Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,850 products)
- Apoptosis(6,367 products)
- Cell Cycle/Checkpoint(4,909 products)
- Chromatin/Epigenetics(2,631 products)
- Cytoskeletal Signaling(1,586 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,765 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,053 products)
- Immunology and Inflammation(3,946 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,163 products)
- Metabolism(10,156 products)
- Microbiology/Virology(7,671 products)
- Neuroscience(10,551 products)
- Other Inhibitors(35,855 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,435 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,989 products)
- Ubiquitination(1,744 products)
Show 16 more subcategories
Found 66515 products of "Inhibitors"
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S-Adenosyl-L-methionine (1,4-butanedisulfonate)
CAS:S-Adenosyl-L-methionine (SAMe) 1,4-butanedisulfonate functions as an orally active methyl group donor and serves as a dietary supplement known for itsFormula:C19H32N6O11S3Purity:98%Color and Shape:SolidMolecular weight:616.69Cimicoxib
CAS:Cimicoxib (UR8880) is a potent and selective inhibitor of COX-2 with anti-inflammatory and analgesic activity.Formula:C16H13ClFN3O3SPurity:98.22%Color and Shape:SolidMolecular weight:381.81Ref: TM-T30937
1mg44.00€2mg55.00€5mg79.00€1mL*10mM (DMSO)96.00€10mg105.00€25mg170.00€50mg255.00€100mg379.00€LY-393675
CAS:LY-393675 is an antagonist of metabotropic glutamate receptor (mGluR).Formula:C21H21NO4SColor and Shape:SolidMolecular weight:383.46RP-001
CAS:RP-001 is a selective agonist of picomolar short-acting S1P1 (EDG1)(EC50 of 9 pM), has little activity on S1P2-S1P4 and only moderate affinity for S1P5.Formula:C24H24N4O4Purity:98%Color and Shape:SolidMolecular weight:432.47UPCDC30766
CAS:UPCDC30766, a potent allosteric inhibitor of p97, exhibits an IC50 of 12 nM and is applicable for colon cancer research [1].Formula:C30H32F2N6O3SPurity:98%Color and Shape:SolidMolecular weight:594.68XR9051
CAS:XR9051, a synthetic derivative of a natural compound, potently reverses P-glycoprotein MDR (EC50 = 1.4 nM) by inhibiting cytotoxic binding.Formula:C39H38N4O5Color and Shape:SolidMolecular weight:642.74CeMMEC1 HCl
CAS:CeMMEC1 is a compound derived from N-methylisoquinolinone that inhibits the second bromodomain of TAF1.Formula:C19H17ClN2O4Color and Shape:SolidMolecular weight:372.8N-Benzylnaltrindole hydrochloride
CAS:δ2 opioid receptor antagonistFormula:C33H33ClN2O3Purity:98%Color and Shape:SolidMolecular weight:541.08TASP0412098
CAS:TASP0412098 is a potent, selective CRTH2 antagonist with oral activity.Formula:C27H23ClN2O3Purity:98%Color and Shape:SolidMolecular weight:458.94dBRD4-BD1
CAS:dBRD4-BD1 selectively inhibits and degrades BRD4 (DC50=280nM), upregulates BRD2/3, and aids in creating BRD4-specific probes.Formula:C50H53F3N8O9Color and Shape:SolidMolecular weight:967VCH-286
CAS:VCH-286 is a C-C chemokine receptor type 5 (CCR5) receptor antagonist.Formula:C34H50F2N4O3Purity:98%Color and Shape:SolidMolecular weight:600.78YM49598
CAS:YM49598 is a tachykinin receptor antagonist with high affinity for NK(1) and NK(2). It inhibits rat bladder contraction induced by NK(1) agonists.Formula:C36H45Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:608.66WAY-604603
CAS:WAY-604603 is an active molecule, demonstrating inhibitory activity on the enzyme cholinesterase, more specifically on acetylcholinesterase (AChE), whileFormula:C15H10ClNO4SColor and Shape:SolidMolecular weight:335.76GSK-2485852
