Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,789 products)
- Chromatin/Epigenetics(2,437 products)
- Cytoskeletal Signaling(1,525 products)
- DNA Damage/DNA Repair(2,967 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,000 products)
- Immunology and Inflammation(3,869 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,249 products)
- Membrane Transporter/Ion Channel(3,029 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,583 products)
- Neuroscience(10,380 products)
- Other Inhibitors(36,059 products)
- Oxidation-Reduction(43 products)
- PI3K/Akt/mTOR Signaling(1,445 products)
- Proteases/Proteasome(1,725 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,037 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66687 products of "Inhibitors"
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5-HT7 agonist 2
CAS:Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.Formula:C23H29N3OColor and Shape:SolidMolecular weight:363.5DHP-218
CAS:DHP-218, a calcium channel blocker, inhibits rat aorta contractions; pA2: 9.11, IC50: 6.3 nmol/L (high K+) & 66 nmol/L (phenylephrine).Formula:C18H21N2O7PPurity:98%Color and Shape:SolidMolecular weight:408.34ICI-170809
CAS:ICI-170809 is a 5-HT2 receptor antagonist.Formula:C21H24N2SColor and Shape:SolidMolecular weight:336.49MMP-9-IN-3
CAS:MMP-9-IN-3: MMP-9/AKT inhibitor (IC50: 5.56/2.11 nM), forms H-bonds, cytotoxic, induces apoptosis, used in cancer research.Formula:C29H25N3O4Color and Shape:SolidMolecular weight:479.53Fallypride
CAS:Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.Formula:C20H29FN2O3Purity:98.97% - >99.99%Color and Shape:SolidMolecular weight:364.45NSC 601980
CAS:NSC601980, an antitumor agent, inhibits COLO 205 and HT29 cell growth with Log GI50s of -6.6 and -6.9.Formula:C15H12N4Purity:98%Color and Shape:SolidMolecular weight:248.28CI 951
CAS:CI 951 is a novel dihydronaphthyl Ca2+ antagonist and channel blocker.Formula:C22H23F3N2O3Color and Shape:SolidMolecular weight:420.42Ro 24-6392
CAS:Ro 24-6392, an ester co-drug of ciprofloxacin and desacetylcefotaxime, combats various aerobic bacteria.Formula:C31H31FN8O8S2Purity:98%Color and Shape:SolidMolecular weight:726.76Liothyronine HCl
CAS:Liothyronine is a T3 thyroid hormone normally synthesized and secreted by the thyroid gland in much smaller quantities than thyroxine.Formula:C15H13ClI3NO4Purity:98%Color and Shape:SolidMolecular weight:687.43IRAK4-IN-13
CAS:IRAK4-IN-13 (compound 21) is a potent IRAK4 inhibitor, IC50 0.6 nM, with high HLM clearance at 96 μL/min/mg.Formula:C24H27N9OColor and Shape:SolidMolecular weight:457.53ETB067
CAS:ETB067 is a PKA and AKT1 inhibitor, does not hinder CAMK2B or harm mice tissue at tested doses.Formula:C21H22BrN3O2SPurity:98%Color and Shape:SolidMolecular weight:460.39Ketocaine
CAS:Ketocaine（Rec 7-0518） is a local anesthetic commonly used in animal experiments with potential antitumor activity for pain relief.Formula:C18H29NO2Purity:98.59%Color and Shape:SolidMolecular weight:291.43GNF-2-PEG-acid
GNF-2-PEG-acid is usually used as a fluorescent probe.Formula:C26H27F3N4O7Purity:98%Color and Shape:SolidMolecular weight:564.51Setoperone
CAS:Setoperone, as a sensitive radioligand, can be commonly used in position emission tomography (PET) imaging.Formula:C21H24FN3O2SColor and Shape:SolidMolecular weight:401.5D719
