Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,834 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,613 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,015 products)
- Immunology and Inflammation(3,904 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,257 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,137 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,423 products)
- Other Inhibitors(35,848 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,429 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(732 products)
- Tyrosine Kinase/Adaptors(1,982 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66516 products of "Inhibitors"
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U 104489
CAS:U 104489 (PNU-104489) is a novel specific inhibitor of human immunodeficiency virus 1 (HIV-1), showing effective activity against BHA-P-resistant HIV-1MF.Formula:C26H36N6O3SColor and Shape:SolidMolecular weight:512.67PRMT6-IN-3
CAS:PRMT6-IN-3 is a selective PRMT6 inhibitor with an IC50 value of 192 nM.PRMT6-IN-3 has anticancer activity and induces apoptosis in cancer cells.Formula:C19H26N4O2SPurity:98.12%Color and Shape:SolidMolecular weight:374.5SHP2-IN-20
CAS:SHP2-IN-20 (compound 193), a potent SHP2 inhibitor, exhibits an IC50 of 3 nM, making it suitable for glioblastoma research [1].Formula:C25H24F2N6Color and Shape:SolidMolecular weight:446.5RASP-IN-1
CAS:RASP-IN-1 (Compound A), a lipophilic compound, serves as an inhibitor for macular degeneration and exhibits biological activity within the rabbit retina.Formula:C16H16N2O2Color and Shape:SolidMolecular weight:268.31DDR1/2 inhibitor-2
CAS:DDR1/2 Inhibitor-2 (Example 31) serves as an inhibitor of DDR1/DDR2, exhibiting IC50 values below 100 nM.Formula:C25H19F3N6O2Color and Shape:SolidMolecular weight:492.45Stafib-2
CAS:Stafib-2 is a potent and selective inhibitor of the transcription factor STAT5b.Stafib-2 inhibits STAT5b and STAT5a with IC50 values of 82 nM and 1.7 μM,
Formula:C28H26N2O12P2Purity:98.48%Color and Shape:SolidMolecular weight:644.46PD-L1-IN-2
CAS:PD-L1-IN-2, a Naamidine J derivative, serves as a promising antineoplastic immunomodulator by hindering PD-L1 activity.Formula:C33H38N4O6Purity:98%Color and Shape:SolidMolecular weight:586.68MK-0493
CAS:MK-0493 is an effective and selective agonist of the melanocortin receptor 4 (MC4R). It also demonstrated significant reductions in energy intake.Formula:C30H38ClF2N3O2Purity:98%Color and Shape:SolidMolecular weight:546.09PBR28
CAS:PBR28, a TSPO modulator, holds potential for preventative research in Pulmonary Arterial Hypertension (PAH) and is instrumental in brain positron emissionFormula:C21H20N2O3Purity:98%Color and Shape:SolidMolecular weight:348.4Barzuxetan
CAS:Barzuxetan is a potential research tool in oncology [1].Formula:C26H34N4O10SColor and Shape:SolidMolecular weight:594.63CGA-JK3
CAS:CGA-JK3 is an IkappaB kinase inhibitor in innate immune process.Formula:C15H19NO3Purity:98%Color and Shape:SolidMolecular weight:261.32ZINC03129319
CAS:ZINC03129319 is an inhibitor of dengue virus (DENV) NS2B-NS3 protease.Formula:C24H14N2O6S2Purity:90%Color and Shape:SolidMolecular weight:490.51Caerulomycin A
CAS:Caerulomycin A (Caerulomycin) (Cerulomycin; Caerulomycin) is an antifungal compound.Formula:C12H11N3O2Purity:99.28%Color and Shape:SolidMolecular weight:229.23Ref: TM-T14854
1mg145.00€5mg284.00€10mg424.00€25mg730.00€50mg1,064.00€100mg1,406.00€200mg1,863.00€1mL*10mM (DMSO)261.00€Pumaprazole
CAS:Pumaprazole (BY-841) is an antagonist of a reversible proton pump.Formula:C19H22N4O2Purity:99.91%Color and Shape:SolidMolecular weight:338.4Ref: TM-T16682
1mg87.00€5mg178.00€10mg295.00€25mg602.00€50mg964.00€100mg1,558.00€200mg2,097.00€1mL*10mM (DMSO)203.00€Arbemnifosbuvir
CAS:Arbemnifosbuvir, a drug interfering with the nidovirus DdRp-associated nucleotidyltransferase (NiRAN) domain of non-structural protein 12 (nsp12), is utilizedFormula:C24H33FN7O7PPurity:98%Color and Shape:SolidMolecular weight:581.53MDK-5432
CAS:MDK-5432, also known as AMPA stabilizer (R,R)-2a, is the most potent AMPA stabilizer.Formula:C20H28N2O4S2Color and Shape:SolidMolecular weight:424.58GSK1842799
CAS:GSK1842799 is a selective S1P1 receptor agonist with good oral bioavailability.Formula:C24H30F9N3O6SColor and Shape:SolidMolecular weight:659.56MK-8666
CAS:MK-8666, a partial GPCR agonist targeting GPR40, may treat type 2 diabetes by enhancing insulin secretion and lowering glucose safely.Formula:C29H31NO6SColor and Shape:SolidMolecular weight:521.62MRS 1754
CAS:MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.
