Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,789 products)
- Chromatin/Epigenetics(2,437 products)
- Cytoskeletal Signaling(1,525 products)
- DNA Damage/DNA Repair(2,967 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,000 products)
- Immunology and Inflammation(3,869 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,249 products)
- Membrane Transporter/Ion Channel(3,029 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,583 products)
- Neuroscience(10,380 products)
- Other Inhibitors(36,059 products)
- Oxidation-Reduction(43 products)
- PI3K/Akt/mTOR Signaling(1,445 products)
- Proteases/Proteasome(1,725 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,037 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66687 products of "Inhibitors"
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Cemadotin hydrochloride
CAS:Cemadotin hydrochloride (LU103793) is a synthetic mitosis inhibitor derived from Dolastatin 15 for treating solid tumors.Formula:C35H57ClN6O5Color and Shape:SolidMolecular weight:677.33Pralidoxime
CAS:Pralidoxime reactivates AChE blocked by nerve agents, aiding as an organophosphate poisoning antidote.Formula:C7H9N2OColor and Shape:SolidMolecular weight:137.16Kongensin A
CAS:Kongensin A is an effective heat shock protein 90 (HSP90) inhibitor that has potential anti-necroptosis and anti-inflammation applications.Formula:C22H30O5Purity:98%Color and Shape:SolidMolecular weight:374.47JNJ-4929821
CAS:JNJ-4929821 is a potent, reversible methionine aminopeptidase-2 (MetAP-2) inhibitor with IC50 of 8 nM.Formula:C14H13FN4O2S2Color and Shape:SolidMolecular weight:352.41Tau-aggregation-IN-1
CAS:Tau-aggregation-IN-1 is a dopamine D2 and D3 receptor agonist and an inhibitor of tau441 protein aggregation (IC50: 21 μM).Formula:C28H37N5O2SColor and Shape:SolidMolecular weight:507.69BET bromodomain inhibitor 2
CAS:BET bromodomain inhibitor 2 is a potent inhibitor of the BET-type bromodomain (IC50: 14.1 μM).Formula:C23H30N2O5SColor and Shape:SolidMolecular weight:446.56Reteplase
CAS:Reteplase, a recombinant plasminogen activator from t-PA's domains, is made via DNA tech in E. coli.Color and Shape:SolidGSI-136
CAS:GSI-136 is a gamma secretase inhibitor.Formula:C11H18ClNO3S2Color and Shape:SolidMolecular weight:311.857-Methotrexate
CAS:7-Methotrexate: chemotherapy, treats cancer, autoimmune disorders, ectopic pregnancy and aids medical abortions.Formula:C20H22N8O5Color and Shape:SolidMolecular weight:454.44(Rac)-CFT7455
CAS:(Rac)-CFT7455 degrades Ikaros/Aiolos via ubiquitin pathway, effective on NCIH929.1 (GI50: 0.05 nM), racemic with anticancer properties.Formula:C28H27N3O4Color and Shape:SolidMolecular weight:469.53GTC365
CAS:GTC365 is an hTERT transcriptional repressor that acts in the early stages of the G-quadruplex folding pathway.Formula:C23H25Cl2N7O4SColor and Shape:SolidMolecular weight:566.46NGB-2849
CAS:NGB-2849 is a selective dopamine D3 receptor antagonist.Formula:C29H29Cl2N3OColor and Shape:SolidMolecular weight:506.47DHODH-IN-21
CAS:DHODH-IN-21, orally active DHODH blocker with 1.1 nM IC50, shows anticancer activity, potential for AML research.Formula:C20H19ClF4N6O4Color and Shape:SolidMolecular weight:518.85AHR-16329
CAS:AHR-16329 can be used in ocular pharmacology.Formula:C11H14ClN3O4SColor and Shape:SolidMolecular weight:319.77Transketolase-IN-4
