Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,832 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,611 products)
- Cytoskeletal Signaling(1,563 products)
- DNA Damage/DNA Repair(2,873 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,900 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,141 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,369 products)
- Other Inhibitors(35,851 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,690 products)
- Stem Cell and Derivatives(735 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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Abaperidone
CAS:Abaperidone is an atypical antipsychotic, antagonizes 5-HT2A (IC50=6.2 nM) and D2 receptors (IC50=17 nM), reduces hsp70 mRNA in rat brains.Formula:C25H25FN2O5Purity:99.77%Color and Shape:SolidMolecular weight:452.47Dibenamine hydrochloride
CAS:Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.Formula:C16H19Cl2NPurity:96.43%Color and Shape:Oily Liquid SolidMolecular weight:296.23Erigeside I
CAS:Erigeside I is a radical scavenger.Formula:C20H20O11Purity:98%Color and Shape:SolidMolecular weight:436.37Antifungal agent 49
CAS:Antifungal agent 49 (Example 112) exhibits activity against Cryptococcus neoformans, demonstrating a minimum inhibitory concentration (MIC) of 49 μM [1].Formula:C15H12O4Color and Shape:SolidMolecular weight:256.25BTK inhibitor 13
CAS:BTK inhibitor 13 (compound 8) is an effective and selective BTK inhibitor(IC50: 1.2 nM).Formula:C29H26FN5O3Purity:98%Color and Shape:SolidMolecular weight:511.55Sunepitron Free Base
CAS:Sunepitron Free Base, a 5-HT1A agonist/α₂-antagonist, halted in Phase III for depression/anxiety.Formula:C17H23N5O2Color and Shape:SolidMolecular weight:329.4Mal-Pc
CAS:Mal-Pc, a maleimide phthalocyanine, depletes GSH to reduce aggregation and boost ROS, improving PDT against cancer.Formula:C46H28N10O8SiPurity:98%Color and Shape:SolidMolecular weight:876.86RO5527239
CAS:RO5527239 is a potent, orally available GPBAR1 agonist agent.Formula:C28H31N3O3Purity:98%Color and Shape:SolidMolecular weight:457.56CB-25
CAS:CB-25 is a partial agonist ligand of CB1 cannabinoid receptors, augmenting Forskolin-induced cAMP formation in cancer cells, though not affecting hCB1-CHO cellsFormula:C25H41NO3Purity:98%Color and Shape:SolidMolecular weight:403.6Fiduxosin hydrochloride
CAS:Fiduxosin hydrochloride is an alpha 1a-adrenoceptor antagonist that may be useful in the treatment of Benign Prostatic Hyperplasia.Formula:C30H30ClN5O4SColor and Shape:SolidMolecular weight:592.11KM05382
CAS:KM05382 inhibits CDK9 and the transcription of GAPDH.Formula:C20H19ClN2O3S2Color and Shape:SolidMolecular weight:434.96Bay 65-1942 (R form)
CAS:Bay 65-1942 R form is the less active R-form of Bay 65-1942. Bay 65-1942 is a selective and ATP-competitive IKKβ inhibitor.Formula:C22H25N3O4Purity:98%Color and Shape:SolidMolecular weight:395.45Antitumor agent-38
CAS:Antitumor agent-38 inhibits cancer cell growth, causing cell cycle arrest at the S/G2/M phase without affecting microtubules or cell shape.Formula:C22H24N2O4Color and Shape:SolidMolecular weight:380.44TASP0412098
CAS:TASP0412098 is a potent, selective CRTH2 antagonist with oral activity.Formula:C27H23ClN2O3Purity:98%Color and Shape:SolidMolecular weight:458.94Bocodepsin hydrochloride
CAS:Bocodepsin hydrochloride (OKI-179) is a selective HDAC inhibitor with antitumor properties, efficacious via oral administration.Formula:C26H40ClN5O6S2Purity:98%Color and Shape:SolidMolecular weight:618.21Ro-70-0004
