Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,763 products)
- Apoptosis(6,207 products)
- Cell Cycle/Checkpoint(4,810 products)
- Chromatin/Epigenetics(2,547 products)
- Cytoskeletal Signaling(1,520 products)
- DNA Damage/DNA Repair(2,908 products)
- Endocrinology/Hormones(3,703 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(9,002 products)
- Immunology and Inflammation(3,751 products)
- Influenza Virus(298 products)
- JAK/STAT signaling(416 products)
- MAPK Signaling(1,245 products)
- Membrane Transporter/Ion Channel(3,103 products)
- Metabolism(10,129 products)
- Microbiology/Virology(7,570 products)
- Neuroscience(10,343 products)
- Other Inhibitors(35,810 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,412 products)
- Proteases/Proteasome(1,682 products)
- Stem Cell and Derivatives(757 products)
- Tyrosine Kinase/Adaptors(1,954 products)
- Ubiquitination(1,715 products)
Show 16 more subcategories
Found 66606 products of "Inhibitors"
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PD-156707
CAS:PD-156707 is a selective antagonist of endothelin A receptor.Formula:C28H26NaO9Purity:98%Color and Shape:SolidMolecular weight:529.497JMX0293
JMX0293, a salicylamide derivative, inhibits STAT3, inducing MDA-MB-231 cell apoptosis with IC50=3.38μM, while sparing MCF-10A (IC50>60μM).Formula:C25H30Cl2N4O7Color and Shape:SolidMolecular weight:569.43CAP-1
CAS:CAP-1 is an inhibitor of HIV-1 capsid formation.Formula:C18H24ClN3O2SColor and Shape:SolidMolecular weight:381.92CAY10701
CAS:CAY10701, a 7-deazahypoxanthine, impedes cell growth (GI50: 9-38 nM) while sparing normal fibroblasts (>1,500-fold), and shrinks mouse colorectal tumors.Formula:C24H19N3O2Color and Shape:SolidMolecular weight:381.43Anticancer agent 60
CAS:Anticancer agent 60 hinders HepG2 cell growth with IC50 of 4.13 μM and suppresses tumors in HepG2 mouse model.Formula:C27H33N5O4SColor and Shape:SolidMolecular weight:523.65NSC1008
CAS:NSC1008 is an inhibitor of the Ras Converting Enzyme 1 (Rce1) protease that disrupts Ras membrane localization in human cells.Formula:C22H18N2OColor and Shape:SolidMolecular weight:326.39Antitumor agent-88
CAS:Antitumor agent-88, a potent antimitotic, arrests G2/M phase, disrupts microtubules in breast cancer, and inhibits CYP1A1 (Ki: 1.4 μM).Formula:C23H30N2O7SColor and Shape:SolidMolecular weight:478.56Cap-dependent endonuclease-IN-3
CAS:Cap-dependent endonuclease-IN-3 inhibits CEN, promising for studying influenza A/B. (Patent WO2019141179A1, compound III-2)Formula:C29H25F2N3O7SColor and Shape:SolidMolecular weight:597.59AChE/BChE-IN-4
CAS:AChE/BChE-IN-4 (BMC-3) crosses the BBB; IC50: hAChE 792 nM, hBChE 2.2 nM. Dual AChE/BChE inhibitor.Formula:C17H26N2O3Color and Shape:SolidMolecular weight:306.4Seladelpar Lysine dihydrate
CAS:Seladelpar lysine, a selective PPAR-δ agonist, is used for the therapy of Homozygous Familial Hypercholesterolemia (HoFH).Formula:C27H41F3N2O9SPurity:98%Color and Shape:SolidMolecular weight:626.68T-1095A
CAS:T-1095A, a T-1095 metabolite, inhibits SGLTs, lowers blood glucose, improves glucose intolerance in mice, and prevents neuropathy in diabetic rats.Formula:C24H26O9Purity:98%Color and Shape:SolidMolecular weight:458.46(+/-)-PPCC oxalate
CAS:Sigma receptor ligand with high sigma-1 affinity; binds sigma-2 as well (Ki = 1.5 & 50.8 nM). Selective over dopaminergic, muscarinic receptors, DAT, SERT.Formula:C50H60N2O10Color and Shape:SolidMolecular weight:849.034Lysinenorleucine
