Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,838 products)
- Apoptosis(6,316 products)
- Cell Cycle/Checkpoint(4,881 products)
- Chromatin/Epigenetics(2,615 products)
- Cytoskeletal Signaling(1,570 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,753 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,023 products)
- Immunology and Inflammation(3,903 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,258 products)
- Membrane Transporter/Ion Channel(3,159 products)
- Metabolism(10,130 products)
- Microbiology/Virology(7,618 products)
- Neuroscience(10,516 products)
- Other Inhibitors(35,844 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,431 products)
- Proteases/Proteasome(1,688 products)
- Stem Cell and Derivatives(729 products)
- Tyrosine Kinase/Adaptors(1,983 products)
- Ubiquitination(1,727 products)
Show 16 more subcategories
Found 66513 products of "Inhibitors"
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FR-194921
CAS:FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.Formula:C23H23N5OColor and Shape:SolidMolecular weight:385.46HEAT hydrochloride
CAS:HEAT hydrochloride is an α1-adrenoceptor antagonist.Formula:C19H22ClNO2Purity:98%Color and Shape:SolidMolecular weight:331.84Emiglitate
CAS:Emiglitate is a selective and competitive α-glucoside hydrolase inhibitor.Formula:C17H25NO7Purity:98%Color and Shape:SolidMolecular weight:355.38Pulrodemstat Methylbenzenesulfonate
CAS:LSD1-IN-7 Methylbenzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.Formula:C31H31F2N5O5SPurity:98%Color and Shape:SolidMolecular weight:623.67Hydrocarbon chain derivative 1
CAS:Hydrocarbon chain derivative 1 has inhibitory activities against lipid synthesis.Formula:C16H34O3Purity:98%Color and Shape:SolidMolecular weight:274.44MNI-caged-L-glutamate
CAS:rapidly and efficiently releases glutamateFormula:C14H17N3O6Purity:98%Color and Shape:SolidMolecular weight:323.3S 14506 hydrochloride
CAS:S 14506 hydrochloride is a 5-HT1A receptor full agonist.Formula:C24H27ClFN3O2Purity:99.92%Color and Shape:SolidMolecular weight:443.94Eggmanone
CAS:EGM1: potent PDE4D3 inhibitor, IC50=72 nM, 40-50x selectivity over other PDEs, activates PKA, blocks Hh.Formula:C20H20N2O2S3Color and Shape:SolidMolecular weight:416.58BO3482
CAS:BO3482 is an antimicrobial compound and can inhibit the growth of methicillin-resistant Staphylococci (MIC90: 6.25 mg/mL).Formula:C14H20N2NaO5S2Purity:98%Color and Shape:SolidMolecular weight:383.43Tubulin polymerization-IN-22
CAS:Tubulin polymerization-IN-22 inhibits tubulin (IC50=8.1μM), blocks G2/M phase, and triggers apoptosis.Formula:C19H16O4Color and Shape:SolidMolecular weight:308.33Demethoxyviridiol
CAS:Demethoxyviridiol is a mycotoxin that inhibits phosphatidylinositol 3-kinase (PI3K).Formula:C19H16O5Color and Shape:SolidMolecular weight:324.33iNOs-IN-3
CAS:iNOs-IN-3: oral iNOS inhibitor, IC50 = 3.342 μM, anti-inflammatory, for LPS-induced ALI study.Formula:C27H24N2O5SColor and Shape:SolidMolecular weight:488.55PKI-179
CAS:PKI-179: Dual PI3K/mTOR inhibitor, orally active, IC50s: 0.42-77 nM, targets E545K and H1047R, antitumor in vivo.Formula:C25H28N8O3Color and Shape:SolidMolecular weight:488.54FR-182024
CAS:FR-182024 is a novel cephem derivative, it has potent anti-Helicobacter pylori activity.Formula:C18H16N4O4S3Color and Shape:SolidMolecular weight:448.54Resminostat
