Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,789 products)
- Chromatin/Epigenetics(2,437 products)
- Cytoskeletal Signaling(1,525 products)
- DNA Damage/DNA Repair(2,967 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,000 products)
- Immunology and Inflammation(3,869 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,249 products)
- Membrane Transporter/Ion Channel(3,029 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,583 products)
- Neuroscience(10,380 products)
- Other Inhibitors(36,059 products)
- Oxidation-Reduction(43 products)
- PI3K/Akt/mTOR Signaling(1,445 products)
- Proteases/Proteasome(1,725 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,037 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66687 products of "Inhibitors"
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NBC 6
CAS:NLRP3-IN-NBC6: potent NLRP3 inflammasome inhibitor, IC50 574 nM, Ca2+ independent, inhibits inflammasome in THP-1 cells/BMDMs.Formula:C18H16BCl3N2O2Color and Shape:SolidMolecular weight:409.5AQX-016A
CAS:AQX-016A, a potent SHIP1 agonist, is an oral analog of pelorol, 3x stronger, inhibits PI3K, TNFa, for inflammation research.Formula:C22H32O2Color and Shape:SolidMolecular weight:328.49CT-1
CAS:<p>CT-1 is a DNA minor groove ligand and causes p53-dependent breast cancer cell apoptosis.</p>Formula:C29H23F3N4OPurity:99.79%Color and Shape:SolidMolecular weight:500.51B 4310
CAS:B 4310 is a bradykinin inhibitor.Formula:C62H95N19O14S2Color and Shape:SolidMolecular weight:1394.67Lenperone
CAS:Lenperone is a butyrophenone antipsychotic. Like other major tranquilizers, It has some alpha-adrenergic blocking action and is antiemetic.Formula:C22H23F2NO2Color and Shape:SolidMolecular weight:371.42PKM2 activator 3
CAS:PKM2 activator 3, with 90 nM AC50, enhances PKM2. It has good Caco-2 permeability, stable, and aids cancer research.Formula:C15H11ClF2N2O3SColor and Shape:SolidMolecular weight:372.77P2X3 antagonist 36
CAS:P2X3 antagonist 36 is a P2X3 antagonist.Formula:C20H18ClF3N6O3Color and Shape:SolidMolecular weight:482.84HDAC3-IN-T326
CAS:HDAC3-IN-T326: potent, selective HDAC3 inhibitor, boosts NF-κB acetylation, activates latent HIV gene expression.Formula:C21H18N6O3SPurity:98%Color and Shape:SolidMolecular weight:434.4714-(Fmoc-amino)-tetradecanoic acid
CAS:14-(Fmoc-amino)-tetradecanoic acid: a PROTAC linker with Fmoc-protected amine and carboxylic end-groups, used in amide bond formation.Formula:C29H39NO4Color and Shape:SolidMolecular weight:465.62BTK-IN-22
CAS:BTK-IN-22 is a selective BTK inhibitor with IC50 of 0.9 nM; also targets BLX, BMX (IC50s: 1.4, 1.2 nM); better selectivity than Ibrutinib.Formula:C26H26N6O2Color and Shape:SolidMolecular weight:454.52KR-31378
CAS:KR-31378, a K(ATP) channel activator, is used potentially for the treatment of ocular hypertension and glaucoma.Formula:C22H27N5O4Color and Shape:SolidMolecular weight:425.48Y06036
CAS:Y06036, a potent and selective BET inhibitor, can bind to the BRD4(1) bromodomain (Kd: 82 nM).Formula:C16H15BrN2O5SPurity:99.97%Color and Shape:SolidMolecular weight:427.27PU-H54-iso
CAS:PU-H54-iso is a novel Hsp90- and Grp94-selective inhibitor.Formula:C18H19N5SPurity:98%Color and Shape:SolidMolecular weight:337.44Tetridamine
