Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,797 products)
- Apoptosis(6,257 products)
- Cell Cycle/Checkpoint(4,836 products)
- Chromatin/Epigenetics(2,592 products)
- Cytoskeletal Signaling(1,534 products)
- DNA Damage/DNA Repair(2,880 products)
- Endocrinology/Hormones(3,748 products)
- Enzyme(3,670 products)
- GPCR/G-Protein(8,985 products)
- Immunology and Inflammation(3,794 products)
- Influenza Virus(299 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,250 products)
- Membrane Transporter/Ion Channel(3,148 products)
- Metabolism(10,144 products)
- Microbiology/Virology(7,591 products)
- Neuroscience(10,345 products)
- Other Inhibitors(35,829 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,421 products)
- Proteases/Proteasome(1,680 products)
- Stem Cell and Derivatives(748 products)
- Tyrosine Kinase/Adaptors(1,960 products)
- Ubiquitination(1,721 products)
Show 16 more subcategories
Found 66564 products of "Inhibitors"
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OSI-296
CAS:OSI-296: potent cMET/RON inhibitor (IC50: 42/200 nM), effective in tumor models, tolerable, oral, reduces bone tumor growth.Formula:C21H19Cl2FN4O3Purity:98%Color and Shape:SolidMolecular weight:465.3ICMT-IN-42
CAS:ICMT-IN-42 (compound 21) serves as an ICMT inhibitor, demonstrating potency with an IC50 of 0.054 μM [1].Formula:C23H31NOColor and Shape:SolidMolecular weight:337.5Antitumor agent-110
CAS:Antitumor Agent-110 (Compound 13), an imidazotetrazine anticancer agent, exhibits excellent permeability.Formula:C10H6N6OSPurity:98%Color and Shape:SolidMolecular weight:258.26mGAT-IN-1
CAS:mGAT-IN-1 is a potent, non-selective GAT inhibitor that inhibits mGAT3 activity well (IC50: 2.5 μM, pIC50: 5.61).Formula:C28H34ClN3O2S2Color and Shape:SolidMolecular weight:544.171-Palmitoyl-sn-glycerol 3-phosphate
CAS:1-Palmitoyl-sn-glycerol 3-phosphate (1-P-GPA), an endogenous metabolite, is utilized in the research of non-alcoholic fatty liver disease [1].Formula:C19H39O7PColor and Shape:SolidMolecular weight:410.48Bay 65-1942 (R form)
CAS:Bay 65-1942 R form is the less active R-form of Bay 65-1942. Bay 65-1942 is a selective and ATP-competitive IKKβ inhibitor.Formula:C22H25N3O4Purity:98%Color and Shape:SolidMolecular weight:395.45(-)-15-Deoxyspergualin trihydrochloride
CAS:(-)-15-Deoxyspergualin trihydrochloride exhibits potent antitumor properties and demonstrates significant inhibition activity against mouse leukemia L-1210 [1].Formula:C17H40Cl3N7O3Color and Shape:SolidMolecular weight:496.9Protopanaxatriol
CAS:Protopanaxatriol (20(R)-APPT), a major ginseng constituent, is a novel PPARγ antagonist.Formula:C30H52O4Purity:99.89%Color and Shape:SolidMolecular weight:476.73Etiroxate
CAS:Etiroxate (CG-635) is a lipid-lowering agent utilized in hyperlipoproteinemia studies [1].Formula:C18H17I4NO4Color and Shape:SolidMolecular weight:818.95AL-38022A
CAS:AL-38022A: selective 5-HT2 ligand, Ki ≤2.2 nM; >100-fold less binding to other 5-HT; minimal interaction with non-5-HT targets; full agonist.Formula:C13H17N3OColor and Shape:SolidMolecular weight:231.29ICMT-IN-23
CAS:ICMT-IN-23 (compound 36) serves as an inhibitor of ICMT, exhibiting a half-maximal inhibitory concentration (IC50) of 0.123 μM [1].Formula:C22H26N2OColor and Shape:SolidMolecular weight:334.45DC 432
CAS:DC 432, a potent peptidomimetic inhibitor of N-terminal methyltransferase 1/2 (NTMT1/2) with an IC50 value of 54 nM, incorporates a BM30 peptide enhanced byFormula:C55H100N28O10Color and Shape:SolidMolecular weight:1313.59BI 7446
CAS:BI 7446 is a potent and selective cyclic dinucleotide (CDN)-based stimulator of interferon genes (STING) agonist capable of activating all five STING variantsFormula:C20H22FN9O10P2S2Purity:98%Color and Shape:SolidMolecular weight:693.52MALT1-IN-6
