Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,853 products)
- Apoptosis(6,368 products)
- Cell Cycle/Checkpoint(4,909 products)
- Chromatin/Epigenetics(2,633 products)
- Cytoskeletal Signaling(1,587 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,765 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,054 products)
- Immunology and Inflammation(3,952 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,163 products)
- Metabolism(10,156 products)
- Microbiology/Virology(7,674 products)
- Neuroscience(10,550 products)
- Other Inhibitors(35,855 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,437 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,992 products)
- Ubiquitination(1,744 products)
Show 16 more subcategories
Found 66513 products of "Inhibitors"
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Glucocorticoid receptor agonist
CAS:Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.Formula:C20H20F4N2O2Purity:98%Color and Shape:SolidMolecular weight:396.38K-Ras G12C-IN-2
CAS:K-Ras G12C-IN-2 is a covalent kras g12c inhibitor.Formula:C21H27ClN4O3Purity:98%Color and Shape:SolidMolecular weight:418.92NLRP3-IN-22
CAS:NLRP3-IN-22 (Compound II-4) is an inhibitor of NLRP3, exhibiting a 67% inhibition rate at a concentration of 10 μM [1].Formula:C19H12F3NO4SPurity:98%Color and Shape:SolidMolecular weight:407.36Fosfluridine tidoxil
CAS:Fosfluridine tidoxil, a thymidylate synthase inhibitor, is used potentially for the treatment of colorectal cancer, and breast cancer.Formula:C34H62FN2O10PSColor and Shape:SolidMolecular weight:740.95-HT2A receptor agonist-3
CAS:5-HT2A receptor agonist-3 represents the highest selectivity for the human 5-HT2A receptor currently identified, exhibiting a K i of 2.5 nM.Formula:C21H26BrNO3Purity:98%Color and Shape:SolidMolecular weight:420.34WRNA10
CAS:WRNA10 is a potent binding agent for HIV-1TAR RNA (IC50: 10 μM, CC50: 40 μM).Formula:C25H32N4O4Color and Shape:SolidMolecular weight:452.55S-Benzylglutathione
CAS:S-Benzylglutathione acts as a competitive inhibitor of glutathionase and undergoes conversion by rat kidney microsomes into its cysteine derivatives.Formula:C17H23N3O6SColor and Shape:SolidMolecular weight:397.45TNFalpha-IN-S10
CAS:TNFalpha-IN-S10 is an inhibitor of TNF-α.Formula:C21H14N2O3SColor and Shape:SolidMolecular weight:374.41Gö 7874
CAS:Gö 7874 is a potent, reversible, ATP-competitive, and selective inhibitor of protein kinase C (IC50 = 4 nM for rat brain PKC).Formula:C27H26N4O4Color and Shape:SolidMolecular weight:470.52AY 31906
CAS:AY 31906: High ceiling diuretic, boosts sodium/chloride excretion without affecting potassium, GFR, or renal flow in dogs.Formula:C15H24N6O3SColor and Shape:SolidMolecular weight:368.45EML631
CAS:EML631 is a potent and selective SPIN1 inhibitor (SPIN1 Kd= 3 microM).Formula:C41H60N6O3Color and Shape:SolidMolecular weight:684.95Luminespib mesylate
CAS:Luminespib (AUY-922) is a 3rd-gen Hsp90 inhibitor, disrupting tumor cell proliferation & oncogenic proteins, raising Hsp72 levels.Formula:C27H33N3O5Color and Shape:SolidMolecular weight:479.57TP0480066
CAS:TP0480066 inhibits topoisomerase II, DNA gyrase (IC50=1.1nM), topo IV (IC50=62.89nM), effective against drug-resistant bacteria and N. gonorrhoeae.Formula:C18H14FN3O5Color and Shape:SolidMolecular weight:371.32Tarazepide
CAS:Tarazepide is a potent and specific antagonist of CCK-A receptor.Formula:C28H24N4O2Purity:98%Color and Shape:SolidMolecular weight:448.52PD-140548