CAS:Lysinenorleucine s a Lysine and hydroxylysine derivatives that can be used for the treatment of malignant and benign tumors.Formula:C12H25N3O4Color and Shape:SolidMolecular weight:275.34N-Boc-15-aminopentadecanoic acid
CAS:N-Boc-15-aminopentadecanoic acid, an alkane with carboxylic end and Boc-protected amine, useful as a PROTAC linker.Formula:C20H39NO4Color and Shape:SolidMolecular weight:357.53Adrafinil, (R)-
CAS:Adrafinil (R)-isomer, former eugeroic for enhancing alertness, attention, and mood in elderly.Formula:C15H15NO3SColor and Shape:SolidMolecular weight:289.35Naftidrofuryl
CAS:Naftidrofuryl treats peripheral and cerebral vascular issues, boosts cell oxidation, and relaxes muscles.Formula:C24H33NO3Color and Shape:SolidMolecular weight:383.52Rimiterol
CAS:Rimiterol, a beta 2 stimulant, therefore affects the cardiovascular system less than isoproterenol.Formula:C12H17NO3Color and Shape:SolidMolecular weight:223.27CGP60474
CAS:CGP60474 is an inhibitor of VEGFR-2 (IC50 = 84 nM) and an inhibitor of ATP-competitive PKC.Formula:C18H18ClN5OPurity:98.81%Color and Shape:SolidMolecular weight:355.82Ref: TM-T14943
1mg34.00€2mg46.00€5mg71.00€10mg92.00€25mg177.00€50mg314.00€100mg518.00€1mL*10mM (DMSO)78.00€BI-831266
CAS:BI-831266 is a potent and selective Aurora kinase B inhibitor.Formula:C27H38ClN7O2Color and Shape:SolidMolecular weight:528.09HPK1-IN-28
CAS:HPK1-IN-28 inhibits HPK1, boosts anti-tumor immunity, and shows promise in immune disease research per patent WO2021175270A1.Formula:C25H22F3N5O4Color and Shape:SolidMolecular weight:513.47FMS586
CAS:FMS586 is a selective antagonist of neuropeptide Y Y5 receptor with oral activity.Formula:C24H30N4OPurity:98%Color and Shape:SolidMolecular weight:390.52U 84569
CAS:U-84569 blocks human platelet clustering by reducing cAMP phosphodiesterase activity and platelet PLC activity.Formula:C25H23NO4Color and Shape:SolidMolecular weight:401.45Fluproquazone
CAS:Fluproquazone: a quinazolinone with strong antipyretic, analgesic effects; scrapped for liver toxicity.Formula:C18H17FN2OPurity:98%Color and Shape:SolidMolecular weight:296.34BKM-570
CAS:BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.Formula:C34H34Cl2F5N3O3Purity:98%Color and Shape:SolidMolecular weight:698.55Amisometradine
CAS:Amisometradine is a diuretic which may be used in the treatment of congestive heart failure.Formula:C9H13N3O2Color and Shape:SolidMolecular weight:195.22FR-48217
CAS:FR-48217 is an immunoactive peptide that inhibits multiplication of HSV-1 and HSV-2.Formula:C40H73N5O10Color and Shape:SolidMolecular weight:784.04RPT193
CAS:RPT193 is an oral CCR4 inhibitor reducing Th2 cell migration in atopic dermatitis, asthma, and allergies.Formula:C27H34Cl3N5O2Color and Shape:SolidMolecular weight:566.95DOV-216,303 Free Base
CAS:DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.Formula:C11H11Cl2NPurity:96.7%Color and Shape:SolidMolecular weight:228.125-(4-amino-2-methoxyphenoxy)-1-phenylpentan-1-ol
CAS:Benzyl alcohol, alpha-(4-(4-amino-2-methoxyphenoxy)butyl)- is a bioactive chemical.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.38Lanceotoxin A
CAS:Lanceotoxin A is a potent Ip blocker.Formula:C32H44O12Purity:98%Color and Shape:SolidMolecular weight:620.68BET-IN-2
CAS:BET-IN-2 is a BET inhibitor (IC50: 52 nM for BRD4-BD1).Formula:C23H29N3OPurity:98%Color and Shape:SolidMolecular weight:363.5Zinterol hydrochloride