CAS:MALT1-IN-6 is a MALT1 protease inhibitor (Ki: 9 nM) that exhibits anticancer activity.Formula:C18H12Cl2F3N9OColor and Shape:SolidMolecular weight:498.25USP1-IN-5
CAS:USP1-IN-5 (compound 10) is a potent inhibitor of both USP1, with an IC50 of less than 50 nM, and MDA-MB-436 cells, where it also exhibits an IC50 of less thanFormula:C27H23F3N8OColor and Shape:SolidMolecular weight:532.52MC-VC-PAB-Cyclohexanediamine-Thailanstatin A
CAS:MC-VC-PAB-Cyclohexanediamine-Thailanstatin A is a spliceostatin analog and a drug-linker conjugate for antibody-drug conjugates (ADC), comprising the cytotoxicFormula:C63H91N9O16Purity:98%Color and Shape:SolidMolecular weight:1230.45Fiduxosin hydrochloride
CAS:Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.Formula:C30H30ClN5O4SColor and Shape:SolidMolecular weight:592.11Kelatorphan
CAS:Kelatorphan is an enkephalin degrading enzyme full inhibitor.Formula:C14H18N2O5Purity:98%Color and Shape:SolidMolecular weight:294.3Dexamethasone palmitate
CAS:DXP, a lipophilic prodrug of Dexamethasone, has 47x less glucocorticoid receptor affinity; it's an agonist & anti-inflammatory.Formula:C38H59FO6Purity:99.28%Color and Shape:SolidMolecular weight:630.87WAY-608094
CAS:WAY-608094 is an active compound.Formula:C23H14N2O3Color and Shape:SolidMolecular weight:366.37BRD5648
CAS:BRD5648 ((R)-BRD0705) is an inactive (R)-enantiomer of BRD0705.Formula:C20H23N3OPurity:99.89%Color and Shape:SolidMolecular weight:321.42NGD 98-2 hydrochloride
corticotropin-releasing factor receptor 1 (CRF1) antagonistFormula:C19H24F3N3O3·HClPurity:98%Color and Shape:SolidMolecular weight:435.87KRAS G12C inhibitor 59
CAS:KRAS G12C Inhibitor 59 is a compound with anticancer properties.Formula:C32H39F6N7O5Purity:98%Color and Shape:SolidMolecular weight:715.69YG1702
CAS:YG1702, a potent inhibitor specific to ALDH18A1, suppresses the proliferation of MYCN-amplified neuroblastoma (NB) and reduces MYCN expression.Formula:C23H30N2O7SColor and Shape:SolidMolecular weight:478.56β-Catenin modulator-5
CAS:β-Catenin Modulator-5 (Compound IIa-84), an oxazole and thiazole-based compound, serves as a potent and selective modulator of β-Catenin [1].Formula:C21H22N2O2SColor and Shape:SolidMolecular weight:366.48KRAS G12C inhibitor 17
CAS:KRAS G12C inhibitor 17 is a potent KRAS G12C inhibitor.Formula:C24H20ClF2N3O3Purity:98%Color and Shape:SolidMolecular weight:471.88KNI 174
CAS:KNI 174 is a new type of anti‐AIDS drug used as an HIV‐1 protease inhibitorFormula:C36H45N5O7SColor and Shape:SolidMolecular weight:691.84MMV009085
CAS:MMV009085 is a potent inhibitor of the Plasmodium falciparum hexose transporter (Pf HT1), with potential as an anti-malarial agent.Formula:C22H22N2O6Color and Shape:SolidMolecular weight:410.42EAD1 TFA(1644388-26-0 Free base)
CAS:EAD1 HCL is a potent autophagy inhibitor with antiproliferative activity in lung and pancreatic cancer cells. EAD1 HCL also induces apoptosis
Formula:C26H28Cl2F3N7O2Purity:97.41%Color and Shape:SolidMolecular weight:598.45AM841
CAS:AM841, a high-affinity electrophilic ligand, covalently interacts with a cysteine residue in helix six, thus activating the CB1 cannabinoid receptor.Formula:C26H39NO3SPurity:98%Color and Shape:SolidMolecular weight:445.66hDDAH-1-IN-2
CAS:hDDAH-1-IN-2 is an orally active human dimethylarginine dimethylaminohydrolase-1 (hDDAH-1) inhibitor.Formula:C8H20N4O2Purity:98%Color and Shape:SolidMolecular weight:204.27PD 125754
CAS:PD 125754 is a Renin inhibitor, which represents a group of pharmaceutical drugs used primarily to treat essential hypertension.Formula:C42H65N5O7Purity:98%Color and Shape:SolidMolecular weight:751.99Duocarmycin MB
