Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,781 products)
- Apoptosis(6,260 products)
- Cell Cycle/Checkpoint(4,789 products)
- Chromatin/Epigenetics(2,437 products)
- Cytoskeletal Signaling(1,525 products)
- DNA Damage/DNA Repair(2,967 products)
- Endocrinology/Hormones(3,706 products)
- Enzyme(3,667 products)
- GPCR/G-Protein(9,000 products)
- Immunology and Inflammation(3,869 products)
- Influenza Virus(301 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,249 products)
- Membrane Transporter/Ion Channel(3,029 products)
- Metabolism(10,207 products)
- Microbiology/Virology(7,583 products)
- Neuroscience(10,380 products)
- Other Inhibitors(36,059 products)
- Oxidation-Reduction(43 products)
- PI3K/Akt/mTOR Signaling(1,445 products)
- Proteases/Proteasome(1,725 products)
- Stem Cell and Derivatives(825 products)
- Tyrosine Kinase/Adaptors(2,037 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66687 products of "Inhibitors"
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3,3-Dimethyl-1-butanol
CAS:3,3-Dimethyl-1-butanol (DMB) inhibits TMA/TMAO and affects p65 NF-κB, TGF-β1/Smad3 signaling; potential for CVD treatment.Formula:C6H14OColor and Shape:SolidMolecular weight:102.17DNMT3A-IN-1
CAS:DNMT3A-IN-1 is a potent, selective DNMT3A inhibitor with KI 9.16-18.85 μM (AdoMet) and 11.37-23.34 μM (poly dI-dC).Formula:C30H38N6O4Color and Shape:SolidMolecular weight:546.66PA1 2HCl
CAS:PA1 2HCl is a blocker of photoswitchable epithelial sodium channel (ENaC).Formula:C18H16ClN9OColor and Shape:SolidMolecular weight:409.83Briciclib Na
CAS:Briciclib Na inhibits benzylstyryl sulfone kinase and is use for the treatment of CancerFormula:C19H21Na2O10PSColor and Shape:SolidMolecular weight:518.38HLI 373
CAS:HLI373: potent Hdm2 (ubiquitin ligase) inhibitor, induces apoptosis in tumor cells, has antimalarial properties.Formula:C18H23N5O2Color and Shape:SolidMolecular weight:341.41PU-H39
CAS:PU-H39 is a specific inhibitor of Hsp90b1.Formula:C16H13Cl2N5SPurity:98%Color and Shape:SolidMolecular weight:378.28Tenofovir maleate
CAS:Tenofovir Disoproxil Fumarate is a nucleotide reverse transcriptase inhibitor used in the treatment of HIV and chronic Hepatitis B.Formula:C13H18N5O8PColor and Shape:SolidMolecular weight:403.28Type II topoisomerase inhibitor 1
CAS:Potent E. coli DNA gyrase inhibitor (IC50: 1.7 nM), targets Asp73; weak topoisomerase IV inhibitor (IC50: 0.98 μM).Formula:C18H15N3O4Color and Shape:SolidMolecular weight:337.33Salazopyridazine
CAS:Salazopyridazine is an antibacterial agent that inhibits ulcerative colitis. salazopyridazine can be used in the study of rheumatic diseases.Formula:C18H15N5O6SColor and Shape:SolidMolecular weight:429.41BTG-1640
CAS:BTG-1640 is used potentially for the treatment of anxiety and panic disorder.Formula:C15H19NO2Color and Shape:SolidMolecular weight:245.32hGGPPS-IN-1
CAS:HGGPPS-IN-1: analog of C2-ThP-BPs, inhibits hGGPPS, triggers apoptosis in MM cells, shows anti-myeloma effects in vivo.Formula:C13H13N3O6P2SColor and Shape:SolidMolecular weight:401.27NMDA receptor modulator 2
CAS:NMDA receptor modulator 2 (Compound 1) is a potent modulator of the NMDA receptor that can be used for neurological disorder research [1].Formula:C13H11F3N2O2Color and Shape:SolidMolecular weight:284.23Allantoin polygalacturonic acid
CAS:Allantoin polygalacturonic acid is a protein aggregate suppressor.Formula:C10H16N4O10Color and Shape:SolidMolecular weight:352.256SP-471P
CAS:SP-471P inhibits DENV protease; EC50: DENV1-5.9 μM, DENV2-1.4 μM, DENV3-5.1 μM, DENV4-1.7 μM; CC50 >100 μM; lowers viral RNA synthesis.Formula:C33H26BrN5O2Color and Shape:SolidMolecular weight:604.5Supradamal
