Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,754 products)
- Apoptosis(6,186 products)
- Cell Cycle/Checkpoint(4,807 products)
- Chromatin/Epigenetics(2,573 products)
- Cytoskeletal Signaling(1,503 products)
- DNA Damage/DNA Repair(2,893 products)
- Endocrinology/Hormones(3,702 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,963 products)
- Immunology and Inflammation(3,697 products)
- Influenza Virus(296 products)
- JAK/STAT signaling(414 products)
- MAPK Signaling(1,246 products)
- Membrane Transporter/Ion Channel(3,137 products)
- Metabolism(10,096 products)
- Microbiology/Virology(7,552 products)
- Neuroscience(10,302 products)
- Other Inhibitors(35,769 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,402 products)
- Proteases/Proteasome(1,670 products)
- Stem Cell and Derivatives(742 products)
- Tyrosine Kinase/Adaptors(1,921 products)
- Ubiquitination(1,716 products)
Show 16 more subcategories
Found 66573 products of "Inhibitors"
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MC-70 hydrochloride
CAS:MC-70 hydrochloride inhibits P-gp and BCRP strongly (EC50: Caco-2 0.05μM, MDR1 0.69μM, MRP1 9.3μM, BCRP 73μM).Formula:C24H26ClNO3Color and Shape:SolidMolecular weight:411.926Gemcabene
CAS:Gemcabene (PD-72953) lowers LDL and triglycerides, boosts HDL, and reduces inflammation by decreasing C-reactive protein.Formula:C16H30O5Purity:≥98%Color and Shape:SolidMolecular weight:302.41S-15535
CAS:S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.Formula:C21H24N2O2Purity:98%Color and Shape:SolidMolecular weight:336.43CM764
CAS:CM764 is a potent and selective antagonist of sigma-2 receptors, a novel derivative of SN79.Formula:C23H27FN4O3Color and Shape:SolidMolecular weight:426.48Cemadotin hydrochloride
CAS:Cemadotin hydrochloride (LU103793) is a synthetic mitosis inhibitor derived from Dolastatin 15 for treating solid tumors.Formula:C35H57ClN6O5Color and Shape:SolidMolecular weight:677.33Pralidoxime
CAS:Pralidoxime reactivates AChE blocked by nerve agents, aiding as an organophosphate poisoning antidote.Formula:C7H9N2OColor and Shape:SolidMolecular weight:137.16Gilteritinib hemifumarate
CAS:Gilteritinib hemifumarate (ASP2215 hemifumarate) is a potent ATP-competitive dual FLT3 (IC50: 0.29 nM) and AXL (IC50: 0.73 nM) inhibitor for the treatment of
Formula:C29H44N8O3C4H4O4Purity:99.78%Color and Shape:SolidMolecular weight:610.75JNJ-4929821
CAS:JNJ-4929821 is a potent, reversible methionine aminopeptidase-2 (MetAP-2) inhibitor with IC50 of 8 nM.Formula:C14H13FN4O2S2Color and Shape:SolidMolecular weight:352.41Tau-aggregation-IN-1
CAS:Tau-aggregation-IN-1 is a dopamine D2 and D3 receptor agonist and an inhibitor of tau441 protein aggregation (IC50: 21 μM).Formula:C28H37N5O2SColor and Shape:SolidMolecular weight:507.69BET bromodomain inhibitor 2
CAS:BET bromodomain inhibitor 2 is a potent inhibitor of the BET-type bromodomain (IC50: 14.1 μM).Formula:C23H30N2O5SColor and Shape:SolidMolecular weight:446.56GEM144
CAS:GEM144: oral POLA1/HDAC11 inhibitor; boosts p53, p21; halts G1/S cycle; triggers cell death.Formula:C28H31NO5Color and Shape:SolidMolecular weight:461.55Reteplase
CAS:Reteplase, a recombinant plasminogen activator from t-PA's domains, is made via DNA tech in E. coli.Color and Shape:SolidP2X2/3 modulator-1
CAS:Compound 46, a P2X2/3 modulator, could aid in research of pain, CNS disorders, and inflammation.Formula:C26H21N5OColor and Shape:SolidMolecular weight:419.487-Methotrexate