CAS:Duocarmycin MB, an ADC toxin and DNA alkylating agent, combats multi-drug resistant cells.Formula:C27H26ClN3O4Purity:98%Color and Shape:SolidMolecular weight:491.97SDZ-NVI-085
CAS:SDZ-NVI-085 is an α1 adrenergic receptor agonist and a competitive antagonist of 5-hydroxytryptamine.Formula:C15H21NO2SColor and Shape:SolidMolecular weight:279.42-Methoxyestrone
CAS:2-Methoxyestrone is a methoxylated catechol estrogen and the principal metabolite of 2-hydroxyestrone, a nonuterotropic metabolite of estradiol.Formula:C19H24O3Purity:97.07% - 99.18%Color and Shape:SolidMolecular weight:300.39Ref: TM-T13481
1mg49.00€5mg97.00€10mg160.00€25mg283.00€50mg418.00€100mg615.00€200mg879.00€1mL*10mM (DMSO)106.00€Cbl-b-IN-11
CAS:Cbl-b-IN-11 (Compound 466) is an inhibitor of both casitas B-lineage lymphoma-b (Cbl-b) and c-Cbl, exhibiting half-maximal inhibitory concentrations (IC50s) ofFormula:C31H35F5N6OPurity:98%Color and Shape:SolidMolecular weight:602.64Onchidal
CAS:Onchidal is a key lipid-soluble defense compound from Onchidella binneyi's secretion for chemical protection.Formula:C17H24O3Color and Shape:SolidMolecular weight:276.37CDK9-IN-19
CAS:CDK9-IN-19: Potent CDK9 inhibitor, anti-cancer, moderate pharmacokinetics, low hERG impact, effective in AML research.Formula:C26H22F2N4O5Color and Shape:SolidMolecular weight:508.47GAT100
CAS:GAT100 is a potent dual-action modulator for CB1R, both covalent NAM and enhancing orthosteric agonist CP55,940 binding.Formula:C25H28N4OSColor and Shape:SolidMolecular weight:432.58Glycolithocholic acid 3-sulfate disodium
CAS:Glycolithocholic acid 3-sulfate (disodium) demonstrates inhibitory effects on in vitro HIV-1 replication and has potential applications in HIV infection andFormula:C26H41NNa2O7SColor and Shape:SolidMolecular weight:557.65OfChi-h-IN-1
CAS:OfChi-h-IN-1 is a potent inhibitor of OfChi-h, exhibiting a K i value of 0.33 μM.Formula:C24H27N5O2Color and Shape:SolidMolecular weight:417.5PNU-103017
CAS:PNU-103017 is an inhibitor of HIV protease.Formula:C28H28N2O5SPurity:98%Color and Shape:SolidMolecular weight:504.6SHP2-IN-18
CAS:SHP2-IN-18 (compound 183) is a potent SHP2 inhibitor, exhibiting an IC50 of 3 nM and applicable to glioblastoma research [1].Formula:C26H27FN6Color and Shape:SolidMolecular weight:442.53DAM-IN-1
CAS:DMA-IN-1 is a DNA adenine methyltransferase (DAM) inhibitor with an IC50 value of 48 μM.Formula:C16H17NO4Purity:98%Color and Shape:SolidMolecular weight:287.315-Azacytidine 5′-triphosphate
CAS:5-Azacytidine 5′-triphosphate (5-aza-CMP), a cytidine analog, selectively inhibits the incorporation of [^3H]CTP into RNA during the DNA-dependent RNAFormula:C8H15N4O14P3Color and Shape:SolidMolecular weight:484.14APS3
CAS:APS3 is an inhibitor of GABA and nACh receptors, exhibiting an LC50 value of 7.2423 μg/mL against Plutella xylostella [1].Formula:C18H7Cl2F6N5O5S2Color and Shape:SolidMolecular weight:622.31Minocromil
CAS:Minocromil is a new agent of Anti-asthmatic.Formula:C18H16N2O6Purity:98%Color and Shape:SolidMolecular weight:356.33(+)-Apogossypol
CAS:(+)-Apogossypol is an antagonist of pan-BCL-2. (+)-Apogossypol binds to Mcl-1(Bcl-2 and Bcl-xL with EC50s of 2.6, 2.8 and 3.69 μM, respectively).Formula:C28H30O6Purity:98%Color and Shape:SolidMolecular weight:462.53Casein kinase 1δ-IN-4
CAS:"Casein kinase 1δ-IN-4 (compound 567) is a potent inhibitor of casein kinase 1δ with potential application in Alzheimer's disease research [1]."Formula:C16H12N6SPurity:98%Color and Shape:SolidMolecular weight:320.37Cobimetinib racemate
CAS:Cobimetinib racemate (Cobimetinib (racemate)) (GDC-0973 racemate) is a selective inhibitor of MEK.Cobimetinib racemate is also known as a mitogen-activatedFormula:C21H21F3IN3O2Purity:98.00% - 99.71%Color and Shape:SolidMolecular weight:531.31