CAS:Tetridamine is an anti-inflammatory and analgesic drug used for the treatment of vaginitis.Formula:C9H15N3Purity:98%Color and Shape:SolidMolecular weight:165.24Oxarbazole
CAS:Oxarbazole is an antagonist of slow-reacting substance of anaphylaxis.Formula:C21H19NO4Color and Shape:SolidMolecular weight:349.38Ac32Az19
CAS:Ac32Az19 is a potent, non-toxic, and highly selective inhibitor of Breast Cancer Resistance Protein (BCRP), demonstrating an EC50 of 13 nM in BCRP-overexpressedFormula:C37H33N3O6Color and Shape:SolidMolecular weight:615.67Fadolmidine
CAS:Fadolmidine is a novel and potent alpha2 -adrenoceptor (alpha2) -AR) agonist developed for spinal analgesia.Formula:C13H14N2OColor and Shape:SolidMolecular weight:214.26CP-53631
CAS:CP-53631 is a selective serotonin reuptake inhibitor (SSRI)Formula:C17H19BrClNColor and Shape:SolidMolecular weight:352.7Benzamide, N-(5-amino-2-(octyloxy)benzyl)-
CAS:Benzamide, N-(5-amino-2-(octyloxy)benzyl)- is a bioactive chemical.Formula:C22H30N2O2Color and Shape:SolidMolecular weight:354.49COX-2-IN-23
CAS:COX-2-IN-23 selectively inhibits COX-2 (IC50=0.28μM), weakly affects COX-1 (IC50=20.14μM), and has anti-inflammatory and low ulcerogenic properties.Formula:C24H25N5O3S2Color and Shape:SolidMolecular weight:495.62Lorzafone
CAS:Lorzafone is used in the detection & analysis of pharmacologically active benzodiazepines.Formula:C18H17Cl2N3O3Color and Shape:SolidMolecular weight:394.25(R)-PF-06256142
CAS:(R)-PF-06256142: low-activity R enantiomer of a potent, selective D1 agonist reducing receptor desensitization.Formula:C21H16N4O2Color and Shape:SolidMolecular weight:356.38AHR-10718
CAS:AHR-10718 has an antiarrhythmic effect.Formula:C22H35N3O7SPurity:98%Color and Shape:SolidMolecular weight:485.6sEH inhibitor-5
CAS:sEH inhibitor-5 is a potent inhibitor of sEH (soluble epoxide hydrolase) (IC50: 0.1 nM).Formula:C27H26Cl2N6O3SColor and Shape:SolidMolecular weight:585.5LEO-29102
CAS:LEO-29102: Potent, selective PDE4 inhibitor, promising for treating skin diseases, phase 2 efficacy in atopic dermatitis.Formula:C20H22Cl2N2O5Color and Shape:SolidMolecular weight:441.31Benzoic acid, m-(2-methyl-5-phenylpyrrol-1-yl)-, compd. with 2-aminoethanol (1:1)
CAS:Benzoic acid, m-(2-methyl-5-phenylpyrrol-1-yl)-, compd. with 2-aminoethanol (1:1) is a bioactive chemical.Formula:C20H22N2O3Color and Shape:SolidMolecular weight:338.40Crozbaciclib fumarate
CAS:Crozbaciclib fumarate is a CDK4/6 inhibitor with IC 50 s of 3 and 1 nM, respectively.Formula:C32H34F2N6O4Color and Shape:SolidMolecular weight:604.65NO 756
CAS:NO 756 is a D1 dopamine receptor antagonist.Formula:C19H20ClNOColor and Shape:SolidMolecular weight:313.825BMS-663749 lysine
CAS:BMS-663749 lysine is used as a phosphonooxymethyl prodrug 4 for HIV-1 attachment inhibitor.Formula:C29H39N6O11PPurity:98%Color and Shape:SolidMolecular weight:678.63Efflux inhibitor-1
CAS:Efflux inhibitor-1 is a pyrazolopyrimidine efflux inhibitor.Formula:C28H25N5O3Color and Shape:SolidMolecular weight:479.53PNU-107484A
CAS:PNU-107484A is a unique GABA(A) receptor ligand.Formula:C18H23ClN6Purity:98%Color and Shape:SolidMolecular weight:358.87Trimazosin
