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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66691 products of "Inhibitors"

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  • L 738372

    CAS:
    L 738372 is a non-nucleoside inhibitor of HIV-1 reverse transcriptase.
    Formula:C18H15N3O
    Color and Shape:Solid
    Molecular weight:289.33
  • NCC-149

    CAS:
    NCC-149 is a HDAC8 inhibitor.
    Formula:C16H14N4O2S
    Color and Shape:Solid
    Molecular weight:326.37
  • GLPG3970

    CAS:
    GLPG3970, a pioneering inhibitor of SIK2/SIK3, is utilized in the investigation of inflammation and autoimmune diseases.
    Formula:C25H27F3N4O4
    Purity:99.60% - >99.99%
    Color and Shape:Solid
    Molecular weight:504.5
  • Bezuclastinib

    CAS:
    Bezuclastinib (CGT9486) is a novel, potent and highly selective tyrosine kinase and c-kit D816V inhibitor for the study of advanced mastocytosis.
    Formula:C19H17N5O
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:331.37
  • LP-533401

    CAS:
    LP-533401 is an inhibitor of Tryptophan hydroxylase 1. It is used for regulates serotonin production in the gut.
    Formula:C27H22F4N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:526.48
  • HDAC-IN-31

    CAS:
    HDAC-IN-31: Oral HDAC inhibitor; targets HDAC1, 2, 3; weak on HDAC8; potential in fighting lymphoma.
    Formula:C25H24N4O2
    Color and Shape:Solid
    Molecular weight:412.48
  • ML-243

    CAS:
    inhibitor of cancer stem cells
    Formula:C14H16N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:260.35
  • Vibsanin A

    CAS:
    Vibsanin A, an activator of protein kinase C (PKC) and an inhibitor of HSP90, demonstrates anti-proliferative effects on human cancer cell lines.
    Formula:C25H38O4
    Color and Shape:Solid
    Molecular weight:402.57
  • Satranidazole

    CAS:
    Satranidazole is an anti-bacterial. It is used to treat periodontitis.
    Formula:C8H11N5O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:289.27
  • Radamide

    CAS:
    Radamide is an inhibitor of Grp94.
    Formula:C18H18ClNO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.79
  • Pentachloropseudilin

    CAS:
    Pentachloropseudilin inhibits Myosin-1 and speeds up TGF-β receptor turnover, suppressing TGF-β activity.
    Formula:C10H4Cl5NO
    Purity:98.14%
    Color and Shape:Solid
    Molecular weight:331.41
  • KAA-276 free base

    CAS:
    KAA-276: potent, long-lasting histamine H1 antagonist with minimal irritation; for asthma via inhalation.
    Formula:C31H35FN4O2
    Color and Shape:Solid
    Molecular weight:514.63
  • LGD-2226

    CAS:
    LGD-2226: selective oral androgen receptor modulator, EC50: 0.2nM, Ki: 1.5nM. Treats muscle loss, osteoporosis, sexual issues.
    Formula:C14H9F9N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.22
  • VUF10132

    CAS:
    <p>VUF10132 is a full inverse CXCR3 N3.35A agonist.</p>
    Formula:C19H13BrCl4N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:523.03
  • WAY-260022

    CAS:
    WAY-260022 is the norepinephrine transporter inhibitor.
    Formula:C21H31F3N2O2
    Purity:97.61% - 99.41%
    Color and Shape:Solid
    Molecular weight:400.48
  • AZD2906

    CAS:
    AZD2906: selective GR agonist with human/rat IC50s - 2.2/0.3 nM (PBMC), 41.6/7.5 nM (blood); induces rat bone marrow micronuclei.
    Formula:C26H25FN4O3
    Color and Shape:Solid
    Molecular weight:460.5
  • INU-101