CAS:Transketolase-IN-4: IC50 3.9 μM; targets M. tuberculosis DXS (IC50 114.1 μM) & hinders SW620, LS174T, MIA PaCa-2 tumor cell growth.Formula:C19H14ClN3OPurity:99.52%Color and Shape:SolidMolecular weight:335.792-Pmp-PA
CAS:2-Pmp-PA is a taste modulator that inhibits sweetness.Formula:C10H12O4Color and Shape:SolidMolecular weight:196.2LG-121071
CAS:LG-121071: oral SARM, high-affinity AR full agonist, Ki=17 nM.Formula:C15H15F3N2OPurity:98%Color and Shape:SolidMolecular weight:296.295-Cyclopropylpentanal
CAS:5-Cyclopropylpentanal, an olfactory receptor agonist, effectively enhances OR-I7 activation, demonstrating an EC50 value of 0.3 μM.Formula:C8H14OColor and Shape:SolidMolecular weight:126.2LBW242
CAS:LBW242: oral 3-mer Smac mimetic, IAP inhibitor, targets multiple myeloma, enhances TRAIL/chemo death in ovarian cancer, active on mutant FLT3 cells.Formula:C27H42N4O2Purity:98%Color and Shape:SolidMolecular weight:454.65GX-674
CAS:GX-674 is a highly potent and selective voltage-gated sodium channel 1.7 (Nav1.7) antagonist with an IC50 value of 0.1 nM measured at -40 mV for the study ofFormula:C21H13ClF2N6O3S2Purity:98.60%Color and Shape:SolidMolecular weight:534.95Cgs 22706
CAS:Cgs 22706 is an adenosine A2 receptor antagonist.Formula:C17H22N6O7S2Color and Shape:SolidMolecular weight:486.52CHS-828 nicotinate
CAS:CHS-828, or GMX-1778, is a potent NAMPT inhibitor with anticancer properties, active against tumors and enhanced by certain drugs.Formula:C25H27ClN6O3Color and Shape:SolidMolecular weight:494.97POM2-C-HMBP
CAS:POM2-C-HMBP is a potent Activator of Vγ9Vδ2 T-Lymphocytes. It is also an HMBPP ananlog prodrug.Formula:C18H33O8PColor and Shape:SolidMolecular weight:408.42CYP3A4-IN-1
CAS:CYP3A4-IN-1 is a potent inhibitor of cytochrome P450 3A4 (CYP3A4) (IC50: 0.085 μM).Formula:C31H37N5O3SColor and Shape:SolidMolecular weight:559.72SC-44463
CAS:<p>SC-44463 is an MMP inhibitor, also a collagenase inhibitor , and HDAC inhibitor.</p>Formula:C19H29N3O5Color and Shape:SolidMolecular weight:379.45Mtb-cyt-bd oxidase-IN-4
Mtb-cyt-bd oxidase inhibitor; IC50=0.25μM; MIC=8μM against Mycobacterium tuberculosis; for TB research.Formula:C25H32FNOColor and Shape:SolidMolecular weight:381.53ST-836
CAS:ST-836 is a dopamine receptor ligand; Antiparkinsonian agent .Formula:C23H34N4OSPurity:98%Color and Shape:SolidMolecular weight:414.61(R)-Bambuterol
CAS:Bambuterol is a β2-agonist prodrug for asthma and COPD, taken daily, with a good safety profile and reduces plasma LDL-C and cholesterol.Formula:C18H29N3O5Color and Shape:SolidMolecular weight:367.44SJ-3366
CAS:SJ3366 is a unique and highly potent nonnucleoside reverse transcriptase human immunodeficiency virus type 1 and HIV-2 inhibitor.Formula:C21H24N2O3Color and Shape:SolidMolecular weight:352.43WS 009B
CAS:WS 009B is an antagonist of the endothelin receptor.Formula:C24H25NO11SPurity:98%Color and Shape:SolidMolecular weight:535.52GNE-9822
CAS:GNE-9822 is a potent selective ITK inhibitor that shows favorable ADME properties in preclinical species.Formula:C24H32N6OColor and Shape:SolidMolecular weight:420.55Pipradimadol
CAS:Pipradimadol is a 4,4-disubstituted piperidine derivative with antidepressive and serotonin antagonistic activity.Formula:C24H37ClN2O2Color and Shape:SolidMolecular weight:421.02AChE-IN-9
