Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,828 products)
- Apoptosis(6,305 products)
- Cell Cycle/Checkpoint(4,864 products)
- Chromatin/Epigenetics(2,608 products)
- Cytoskeletal Signaling(1,555 products)
- DNA Damage/DNA Repair(2,875 products)
- Endocrinology/Hormones(3,752 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(9,005 products)
- Immunology and Inflammation(3,869 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(416 products)
- MAPK Signaling(1,253 products)
- Membrane Transporter/Ion Channel(3,156 products)
- Metabolism(10,145 products)
- Microbiology/Virology(7,618 products)
- Neuroscience(10,360 products)
- Other Inhibitors(35,865 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,428 products)
- Proteases/Proteasome(1,688 products)
- Stem Cell and Derivatives(737 products)
- Tyrosine Kinase/Adaptors(1,980 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66541 products of "Inhibitors"
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CGP 20376
CAS:CGP 20376: Benzothiazole anthelmintic, modulates eosinophil burst, antifibrillatory, dose-dependent effects.
Formula:C16H20N2O3S3Purity:95.11%Color and Shape:SolidMolecular weight:384.54GSK-A
CAS:GSK-A is a Histone Lysine Methyltransferase EZH2 inhibitor.Formula:C21H25N5O2Color and Shape:SolidMolecular weight:379.46BIM-46068
CAS:BIM-46068 is a potent inhibitor of human farnesyltransferase with a unique anti-proliferative profile.Formula:C21H42N4O3S3Color and Shape:SolidMolecular weight:494.78N-Acetylpurinomycin
CAS:N-Acetylpurinomycin is a selective agonist of CB2 receptor.Formula:C24H31N7O6Color and Shape:SolidMolecular weight:513.55Bidisomide
CAS:Bidisomide (SC40230) is an agent of class I antiarrhythmic.Formula:C22H34ClN3O2Purity:99.64%Color and Shape:SolidMolecular weight:407.98Ref: TM-T12858
1mg107.00€5mg263.00€10mg386.00€25mg605.00€50mg800.00€100mg1,063.00€500mg2,142.00€1mL*10mM (DMSO)289.00€AC-4
CAS:AC-4 is a blocker of photoswitchable TRPV1 channel.Formula:C26H25F3N4O2SColor and Shape:SolidMolecular weight:514.56AP-C6
CAS:AP-C6 is a potent inhibitor of guanosine 3',5'-cyclic monophosphate (cGMP)-dependent protein kinase II (cGKII), exhibiting a pIC50 of 6.5.Formula:C15H15N5OColor and Shape:SolidMolecular weight:281.31MK-6240
CAS:MK-6240: A tau PET tracer with high specificity for NFTs binding.Formula:C16H11FN4Purity:98%Color and Shape:SolidMolecular weight:278.28Amauromine
CAS:Amauromine is a peripherally selective and potent cannabinoid receptor type 1 (CB1) receptor antagonist, a novel alkaloid with vasodilatory activity.Formula:C32H36N4O2Color and Shape:SolidMolecular weight:508.65Difelikefalin HCl
CAS:Difelikefalin: KOR agonist, EC50=0.16 nM in humans, >1 µM for MOR. Lowers pain/itch in mice, ED50=0.07 mg/kg.Formula:C36H53N7O6·xHClColor and Shape:SolidMolecular weight:789.237PDE4-IN-8
CAS:PDE4-IN-8 is a potent PDE4 inhibitor with IC50 0.93 nM for PDE4B2 and minor impact on IL13, IL4, IFNy (IC50: 4.04, 36.33, 2394 nM).Formula:C18H22BNO4Color and Shape:SolidMolecular weight:327.18Bay 65-1942 (R form)
CAS:Bay 65-1942 R form is the less active R-form of Bay 65-1942. Bay 65-1942 is a selective and ATP-competitive IKKβ inhibitor.Formula:C22H25N3O4Purity:98%Color and Shape:SolidMolecular weight:395.45LY 53857
CAS:LY 53857 is a potent and selective antagonist of 5-HT2 serotonin receptor.Formula:C27H36N2O7Color and Shape:SolidMolecular weight:500.592Zndm19
CAS:Zndm19 is an inhibitor of New Delhi Metallo-β-lactamase-1 (NDM-1), utilized in researching drug-resistant bacterial infections [1].Formula:C13H13N3OS2Color and Shape:SolidMolecular weight:291.39ArgTX-48 TFA