CAS:D719 is a novel inhibitor of integrase nuclear translocation, showing significant inhibition on virus p24 antigen production.Formula:C21H20N2O5SColor and Shape:SolidMolecular weight:412.46R 836
CAS:R 836 has bronchodilator effects.Formula:C13H19N5SColor and Shape:SolidMolecular weight:277.39Niguldipine hydrochloride
CAS:Niguldipine is a calcium channel antagonist. Niguldipine shows high affinity to Ca2+ channels and to a subtype of alpha 1-adrenoceptors.Formula:C36H40ClN3O6Purity:98%Color and Shape:SolidMolecular weight:646.18Ranimustine
CAS:Ranimustine (MCNU) can be used for polycythemia vera and chronic myelogenous leukemia research, which is a nitrosourea alkylating agent [1] [3] [4].Formula:C10H18ClN3O7Color and Shape:SolidMolecular weight:327.72Opc 4392
CAS:Opc 4392 is an agonist of presynaptic dopamine D(2) receptor.Formula:C24H29N3O2Color and Shape:SolidMolecular weight:391.51PIK-C98
CAS:PIK-C98 is an inhibitor of PI3K that acts by displaying potent preclinical activity against multiple myeloma.Formula:C16H10Cl2N2OSPurity:98%Color and Shape:SolidMolecular weight:349.23Mps1-IN-5
CAS:Mps1-IN-5: oral Mps1 inhibitor with 29 nM IC50, induces apoptosis, G2/M arrest, and has anti-tumor properties.Formula:C24H25N9Color and Shape:SolidMolecular weight:439.52BM635
CAS:BM635 is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).Formula:C25H29FN2OColor and Shape:SolidMolecular weight:392.51(R)-Olacaftor
CAS:(R)-Olacaftor (VX-440) is a CFTR modulator with promise for researching cystic fibrosis.Formula:C29H34FN3O4SColor and Shape:SolidMolecular weight:539.66Refortan
CAS:Refortan, as hydroxyethyl starch, can be used in surgery for maintaining hemostasis in patients.Formula:C14H10Cl2O4Color and Shape:SolidMolecular weight:313.13A1/A3 AR antagonist 2
CAS:The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.Formula:C22H16N2O3SColor and Shape:SolidMolecular weight:388.44PI3Kγ inhibitor 7
CAS:PI3Kγ Inhibitor 7 (compound 2) is a potent, orally active agent that selectively inhibits PI3Kγ with an IC50 of 3.42 nM and demonstrates antitumor activity [1].Formula:C31H25N9O2Purity:98%Color and Shape:SolidMolecular weight:555.59Acetaminotadalafil
CAS:Acetaminotadalafil is a new analogue of Tadalafil used for the treatment of erectile dysfunction. It acts as a phosphodiesterase 5 inhibitor.Formula:C23H20N4O5Color and Shape:SolidMolecular weight:432.43Broxaterol
CAS:Broxaterol is a β2 adrenoreceptor agonist. It is part of a class of drugs that affect the smooth muscle receptors in the body.Formula:C9H15BrN2O2Purity:98%Color and Shape:SolidMolecular weight:263.13CFM-2
CAS:CFM-2, a potent and selective non-competitive antagonist of AMPAR (AMPAR), exhibits anticonvulsant activity across various seizure models.Formula:C17H17N3O3Purity:99.84%Color and Shape:SolidMolecular weight:311.34MLS-2064
CAS:MLS-2064 is a STAT3 and Akt signaling inhibitor.Formula:C22H24BrCl2N5O2Color and Shape:SolidMolecular weight:541.27AZ4800
CAS:AZD4800 is a gamma secretase modulators.Formula:C24H29N5O3Color and Shape:SolidMolecular weight:435.52Oxolamine
CAS:Oxolamine is an agent of a cough suppressant.Formula:C14H19N3OPurity:98%Color and Shape:SolidMolecular weight:245.32AHR-5645B fumarate