    CAS:
    INU-101: oral 11β-HSD1 inhibitor improves insulin sensitivity and reduces blood glucose, potential type 2 diabetes treatment.
    Formula:C21H28FN3O4S
    Color and Shape:Solid
    Molecular weight:437.53
  • L 687384

    CAS:
    L 687384 is a high-affinity ligand of sigma receptor.
    Formula:C21H25N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:291.43
  • L-771688 dihydrochloride

    CAS:
    L-771688 is an α1A-adrenoceptor antagonist potentially for the treatment of benign prostatic hyperplasia.
    Formula:C28H35Cl2F2N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:630.51
  • Romifidine

    CAS:
    Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.
    Formula:C9H9BrFN3
    Color and Shape:Solid
    Molecular weight:258.09
  • Butixirate

    CAS:
    Butixirate is a biochemical.
    Formula:C28H33NO2
    Color and Shape:Solid
    Molecular weight:415.577
  • BM-131246

    CAS:
    BM-131246 is an orally available and antidiabetic active thiazolidinedione derivative for the study of diabetes.
    Formula:C22H20N2O4S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:408.47
  • JNK3 inhibitor-4

    CAS:
    <p>JNK3 inhibitor-4: potent, selective JNK3 blocker (IC50=1.0nM), neuroprotective, BBB-permeable.</p>
    Formula:C28H27N7O
    Color and Shape:Solid
    Molecular weight:477.56
  • Rotundifuran

    CAS:
    Rotundifuran from Vitex rotundifolia fruit blocks cell cycle, induces apoptosis in leukemia cells.
    Formula:C22H34O4
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:362.5
  • Integrin-IN-2

    CAS:
    Integrin-IN-2, an oral αv integrin blocker, enhances αvβ6/3/5/8 affinities with pIC50s: 7.8/8.4/8.4/7.4.
    Formula:C27H30N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:458.55
  • Benzaldehyde, oxime

    CAS:
    Benzaldehyde, oxime is an intermediate in the synthesis of chromones.
    Formula:C7H7NO
    Purity:97.68%
    Color and Shape:Solid
    Molecular weight:121.14
  • Erythronic acid

    CAS:
    Erythronic acid, an endogenous carbohydrate metabolite, is instrumental for research into metabolism-associated disorders.
    Formula:C4H8O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:136.1
  • TBC3711

    CAS:
    TBC3711 is an endothelin receptor modulator. It is used for the research of endothelin-mediated disorders.
    Formula:C20H21N3O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:447.53
  • IKKß-IN-124

    CAS:
    IKKβ-IN-124 blocks NF-κB by inhibiting IκBα phosphorylation and securing IKKβ in inactive form.
    Formula:C17H26Cl2N2O3S
    Color and Shape:Solid
    Molecular weight:409.37
  • Lu AE98134

    CAS:
    Lu AE98134 enhances Nav1.1, Nav1.2, and Nav1.5 sodium channels, but not Nav1.4/1.6/1.7; studied in CNS diseases like schizophrenia.
    Formula:C21H23N5O3S
    Color and Shape:Solid
    Molecular weight:425.5
  • PRMT5-IN-10

    CAS:
    PRMT5-IN-10 exhibits promising structure-dependent inhibitory effect on the protein methyltransferase PRMT5:MEP50 complex.
    Formula:C13H17N5O4
    Color and Shape:Solid
    Molecular weight:307.31
  • TB 21007

    CAS:
    GABAA receptor inverse agonist
    Formula:C15H17NO2S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:339.5
  • BRD9185

    CAS:
    BRD9185 is an inhibitor of Dihydroorotate dehydrogenase (DHODH) with an EC50 of 16 nM against multidrug-resistant blood-stage parasites in vitro.
    Formula:C23H21F6N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:485.42
  • NSC260594

    CAS:
    NSC260594 is a chemical compound that promotes apoptosis by binding to the shallow groove of the Mcl-1 protein and suppressing its expression through down-
    Formula:C29H24N6O3
    Color and Shape:Solid
    Molecular weight:504.54
  • SDZ NKT 343