CAS:Supradamal is a potent Inhibitor of Plasmodium FK506 Binding Protein 35 (FKBD35). It also acts as an HIV inhibitor.Formula:C17H21N3O2Color and Shape:SolidMolecular weight:299.37Isomolpan hydrochloride
CAS:Isomolpan hydrochloride is a dopamine receptor D2 agonist.Formula:C15H22ClNO2Color and Shape:SolidMolecular weight:283.79SARS-CoV-2 nsp13-IN-3
CAS:SARS-CoV-2 nsp13-IN-3 (Compound C3) is a small molecule inhibitor of SARS-CoV-2 non-structural protein 13 (nsp13) that acts on nsp13 ssDNA+ATPase (IC50: 32 μM).Formula:C24H27N7OColor and Shape:SolidMolecular weight:429.52Tubulin inhibitor 26
CAS:Compound 3c, a potent indazole-based tubulin inhibitor, halts G2/M phase and induces apoptosis in various cancers without weight loss in mice.Formula:C17H19N3O3Color and Shape:SolidMolecular weight:313.35HP1328
CAS:HP1328: potent FLT3/ITD inhibitor, reduces leukemia, extends survival in mice, belongs to benzoimidazole family.Formula:C23H23N3O3Color and Shape:SolidMolecular weight:389.45Alteminostat
CAS:Alteminostat is used as a histone deacetylase inhibitor and is an antineoplastic drug candidate.Formula:C27H36N6O3Color and Shape:SolidMolecular weight:492.61(-)-Pinocembrin
CAS:(-)-Pinocembrin: Anti-tuberculosis (IC50: 1.11 mg/mL dormant, 1.21 mg/mL active), antiproliferative (IC50: 1.88-11 mg/mL on various cell lines).Formula:C15H12O4Color and Shape:SolidMolecular weight:256.25ALK4290
CAS:ALK4290 (AKST4290), a potent oral CCR3 inhibitor with a Ki of 3.2 nM, may treat macular degeneration and Parkinsonism.Formula:C27H34ClN5O3Color and Shape:SolidMolecular weight:512.04CC-3052
CAS:CC-3052: water-soluble thalidomide analogue, inhibits HIV-1 and TNF-α in PBMC and monocyte adhesion.Formula:C20H21NO5Color and Shape:SolidMolecular weight:355.38PDGFRα/FLT3-ITD-IN-1
CAS:PDGFRα/FLT3-ITD-IN-1 are potent inhibitors of PDGFRα/FLT3, and their IC50 values are greater than 0.036 and 0.003 μM, respectively.Formula:C27H39N9OColor and Shape:SolidMolecular weight:505.66Alcuronium free base
CAS:Alcuronium free base is a non-depolarizing skeletal muscle relaxant similar to Tubocurarine. It is used as an anesthesia adjuvant.Formula:C44H50N4O2Color and Shape:SolidMolecular weight:666.9(R)-Bromoenol lactone
CAS:(R)-Bromoenol lactone (BEL) irreversibly inhibits iPLA2γ with 0.6 μM IC50, not affecting iPLA2β unless at 20-30 μM doses.Formula:C16H13BrO2Color and Shape:SolidMolecular weight:317.18Xanthine oxidase-IN-5
CAS:Xanthine oxidase-IN-5: oral XO inhibitor, IC50 = 0.70 μM, LE = 0.33, LLE = 3.41, reduces uric acid in rats.Formula:C18H16FN3O3Color and Shape:SolidMolecular weight:341.34JO146
CAS:JO146为针对沙眼衣原体高温需要蛋白A(CtHtrA)的蛋白酶抑制剂，其对CtHtrA和人中性粒细胞弹性蛋白酶(HNE)的IC50值分别为21.86 μM和1.15 μM，可应用于细菌感染的抑制。Formula:C31H44N3O7PColor and Shape:SolidMolecular weight:601.67Pildralazine
CAS:Pildralazine, also Propyldazine, is an oral, non-carcinogenic antihypertensive vasodilator similar to hydralazine.Formula:C8H15N5OColor and Shape:SolidMolecular weight:197.24AHR-5645B fumarate
CAS:AHR-5645B fumarate is a substituted benzamide that has been shown to inhibit 3H-spiperone binding to bovine anterior pituitary membranes.Formula:C22H31N3O5Color and Shape:SolidMolecular weight:417.5(6R)-ML753286
(6R)-ML753286, an ML753286 isomer, selectively inhibits BCRP (IC50: 0.6μM), has high permeability, and is stable in plasma.Formula:C20H25N3O3Color and Shape:SolidMolecular weight:355.43m-Toluidine, α-methoxy-4-(octyloxy)-, hydrochloride