CAS:PD-140548 is a potent, CCKA receptor-selective antagonist.Formula:C33H39N3O5Purity:98%Color and Shape:SolidMolecular weight:557.68ICMT-IN-33
CAS:ICMT-IN-33 (compound 73) functions as an ICMT inhibitor with an IC50 value of 0.46 μM [1].Formula:C20H24ClNOColor and Shape:SolidMolecular weight:329.865-HT2A&5-HT2C agonist-1
CAS:5-HT2A&5-HT2C agonist-1 (Example 2) is a dual-acting agent targeting the 5-HT2A and 5-HT2C receptors with respective IC50 values of 196 nM and 0.9 nM.Formula:C14H20N2OPurity:98%Color and Shape:SolidMolecular weight:232.32Levocabastine hydrochloride
CAS:Levocabastine HCl is an agent with antihistaminic activity.Formula:C26H30ClFN2O2Color and Shape:SolidMolecular weight:456.98CP-664511
CAS:CP-664511 is an alpha4beta1/ vascular cell adhesion molecule-1 (VCAM-1) inhibitor with therapeutic potential for allergic airway disease.Formula:C28H34N4O6Color and Shape:SolidMolecular weight:522.59Amentoflavone hexaacetate
CAS:Amentoflavone hexaacetate is a 3,5-cyclic nucleotide phosphodiesterase inhibitor. It has anti-angiogenic and anti-metastatic effects.Formula:C42H30O16Color and Shape:SolidMolecular weight:790.68L 687306
CAS:L 687306 is a partial agonist of muscarinic M1 receptors. It is also a highly competitive antagonist at cardiac M2 receptors and ileal M3 muscarinic receptors.Formula:C11H15N3OColor and Shape:SolidMolecular weight:205.26IIIM-290
CAS:IIIM-290 is an oral CDK inhibitor (IC50s: 90 and 94 nM for CDK2/A and CDK9/T1).Formula:C23H21Cl2NO5Purity:98%Color and Shape:SolidMolecular weight:462.323-Acetyl-6-bromocoumarin
CAS:3-Acetyl-6-bromocoumarin is a coumarin derivative that has exhibited potent antioxidant activity, demonstrated at a rate of 56% [1].Formula:C11H7BrO3Color and Shape:SolidMolecular weight:267.08Anticancer agent 61
CAS:Anticancer agent 61, an oral drug, inhibits HepG2, Bel-7402, MCF-7 cell growth; IC50: 1.12, 1.97, 1.08 μM respectively. Stops tumor growth.Formula:C22H22N3Na2O8PSColor and Shape:SolidMolecular weight:565.45PIM1-IN-4
CAS:PIM1-IN-4: strong PIM1 inhibitor, also blocks SGK-1, PKA, CaMK-1, GSK3β, MSK1; promising for cancer studies.Formula:C27H25BrCl2CuN6OPurity:98%Color and Shape:SolidMolecular weight:663.88L-796568 free base
CAS:L-796568 is a potent β3 agonist for obesity with 600x selectivity over β1/β2 receptors (EC50: 3.6 nM).Formula:C31H27F3N4O3S2Color and Shape:SolidMolecular weight:624.7PI3Kγ inhibitor 2
CAS:PI3Kγ inhibitor 2 is an orally bioavailable inhibitor of PI3Kγ(Ki of 4 nM).Formula:C20H18F3N5O3Purity:98%Color and Shape:SolidMolecular weight:433.38CYP3A4-IN-2
CAS:CYP3A4-IN-2, a potent CYP3A4 inhibitor (IC50: 0.055 μM), is a hydrophobic ritonavir analog with immunosuppressive and antiviral properties.Formula:C33H38N4O3SColor and Shape:SolidMolecular weight:570.74SDZ SER 082 fumarate
CAS:5-HT2B/2C receptor antagonistFormula:C15H20N2Purity:98%Color and Shape:SolidMolecular weight:228.33WAY-620445
CAS:WAY-620445 is an active molecule.Formula:C19H17NO4S2Color and Shape:SolidMolecular weight:387.47Antitumor agent-93
CAS:Antitumor agent-93 (compound 7D) effectively inhibits the proliferation of multiple tumor cell lines, including MDA-MB-231 and HCT-116 [1].Formula:C22H20O8Color and Shape:SolidMolecular weight:412.39N,N-Dimethyldoxorubicin
CAS:N,N-Dimethyldoxorubicin, a Doxorubicin analogue, exhibits cytotoxicity against a range of tumor cell lines with IC50 values below 0.3 μM [1].Formula:C29H33NO11Color and Shape:SolidMolecular weight:571.57CMB-087229