CAS:7-Methotrexate: chemotherapy, treats cancer, autoimmune disorders, ectopic pregnancy and aids medical abortions.Formula:C20H22N8O5Color and Shape:SolidMolecular weight:454.44(Rac)-CFT7455
CAS:(Rac)-CFT7455 degrades Ikaros/Aiolos via ubiquitin pathway, effective on NCIH929.1 (GI50: 0.05 nM), racemic with anticancer properties.Formula:C28H27N3O4Color and Shape:SolidMolecular weight:469.53GTC365
CAS:GTC365 is an hTERT transcriptional repressor that acts in the early stages of the G-quadruplex folding pathway.Formula:C23H25Cl2N7O4SColor and Shape:SolidMolecular weight:566.46NGB-2849
CAS:NGB-2849 is a selective dopamine D3 receptor antagonist.Formula:C29H29Cl2N3OColor and Shape:SolidMolecular weight:506.47DHODH-IN-21
CAS:DHODH-IN-21, orally active DHODH blocker with 1.1 nM IC50, shows anticancer activity, potential for AML research.Formula:C20H19ClF4N6O4Color and Shape:SolidMolecular weight:518.85AHR-16329
CAS:AHR-16329 can be used in ocular pharmacology.Formula:C11H14ClN3O4SColor and Shape:SolidMolecular weight:319.77Antimycobacterial agent-2
CAS:Antimycobacterial agent-2 has MIC99 0.8 μM vs M.tb H37Rv; cytotoxic with IC50 48.1 μM on CHO cells.Formula:C31H50O5Color and Shape:SolidMolecular weight:502.73AVN-101 free base
CAS:AVN-101: potent 5-HT7 antagonist, also targets 5-HT6, 5-HT2A, 5-HT2C. Aims to treat CNS disorders.Formula:C21H24N2Color and Shape:SolidMolecular weight:304.43PI3Kδ-IN-11
CAS:PI3Kδ-IN-11 is a potent and selective PI3Kδ inhibitor (IC50: 27.5 nM) that dose-dependently blocks PI3K/Akt pathway activity.Formula:C27H21N5OColor and Shape:SolidMolecular weight:431.49HIF-PHD-IN-2
CAS:HIF-PHD-IN-2 (compound 25) is a highly effective PHD inhibitor, displaying IC50 values below 100 nM for PHD1, PHD2, and PHD3 [1].Formula:C17H15N5O3SColor and Shape:SolidMolecular weight:369.4BTK-IN-9
CAS:BTK-IN-9 reversibly inhibits BTK, disrupts mitochondria, boosts ROS, and triggers apoptosis in Z138 cells, impeding condyloma cell growth.Formula:C25H19N7O4Color and Shape:SolidMolecular weight:481.46ER-38925
CAS:ER-38925 is a retinoic acid receptor (rar) subtype α-selective agonistFormula:C21H17NO3Color and Shape:SolidMolecular weight:331.36Intiquinatine
CAS:Intiquinatine (Tiliquinatine) may have potential anticancer activity.Formula:C18H14BrNO4Color and Shape:SolidMolecular weight:388.21(S)-Gyramide A
CAS:(S)-Gyramide A is a bacterial DNA gyrase inhibitor that acts by exhibiting antimicrobial activity and inhibiting bacterial cell division.Formula:C21H27FN2O3SPurity:98%Color and Shape:SolidMolecular weight:406.51SK 946
CAS:SK 946 is a cognition activator.Formula:C15H21N3O2Color and Shape:SolidMolecular weight:275.352PC170942 Sodium
CAS:PC170942 Sodium is a water-soluble bacterial cytokinesis inhibitor that acts by inhibiting FtsZ.Formula:C24H24ClNO2SPurity:98%Color and Shape:SolidMolecular weight:425.97SC 11927
CAS:SC 11927 is an aldosterone antagonist.Formula:C22H30FKO5Color and Shape:SolidMolecular weight:432.57Silatrane
CAS:Silatrane is a reversible cholinesterase inhibitor and anti-tumor agent.Formula:C6H13NO3SiColor and Shape:SolidMolecular weight:175.26Stampidine
CAS:Stampidine prevents HIV-1, effective against resistant strains at subnanomolar levels.Formula:C20H23BrN3O8PPurity:98%Color and Shape:SolidMolecular weight:544.29hClpP-activator-D9
