Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,833 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,612 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,901 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,139 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,377 products)
- Other Inhibitors(35,852 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,430 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,983 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
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(S)-FTY-720 Vinylphosphonate
CAS:(S)-FTY-720 Vinylphosphonate blocks sphingosine kinase 1 and aids its breakdown in various human cancer cells.Formula:C20H34NO4PColor and Shape:SolidMolecular weight:383.46ICMT-IN-13
CAS:ICMT-IN-13 (compound 49) functions as an inhibitor of ICMT, exhibiting an IC50 value of 0.47 μM [1].Formula:C21H25ClFNOColor and Shape:SolidMolecular weight:361.88VT-102 free base
CAS:VT-102 inhibits TEAD autopalmitoylation, blocking NF2-deficient mesothelioma growth, affecting firefly luciferase, not Renilla.Formula:C21H20BrN5OSColor and Shape:SolidMolecular weight:470.39Niceritrol
CAS:Niceritrol (Cardiolipol) is a niacin ester that reduces cholesterol and triglycerides in total plasma and in the VLD and LD lipoprotein fractions.Formula:C29H24N4O8Purity:97.02%Color and Shape:SolidMolecular weight:556.52Ref: TM-T19861
1mg57.00€2mg80.00€5mg103.00€10mg147.00€25mg255.00€50mg384.00€100mg567.00€1mL*10mM (DMSO)142.00€MONIRO-1
CAS:MONIRO-1 blocks T/N-type Ca²⁺ channels: hCav2.2 (IC50: 34μM), hCav3.1 (3.3μM), hCav3.2 (1.7μM), hCav3.3 (7.2μM).Formula:C23H24ClFN4O3Color and Shape:SolidMolecular weight:458.92HOE961
CAS:HOE961, a diacetate ester prodrug of S2242, is an oral anti-orthopoxvirus agent effective against cowpox.Formula:C13H17N5O5Color and Shape:SolidMolecular weight:323.3FGFR3-IN-7
CAS:FGFR3-IN-7 is a potent, selective inhibitor of FGFR 3, demonstrating an IC50 value of less than 350 nM , and is utilized in cancer research [1].Formula:C25H24FN9OPurity:98%Color and Shape:SolidMolecular weight:485.52SQ 26655
CAS:SQ 26655 is an antagonist of thromboxane A2/prostaglandin H2.Formula:C21H34O4Purity:98%Color and Shape:SolidMolecular weight:350.49SKI2496
CAS:SKI2496: potent, oral GnRH receptor antagonist, hGnRHR IC50=0.46nM, 84% LH inhibition at 12h, 76% at 24h, selective for humans over monkeys/rats.Formula:C35H36F7N5O5Color and Shape:SolidMolecular weight:739.68Dersalazine sodium
CAS:Dersalazine, potential ulcerative colitis drug, inhibits PAF & TNFα, reduces inflammation and MPO activity in rats.Formula:C35H32N6NaO4Purity:98%Color and Shape:SolidMolecular weight:623.669SARS-CoV-2-IN-66
CAS:SARS-CoV-2-IN-66 (1), a derivative of vitamin K, functions as an inhibitor of SARS-CoV-2, exhibiting an effective concentration (EC50) of 70.8 μM in VeroE6/Formula:C28H30O2Purity:98%Color and Shape:SolidMolecular weight:398.54Tomaymycin DM
CAS:Tomaymycin DM, a derivative of Tomaymycin, functions as a DNA alkylator and PBD dimer.Formula:C14H14N2O3Color and Shape:SolidMolecular weight:258.27PD 109488
CAS:PD 109488 is a metabolite of quinapril and is a derivative of Quinapril that acts as an ACE inhibitor.Formula:C25H28N2O4Purity:98%Color and Shape:SolidMolecular weight:420.5NF 023
CAS:NF 023 is a potent, selective P2X1 purinoceptor antagonist.Formula:C35H26N4O21S6Color and Shape:SolidMolecular weight:1030.99Keap1-Nrf2-IN-10
CAS:Keap1-Nrf2-IN-10 (compound 15) is a potent inducer of NQO1 and efficaciously mitigates oxidative stress in gamma-irradiated mice by reducing MDA and ROS levelsFormula:C25H22I2N4O7S2Color and Shape:SolidMolecular weight:808.4Fomocaine
