet phosphodiesterase, with antithrombotic properties.Formula:C12H12BrN3OPurity:98%Color and Shape:SolidMolecular weight:294.15Immepip dihydrobromide
CAS:Immepip dihydrobromide is a histamine H3 receptor agonist.Formula:C9H17Br2N3Purity:98%Color and Shape:SolidMolecular weight:327.059(BrMT)2
CAS:(BrMT)2 is an activator of the Kv1.1 potassium ion channel.Formula:C20H20Br2N4S2Color and Shape:SolidMolecular weight:540.34Buclosamide
CAS:Buclosamide is a topical antimycotic agent that can be used in dermatomycoses [1].Formula:C11H14ClNO2Color and Shape:SolidMolecular weight:227.69SIRT6 activator 12q
CAS:SIRT6 activator 12q: potent, selective, oral; IC50 - SIRT1: 171.20μM, SIRT6: 0.58μM; halts cell growth/migration, induces apoptosis, G2 arrest, anticancer.Formula:C31H22N2O2Color and Shape:SolidMolecular weight:454.52MRT80
CAS:MRT80 is an inhibitor of GSK-3 in vitro. MRT80 de-stabilizes MDM2 and stabilizes p53 protein and E2F-1.Formula:C15H15N5OPurity:98%Color and Shape:SolidMolecular weight:281.31MDL-73669
CAS:MDL-73669 is a macrocyclic HIV-protease inhibitor that contains a difluorostatone peptide mimetic.Formula:C38H39F2N3O6Color and Shape:SolidMolecular weight:671.73Kurasoin B
CAS:Kurasoin B is an inhibitor of protein farnesyltransferase.Formula:C18H17NO2Color and Shape:SolidMolecular weight:279.33S-5751
CAS:S-5751, a prostanoid DP (DP1) antagonist, is used potentially for the treatment of bronchial asthma.Formula:C25H31NO4SColor and Shape:SolidMolecular weight:441.58AChE/BChE-IN-5
CAS:AChE/BChE-IN-5 (BMC-16) crosses BBB; IC50: hAChE 266 nM, hBChE 10.6 nM. Dual AChE/BChE inhibitor.Formula:C17H26N2O3Color and Shape:SolidMolecular weight:306.4Gyki 32887
CAS:Gyki 32887 is a dopamine agonist.Formula:C23H28N6O6SPurity:98%Color and Shape:SolidMolecular weight:516.57BI8622
CAS:BI8622 is a HUWE1 antagonist that restores levels of RP2 mutants in retinal cell lines and inhibits cellular activation of NLRP3 and AIM2 inflammatory vesicles.Formula:C25H26N6OPurity:98.28% - 98.28%Color and Shape:SolidMolecular weight:426.51YM-341619
CAS:YM-341619 (AS1617612), potent STAT6 inhibitor; IC50: 0.70 nM; hinders IL-4-induced Th2 in mice; may aid allergic disease research.Formula:C22H21F3N6O2Color and Shape:SolidMolecular weight:458.44TMV-IN-1
CAS:TMV-IN-1: a chalcone inhibits TMV with EC50s of 70.7 and 60.8 μg/mL, applicable in infection and tumor studies.Formula:C28H26O4Color and Shape:SolidMolecular weight:426.5MCC-134
CAS:MCC-134 is an inverse agonist for the pancreatic-type ATP-sensitive K(+) channel. It also used as a vascular relaxing agent.Formula:C16H17N3OSColor and Shape:SolidMolecular weight:299.39Clopenthixol decanoate
CAS:Clopenthixol decanoate: thioxanthene, akin to phenothiazine antipsychotics, blocks D1/D2 dopamine receptors.Formula:C32H43ClN2O2SColor and Shape:SolidMolecular weight:555.21Ecadotril
CAS:Ecadotril is a neutral endopeptidase (NEP) inhibitor, which plays an anti hypertensive role.Formula:C21H23NO4SColor and Shape:SolidMolecular weight:385.48Carburazepam
CAS:Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.Formula:C17H16ClN3O2Purity:98%Color and Shape:SolidMolecular weight:329.78Bezuclastinib
CAS:Bezuclastinib (CGT9486) is a novel, potent and highly selective tyrosine kinase and c-kit D816V inhibitor for the study of advanced mastocytosis.Formula:C19H17N5OPurity:99.55%Color and Shape:SolidMolecular weight:331.37TPN729
CAS:TPN729, a PDE5 inhibitor, has an IC50 of 2.28 nM, used to research erectile dysfunction.Formula:C25H36N6O4SColor and Shape:SolidMolecular weight:516.66S 8308
CAS:S 8308 is a weak, but specific and competitive, non-peptide antagonist of AII exerting its inhibitory action at the receptor level.Formula:C16H17ClN3NaO4Color and Shape:SolidMolecular weight:373.76KRAS G12C inhibitor 45
CAS:KRAS G12C inhibitor 45 is a potent KRAS G12C inhibitor .Formula:C32H33F2N5O5SColor and Shape:SolidMolecular weight:637.7LP-533401