AChE-IN-9: Tacrine-β-glucose glycoconjugate; IC50 0.4μM; reduced hepatotoxicity; Alzheimer's research.Formula:C30H35N5O9Color and Shape:SolidMolecular weight:609.63R140309
CAS:R140309 is an UCHL3 inhibitor.Formula:C22H17FN2O4Color and Shape:SolidMolecular weight:392.38Fenoldopam hydrobromide
CAS:<p>Fenoldopam hydrobromide is a Dopamine D1-receptor agonist that acts as an antihypertensive.</p>Formula:C16H17BrClNO3Color and Shape:SolidMolecular weight:386.67Nω-Propyl-L-arginine hydrochloride
CAS:Highly selective and potent inhibitor of nNOS (Ki = 57 nM). Displays 3158-fold and 149-fold selectivity over iNOS and eNOS respectively. Hypotensive in vivo.Formula:C9H21ClN4O2Color and Shape:SolidMolecular weight:252.74Odelepran
CAS:Odelepran (LY2196044) is an opioid receptor antagonist under development for the treatment of alcohol dependence.Formula:C20H24FN3O3Color and Shape:SolidMolecular weight:373.42ML299
CAS:ML299 (VU0463568) is a dual PLD1/2 inhibitor (PLD1 and PLD2, IC50 of 6 nM, 20 nM, respectively).Formula:C23H26BrFN4O2Purity:98%Color and Shape:SolidMolecular weight:489.38L-701252
CAS:L-701252, a potent glycine site NMDA receptor antagonist, exhibits an inhibition concentration (IC50) of 420 nM.Formula:C13H10ClNO3Purity:97.7%Color and Shape:White Crystalline SolidMolecular weight:263.68ANEB-001
CAS:ANEB-001 is an orally active CB1 inhibitor that can be used in studies of acute cannabinoid intoxication.Formula:C22H24ClF3N2O2Color and Shape:SolidMolecular weight:440.89AK301
CAS:AK301 is a potent and selective inhibitor of tubulin polymerization and an effective sensitizer of cancer cells to apoptotic ligands (EC50 < 200 nM).Formula:C19H21ClN2O2Purity:99.75%Color and Shape:SolidMolecular weight:344.84YM-75466
CAS:YM-75466 is a factor Xa inhibitor reducing TAT in plasma dose-dependently without prolonging coagulation.Formula:C28H35N5O8S2Color and Shape:SolidMolecular weight:633.74Cgp 28861
CAS:Cgp 28861 reverses the effects of calcium channel blockaders in the frog heart.Formula:C18H17F2NO5Color and Shape:SolidMolecular weight:365.33MIPS1455
CAS:MIPS1455 is a photoactivatable allosteric M1 muscarinic acetylcholine receptor ligand.Formula:C24H17NO4Purity:98%Color and Shape:SolidMolecular weight:383.4AZD 1152 (hydrochloride)
CAS:AZD 1152, an oral prodrug, becomes AZD 1152-HQPA in plasma, selectively inhibits Aurora kinase B (IC50=0.36 nM), and blocks tumor growth.Formula:C26H33Cl2FN7O6PColor and Shape:SolidMolecular weight:660.47RK-52
CAS:RK-52: synthetic rhodesain inhibitor; ksecond = 67M min^-1, Ki = 38 pM, high affinity for trypanosomal protease.Formula:C30H32N2O4Color and Shape:SolidMolecular weight:484.59BMS-663749
CAS:BMS-663749 is an attachment inhibitor of human immunodeficiency virus type 1 (HIV-1).Formula:C23H25N4O9PColor and Shape:SolidMolecular weight:532.44Hepta-histidine
CAS:Hepta-histidine is a novel inhibitor of Tau aggregation against Tau-related neurodegenerative diseases including Alzheimer's disease (AD).Formula:C42H51N21O8Color and Shape:SolidMolecular weight:977.99sEH inhibitor-6
CAS:sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].Formula:C21H14ClN3O2Color and Shape:SolidMolecular weight:375.81IM-93
CAS:IM-93 inhibits ferroptosis and NETosis with an IC< sub>50 of 0.45 μM for cell death inhibition [1].Formula:C21H28N4O2Color and Shape:SolidMolecular weight:368.47