CAS:AHR-5645B fumarate is a substituted benzamide that has been shown to inhibit 3H-spiperone binding to bovine anterior pituitary membranes.Formula:C22H31N3O5Color and Shape:SolidMolecular weight:417.5(6R)-ML753286
(6R)-ML753286, an ML753286 isomer, selectively inhibits BCRP (IC50: 0.6μM), has high permeability, and is stable in plasma.Formula:C20H25N3O3Color and Shape:SolidMolecular weight:355.43GSK926
CAS:GSK926 is a selective, SAM-competitive, and cell-active EZH2 inhibitor.Formula:C29H35N7O2Color and Shape:SolidMolecular weight:513.63Rucaparib camsylate
CAS:Rucaparib camsylate, a PARP-1, -2, -3 inhibitor (Ki=1.4 nM for PARP-1) & H6PD blocker, may treat resistant prostate cancer.Formula:C19H18FN3O·xC10H16O4SColor and Shape:SolidRociverine
CAS:Rociverine is an anticholinergic compound used as a smooth muscle relaxant.Formula:C20H37NO3Color and Shape:SolidMolecular weight:339.51RP-101075
CAS:RP-101075, Ozanimod metabolite, mirrors its specificity and effects on S1P receptors in vitro and in vivo.Formula:C21H20N4O2Color and Shape:SolidMolecular weight:360.41Butopamine
CAS:Butopamine differs from dobutamine in location of only one hydroxyl group, but is no longer a catecholamine.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.38RET-IN-16
CAS:RET-IN-16: Selective RET inhibitor, IC50s 3.98-15.05 nM for various RET mutations; anticancer properties.Formula:C31H29F3N8O2Color and Shape:SolidMolecular weight:602.61MCI826
CAS:MCI826 is a potent and selective antagonist of P-glycoprotein (P-gp) and peptide leukotrienes (p-LTs), showing anti-asthmatic activity in a guinea pig model ofFormula:C22H28N2O3SPurity:98.73%Color and Shape:SolidMolecular weight:400.53m-Toluidine, α-methoxy-4-(octyloxy)-, hydrochloride
CAS:m-Toluidine, alpha-methoxy-4-(octyloxy)-, hydrochloride is a bioactive chemcial.Formula:C16H28ClNO2Color and Shape:SolidMolecular weight:301.85Nemiralisib
CAS:Nemiralisib (GSK-2269557) is an oral PI3Kδ inhibitor (pKi 9.9) for treating respiratory diseases like COPD.Formula:C26H28N6OPurity:99.91%Color and Shape:SolidMolecular weight:440.54Choline theophyllinate
CAS:Choline theophyllinate (Oxtriphylline) is the choline salt of theophylline, a small molecule PDE inhibitor that can be used to treat immune system disorders andFormula:C12H21N5O3Purity:98%Color and Shape:SolidMolecular weight:283.33GI-129471
CAS:GI-129471 is a metalloproteinase inhibitor, specifically blocking TNF-alpha secretion both in vitro and in vivo.Formula:C25H33N3O4SColor and Shape:SolidMolecular weight:471.61DBHDA
CAS:DBHDA transforms C-terminal Cys into Dha in Ubl G76C mutant probes.Formula:C6H10Br2N2O2Color and Shape:SolidMolecular weight:301.96L-CCG-l
CAS:group II metabotropic glutamate receptor agonistFormula:C6H9NO4Purity:98%Color and Shape:SolidMolecular weight:159.14Valategrast hydrochloride
CAS:Valategrast hydrochloride (R411), a dual antagonist of integrin α4β1 (VLA-4), is used for the potential treatment of asthma.Formula:C30H33Cl4N3O4Purity:98%Color and Shape:SolidMolecular weight:641.41Gallamine
CAS:Gallamine is an allosteric antagonist at muscarinic M2 acetylcholine receptors and an inhibitor of acetylcholinesterase.Formula:C24H45N3O3Color and Shape:SolidMolecular weight:423.63ONO-2921
CAS:ONO-2921 is a Novel N-Type Ca Channel BlockerFormula:C31H48N4O4S2Color and Shape:SolidMolecular weight:604.87