CAS:GSK-2485852, a NS5B inhibitor, is used potentially for treatment of HCV infection.Formula:C27H25BF2N2O6SColor and Shape:SolidMolecular weight:554.37GGFG-amide-glycol-amide-Exatecan
CAS:Exatecan (Intermediate 2), a derivative of GGFG-amide-glycol-amide-Exatecan, facilitates the synthesis of antibody-drug conjugates (ADCs) [1].Formula:C43H47FN8O11Color and Shape:SolidMolecular weight:870.88Hydroxy Darunavir
CAS:Hydroxy darunavir, a metabolite of the HIV-1 protease inhibitor darunavir, is generated through isobutyl aliphatic hydroxylation of darunavir.Formula:C27H37N3O8SColor and Shape:SolidMolecular weight:563.66HPK1-IN-10
CAS:HPK1-IN-10 inhibits HPK1, a MAP4K kinase from progenitor cells, with potential in treating HPK1 diseases, detailed in patent WO2021213317A1.Formula:C31H34N6O2Color and Shape:SolidMolecular weight:522.64PHD2/HDACs-IN-1
CAS:PHD2/HDACs-IN-1: strong PHD2/HDAC inhibitor (IC50: 1.15-26.60 μM), low-toxicity, protects kidneys from cisplatin-induced AKI.Formula:C18H19N9O4Color and Shape:SolidMolecular weight:425.4AR-C141990
CAS:AR-C141990 is a lactate transporters inhibitor.Formula:C26H28N4O4SColor and Shape:SolidMolecular weight:492.59DUB-IN-7
CAS:DUB-IN-7 (compound 43), a deubiquitinating enzyme (DUB) inhibitor, has utility in researching diseases driven by aberrant JAK2 activity, including leukemia [1].Formula:C17H19N5OColor and Shape:SolidMolecular weight:309.37AS6
CAS:AS6 is an ABA-induced PYL-PP2C interaction antagonist in a dose-dependent manner.Formula:C21H32O4SPurity:98%Color and Shape:SolidMolecular weight:380.54KFM19
CAS:KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.Formula:C16H22N4O3Purity:98.62%Color and Shape:SolidMolecular weight:318.37GLP-1R agonist 9
CAS:GLP-1R agonist 9 acts as a GLP-1R agonist, demonstrating efficacy with EC50 values of 1.1 nM and 11 nM against CHO GLP-1R Clone H6 and Clone C6, respectively.Formula:C32H30ClF2N3O5Color and Shape:SolidMolecular weight:610.057-Deaza-2′-deoxyguanosine 5′-triphosphate
CAS:7-Deaza-2′-deoxyguanosine 5′-triphosphate (7-Deaza-2'-dGTP), a nucleotide analogue, functions as a telomerase inhibitor with an IC50 value of 11 μM [1].Formula:C11H17N4O13P3Purity:98%Color and Shape:SolidMolecular weight:506.19GALK1-IN-1
CAS:Compound 4, known as GALK1-IN-1, is a potent inhibitor of galactokinase, exhibiting an IC50 value of 4.2129 μM [1].Formula:C19H20N4O2Purity:98%Color and Shape:SolidMolecular weight:336.39ASN 07115873
CAS:ASN 07115873 is an anti-Zika virus (ZIKV) compound with an inhibitory concentration (IC50) of 189.2 picomolar (pM), suitable for antiviral research [1].Formula:C12H11ClN4OS2Color and Shape:SolidMolecular weight:326.83MKA031
CAS:MKA031 (compound 6y) is a non-competitive inhibitor of macrophage migration inhibitory factor (MIF), exhibiting an IC50 of 1.7 μM.Formula:C21H17N5O2SColor and Shape:SolidMolecular weight:403.46PAK1-IN-1
CAS:PAK1-IN-1: PAK1 inhibitor, IC50 9.8 nM, hinders tumor cell migration and invasion dose-dependently.Formula:C26H20ClN5O2Color and Shape:SolidMolecular weight:469.92FR-186054
CAS:FR-186054, a potent ACAT inhibitor with high oral efficacy, outperforms others in vitro regardless of dosage.Formula:C26H27N5OS2Purity:98%Color and Shape:SolidMolecular weight:489.66ICy-Q
CAS:ICy-Q, a NIR reagent activated by NQO-1, triggers pyroptosis in pancreatic cancer cells, aiding diagnosis.Formula:C48H50I2N2O5Purity:98%Color and Shape:SolidMolecular weight:988.73S-Fcme
CAS:S-Fcme activates multidrug resistance transporter by boosting ATPase activity and competing for drug binding.Formula:C19H33NO2SColor and Shape:SolidMolecular weight:339.54HDAC-IN-55