CAS:Ro-70-0004 is a selective antagonist of alpha1A-adrenoceptor.Formula:C20H24F4N4O3Color and Shape:SolidMolecular weight:444.42CH-5137291
CAS:CH-5137291 is a pure AR antagonist with AR nuclear translocation inhibition activity. It suppresses castration and prevents the growth of prostate cancer cells.Formula:C18H14F3N5O3S2Color and Shape:SolidMolecular weight:469.46KRAS G12C inhibitor 35
CAS:KRAS G12C inhibitor 35 targets KRAS G12C in cancer research (CN112920183A, compound 3).Formula:C31H27ClF2N6O3Color and Shape:SolidMolecular weight:605.03ICMT-IN-54
CAS:ICMT-IN-54 (compound 7c), an adamantyl analogue, serves as an ICMT inhibitor with an IC50 value of 12.4 μM, targeting the methylation process facilitated byFormula:C29H45NO3SColor and Shape:SolidMolecular weight:487.74PHD-IN-2
CAS:PHD-IN-2 (Compound 91), a potent PHD antagonist with an IC50 of less than 5 nM, effectively stimulates erythropoietin synthesis in HEP3B cells with an EC50 ofFormula:C26H27N7O4Purity:98%Color and Shape:SolidMolecular weight:501.541-Methoxyphaseollidin
CAS:1-Methoxyphaseollidin exhibits anti-Helicobacter pylori activity against the CLAR and AMOX-resistant strain as well as four CLAR (AMOX)-sensitive strains.Formula:C21H22O5Purity:98%Color and Shape:SolidMolecular weight:354.42-Thiophenecarboxamide, N-(5-(p-aminophenoxy)pentyl)-
CAS:2-Thiophenecarboxamide, N-(5-(p-aminophenoxy)pentyl)- is a bioactive chemical.Formula:C16H20N2O2SColor and Shape:SolidMolecular weight:304.41Isopropyl dodec-11-enylfluorophosphonate
CAS:Isopropyl dodec-11-enylfluorophosphonate (IDEFP) is an organophosphorus ester functioning as a central cannabinoid receptor (CB1) antagonist and exhibitsFormula:C15H30FO2PPurity:98%Color and Shape:SolidMolecular weight:292.37Itch-Targeting Compound 1
CAS:Compound 1: Anti-itch, combats bites, allergens, infections, vermination, dialysis-related itching.Formula:C25H36ClN3O3Purity:98%Color and Shape:SolidMolecular weight:462.03ICMT-IN-40
CAS:ICMT-IN-40 (compound 19) is a potent inhibitor of ICMT, exhibiting an IC50 value of 0.031 μM [1].Formula:C22H29NOColor and Shape:SolidMolecular weight:323.47Cgs 18102A (HCl)
CAS:Cgs 18102A (HCl) has 5-HT(1) agonist & 5-HT(2) antagonist properties.Formula:C16H24ClNO2Color and Shape:SolidMolecular weight:297.82MALT1-IN-7
CAS:MALT1-IN-7 (compound 142b) is a potent inhibitor of MALT1 protease with potential for cancer research.Formula:C19H17F3N8O2SColor and Shape:SolidMolecular weight:478.45ICMT-IN-52
CAS:ICMT-IN-52 (compound 44) serves as an ICMT inhibitor with an IC50 value of 0.052 μM [1].Formula:C21H26FNOColor and Shape:SolidMolecular weight:327.44Protopanaxatriol
CAS:Protopanaxatriol (20(R)-APPT), a major ginseng constituent, is a novel PPARγ antagonist.Formula:C30H52O4Purity:99.89%Color and Shape:SolidMolecular weight:476.73hDHODH-IN-1
CAS:hDHODH-IN-1 is an inhibitor of human dihydroorotate dehydrogenase (hDHODH) with an anti-inflammatory effect.Formula:C17H14N2O2Purity:99.97%Color and Shape:SolidMolecular weight:278.31Ref: TM-T11546
1mg34.00€5mg71.00€10mg103.00€25mg200.00€50mg290.00€100mg404.00€200mg545.00€1mL*10mM (DMSO)78.00€NBI-6024
CAS:NBI-6024, an altered peptide ligand (APL), serves as an epitope for interferon-gamma-producing T helper lymphocytes associated with inflammation in patientsFormula:C66H112N20O21Color and Shape:SolidMolecular weight:1521.72NorA-IN-1
CAS:NorA-IN-1 is a NorA efflux inhibitor, which can be used to study overcoming multidrug resistance based on microbial efflux transporter proteins.
