Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,856 products)
- Apoptosis(6,375 products)
- Cell Cycle/Checkpoint(4,913 products)
- Chromatin/Epigenetics(2,633 products)
- Cytoskeletal Signaling(1,590 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,765 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,055 products)
- Immunology and Inflammation(3,957 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,162 products)
- Metabolism(10,157 products)
- Microbiology/Virology(7,674 products)
- Neuroscience(10,550 products)
- Other Inhibitors(35,861 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,438 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,992 products)
- Ubiquitination(1,744 products)
Show 16 more subcategories
Found 66511 products of "Inhibitors"
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GSK-3β inhibitor 8
CAS:GSK-3β inhibitor 8 (GSK3β Inhibitor XVIII) is a potent and selective GSK-3β inhibitor with an IC50 value of 64 nM.GSK-3β inhibitor 8 is a thienopyrimidineFormula:C20H20ClN5OSPurity:98.46%Color and Shape:SolidMolecular weight:413.92Bactobolamine
CAS:Bactobolamine, an immunosuppressant, suppresses IL-2 production in CTLL cells at a concentration of 200 µg/ml and extends heart allograft survival in both MHC-Formula:C11H15Cl2NO5Color and Shape:SolidMolecular weight:312.15NSC309401
CAS:NSC309401 is an E. coli dihydrofolate reductase inhibitor, displaying potency with an IC50 value of 189 nM and a dissociation constant (KD) of 14.57 nM [1].Formula:C17H16N6Color and Shape:SolidMolecular weight:304.35VU0360172
CAS:VU0360172 is a positive allosteric modulator of mGlu5 receptors (EC50 = 16 nM; Ki = 195 nM).Formula:C18H15FN2OPurity:99.56%Color and Shape:SolidMolecular weight:294.32ICMT-IN-5
CAS:ICMT-IN-5 (compound 46) is an ICMT inhibitor with an IC50 value of 0.3 μM [1].Formula:C22H28FNOColor and Shape:SolidMolecular weight:341.46KS I
CAS:KS I is a gonadotropin antagonist and is a cyclolignan isolated from extracts of Lycopus and Lithosperum after oxidation with caffeic acid.Formula:C18H14O8Color and Shape:SolidMolecular weight:358.3Luminespib mesylate
CAS:Luminespib (AUY-922) is a 3rd-gen Hsp90 inhibitor, disrupting tumor cell proliferation & oncogenic proteins, raising Hsp72 levels.Formula:C27H33N3O5Color and Shape:SolidMolecular weight:479.57T145
CAS:T145 halts key bacteria growth at sub μg/ml, deters resistance, and may enhance drug lifespan.Formula:C18H16N2O5Purity:98%Color and Shape:SolidMolecular weight:340.33EGGGG-PEG8-amide-bis(deoxyglucitol)
CAS:EGGGG-PEG8-amide-bis(deoxyglucitol) constitutes a cleavable linker utilized in Antibody-Drug Conjugates (ADCs).Formula:C49H91N9O28Color and Shape:SolidMolecular weight:1254.29L-ANAP hydrochloride (1313516-26-5 free base)
L-ANAP hydrochloride is a polarity-sensitive and genetically encodable fluorescent unnatural amino acid.Formula:C15H17ClN2O3Purity:98%Color and Shape:SolidMolecular weight:308.76ALM301
CAS:ALM301: oral AKT inhibitor targeting AKT1, AKT2, AKT3; blocks AKT phosphorylation, curbs cancer cell growth.Formula:C25H25N3O3Color and Shape:SolidMolecular weight:415.48LY2780301
CAS:LY2780301, an oral Akt (protein kinase B) inhibitor, may hinder cancer cell growth and trigger apoptosis by blocking the PI3K/Akt pathway.Formula:C25H27F4N7OColor and Shape:SolidMolecular weight:517.52KRAS inhibitor-12
CAS:KRAS inhibitor-12 blocks KRAS G12C (IC50: 0.537 μM) and p-ERK in cancer cells; promising for pancreatic, colorectal, lung cancer study.Formula:C19H16Cl2FN5OSColor and Shape:SolidMolecular weight:452.33AAK1-IN-4
CAS:AAK1-IN-4 selectively inhibits AAK1 with IC50 of 4.6 nM; penetrates CNS, oral bioactive, potential for studying neuropathic pain.Formula:C20H28N4O3Color and Shape:SolidMolecular weight:372.46PPARγ agonist 7