CAS:hClpP-activator-D9 is a novel potent and species-selective activator of human ClpP (hClpP).Formula:C18H13ClFN3O4Color and Shape:SolidMolecular weight:389.76LR 16
CAS:LR 16 has potent effects on oxygen affinity of hemoglobin, on blood cholesterol and on low density lipoprotein.Formula:C17H16Cl2N2O4Color and Shape:SolidMolecular weight:383.23(2R,5S)-Ritlecitinib
CAS:(2R,5S)-Ritlecitinib ((2R,5S)-PF-06651600) is a potent and selective inhibitor of JAK3 with IC 50 of 144.8 nM[1].Formula:C15H19N5OColor and Shape:SolidMolecular weight:285.34SWE101
CAS:SWE101 is a potent human and rat soluble epoxide hydrolase (sEH)-P inhibitor(IC50s of 4 μM and 2.8 μM, respectively).Formula:C19H15Cl2NO3Purity:98%Color and Shape:SolidMolecular weight:376.23Albaconazole
CAS:Albaconazole, a small fungal CYP51A1 inhibitor, treats fungal infections and some musculoskeletal disorders.Formula:C20H16ClF2N5O2Purity:99.27%Color and Shape:SolidMolecular weight:431.82Ref: TM-T7725
1mg315.00€5mg745.00€10mg1,018.00€25mg1,431.00€50mg1,783.00€100mg2,250.00€500mg4,410.00€trans-Cephalosporin
CAS:Trans-substituted cephalosporin is an efficient inhibitor of NDM-1, demonstrating an IC50 value of 0.13 μM.Formula:C16H14N2O4S3Color and Shape:SolidMolecular weight:394.49Talarozole (R enantiomer)
CAS:Talarozole R enantiomer is a potent and selective inhibitor of cytochrome P450 26-mediated breakdown of endogenous all-trans retinoic acid.Formula:C21H23N5SPurity:98%Color and Shape:SolidMolecular weight:377.51Acetamide, N-(5-(p-aminophenoxy)pentyl)-2-cyano-
CAS:Acetamide, N-(5-(p-aminophenoxy)pentyl)-2-cyano- is a Drug / Therapeutic Agent.Formula:C14H19N3O2Color and Shape:SolidMolecular weight:261.32VUF14862
CAS:VUF14862 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Formula:C26H32N4O2Color and Shape:SolidMolecular weight:432.56AZD 1152 (hydrochloride)
CAS:AZD 1152, an oral prodrug, becomes AZD 1152-HQPA in plasma, selectively inhibits Aurora kinase B (IC50=0.36 nM), and blocks tumor growth.Formula:C26H33Cl2FN7O6PColor and Shape:SolidMolecular weight:660.47RK-52
CAS:RK-52: synthetic rhodesain inhibitor; ksecond = 67M min^-1, Ki = 38 pM, high affinity for trypanosomal protease.Formula:C30H32N2O4Color and Shape:SolidMolecular weight:484.59Tec-IN-21
CAS:Tec-IN-21 is an inhibitor of Tec kinase, it also blocks unconventional secretion of fibroblast growth factor 2 (FGF2).Formula:C16H15ClN4O2SPurity:98%Color and Shape:SolidMolecular weight:362.83sEH inhibitor-6
CAS:sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].Formula:C21H14ClN3O2Color and Shape:SolidMolecular weight:375.81IM-93
CAS:IM-93 inhibits ferroptosis and NETosis with an IC< sub>50 of 0.45 μM for cell death inhibition [1].Formula:C21H28N4O2Color and Shape:SolidMolecular weight:368.47GPR35 agonist 1
CAS:GPR35 agonist 1 is a highly effective and specific GPR35/CXCR8 agonist (EC50: 5.8 nM).Formula:C10H4BrN5O5Purity:98%Color and Shape:SolidMolecular weight:354.07ROCK-IN-D3
CAS:ROCK-IN-D3 is an effective and selective inhibitor of ROCK.Formula:C20H22N4OPurity:98%Color and Shape:SolidMolecular weight:334.41ABT-770
CAS:ABT-770: an orally potent and selective MMP inhibitor, shown to reduce tumor growth in animal models.Formula:C22H22F3N3O6Color and Shape:SolidMolecular weight:481.42(R)-SKF-82957 hydrobromide
CAS:(R)-SKF-82957 hydrobromide is a selective D1 dopamine receptor agonistFormula:C17H19BrClNO2Color and Shape:SolidMolecular weight:384.7
