Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,849 products)
- Apoptosis(6,366 products)
- Cell Cycle/Checkpoint(4,907 products)
- Chromatin/Epigenetics(2,625 products)
- Cytoskeletal Signaling(1,585 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,759 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,051 products)
- Immunology and Inflammation(3,945 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,163 products)
- Metabolism(10,148 products)
- Microbiology/Virology(7,672 products)
- Neuroscience(10,549 products)
- Other Inhibitors(35,858 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(734 products)
- Tyrosine Kinase/Adaptors(1,991 products)
- Ubiquitination(1,744 products)
Show 16 more subcategories
Found 66516 products of "Inhibitors"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Dapaconazole
CAS:Dapaconazole is used as a drug candidate for antifungals.Formula:C19H15Cl2F3N2OColor and Shape:SolidMolecular weight:415.24GF 15
CAS:GF 15 is a potent inhibitor of centrosomal clustering in tumor cells.Formula:C23H21ClO6Purity:98%Color and Shape:SolidMolecular weight:428.86Clentiazem maleate
CAS:Clentiazem maleate is a calcium channel antagonist .Formula:C26H29ClN2O8SColor and Shape:SolidMolecular weight:565.034OKY 1581
CAS:OKY 1581 is a new thromboxane synthetase inhibitorFormula:C16H14NNaO2Color and Shape:SolidMolecular weight:275.28Benamocaine
CAS:Benamocaine is a biochemical.Formula:C19H21NO2Color and Shape:SolidMolecular weight:295.38Pomisartan
CAS:Pomisartan (BIBR-363) is a small molecule angiotensin type 1 receptor (AT1R) antagonist that is used in the treatment of cardiovascular disease, studying heartFormula:C31H30N4O2Purity:>99.99%Color and Shape:SolidMolecular weight:490.6Lidoflazine
CAS:Lidoflazine: antianginal, blocks HERG K+ & Ca channels, risks QT prolongation & arrhythmia.Formula:C30H35F2N3OPurity:98%Color and Shape:SolidMolecular weight:491.62ER21355
CAS:ER21355, utilized for the treatment of prostatic diseases, acts as a phosphodiesterase 5 (PDE5) inhibitor.Formula:C22H21ClN4O4Purity:98%Color and Shape:SolidMolecular weight:440.88DAT 582
CAS:DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agentFormula:C22H28ClN5OPurity:98%Color and Shape:SolidMolecular weight:413.95NHE3-IN-3
CAS:NHE3-IN-3 inhibits human/rat NHE3 with pIC50s 6.2/6.6; 98% oral bioavailability in rats.Formula:C16H16Cl2N2O2SColor and Shape:SolidMolecular weight:371.28Bromodomain inhibitor-9
CAS:Bromodomain inhibitor-9 selectively targets BRD4-1 (Kd 12 nM), used in metabolic, inflammatory, fibrotic, and autoimmune disease studies.Formula:C24H28N4O5SColor and Shape:SolidMolecular weight:484.57AM-206
CAS:AM-206 is a bio-active chemical.Formula:C25H22F3N2NaO4Color and Shape:SolidMolecular weight:494.44CDMG1
CAS:CDMG1: Novel Wnt inhibitor that aids heart repair and growth by increasing cardiac progenitor cells.Formula:C14H15N5SColor and Shape:SolidMolecular weight:285.37Cgs 27830
CAS:Cgs 27830 is an Endothelin Receptor Antagonist.Formula:C32H30N4O11Color and Shape:SolidMolecular weight:646.6NBOH-2C-CN hydrochloride
CAS:5-HT2A agonistFormula:C18H21ClN2O3Purity:98%Color and Shape:SolidMolecular weight:348.82Dehydrodeoxy donepezil
CAS:Dehydrodeoxy donepezil is an inhibitor of acetylcholinesterase (AChE)Formula:C24H29NO2Color and Shape:SolidMolecular weight:363.49BI-4834
CAS:BI-4834, a potent PLK1 inhibitor with high selectivity, IC50: 7.6 nm. More selective than BI-2536, especially against PLK3.Formula:C32H47N7O4Color and Shape:SolidMolecular weight:593.76CT-1
CAS:CT-1 is a DNA minor groove ligand and causes p53-dependent breast cancer cell apoptosis.