CAS:ArgTX-48 is a highly potent and subfamily selective antagonist of the NMDARs and AMPARs.Formula:C40H62F9N11O14Color and Shape:SolidMolecular weight:1091.9846h15-LOX-2 inhibitor 1
CAS:Compound 105 (h15-LOX-2 inhibitor 1) is a potent inhibitor of human epithelial 15-lipoxygenase-2 (h15-LOX-2), exhibiting an IC50 of 0.34 μM [1].Formula:C17H13F3N2SPurity:98%Color and Shape:SolidMolecular weight:334.36Cgp 57813
CAS:CGP 57813 is a lipophilic compound, which can be used as an inhibitor of HIV-1 protease.Formula:C43H58N4O8Color and Shape:SolidMolecular weight:758.94Ronopterin
CAS:Ronopterin is a potent Nitric oxide synthase inhibitor and Neuroprotectant.Formula:C9H16N6O2Color and Shape:SolidMolecular weight:240.26Adam-20-S
CAS:Adam-20-S is a potent inhibitor of glucosinolate sulfatase, exhibiting an IC50 of 9.04 μg/mL.Formula:C17H21FN2O4SColor and Shape:SolidMolecular weight:368.42MEL24
CAS:MEL24, an Mdm2 E3 ligase inhibitor, diminishes cell viability and enhances sensitivity to DNA-damaging agents in a p53-dependent manner, suggesting itsFormula:C17H18N4O3Purity:98%Color and Shape:SolidMolecular weight:326.35PARPYnD
CAS:PARPYnD: Photoaffinity PARP probe; inhibits PARP2, PARP1, PARP6 (IC50: 6, 38, 230 nM); tags PARP1/2 with N3 fluorescent probe.Formula:C34H31N9O3Color and Shape:SolidMolecular weight:613.67DC-120
CAS:DC-120: ATP-competitive AKT inhibitor, hinders liver cancer growth, triggers apoptosis, blocks AKT pathway, effective in vivo/vitro with EC50 of 153 nM.Formula:C18H18Cl2N6OSColor and Shape:SolidMolecular weight:437.35NMS-P515
CAS:NMS-P515 is an effective, orally active, and stereospecific PARP-1 inhibitor (Kd: 16 nM and an IC50: 27 nM (in Hela cells)). It has anti-tumor activity.Formula:C21H29N3O2Purity:98%Color and Shape:SolidMolecular weight:355.47GNE-3476
CAS:GNE-3476 is an NMDA PAM with low GluN2A efficacy, AMPAR activity, and weak at GluN2B receptors.Formula:C18H22N4OSColor and Shape:SolidMolecular weight:342.46Mioflazine hydrochloride anhydrous
CAS:Mioflazine hydrochloride anhydrous is a nucleoside transport inhibitor that acts on adenosine to improve sleep.Formula:C29H32Cl4F2N4O2Color and Shape:SolidMolecular weight:648.4Murabutide
CAS:Murabutide, a safe synthetic immunomodulator, diminishes the expression of CD4 and CCR5 receptors and promotes the secretion of high levels of beta-chemokines,Formula:C23H40N4O11Color and Shape:SolidMolecular weight:548.58SNIPER(TACC3)-11
CAS:SNIPER(TACC3)-11 is a powerful FGFR3-TACC3 protein degrader, reducing its amount and hindering FGFR3-TACC3+ cancer cell growth.Formula:C51H66N10O7S2Color and Shape:SolidMolecular weight:995.26GSK2163632A
CAS:GSK2163632A is an insulin-like growth factor 1 receptor inhibitor that acts by binding to a novel region of the GRK active site cleft.Formula:C27H32N8O3SColor and Shape:SolidMolecular weight:548.66VPC 32183 (S)
CAS:VPC 32183 (S) is an LPA1/LPA3 antagonist with no agonist effect on human/mammal LPA receptors.Formula:C33H54N3O6PColor and Shape:SolidMolecular weight:619.78Ac-Lys-Val-Cit-PABC-MMAE
CAS:Ac-Lys-Val-Cit-PABC-MMAE is a conjugate comprising an antibody-drug conjugate (ADC) linker (peptide Ac-Lys-Val-Cit-PABC) and the cytotoxic agent monomethylFormula:C66H108N12O14Color and Shape:SolidMolecular weight:1293.64ASS234
CAS:ASS234 is a multi-target propylamine used in the treatment of Alzheimer's disease.Formula:C29H37N3OColor and Shape:SolidMolecular weight:443.62Antitumor agent-110