CAS:m-Toluidine, alpha-methoxy-4-(octyloxy)-, hydrochloride is a bioactive chemcial.Formula:C16H28ClNO2Color and Shape:SolidMolecular weight:301.85DBHDA
CAS:DBHDA transforms C-terminal Cys into Dha in Ubl G76C mutant probes.Formula:C6H10Br2N2O2Color and Shape:SolidMolecular weight:301.96Falimint
CAS:Falimint is a compound with antipyretic and analgesic activity [1].Formula:C11H14N2O4Color and Shape:SolidMolecular weight:238.24Carbazomycin C
CAS:Carbazomycin C, from Streptomyces, targets S. aureus, B. anthracis, fungi, P. falciparum, and is cytotoxic to several cancer cells, inhibiting 5-LO.Formula:C16H17NO3Color and Shape:SolidMolecular weight:271.31Antitrypanosomal agent 7
CAS:Compound 18c, an antitrypanosomal, is twice as potent as Nifurtimox against T. brucei (IC50: 0.71 μM), with favorable ADME and AT-DNA binding affinity.Formula:C23H29N5O2Color and Shape:SolidMolecular weight:407.51WNK1-IN-1
CAS:WNK1-IN-1, a WNK1 inhibitor (IC50: 1.6 μM), also inhibits OSR1 phosphorylation (IC50: 4.3 μM), used in blood pressure and cancer research.Formula:C13H15BrCl2N2O4SPurity:98.09%Color and Shape:SolidMolecular weight:446.14ts-SA
CAS:ts-SA is a metalloenzyme carbonic anhydrase (CA) inhibitor. It is active against 7 out of 10 human CA isoforms.Formula:C14H15N3O5S2Purity:98%Color and Shape:SolidMolecular weight:369.42Ro 04-5595 free base
CAS:"Ro 04-5595: Selective NMDA NR2B antagonist, EC50 186nmol/L; binds EVT-101 site; hierarchy of inhibition affinity observed."Formula:C19H22ClNO2Color and Shape:SolidMolecular weight:331.84NY0173
CAS:NY0173 is a potent exchange protein activated by cAMP antagonists.Formula:C18H15Cl3N4O2Color and Shape:SolidMolecular weight:425.7IAA-94
CAS:IAA-94 is an inhibitor of chloride channels, it binds channels in bovine kidney cortex microsomes with a Ki value of 1 µM.Formula:C17H18Cl2O4Color and Shape:SolidMolecular weight:357.232'-Deoxy-L-guanosine
CAS:2'-Deoxy-L-guanosine is a nucleoside that shows antibiotic properties by inhibiting protein synthesis, leading to cell death.Formula:C10H13N5O4Color and Shape:SolidMolecular weight:267.24FUBP1-IN-2
CAS:FUBP1-IN-2 hinders FUBP1, affects c-Myc and p21 expression, and depletes polyamines.Formula:C26H26ClN3O4Color and Shape:SolidMolecular weight:479.96Ro 7-0213
CAS:RO 7-0213 is a novel benzodiazepine (RO7-0213) containing a fully positive quaternary ammonium component.Formula:C20H23ClN3OColor and Shape:SolidMolecular weight:356.87ATX inhibitor 16
CAS:ATX inhibitor 16 is a potent inhibitor of ATX (IC50: 0.0021 μM). ATX inhibitor 16 exhibits a significant anti-proliferative effect on breast cancer cells.Formula:C28H27F3N6OS2Color and Shape:SolidMolecular weight:584.68FAUC-299
CAS:FAUC-299 is a dopamine D4 receptor agonist.Formula:C20H20N4Color and Shape:SolidMolecular weight:316.4Nampt activator-3
CAS:NAMPT activator-3: a NAT derivative, EC50 of 2.6 μM, KD 132 nM, protects cells, prevents FK866 toxicity, and is neuroprotective in CIPN mice.Formula:C19H20N2O3Color and Shape:SolidMolecular weight:324.37Lumefantrine Impurity A
CAS:2-(Dibutylamino)-2-(2,7-dichloro-9-(4-chlorobenzylidene)-9H-fluoren-4-yl)ethanol, (RS, Z)- is a bioactive chemical.Formula:C30H32Cl3NOColor and Shape:SolidMolecular weight:528.94Oxyfedrine
CAS:Oxyfedrine: oral β-adrenoreceptor agonist, vasodilator for cardiovascular research.Formula:C19H23NO3Color and Shape:SolidMolecular weight:313.39JS1310
CAS:JS1310 is a selective PRMT7 inhibitor (IC50: 5 μM against human PRMT7). JS1310 has shown anti-cancer effects on different cancer cells.Formula:C23H22FN5O3Color and Shape:SolidMolecular weight:435.45