CAS:LP-533401 is an inhibitor of Tryptophan hydroxylase 1. It is used for regulates serotonin production in the gut.Formula:C27H22F4N4O3Purity:98%Color and Shape:SolidMolecular weight:526.48Bifenazate
CAS:Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.Formula:C17H20N2O3Purity:99.62%Color and Shape:Solid CrystallineMolecular weight:300.35FFN200 dihydrochloride
CAS:FFN200 is a vesicular monoamine transporter 2 (VMAT2) substrate that selectively traces monoamine exocytosis in both neuronal cell culture and brain tissue.Formula:C11H14Cl2N2O2Color and Shape:SolidMolecular weight:277.15Keap1-Nrf2-IN-12
CAS:eap1-Nrf2-IN-12 is a potent inhibitor of Keap1-Nrf2 (IC50: 2.30 μM). eap1-Nrf2-IN-12 is metabolically stable in human liver microsomes.Formula:C26H28N2O10S2Color and Shape:SolidMolecular weight:592.64Hexestrol dibutyrate
CAS:Hexestrol dibutyrate: Synthetic ER activator, microtubule blocker, possible carcinogen, causes mitotic arrest, aneuploidy, and DNA adducts.Formula:C26H34O4Color and Shape:SolidMolecular weight:410.55(S)-Lercanidipine hydrochloride
CAS:(S)-Lercanidipine hydrochloride is the S-enantiomer of Lercanidipine hydrochloride. (S)-lercanidipine hydrochloride is a potent blocker of calcium channel.Formula:C36H42ClN3O6Purity:98%Color and Shape:SolidMolecular weight:648.19c-Kit-IN-3
CAS:c-Kit-IN-3 is a selective inhibitor of c-KIT kinase with IC50s of 4 nM and 8 nM for c-Kit (wt) and c-Kit (T670I).Formula:C26H20ClF3N2O4Purity:99.94%Color and Shape:SolidMolecular weight:516.9Ref: TM-T10651
1mg87.00€5mg162.00€10mg254.00€25mg419.00€50mg562.00€100mg787.00€500mg1,578.00€1mL*10mM (DMSO)334.00€CP-94707
CAS:CP-94707 is a new inhibitor of nonnucleoside reverse transcriptase (NNRTI).Formula:C21H16N4OSColor and Shape:SolidMolecular weight:372.44iBAP-II
CAS:iBAP-II suppresses ASCL1/MYCL/E2F in SCLC, reducing cell viability and tumor growth.Formula:C18H16N2O3Color and Shape:SolidMolecular weight:308.33AqB007
CAS:AqB007 is a selective blocker of the Aquaporin-1 ion channel conductance, thereby slowing cancer cell migration.Formula:C24H35N5O4SColor and Shape:SolidMolecular weight:489.63Vapendavir
CAS:Vapendavir binds enterovirus capsids; effective against EV71 with EC50 of 0.5-1.4 μM.Formula:C21H26N4O3Purity:98%Color and Shape:SolidMolecular weight:382.46TIE-2/VEGFR-2 kinase-IN-1
CAS:TIE-2/VEGFR-2 kinase-IN-1 synthesizes inhibitors for angiogenesis-related disease research.Formula:C13H11N3O2Color and Shape:SolidMolecular weight:241.25DNAC-1
CAS:DNAC-1 is against Gram-positive and Gram-negative pathogens potentiator of β-lactam activity.Formula:C11H9BrN2S2Purity:98%Color and Shape:SolidMolecular weight:313.24CGP 35949
CAS:CGP 35949 is an LTD4 antagonist with phospholipase inhibitory activity.Formula:C23H25ClN5NaO5Purity:99.62%Color and Shape:SolidMolecular weight:509.92Ref: TM-T30828
1mg77.00€5mg158.00€10mg225.00€25mg338.00€50mg472.00€100mg645.00€200mg869.00€1mL*10mM (DMSO)To inquireIprindole
CAS:Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].Formula:C19H28N2Purity:99.54%Color and Shape:SolidMolecular weight:284.44Ref: TM-T37015
2mg37.00€5mg52.00€10mg80.00€25mg154.00€50mg266.00€100mg455.00€200mg652.00€1mL*10mM (DMSO)84.00€APC-0576
CAS:APC-0576, an (S,S)-isomer, blocks NF-kappaB gene activation and may reduce inflammation in human cells.Formula:C23H27N3O3Color and Shape:SolidMolecular weight:393.48PI3K-IN-28
CAS:PI3K-IN-28, a potent PI3K inhibitor with low toxicity in MCF-10a, has IC50 values of 5.8, 2.3, 7.9 μM and high selectivity index of 39.Formula:C26H16F9N3O3S2Color and Shape:SolidMolecular weight:653.54CFI-400936
CAS:CFI-400936: potent TTK inhibitor (IC50=3.6nM), potential anticancer, active in cell assays, selective vs. human kinases.Formula:C25H27N5O3SColor and Shape:SolidMolecular weight:477.58CB1R Allosteric modulator 1
CAS:CB1R modulator 1 (compound 11), a potent CB1R inhibitor, decreases activity of orthosteric ligands.Formula:C24H24ClN3OColor and Shape:SolidMolecular weight:405.92