CAS:Trimazosin, a quinazoline derivative and prazosin relative, lowers blood pressure by blocking alpha1-adrenoceptors.Formula:C20H29N5O6Color and Shape:SolidMolecular weight:435.47RP101988
RP101988, a potent Ozanimod metabolite, selectively targets S1PR1 with EC50 of 0.19 nM and S1PR5 at 32.8 nM.Formula:C23H22N4O4Color and Shape:SolidMolecular weight:418.45RO314724
CAS:RO314724: HDAC & reversible MMP inhibitor, Ki=26 nm, protects cartilage by inhibiting MMP-related breakdown.Formula:C19H35N3O6Color and Shape:SolidMolecular weight:401.5Tyrosinase-IN-11
CAS:Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.Formula:C15H14O5Color and Shape:SolidMolecular weight:274.27Tisopurine
CAS:Tisopurine is a drug used in the treatment of gout in some countries. It reduces uric acid production through inhibiting an early stage in its production.Formula:C5H4N4SColor and Shape:SolidMolecular weight:152.18Aurora kinase-IN-1
Aurora kinase-IN-1: potent aurora kinase inhibitor, alters G1 cycle proteins, induces G1/S arrest and apoptosis, potential chemotherapy lead.Formula:C30H25Br2N3O5Color and Shape:SolidMolecular weight:667.34CB10-277
CAS:CB10-277 is a synthetic anti-cancer drug related to dacarbazine that alkylates DNA, inhibits DNA replication and repair, and may block DNA synthesis.Formula:C9H11N3O2Color and Shape:SolidMolecular weight:193.2ORY-1001 free base
CAS:ORY-1001: potent KDM1A inhibitor (IC50 <20nM), selective, affects THP-1 cell gene regulation and apoptosis, hinders MV(4;11) cell growth (EC50 <1nM).Formula:C15H22N2Purity:98%Color and Shape:SolidMolecular weight:230.35SQ 32602
CAS:SQ 32602 is a cathepsin E inhibitor.Formula:C32H52N3O7PColor and Shape:SolidMolecular weight:621.74Laropiprant analog
CAS:Laropiprant analog is an antagonist of the prostaglandin PGD2 receptor DP1.Formula:C20H18ClFN2O4SColor and Shape:SolidMolecular weight:436.88FK-386 HCl
CAS:FK-386 HCl is an inhibitor of chymotrypsin.Formula:C32H39Cl2N3O5Color and Shape:SolidMolecular weight:616.58CPI-905
CAS:CPI-905 is a potent and selective EZH2 inhibitor with IC50 value of 39.5 nM.Formula:C18H20N2O5Color and Shape:SolidMolecular weight:344.36BR103
CAS:BR103 is a C3aR-selective agonist that is metabolically stable.Formula:C24H28N6O3Color and Shape:SolidMolecular weight:448.52BE 2254
CAS:BE 2254 is an antagonist of central noradrenergic receptor.Formula:C19H21NO2Color and Shape:SolidMolecular weight:295.38CAY10761
CAS:CAY10761 inhibits ENPP1 (IC50: 467 μM human, 429 μM snake), mushroom tyrosinase (Ki: 1.9 μM), and urease from different sources (IC50: 0.093-<0.125 mM).Formula:C7H8N4O2S2Color and Shape:SolidMolecular weight:244.29Pirandamine Free Base
CAS:Pirandamine Free Base is a tricyclic derivative which acts as a selective serotonin reuptake inhibitorFormula:C17H23NOColor and Shape:SolidMolecular weight:257.37BMS-955829
CAS:BMS-955829 is a positive allosteric modulator (PAM).Formula:C22H14F2N2O2Color and Shape:SolidMolecular weight:376.36BuChE-IN-1
CAS:BuChE-IN-1 is a potent BBB-permeable, low-toxic BuChE inhibitor with potential for AD research.Formula:C23H23FN2O4SColor and Shape:SolidMolecular weight:442.5Alinastine
CAS:Alinastine is a noncompetitive histamine H1 receptor antagonist.Formula:C28H39N3OColor and Shape:SolidMolecular weight:433.63