CAS:Fomocaine (P 652), an orally active local anesthetic, also exhibits antiarrhythmic activity [1] [2].Formula:C20H25NO2Color and Shape:SolidMolecular weight:311.42VU0360172
CAS:VU0360172 is a positive allosteric modulator of mGlu5 receptors (EC50 = 16 nM; Ki = 195 nM).Formula:C18H15FN2OPurity:99.56%Color and Shape:SolidMolecular weight:294.32YUN90389
CAS:YUN90389 (CAS#1673590-38-9) is the first pparα/δ dual antagonist, as reported in 2019.Formula:C34H29F4N3O4Color and Shape:SolidMolecular weight:619.61BDM91270
CAS:BDM91270 (compound 29) serves as an inhibitor of the E.Formula:C17H21Cl3N4O2Color and Shape:SolidMolecular weight:419.73Henatinib
CAS:Henatinib: orally active multi-kinase inhibitor targeting VEGFR-2, c-kit, PDGFR with antitumor effects.Formula:C25H29FN4O4Color and Shape:SolidMolecular weight:468.52Aurora Kinases-IN-4
CAS:Aurora Kinases-IN-4 (Compound 11c) is a covalent, ATP-competitive inhibitor of aurora kinase A with an IC50 value of 1.7 nM.Formula:C26H28N8OPurity:98%Color and Shape:SolidMolecular weight:468.55MGAT2-IN-2
CAS:MGAT2-IN-2 is a potent inhibitor of acyl CoA:monoacylglycerol acyltransferase 2 (MGAT2) (IC50 of 3.4 nM).Formula:C26H21F5N4O4SPurity:98%Color and Shape:SolidMolecular weight:580.53NUC-7738
CAS:NUC-7738 is a 5'-aryloxyphosphoamidoester prodrug of 3'-dA, which regulates 尾-catenin signaling and can be used in cancer research.Formula:C26H29N6O7PPurity:97.32% - 97.32%Color and Shape:SolidMolecular weight:568.52Hydroxy Darunavir
CAS:Hydroxy darunavir, a metabolite of the HIV-1 protease inhibitor darunavir, is generated through isobutyl aliphatic hydroxylation of darunavir.Formula:C27H37N3O8SColor and Shape:SolidMolecular weight:563.66BX-320
CAS:BX-320, a PDK1 inhibitor (IC50=30nM), selectively blocks Akt/p70S6K1 phosphorylation, induces apoptosis, and inhibits cancer cell growth.Formula:C23H31BrN8O3Color and Shape:SolidMolecular weight:547.45GW-813893
CAS:GW-813893: potent, selective oral factor Xa inhibitor; Ki 4.0 nM (FXa), 9.7 nM (prothrombinase).Formula:C17H22ClN3O5S2Purity:98%Color and Shape:SolidMolecular weight:447.96S-Benzylglutathione
CAS:S-Benzylglutathione acts as a competitive inhibitor of glutathionase and undergoes conversion by rat kidney microsomes into its cysteine derivatives.Formula:C17H23N3O6SColor and Shape:SolidMolecular weight:397.45ICMT-IN-33
CAS:ICMT-IN-33 (compound 73) functions as an ICMT inhibitor with an IC50 value of 0.46 μM [1].Formula:C20H24ClNOColor and Shape:SolidMolecular weight:329.86Naxagolide free base
CAS:Naxagolide is a sustained release formulation. It is a dopamine agonist.Formula:C15H21NO2Purity:98%Color and Shape:SolidMolecular weight:247.33Bcl-2-IN-16
CAS:Bcl-2-IN-16 is a Bcl-2 (B-cell lymphoma 2) inhibitor [1].Formula:C53H63ClN8O10SColor and Shape:SolidMolecular weight:1039.63Solimastat
CAS:Solimastat: oral MMPI, >10x active than marimastat, inhibits cell-bound TNF-alpha processing.Formula:C20H32N4O5Color and Shape:SolidMolecular weight:408.49EGGGG-PEG8-amide-bis(deoxyglucitol)
CAS:EGGGG-PEG8-amide-bis(deoxyglucitol) constitutes a cleavable linker utilized in Antibody-Drug Conjugates (ADCs).Formula:C49H91N9O28Color and Shape:SolidMolecular weight:1254.29ALM301
CAS:ALM301: oral AKT inhibitor targeting AKT1, AKT2, AKT3; blocks AKT phosphorylation, curbs cancer cell growth.Formula:C25H25N3O3Color and Shape:SolidMolecular weight:415.48KRAS inhibitor-12