CAS:Resminostat (4SC-201) is an orally bioavailable inhibitor of histone deacetylases (HDACs) with potential antineoplastic activity.Formula:C16H19N3O4SPurity:99.46%Color and Shape:SolidMolecular weight:349.4AMP-Deoxynojirimycin
CAS:AMP-Deoxynojirimycin (AMP-DNM) is a ceramide glucosyltransferase and GCase 2 inhibitor for the study of Parkinson's and diabetes.Formula:C22H39NO5Purity:>99.99%Color and Shape:SolidMolecular weight:397.55TMB 8 (hydrochloride)
CAS:TMB 8 blocks nAChRs (IC50: 390-480 nM), reduces Ca2+ in muscles, hinders rabbit aorta contraction at 50 μM, and inhibits PKC dose-dependently.Formula:C22H38ClNO5Color and Shape:White SolidMolecular weight:431.99DA 3505
CAS:DA 3505, a feprazone metabolite, detectable at 0.1μg/ml (feprazone) & 0.2μg/ml (metabolite) via HPLC, 0.5μg/ml with TLC.Formula:C20H20N2O3Color and Shape:SolidMolecular weight:336.38SCH-23985
CAS:SCH-23985 is an antagonist of D1 dopamine receptor.Formula:C18H20ClNOPurity:98%Color and Shape:SolidMolecular weight:301.81Bepotastine tosylate
CAS:Bepotastine tosylate: Oral 2nd-gen H1 antagonist, inhibits histamine effects on NGF; treats conjunctivitis, urticaria.Formula:C28H33ClN2O6SColor and Shape:SolidMolecular weight:561.09COX-1/2-IN-1
CAS:"COX-1/2-IN-2: Strong dual inhibitor of COX-1 (IC50 = 13.9 μM) and COX-2 (IC50 = 6.4 μM)."Formula:C15H10BrClN2OColor and Shape:SolidMolecular weight:349.61Anisodine hydrobromide
CAS:Anisodine hydrobromide is an inhibitor of adenosine kinase.Formula:C17H22BrNO5Color and Shape:White Crystals Or Crystalline PowderMolecular weight:400.27PXYC13
CAS:PXYC13 inhibits Mtb RpsA essential for trans-translation with Kd of 7.61 μM; less effective on RpsA-CTD Δ438A (Kd 8.50 μM).Formula:C15H15N5O2SColor and Shape:SolidMolecular weight:329.38DSM74
CAS:DSM74 is a metabolically stable dihydroorotate dehydrogenase inhibitor that has antimalarial activity.Formula:C13H10F3N5Purity:98%Color and Shape:SolidMolecular weight:293.25PHA-680626
CAS:PHA-680626 is a PLK inhibitor, effective on resistant leukemia cells, with IC50: Plk1 (0.53 μM), Plk2 (0.07 μM), Plk3 (1.61 μM).Formula:C23H26N6O2SColor and Shape:SolidMolecular weight:450.56Carbuterol hydrochloride
CAS:Carbuterol hydrochloride is a short-acting β2 adrenoreceptor agonist.Formula:C13H22ClN3O3Color and Shape:SolidMolecular weight:303.79Sortin1
CAS:Sortin1, a chemical genetic-hit compound, specifically induces mislocalization of both soluble and membrane-associated vacuolar markers in plants and yeast.Formula:C26H19NO6Purity:98%Color and Shape:SolidMolecular weight:441.43Btm 1042
CAS:Btm 1042 is an antispasmodic drug. It has been found to depress twitch responses in the ileum of guinea pigs.Formula:C21H26ClN3OSColor and Shape:SolidMolecular weight:403.97Famiraprinium
CAS:Famiraprinium is a competitive antagonist at the GABA receptor site.Formula:C15H17N3O2Color and Shape:SolidMolecular weight:271.31NVS-CRF38
CAS:NVS-CRF38 is an antagonist of corticotropin-releasing factor receptor 1 (CRF1).Formula:C19H21N5O2Purity:98%Color and Shape:SolidMolecular weight:351.4CRA1000
CAS:CRA1000, a CRF1 receptor antagonist, involved in the regulation of stress response.Formula:C28H33FN4SPurity:98%Color and Shape:SolidMolecular weight:476.65WNK-IN-3
CAS:WNK-IN-3 is a novel allosteric inhibitor of WNK kinase.Formula:C27H32F3N7O2Color and Shape:SolidMolecular weight:543.58HAT-IN-1