CAS:PPARγ agonist 7 (Compound 3a) is a highly potent and selective agonist of the peroxisome proliferator-activated receptor gamma (PPARγ).Formula:C20H30O6Color and Shape:SolidMolecular weight:366.45MSC2360844
CAS:MSC2360844 is a potent, orally active and selective inhibitor of PI3Kδ(IC50 of 145 nM).Formula:C26H27FN4O5SPurity:99.54% - 99.9%Color and Shape:SolidMolecular weight:526.58Ref: TM-T12115
1mg52.00€5mg116.00€1mL*10mM (DMSO)135.00€10mg182.00€25mg354.00€50mg568.00€100mg900.00€200mg1,206.00€ZL-2201
CAS:ZL-2201 is a potent inhibitor of DNA-PK, demonstrating an IC50 value of 1 nM.Formula:C20H25N9O5SPurity:98%Color and Shape:SolidMolecular weight:503.54Diethyl-pythiDC
CAS:Diethyl-pythiDC is an collagen prolyl 4-hydroxylase inhibitor.Formula:C14H14N2O4SPurity:99.98%Color and Shape:SolidMolecular weight:306.34HDAC/HSP90-IN-3
CAS:HDAC/HSP90-IN-3, a dual inhibitor targeting fungal Hsp90 (IC50: 0.83 μM) & HDAC (IC50: 0.91 μM), counters azole-resistant C. albicans.Formula:C26H33N5O6Color and Shape:SolidMolecular weight:511.57XZ426
CAS:XZ426 is a potent integrase strand transfer inhibitor with anti- HIV activity .Formula:C22H24F2N4O4Color and Shape:SolidMolecular weight:446.45CRF1 receptor antagonist-1
CAS:CRF1 Receptor Antagonist-1 (Compound 2), a CRF1 receptor antagonist, is utilized in research pertaining to congenital adrenal hyperplasia (CAH) [1].Formula:C27H28ClFN2O2SPurity:98%Color and Shape:SolidMolecular weight:499.04DU172
CAS:DU172 is the tyrosine-targeted covalent adenosine A1 receptor antagonist.Formula:C24H30FN5O5SColor and Shape:SolidMolecular weight:519.59PPO-IN-3
CAS:PPO-IN-3 (Compound 8ad) is a potent PPO inhibitor, exhibiting a Ki value of 0.67 nM and possessing post-emergence herbicidal properties suitable for weedFormula:C19H19ClFN3O2S2Color and Shape:SolidMolecular weight:439.95UNC-2170
CAS:UNC-2170 (UNC2170 Maleate) is the methyl-lysine binding protein, 53BP1 ligand.Formula:C14H21BrN2OPurity:97.44%Color and Shape:SolidMolecular weight:313.23Ref: TM-T24925
5mg46.00€1mL*10mM (DMSO)57.00€10mg71.00€25mg138.00€50mg200.00€100mg284.00€200mg391.00€K145 hydrochloride
CAS:K145 hydrochloride is a selective sphk2 inhibitor with substrate competitiveness and oral activity, with IC50 of 4.3 µM and Ki of 6.4 µM.Formula:C18H25ClN2O3SPurity:99.8%Color and Shape:SolidMolecular weight:384.92OB 24 hydrochloride
CAS:OB 24 hydrochloride inhibits HO-1 (IC50 = 1.9 μM), not HO-2, and curbs PCA cell growth, carbonylation, ROS; also reduces tumor/metastases with Taxol.Formula:C15H18BrClN2O2Purity:99.98%Color and Shape:SolidMolecular weight:373.68Ref: TM-T41175
1mgTo inquire25mgTo inquire50mgTo inquire1mL*10mM (DMSO)To inquire5mg103.00€10mg164.00€100mg1,009.00€LY108742
CAS:LY108742 is an antagonist of 5-HT2.Formula:C21H28N2O3Purity:98%Color and Shape:SolidMolecular weight:356.46SD 1008
CAS:SD 1008 is a JAK2/STAT3 signaling pathway inhibitor. SD 1008 inhibits activation of STAT3, JAK2, and Src.Formula:C18H19NO5Purity:98%Color and Shape:SolidMolecular weight:329.35PF-04957325
CAS:PF-04957325 is an inhibitor of PDE8.PF-04957325 has an IC50 of 0.7 nM for PDE8A.PF-04957325 can be used for the study of autoimmune encephalomyelitis.Formula:C14H15F3N8OSPurity:99.02%Color and Shape:SolidMolecular weight:400.38Ref: TM-T12422
1mg130.00€1mL*10mM (DMSO)195.00€5mg222.00€10mg334.00€25mg578.00€50mg838.00€100mg1,251.00€Satigrel
CAS:Satigrel is a new antiplatelet agent. It also inhibits platelet accumulation in prosthetic arterial grafts.Formula:C20H19NO4Purity:98%Color and Shape:SolidMolecular weight:337.37Aurora kinase inhibitor-8
CAS:Aurora kinase inhibitor-8 is a highly selective inhibitor of Aurora kinase.Formula:C30H29N7O3Color and Shape:SolidMolecular weight:535.6AMD-3329 free base