    CAS:
    human tachykinin NK1 receptor antagonist
    Formula:C33H33N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:579.65
  • ARI-3531

    CAS:
    ARI-3531 is a selective prolyl endopeptidase inhibitor.
    Formula:C15H22BN3O4
    Color and Shape:Solid
    Molecular weight:319.16
  • BuChE-IN-2

    CAS:
    BuChE-IN-2 inhibits BuChE (IC50: 1.28 μM), NO (0.67 μM), Aβ, ROS, chelates Cu2+, penetrates BBB, used in Alzheimer's research.
    Formula:C28H20F4N6O3
    Color and Shape:Solid
    Molecular weight:564.49
  • Trotabresib

    CAS:
    Trotabresib (CC-90010) is an orally active inhibitor of BET and can be used in studies about advanced solid tumors.
    Formula:C21H21NO4S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:383.46
  • Enpp-1-IN-17

    CAS:
    Enpp-1-IN-17 (example 274) is a potent inhibitor of ENPP1, exhibiting inhibition constants (Ki values) of 100 nM-1 μM for cGAMP hydrolysis and >1 μM for ATP
    Formula:C18H24N4O2
    Color and Shape:Solid
    Molecular weight:328.41
  • Coldephnine

    CAS:
    Coldephnine is a aconitine-type norditerpenoid alkaloid used as a nicotinic acetylcholine (ACh) receptor antagonist.
    Formula:C25H39NO6
    Color and Shape:Solid
    Molecular weight:449.58
  • RP-101075

    CAS:
    RP-101075, Ozanimod metabolite, mirrors its specificity and effects on S1P receptors in vitro and in vivo.
    Formula:C21H20N4O2
    Color and Shape:Solid
    Molecular weight:360.41
  • Seladelpar Lysine dihydrate

    CAS:
    Seladelpar lysine, a selective PPAR-δ agonist, is used for the therapy of Homozygous Familial Hypercholesterolemia (HoFH).
    Formula:C27H41F3N2O9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:626.68
  • SEW-05929

    CAS:
    SEW-05929 is the first effective SecA inhibitor.
    Formula:C28H19ClFN3O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:548.05
  • Orazipone

    CAS:
    Orazipone inhibits cytokine production and histamine release; an NSAID.
    Formula:C13H14O4S
    Color and Shape:Solid
    Molecular weight:266.31
  • Tropodifene

    CAS:
    Tropodifene is an inhibitor of the α-Adrenergic receptor.
    Formula:C25H29NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:407.5
  • AZ8838

    CAS:
    <p>AZ8838 is an effective, competitive, allosteric, orally active non-peptide small molecule antagonist of PAR2 with a pK i of 6.4 for hPAR2 [1].</p>
    Formula:C13H15FN2O
    Color and Shape:Solid
    Molecular weight:234.27
  • Alvameline maleate

    CAS:
    Alvameline maleate is used as a Partial M1 Agonist and M2/M3 Antagonist.
    Formula:C13H19N5O4
    Color and Shape:Solid
    Molecular weight:309.32
  • Butalamine

    CAS:
    Butalamine is a vasodilator (peripheral) with local anesthetic effects. It suppresses state 3 respiration and decreases ADP/O in the rat liver.
    Formula:C18H28N4O
    Color and Shape:Solid
    Molecular weight:316.44
  • Figopitant

    CAS:
    Figopitant is a tachykinin neurokinin-1 antagonist.
    Formula:C27H31F6N3O
    Color and Shape:Solid
    Molecular weight:527.54
  • Way 100135

    CAS:
    WAY-100135: research drug, phenylpiperazine, potent 5-HT1A antagonist, partial 5-HT1D agonist, minor 5-HT1B activity.
    Formula:C24H33N3O2
    Color and Shape:Solid
    Molecular weight:395.54