CAS:HAT-IN-1 is an inhibitor of HAT used in the research of cancer.Formula:C23H18BrF4N3O4Purity:98%Color and Shape:SolidMolecular weight:556.3Suclofenide
CAS:Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.Formula:C16H13ClN2O4SPurity:98%Color and Shape:SolidMolecular weight:364.8ARI-3099
CAS:ARI-3099 inhibits fibroblast activation protein, alpha (FAP).Formula:C13H18BN3O4Color and Shape:SolidMolecular weight:291.11Carboxyamidotriazole
CAS:Carboxyamidotriazole is a cytostatic inhibitor of non-voltage-operated calcium channels and calcium channel-mediated signaling pathways.Formula:C17H12Cl3N5O2Purity:98%Color and Shape:SolidMolecular weight:424.67CDKi Hydrochloride
CAS:CDKi hydrochloride is a potent and selective ATP competitive inhibitor of cycB-CDK1, cycE-CDK2, and cycD1-CDK4.Formula:C4H6N4OColor and Shape:SolidMolecular weight:126.12Aminochlorthenoxazin
CAS:Aminochlorthenoxazin is an antipyretic and analgesic agent.Formula:C10H11ClN2O2Purity:98%Color and Shape:SolidMolecular weight:226.66NPP1-IN-1
CAS:NPP1-IN-1 is a highly potent inhibitor of NPP enzymes, effectively inhibiting NPP1 with an IC 50 value of 0.15 μM and NPP3 with an IC 50 value of 40 μM [1].Formula:C27H21NO2Color and Shape:SolidMolecular weight:391.46Saikosaponin B4
CAS:Saikosaponin B4 is isolated from the MeOH extract of the roots of Bupleurum falcatum L.Formula:C43H72O14Purity:99.03%Color and Shape:SolidMolecular weight:813.02HUHS2002
CAS:HUHS2002 is a free fatty acid derivative that works as a potentiator of GluA1 AMPA receptor responses and α7 ACh receptor responses.Formula:C17H24O3Purity:98%Color and Shape:SolidMolecular weight:276.37LEI-101
CAS:LEI-101: potent CB2 agonist, pEC50=8, bioavailable, >100x selective over CB1, potential for inflammatory diseases.Formula:C23H25FN4O4SPurity:98%Color and Shape:SolidMolecular weight:472.53Tubulin inhibitor 23
CAS:Potent Tubulin inhibitor 23 (IC50: 4.8 μM) induces apoptosis and has dose-dependent antiangiogenic properties, promising for leukemia research.Formula:C26H23NO6SColor and Shape:SolidMolecular weight:477.53DC_M5_2
CAS:DC_M5_2 is a novel inhibitor of wdr5-mll1 interactionFormula:C22H22BrNO5Color and Shape:SolidMolecular weight:460.32ZD7114 free base
CAS:ZD7114 (ICI-D7114) selectively activates brown fat, boosts thermogenesis, and aids in obesity and metabolic disorders.Formula:C22H30N2O6Color and Shape:SolidMolecular weight:418.48CSF1R-IN-14
CAS:CSF1R-IN-14, an isoindolinone derivative, powerfully inhibits CSF1R, with potential in cancer research. See WO2019134662A1, compound 1.Formula:C23H22F3N5OColor and Shape:SolidMolecular weight:441.454-CPI
CAS:4-CPI inhibits non-active site mutants of cytochrome P450 2B4.Formula:C9H7ClN2Purity:98%Color and Shape:SolidMolecular weight:178.62CP94253 hydrochloride
CAS:CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).Formula:C15H20ClN3OPurity:99.78%Color and Shape:SolidMolecular weight:293.79Ref: TM-T22689
5mg66.00€1mL*10mM (DMSO)66.00€10mg90.00€25mg205.00€50mg334.00€100mg537.00€200mg745.00€UNC6212 (Kme2)
UNC6212 (Kme2), a dimethyllysine (Kme2)-containing ligand, has a K D for CBX5 of 5.7 μM .Formula:C39H53N7O11Color and Shape:SolidMolecular weight:795.88Anticancer agent 83
CAS:Anticancer agent 83: potent, GI50 0.15 mM against LOX IMVI, reduces mitochondria potential, DNA damage, induces leukemia apoptosis.Formula:C20H19N5OSColor and Shape:SolidMolecular weight:377.46