CAS:Antitumor Agent-110 (Compound 13), an imidazotetrazine anticancer agent, exhibits excellent permeability.Formula:C10H6N6OSPurity:98%Color and Shape:SolidMolecular weight:258.26GSK1842799 HCl
CAS:GSK1842799, a selective S1P1 agonist for MS, shows >1000x selectivity over S1P3 & good oral bioavailability.Formula:C20H30Cl2F3N3O2SColor and Shape:SolidMolecular weight:504.4342Vadaclidine
CAS:Vadaclidine is an orally acting antinociceptive muscarinic agonist.Formula:C13H21N3S2Color and Shape:SolidMolecular weight:283.46BAY-60-5521
CAS:BAY-60-5521 is an effective cholesterol ester transfer protein (CETP) inhibitor.Formula:C30H37F4NOColor and Shape:SolidMolecular weight:503.61(S)-(-)-Bay-K-8644
CAS:(S)-(-)-Bay-K-8644 ((S)-(-)-Bay K 8644) is an agonist of L-type Ca2+ channel and activates Ba2+ currents with an EC50 of 32 nM.Formula:C16H15F3N2O4Purity:98.28% - 99.37%Color and Shape:SolidMolecular weight:356.3ZL0513
CAS:ZL0513: orally active, BRD4 BD1 inhibitor with strong in vivo results and good pharmacokinetics for treating inflammation.Formula:C27H33NO6Color and Shape:SolidMolecular weight:467.55CC-885-CH2-PEG1-NH-CH3
CAS:CC-885-CH2-PEG1-NH-CH3 is a neoDegrader compound employed for the production of Antibody neoDegrader Conjugate (AnDC) during synthesis.Formula:C26H30ClN5O5Color and Shape:SolidMolecular weight:528.01HBV-IN-17
CAS:HBV-IN-17 (compound 8) is a potent regulator of HBV capsid assembly (EC50: 511 nM).Formula:C17H15F6N5O2Color and Shape:SolidMolecular weight:435.32p38 Kinase inhibitor 4
CAS:Compound 135, also known as p38 Kinase Inhibitor 4, is a potent inhibitor of p38 [1].Formula:C12H9Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:282.13GSK2973980A
CAS:GSK2973980A is a selective Acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1) inhibitor (IC50: 3 nM).Formula:C25H19F5N4O4Purity:98%Color and Shape:SolidMolecular weight:534.43DL-threo dihydrosphingosine
CAS:DL-threo dihydrosphingosine blocks ERK, inhibits smooth muscle proliferation, and works against growth factor/G-protein ERK activation.Formula:C18H39NO2Color and Shape:SolidMolecular weight:301.51HDAC/HSP90-IN-3
CAS:HDAC/HSP90-IN-3, a dual inhibitor targeting fungal Hsp90 (IC50: 0.83 μM) & HDAC (IC50: 0.91 μM), counters azole-resistant C. albicans.Formula:C26H33N5O6Color and Shape:SolidMolecular weight:511.575-n-Heptyl-6-hydroxy-4,7-dioxobenzothiazole
CAS:5-n-Heptyl-6-hydroxy-4,7-dioxobenzothiazole acts as a competitive inhibitor at the Qo site of the cytochrome bc1 complex (cytochrome c oxidoreductase) inFormula:C14H17NO3SColor and Shape:SolidMolecular weight:279.36U 19052
CAS:U 19052 is a Leukotriene D4 antagonist.Formula:C31H42O6SColor and Shape:SolidMolecular weight:542.73LONP1-IN-2
CAS:LONP1-IN-2: Potent LONP1 inhibitor, IC50=0.187μM; weak on 20S proteasome (>10μM); for cancer research.Formula:C16H27BN4O4Color and Shape:SolidMolecular weight:350.22Ardisin
CAS:Ardisin is a Topoisomerase I and II enzyme inhibitor. Ardisin may have antioxidant effects.Formula:C20H32O2Color and Shape:SolidMolecular weight:304.47Ocoteine
CAS:Ocoteine is an alpha 1-adrenoceptor antagonist.Formula:C21H23NO5Color and Shape:SolidMolecular weight:369.42Antioxidant agent-11
CAS:Antioxidant Agent-11 (compound 3d) exhibits weak anti-cancer and antioxidant properties [1].Formula:C23H18N4OColor and Shape:SolidMolecular weight:366.42MT-3014
CAS:MT-3014: Strong, selective brain-penetrating PDE 10A inhibitor; IC50 0.062 nM (human), 0.09 nM (bovine).Formula:C23H25F2N7OPurity:98%Color and Shape:SolidMolecular weight:453.49