CAS:Zinterol HCl is a selective β2-adrenoceptor agonist.Formula:C19H27ClN2O4SColor and Shape:SolidMolecular weight:414.95IDH2R140Q-IN-1
CAS:IDH2R140Q-IN-1 is a potent inhibitor of IDH2R140Q (IC50: 6.1 nM) and can be used in studies of acute myeloid leukemia.Formula:C22H20F6N6Color and Shape:SolidMolecular weight:482.42Talaglumetad hydrochloride
CAS:Talaglumetad hydrochloride, a prodrug of Eglumegad, targets mGluR2/3 to treat psychiatric disorders.Formula:C11H17ClN2O5Color and Shape:SolidMolecular weight:292.72PQ1 Succinate
CAS:PQ1 Succinate boosts GJIC and connexin in breast cancer cells without impacting normal mammary cells.Formula:C25H28F3N3O6Color and Shape:SolidMolecular weight:523.5CS-0045569
CAS:CS-0045569 (ZUN24972) is a drug synthesis intermediate reported in WO 2020086857 as WDR5 inhibitor component.Formula:C12H12O6Color and Shape:SolidMolecular weight:252.22UK 1745
CAS:UK 1745 is a novel drug of cardiotonic.Formula:C16H23ClN2O2Color and Shape:SolidMolecular weight:310.82Quiloflex
CAS:Quiloflex is a central sedative used on animals.Formula:C13H20ClNO3Color and Shape:SolidMolecular weight:273.76Nafazatrom
CAS:Nafazatrom: pyrazolinone lipoxygenase inhibitor, anticancer & antithrombotic, boosts PGI2, reduces arrhythmias.Formula:C16H16N2O2Color and Shape:SolidMolecular weight:268.31CYP3A4-IN-3
CAS:CYP3A4-IN-3, a ritonavir analogue, is a potent CYP3A4 inhibitor with an IC50 of 0.075 μM, used as an antiviral and immunosuppressant.Formula:C34H39N3O3SColor and Shape:SolidMolecular weight:569.76Metanilyl fluoride hydrochloride
CAS:Metanilyl fluoride hydrochloride is a protease inhibitor.Formula:C6H7ClFNO2SColor and Shape:SolidMolecular weight:211.64Grepafloxacin, (S)-
CAS:Grepafloxacin, (S)- is an oral broad-spectrum fluoroquinolone antibacterial used for the treatment of bacterial infections.Formula:C19H22FN3O3Color and Shape:SolidMolecular weight:359.39THIQ-40
CAS:THIQ-40: potent ERα antagonist, oral SERD with antitumor effects.Formula:C28H29NO3Color and Shape:SolidMolecular weight:427.53Dimethenamid
CAS:Dimethenamid is a chloroacetamide herbicide.Formula:C12H18ClNO2SColor and Shape:Yellow-Brown Viscous LiquidMolecular weight:275.80SRTCX1003
CAS:SRTCX1003, a SIRT1 activator, suppresses inflammatory responses through promotion of p65 deacetylation and inhibition of NF-κB activity.Formula:C23H23N5O3SColor and Shape:SolidMolecular weight:449.53Saroglitazar
CAS:Saroglitazar (Lipaglyn) is an agonist of PPAR with EC50 values of 0.65 pM and 3 nM for PPARα and PPARγ.Formula:C25H29NO4SPurity:98.51%Color and Shape:SolidMolecular weight:439.57ERK5-IN-4
CAS:ERK5-IN-4 (34b) is a potent, specific ERK5 inhibitor; IC50: 77 nM full-length, 300 nM ΔTAD in HEK293 cells.Formula:C16H11Cl2FN4O2Color and Shape:SolidMolecular weight:381.19trans-Ned 19
CAS:trans-Ned 19 blocks NAADP and TPC, hindering calcium signaling and aorta relaxation at low histamine levels.Formula:C30H31FN4O3Purity:98%Color and Shape:SolidMolecular weight:514.59TMC310911
CAS:TMC310911 is an oral HIV-1 protease inhibitor with an EC50 of 2.2-14.2 nM, effective against various HIV-1 strains.Formula:C38H53N5O7S2Purity:98%Color and Shape:SolidMolecular weight:755.99INSCoV-601I(1)
CAS:INSCoV-601I(1) is a strong 3CLpro inhibitor, key in SARS-CoV-2 replication; potential for research use - WO2021219089A1.Formula:C23H22ClF2N5O2SColor and Shape:SolidMolecular weight:505.97