CAS:KRAS inhibitor-12 blocks KRAS G12C (IC50: 0.537 μM) and p-ERK in cancer cells; promising for pancreatic, colorectal, lung cancer study.Formula:C19H16Cl2FN5OSColor and Shape:SolidMolecular weight:452.33CPFX2090
CAS:CPFX2090, a cephalosporin antibacterial compound.Formula:C28H28ClNO6Purity:98%Color and Shape:SolidMolecular weight:509.98DA-3934
CAS:DA-3934 targets gastrin/CCK-B receptors, not CCK-A, and reduces rat gastric acid secretion dose-dependently.Formula:C35H35N5O7Purity:98%Color and Shape:SolidMolecular weight:637.681-Palmitoyl-2-succinyl-sn-glycerophosphorylcholine
CAS:1-Palmitoyl-2-succinyl-sn-glycerophosphorylcholine, a glycerophosphorylcholine derivative, comprises glycerol phosphate, choline, and palmitic acid andFormula:C28H54NO10PColor and Shape:SolidMolecular weight:595.7AC-099 hydrochloride
CAS:AC-099 hydrochloride is a full agonist of neuropeptide FF2 receptor NPFF2R and a partial agonist of neuropeptide FF1 receptor NPFF1R.Formula:C9H9Cl2F3N4Purity:99.86%Color and Shape:SolidMolecular weight:301.1AVG-233
CAS:AVG-233 is an RNA-dependent RNA polymerase (RdRp) inhibitor with antiviral activity for the study of respiratory syncytial virus infections.Formula:C26H22ClN5O3Purity:99%Color and Shape:SolidMolecular weight:487.94OB 24 hydrochloride
CAS:OB 24 hydrochloride inhibits HO-1 (IC50 = 1.9 μM), not HO-2, and curbs PCA cell growth, carbonylation, ROS; also reduces tumor/metastases with Taxol.Formula:C15H18BrClN2O2Purity:99.98%Color and Shape:SolidMolecular weight:373.68Ref: TM-T41175
1mgTo inquire5mgTo inquire10mg164.00€25mgTo inquire50mgTo inquire100mgTo inquire1mL*10mM (DMSO)To inquireRS 5773
CAS:RS 5773 is a benzothiazepine derivative with antianginal effects.Formula:C29H33ClN2O4SPurity:98%Color and Shape:SolidMolecular weight:541.1Timepidium bromide
CAS:Timepidium bromide is an agent of anticholinergic.Formula:C17H22BrNOS2Purity:98%Color and Shape:SolidMolecular weight:400.4Dasolampanel etibutil
CAS:Dasolampanel etibutil is a novel selective antagonist of ionotropic glutamate receptor 5 (iGluR5).Formula:C23H32ClN5O3Color and Shape:SolidMolecular weight:461.98Lipid peroxidation inhibitor 1
CAS:Lipid peroxidation inhibitor 1 is an inhibitor of lipid peroxidation (IC50: 0.07 μM).
Formula:C24H32N2OPurity:98%Color and Shape:SolidMolecular weight:364.52Deoxynybomycin
CAS:Deoxynybomycin, a selective anti-tumor agent, inhibits topoisomerase I and induces apoptosis.Formula:C16H14N2O3Purity:98%Color and Shape:SolidMolecular weight:282.29ICI 200355
CAS:ICI 200355 is an inhibitor of human neutrophil elastase.Formula:C30H34BrF3N4O7SPurity:98%Color and Shape:SolidMolecular weight:731.58CHMFL-FLT3-122
CAS:CHMFL-FLT3-122 is a potent and orally available FLT3 kinase inhibitor used to treat FLT3-ITD positive acute myeloid leukemia.
Formula:C26H29N7O2Purity:99.63%Color and Shape:SolidMolecular weight:471.55GABA-IN-2
CAS:GABA-IN-2 (Compound 5), a GABA inhibitor, exhibits both larvicidal and insecticidal properties, achieving an 87% mortality rate at a concentration of 50 mg/L [1Formula:C12H4Cl2F6N4SeColor and Shape:SolidMolecular weight:468.04Lingdolinurad
CAS:Lingdolinurad is a uric acid transporter protein inhibitor targeting hURAT1 for the study of hyperuricemia or gout.Formula:C17H12BrN3O2Purity:96.26%Color and Shape:SolidMolecular weight:370.2Ref: TM-T79854
1mg115.00€5mg275.00€10mg394.00€25mg615.00€50mg848.00€100mg1,121.00€200mg1,510.00€1mL*10mM (DMSO)281.00€Me-Indoxam
CAS:Me-Indoxam is an inhibitor of sPLA2. It has no effect on arachidonic acid release and platelet activating factor synthesis.Formula:C26H22N2O5Purity:98%Color and Shape:SolidMolecular weight:442.46