Formula:C29H23F3N4OPurity:99.79%Color and Shape:SolidMolecular weight:500.51PD-1/PD-L1-IN-NP19
CAS:PD-1/PD-L1-IN-NP19: a PD-1/PD-L1 inhibitor with 12.5 nM IC50, may boost antitumor immunity.Formula:C33H31ClN2O4Purity:96.70%Color and Shape:SolidMolecular weight:555.06Sch 39304
CAS:Sch 39304 is an oral triazole antifungal.Formula:C13H15F2N3O3SColor and Shape:SolidMolecular weight:331.34PIKfyve-IN-2
CAS:PIKfyve-IN-2 is a potent inhibitor of the PIKfyve kinase, with potential applications in cancer and autoimmune disorder research [1].Formula:C22H22N8OColor and Shape:SolidMolecular weight:414.46Apoptosis inducer 8
CAS:Apoptosis inducer 8 is a galectin-1 (gal-1)-mediated apoptosis inducer and a PET imaging agent that significantly reduces gal-1 protein levels and can be usedFormula:C29H22ClN5O2Color and Shape:SolidMolecular weight:507.97CI 924
CAS:CI 924 is a lipid-lowering drug. CI 924 increased anti-atherosclerotic HDL and decreased VLDL at 600 mg/day.Formula:C26H34O6Color and Shape:SolidMolecular weight:442.54CH5164840
CAS:CH5164840: strong HSP90 blocker; excels in NSCLC treatment; boosts erlotinib efficacy on EGFR-mutant tumors.Formula:C19H23N5O2SColor and Shape:SolidMolecular weight:385.48Fenmetozole Tosylate
CAS:Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,Formula:C17H18Cl2N2O4SPurity:98%Color and Shape:SolidMolecular weight:417.31DB-959 (free base)
CAS:DB-959 is a potential agonist of PPAR.Formula:C25H27NO5Color and Shape:SolidMolecular weight:421.49Safusidenib
CAS:Safusidenib, oral mutant IDH1 inhibitor, selectively targets IDH1R132H/C mutations with IC50 of 15/130 nM; impairs chondrosarcoma growth.Formula:C25H18Cl3FN2O4Color and Shape:SolidMolecular weight:535.78U 80816B
CAS:U 80816B is a cholinergic direct agonist.Formula:C12H16BrN3OColor and Shape:SolidMolecular weight:298.184Y06036
CAS:Y06036, a potent and selective BET inhibitor, can bind to the BRD4(1) bromodomain (Kd: 82 nM).Formula:C16H15BrN2O5SPurity:99.97%Color and Shape:SolidMolecular weight:427.27ARN14988
CAS:ARN14988 inhibits human acid ceramidase (IC50 = 12.8 nM), increases C16 ceramides in melanoma cells, and reduces A375/G361 cell growth (EC50 = 41.8/67.7 μM).Formula:C16H24ClN3O5Color and Shape:SolidMolecular weight:373.83Paltusotine HCl
CAS:Paltusotine, also known as CRN00808, is a somatostatin receptor agonist.Formula:C27H24Cl2F2N4OColor and Shape:SolidMolecular weight:529.41LDDN-0003499
CAS:LDDN-0003499 is a novel Src family tyrosine kinase inhibitor with anti-inflammatory effects in response to Aß stimulation of microglia.Formula:C16H13Cl2N3O2Color and Shape:SolidMolecular weight:350.2MP-135
CAS:MP135, a μ-δ opioid receptor agonist, needs refining to reduce classical side effects like respiratory depression.Formula:C32H38FN3O2Color and Shape:SolidMolecular weight:515.66DHFR-IN-1