CAS:AMD-3329 is a potent anti-HIV agent that blocks virus replication by targeting CXCR4, a key receptor for X4 viruses' entry.Formula:C34H50N8Color and Shape:SolidMolecular weight:570.81ThrRS-IN-3
ThrRS-IN-3: Potent inhibitor of Salmonella enterica ThrRS, IC50 = 19 nM, Kd = 34 nM, with antibacterial effects.Formula:C31H30Cl2N6O5Color and Shape:SolidMolecular weight:637.51AGN-201904Z
CAS:AGN-201904Z is a slow-release, acid-resistant pro-PPI that turns into omeprazole, offering extended acid suppression.Formula:C25H25N3NaO8S2Purity:98%Color and Shape:SolidMolecular weight:582.6Anticancer agent 113
CAS:Anticancer agent 113 possesses anticancer activity [1].Formula:C27H31ClN6O2Color and Shape:SolidMolecular weight:507.03TIQ-15
CAS:TIQ-15 is an effective and selective CXCR4 antagonist. It has good drug-like properties.Formula:C23H32N4Purity:98%Color and Shape:SolidMolecular weight:364.53IP7e
CAS:IP7e (isoxazolo-pyridinone 7e) is a Nurr1 activator with an EC50 value of 3.9 nM.Formula:C23H22N2O4Purity:99.86%Color and Shape:SolidMolecular weight:390.43Ref: TM-T27620
1mg52.00€5mg111.00€1mL*10mM (DMSO)124.00€10mg169.00€25mg376.00€50mg617.00€100mg938.00€200mg1,311.00€TIS108
CAS:TIS108为一种抑制三唑型独脚金内酯生物合成的化合物。它抑制拟南芥的胚胎发生并降低水稻中2′-epi-5-deoxystrigol (epi-5DS)的含量。Formula:C20H21N3O2Color and Shape:SolidMolecular weight:335.4RP-001
CAS:RP-001 is a selective agonist of picomolar short-acting S1P1 (EDG1)(EC50 of 9 pM), has little activity on S1P2-S1P4 and only moderate affinity for S1P5.Formula:C24H24N4O4Purity:98%Color and Shape:SolidMolecular weight:432.47PSB-10 hydrochloride
CAS:PSB-10 hydrochloride is a human adenosine A3 receptor antagonist.Formula:C16H15Cl4N5OPurity:98%Color and Shape:SolidMolecular weight:435.14CHM-1
CAS:CHM-1 is an inducer of apoptosis, and displays potent antitumor ability in human hepatocellular carcinoma by activation of Cdc2 kinase activity.Formula:C16H10FNO3Purity:99.839%Color and Shape:SolidMolecular weight:283.25AZD-1656
CAS:AZD-1656 is a glucokinase activator (GKA) that can cause dose-limiting hypoglycemia in normal animals used in embryofetal development studies and type 2Formula:C24H26N6O5Purity:97.07% - 99.37%Color and Shape:SolidMolecular weight:478.5L-054,522
CAS:L-054,522 is potent, selective agonists of somatostatin receptor.Formula:C35H47N7O5Color and Shape:SolidMolecular weight:645.79ZG1077
CAS:ZG1077, a covalent KRAS G12C inhibitor, is utilized in non-small cell lung cancer (NSCLC) research.Formula:C33H33F2N5O5SColor and Shape:SolidMolecular weight:649.71GNE-783
CAS:GNE-783 is a selective inhibitor of CHK1.Formula:C22H20N6Purity:98%Color and Shape:SolidMolecular weight:368.43Atiprimod dimaleate
CAS:Atiprimod Dimaleate is a JAK2 inhibitor.Formula:C30H52N2O8Color and Shape:SolidMolecular weight:568.74Melogliptin
CAS:Melogliptin (EMD-675992, GRC-8200) is a DPP-IV inhibitor for type II diabetes, lowering HbA1c up to 0.75%.Formula:C15H21FN6OColor and Shape:SolidMolecular weight:320.37α-Synuclein inhibitor 9
CAS:α-Synuclein inhibitor 9 (Compound 20C) is a molecule that targets and binds to cavities within mature α-synuclein fibrils, diminishing their β-sheet content.Formula:C27H24O4Color and Shape:SolidMolecular weight:412.48Antiproliferative agent-39
CAS:Antiproliferative Agent-39 (Compound 12) effectively inhibits the proliferation of various cancer cell lines, including A549, SNU-638, Col2, HT1080, and MCF-7,Formula:C22H22N4O3Color and Shape:SolidMolecular weight:390.44LPA1 receptor antagonist 1
CAS:LPA1 receptor antagonist 1(LPA1 R antagonist 1) is a lysophosphatidic acid receptor antagonist for the study of idiopathic pulmonary fibrosis.Formula:C28H26N4O4Purity:99.46% - 99.56%Color and Shape:SolidMolecular weight:482.53