Formula:C18H18O5Purity:95.01%Color and Shape:SolidMolecular weight:314.33BMS-262084
CAS:BMS-262084 is a potent selective β-lactam trypsin inhibitor with therapeutic potential in the treatment of asthma.Formula:C18H31N7O5Color and Shape:SolidMolecular weight:425.48(Rac)-PF-4136309(1341224-83-6 Free base)
CAS:PF-4136309 (INCB8761, PF-04136309) is a highly effective and selective oral CCR2 antagonist with good bioavailability, with an IC50 value of 5.2 nM for humanFormula:C29H31F3N6O3Color and Shape:SolidMolecular weight:568.59Anticancer agent 131
CAS:HCT-116-IN-1, a γ-lactam-fused pyridone derivative, exhibits anticancer properties, demonstrating significant cytotoxicity towards HCT116 cells, with an IC50Formula:C33H24ClN3O5Color and Shape:SolidMolecular weight:578.01BAY-678
CAS:BAY-678: Oral selective human neutrophil elastase inhibitor; IC50: 20 nM; SGC-approved chemical probe.Formula:C20H15F3N4O2Purity:99.36%Color and Shape:SolidMolecular weight:400.35Ref: TM-T10473
5mg37.00€10mg60.00€25mg119.00€50mg173.00€100mg264.00€200mg374.00€1mL*10mM (DMSO)42.00€HIV-1 integrase inhibitor 3
CAS:HIV-1 integrase inhibitor 3 is an HIV-1 integrase strand transfer (INST) inhibitor (IC50: 2.7 nM).Formula:C21H22F2N4O4Purity:98%Color and Shape:SolidMolecular weight:432.42L-783483
CAS:L-783483 is an agonist of PPAR.Formula:C22H21ClF3NO4SPurity:98%Color and Shape:SolidMolecular weight:487.92MN-05
CAS:MN-05 is a neuroprotective and vasodilator for neurodegenerative diseases.Formula:C13H22N2O3Color and Shape:SolidMolecular weight:254.33BF738735
CAS:BF738735 is a selective inhibitor of phosphatidylinositol 4-kinase III beta (PI4KIIIβ, IC50 = 5.7 nM) showing higher activity over α(IC50 = 1.7 μM).Formula:C21H19FN4O3SPurity:90%Color and Shape:SolidMolecular weight:426.46β-Lactamase-IN-2
CAS:β-Lactamase-IN-2 is an inhibitor of β-Lactamase with anti-microbial and anti-bacterial effects.Formula:C11H9FO3Purity:99.52%Color and Shape:SolidMolecular weight:208.19Ref: TM-T35427
2mg39.00€5mg62.00€10mg92.00€25mg155.00€50mg215.00€100mg324.00€200mg460.00€1mL*10mM (DMSO)67.00€Lanabecestat HCl
CAS:Lanabecestat (AZD3293/LY3314814) is a potent oral BACE1 inhibitor that crosses the BBB and reduces Aβ levels.Formula:C26H29ClN4OColor and Shape:SolidMolecular weight:448.995Stafib-2
CAS:Stafib-2 is a potent and selective inhibitor of the transcription factor STAT5b.Stafib-2 inhibits STAT5b and STAT5a with IC50 values of 82 nM and 1.7 μM,
Formula:C28H26N2O12P2Purity:98.48%Color and Shape:SolidMolecular weight:644.46Gö 7874
CAS:Gö 7874 is a potent, reversible, ATP-competitive, and selective inhibitor of protein kinase C (IC50 = 4 nM for rat brain PKC).Formula:C27H26N4O4Color and Shape:SolidMolecular weight:470.52SB1-F-78
CAS:SB1-F-78 is an USP30 inhibitor.Formula:C17H16N6OSColor and Shape:SolidMolecular weight:352.41KRAS G12D modulator-1
CAS:KRAS G12D modulator-1 (compound 6), a potent modulator of KRAS G12D, exhibits IC50 values ranging from 1-10 μM against NEA-G12D, PPI-G12D, and p ERK-AGS, and isFormula:C30H36FN5O4Purity:98%Color and Shape:SolidMolecular weight:549.64NIK-250
CAS:NIK-250 is a P-glycoprotein inhibitor. NIK250 could reverse multidrug resistance in human glioma cells.Formula:C26H25N3O4S2Color and Shape:SolidMolecular weight:507.62Tedizolid HCl (856866-72-3 free base)
Tedizolid HCl, a novel oxazolidinone antibiotic, IC50: MAO-A 8.7 uM, MAO-B 5.7 uM, approved post-linezolid, has a prodrug form tedizolid phosphate.Formula:C17H16ClFN6O3Purity:98%Color and Shape:SolidMolecular weight:406.8WAY-637940
CAS:Sure, here is a clearer and more professional version: "WAY-637940 is an active molecule."Formula:C16H17N3O4SColor and Shape:SolidMolecular weight:347.39