CAS:DHFR-IN-1: selective DHFR blocker, IC50 40.71 nM, antifungal, strong against Gram-positive/negative bacteria, synergizes with Levofloxacin (FIC=0.249).Formula:C22H22N6O4S2Color and Shape:SolidMolecular weight:498.58NV-5440
CAS:NV-5440 is a novel cell penetrant, potent and selective class I glucose transporters (GLUT1) inhibitor, selectively inhibiting mTORC1Formula:C31H36N6O3SColor and Shape:SolidMolecular weight:572.72STING Agonist 1a
CAS:STING agonist 1a activates STING, induces IRF-SEAP, IFN-β, IL-6, CXCL10 (EC50=16.77 µM); effects reversed by STING KO/inhibitor H-151.Formula:C19H11Cl2N5OColor and Shape:SolidMolecular weight:396.23CGP-75254A
CAS:CGP-75254A is a novel oral iron chelator.Formula:C22H28N2NaO6Color and Shape:SolidMolecular weight:439.464Antitubercular agent-24
CAS:Compound 1: Antitubercular, fights M. tuberculosis H37Rv, IC50 - extracellular 0.83 μM, intracellular 0.17 μM.Formula:C18H19N3O2S2Color and Shape:SolidMolecular weight:373.49AHR-10718
CAS:AHR-10718 has an antiarrhythmic effect.Formula:C22H35N3O7SPurity:98%Color and Shape:SolidMolecular weight:485.6CL67
CAS:CL67 is a hypoxia-inducible factor pathway inhibitor. It acts by binding to a G-quadruplex higher-order structure in the HIF promoter sequence in vitro.Formula:C38H42N10O2Color and Shape:SolidMolecular weight:670.81BMS-663749 lysine
CAS:BMS-663749 lysine is used as a phosphonooxymethyl prodrug 4 for HIV-1 attachment inhibitor.Formula:C29H39N6O11PPurity:98%Color and Shape:SolidMolecular weight:678.63Aldose reductase-IN-4
CAS:Aldose reductase-IN-4 (compund IIc) is an inhibitor of aldose reductase with IC50s of 11.70 μM and 0.98 μM for ALR1 and ALR2, respectively [1].Formula:C14H10FNO3SColor and Shape:SolidMolecular weight:291.3PNU-107484A
CAS:PNU-107484A is a unique GABA(A) receptor ligand.Formula:C18H23ClN6Purity:98%Color and Shape:SolidMolecular weight:358.87Zimelidine
CAS:Zimelidine, a withdrawn antidepressant, posed Guillain-Barre risk.Formula:C16H17BrN2Purity:98%Color and Shape:SolidMolecular weight:317.22CInQ-03
CAS:CInQ-03 is a novel and specific MEK inhibitor both in vitro and in vivo.Formula:C22H12ClN5OColor and Shape:SolidMolecular weight:397.82Nizatidine amide
CAS:Nizatidine amide blocks H2 receptors, reducing stomach acid to treat ulcers and GERD.Formula:C11H18N4O3S2Color and Shape:SolidMolecular weight:318.427DG
CAS:7DG is a selective inhibitor of protein kinase R (PKR).Formula:C26H30O5Color and Shape:SolidMolecular weight:422.51DA-7867
CAS:DA-7867, an oxazolidinone, has lower MIC(≤0.25 μg/ml) against aerobic gram-positive bacteria than linezolid, with MIC(90) at 0.125 μg/ml.Formula:C19H18FN7O3Color and Shape:SolidMolecular weight:411.39PCAF-IN-2
CAS:PCAF-IN-2 inhibits PCAF (IC50 = 5.31 µM), induces apoptosis, and halts G2/M cell cycle, showing anti-tumor properties.Formula:C10H7F3N6Color and Shape:SolidMolecular weight:268.2