CAS:CMB-087229 is an inhibitor of mutant superoxide dismutase 1 (SOD1) protein aggregation, exhibiting an IC50 of 67 nM, and holds potential for use in amyotrophicFormula:C10H8Cl2N2O2Color and Shape:SolidMolecular weight:259.09S 16020-2
CAS:S 16020-2 is an olivacine derivative, and DNA topoisomerase II inhibitor endowed with a remarkable antitumor activity against various experimental tumors.Formula:C22H26Cl2N4O2Color and Shape:SolidMolecular weight:449.376Cyclic HPMPC
CAS:Cyclic HPMPC: Potent antiviral, raises O2 in mice with lethal vaccinia, lowers guinea pig CMV replication.Formula:C8H12N3O5PColor and Shape:SolidMolecular weight:261.17Physachenolide C
CAS:Physachenolide C, a selective BET inhibitor, induces apoptosis and arrests the cell cycle at the G0-G1 phase, exhibiting antitumor activity [1].Formula:C30H40O9Purity:98%Color and Shape:SolidMolecular weight:544.63FGFR-IN-8
CAS:FGFR-IN-8, potent oral FGFR inhibitor for wild-type/mutant types, induces apoptosis with anti-cancer properties.Formula:C27H31Cl2N9O2Color and Shape:SolidMolecular weight:584.54-Hydroperoxyifosfamide
CAS:4-Hydroperoxyifosfamide is an anticancer agent capable of penetrating the blood-brain barrier (BBB) [1].Formula:C7H15Cl2N2O4PColor and Shape:SolidMolecular weight:293.09U 66985
CAS:U 66985 is a Platelet-activating factor (PAF) receptor antagonist that inhibit the electrophysiological effects of PAF.Formula:C32H66NO7PColor and Shape:SolidMolecular weight:607.84Efipladib
CAS:Efipladib is a phospholipase inhibitor. Efipladib decreases nociceptive responses without affecting PGE2 levels in the cerebral spinal fluid.Formula:C40H35Cl3N2O4SColor and Shape:SolidMolecular weight:746.14VT-1598
CAS:VT-1598 is a novel, selective, orally active fungal CYP51 inhibitor. VT-1598 exhibits antifungal effects against Candida albicans.Formula:C31H20F4N6O2Color and Shape:SolidMolecular weight:584.52Kras binder 12
CAS:Kras binder 12 can be used in studies about Ras.Formula:C29H47N9O6Color and Shape:SoildMolecular weight:617.74BN 52256
CAS:BN 52256 helps reduce arrhythmias.Formula:C19H19NOSeColor and Shape:SolidMolecular weight:356.32XZ426
CAS:XZ426 is a potent integrase strand transfer inhibitor with anti- HIV activity .Formula:C22H24F2N4O4Color and Shape:SolidMolecular weight:446.45NLRP3-IN-9
CAS:NLRP3-IN-9 (INF-4E) irreversibly inhibits NLRP3 ATPase, caspase-1, and prevents pyroptosis in THP-1 cells.Formula:C12H13ClO3Purity:99.64%Color and Shape:SolidMolecular weight:240.68BMS-763534
CAS:BMS-763534 is a potent antagonist of corticotropin-releasing factor/hormone receptor 1 (CRHR-1).Formula:C18H21ClF2N4O3Color and Shape:SolidMolecular weight:414.83WIN site inhibitor 1 TFA (2407457-36-5 free base)
WIN site inhibitor 1 TFA is a WIN site of chromatin-associated WD repeat-containing protein 5 (WDR5) inhibitor (Kd: 0.1 nM).Formula:C27H23Cl2F4N5O3Purity:98%Color and Shape:SolidMolecular weight:612.4Piperidione
CAS:Piperidione is a cough-suppressing agent [1].Formula:C9H15NO2Color and Shape:SolidMolecular weight:169.22TLR9-IN-18
CAS:TLR9-IN-18 is a potent and selective TLR9 antagonist. TLR9-IN-18 suppresses the production of the proinflammatory cytokine IL-6 in a CpG-induced mouse model.Formula:C25H36N6O2Color and Shape:SolidMolecular weight:452.59β-Catenin modulator-4
CAS:β-Catenin modulator-4 (compound IIa-92), encompassing oxazole and thiazole moieties, acts as a potent and selective modulator of β-Catenin [1].Formula:C21H21ClN2O2SColor and Shape:SolidMolecular weight:400.92