CAS:HDAC-IN-55(8j) is a small-molecule inhibitor that enhances E-cadherin expression and suppresses cancer cell proliferation [1].Formula:C17H17N3O3Purity:98%Color and Shape:SolidMolecular weight:311.348-bromo NAD+ sodium
CAS:8-Bromo NAD+ serves as a prodrug for the cyclic ADP-ribose (cADPR) inhibitor, 8-bromo cADPR, undergoing conversion to its active form by the enzyme CD38.Formula:C21H25BrN7O14P2·NaColor and Shape:SolidMolecular weight:764.30(+/-)- Adomeglivant
CAS:Adomeglivant (LY2409021) is a potent glucagon receptor blocker, reducing blood glucose in type 2 diabetes with minimal side effects.Formula:C32H36F3NO4Color and Shape:SolidMolecular weight:555.63B 581
CAS:B 581 is an inhibitor that specifically blocks farnesylated.Formula:C22H38N4O3S2Purity:98%Color and Shape:SolidMolecular weight:470.693-O-Acetyl-20-Hydroxyecdysone
CAS:3-O-Acetyl-20-Hydroxyecdysone, a steroid extracted from the roots of Cyanotis arachnoidea C.B.Clark, is characterized by its unique structural modifications.Formula:C29H46O8Purity:99.54% - 99.99%Color and Shape:SolidMolecular weight:522.67S-Benzylglutathione
CAS:S-Benzylglutathione acts as a competitive inhibitor of glutathionase and undergoes conversion by rat kidney microsomes into its cysteine derivatives.Formula:C17H23N3O6SColor and Shape:SolidMolecular weight:397.45Phenylpyropene C
CAS:Phenylpyropene C inhibits JAK/STAT and IFN-γ expression (IC50: 5.4-10.8 μM), also blocks acyl CoA (IC50: 16.0 μM).Formula:C28H34O5Color and Shape:SolidMolecular weight:450.57Flovagatran sodium
CAS:Flovagatran sodium, a thrombin inhibitor, is used potentially for the treatment of thrombosis.Formula:C27H36BN3NaO7Purity:98%Color and Shape:SolidMolecular weight:548.4Haloxyfop-P-methyl
CAS:Haloxyfop-P-methyl, an aryloxyphenoxypropionate herbicide, is absorbed through both foliage and roots, where it inhibits lipogenesis and induces oxidativeFormula:C16H13ClF3NO4Color and Shape:SolidMolecular weight:375.73PPACK
CAS:PPACK: synthetic peptide, irreversibly inhibits thrombin (Ki = 0.24 nM), prevents platelet activation.Formula:C21H31ClN6O3Purity:98%Color and Shape:SolidMolecular weight:450.96Me-Indoxam
CAS:Me-Indoxam is an inhibitor of sPLA2. It has no effect on arachidonic acid release and platelet activating factor synthesis.Formula:C26H22N2O5Purity:98%Color and Shape:SolidMolecular weight:442.46RS 17053 hydrochloride
CAS:RS 17053 hydrochloride: selective α1A adrenoceptor antagonist, pKi 9.1, pA2 9.8.Formula:C24H30Cl2N2O2Purity:99.27%Color and Shape:SolidMolecular weight:449.414-Hydroxy-2-methylbenzenesulfonic acid ammonium
CAS:4-Hydroxy-2-methylbenzene ammonium: Policresulen impurity, inhibits NS2B/NS3 protease (IC50: 0.48 μg/mL), hinders DENV2 in BHK-21 cells (IC50: 4.99 μg/mL).Formula:C7H11NO4SPurity:98%Color and Shape:SolidMolecular weight:205.23Emodin-1-O-β-D-glucopyranoside
CAS:1.
Formula:C21H20O10Purity:98.32% - 99.74%Color and Shape:SolidMolecular weight:432.38ICI 200355
CAS:ICI 200355 is an inhibitor of human neutrophil elastase.Formula:C30H34BrF3N4O7SPurity:98%Color and Shape:SolidMolecular weight:731.58N-(2-Hydroxyphenyl)picolinamide
CAS:N-(2-Hydroxyphenyl)picolinamide is an active molecular compound.Formula:C12H10N2O2Color and Shape:SolidMolecular weight:214.22KP496
CAS:KP496 is a selective, dual antagonist for Thromboxane A2 receptor and Leukotriene D4 receptor.Formula:C31H34ClN3O7S3Purity:98%Color and Shape:SolidMolecular weight:692.27ML395
CAS:ML395 is a potent, selective PLD2 allosteric inhibitor with potent antiviral activity (IC50 =360 nM).Formula:C26H29N5O2Purity:98%Color and Shape:SolidMolecular weight:443.54Phosphazide
CAS:Phosphazide is a zidovudine prodrug.Formula:C10H14N5O6PColor and Shape:SolidMolecular weight:331.22