Formula:C26H26N6O4Purity:97.57% - 99.3%Color and Shape:SolidMolecular weight:486.52Raloxifene Bismethyl Ether hydrochloride
CAS:Raloxifene Bismethyl Ether hydrochloride is a Raloxifene metabolite and an estrogen receptor inactive compound on which both hydroxyl groups are absent.Formula:C30H32ClNO4SPurity:98%Color and Shape:SolidMolecular weight:538.1A1/A3 AR antagonist 3
CAS:A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful inFormula:C22H19N5O3Purity:98%Color and Shape:SolidMolecular weight:401.42AM-8735
CAS:AM-8735 is an inhibitor of MDM2 ( IC50: 25 nM).Formula:C27H31Cl2NO6SPurity:98%Color and Shape:SolidMolecular weight:568.51Urease-IN-6
CAS:Urease-IN-6, a potent Urease inhibitor, exhibits an IC50 value of 14.2 μM and is utilized in the research of peptic and gastric ulcers [1].Formula:C18H19N3OSColor and Shape:SolidMolecular weight:325.43Mal-PEG8-Val-Ala-PAB-Exatecan
CAS:Mal-PEG8-Val-Ala-PAB-Exatecan (Compound 9b), an antibody-drug conjugate linker (ADC linker), binds Nectin-4 polypeptides to chemotherapeutic agents for use inFormula:C66H85FN8O20Color and Shape:SolidMolecular weight:1329.42(Rac)-Modipafant
CAS:(Rac)-Modipafantis a PAFR antagonist that inhibits PAF-induced aggregation of washed platelets in rabbits.Formula:C34H29ClN6O3Purity:97.96% - 98.09%Color and Shape:SolidMolecular weight:605.09BMS-639623
CAS:BMS-639623 is a CCR3 antagonist with a picomolar inhibitory effect on eosinophilic chemotaxis and can be used in the treatment of asthma.Formula:C25H32FN7O2Color and Shape:SolidMolecular weight:481.57Tedizolid HCl (856866-72-3 free base)
Tedizolid HCl, a novel oxazolidinone antibiotic, IC50: MAO-A 8.7 uM, MAO-B 5.7 uM, approved post-linezolid, has a prodrug form tedizolid phosphate.Formula:C17H16ClFN6O3Purity:98%Color and Shape:SolidMolecular weight:406.8ZH8659
CAS:ZH8659 is a Gq agonist targeting the trace amine-associated receptor 1 (TAAR1) and has potential applications in schizophrenia research [1].Formula:C12H13NOColor and Shape:SolidMolecular weight:187.24MI-888 free base
CAS:MI-888 is the most potent MDM2 inhibitor (Ki = 0.44 nM), with high oral efficacy in human cancer models and optimal pharmacokinetics.Formula:C28H32Cl2FN3O3Color and Shape:SolidMolecular weight:548.48mp-dLAE-PABC-MMAE
CAS:mp-dLAE-PABC-MMAE is an agent-linker conjugate for antibody-drug conjugates (ADCs) that incorporates the potent tubulin inhibitor Monomethyl auristatin E (MMAEFormula:C68H102N10O17Color and Shape:SolidMolecular weight:1331.59Indinavir lactone
CAS:Indinavir lactone is a protease inhibitor used as a component of highly active antiretroviral therapy to treat HIV/AIDS.Formula:C27H36N4O3Color and Shape:SolidMolecular weight:464.6Demethyleneberberine chloride
CAS:Demethyleneberberine chloride, a natural mitochondria-targeted antioxidant, mitigates colitis in mice and suppresses inflammatory responses by blocking the NF-Formula:C19H18ClNO4Purity:98%Color and Shape:SolidMolecular weight:359.8AM-461 sodium
CAS:AM-461 sodium is the sodium salt of AM-461 --- a novel DP2 receptor antagonistFormula:C25H32NNaO5SColor and Shape:SolidMolecular weight:481.58Fmoc-Gly3-Val-Cit-PAB
CAS:Fmoc-Gly3-Val-Cit-PAB is a cleavable linker utilized in the assembly of antibody-drug conjugates (ADCs).Formula:C39H48N8O9Color and Shape:SolidMolecular weight:772.85BAY-7081
BAY-7081 is a cyanopyridone-based compound that functions as a potent, selective, and orally active PDE9A inhibitor, demonstrating an inhibition concentration (Formula:C19H27ClN4OColor and Shape:SolidMolecular weight:362.9KRAS G12C inhibitor 25
CAS:KRAS G12C inhibitor 25 blocks SOS1-mediated GDP/GTP swap in KRAS-G12C mutants; IC50: 0.48 nM (WO2021216770A1, comp. 3).Formula:C32H41N7O2Color and Shape:SolidMolecular weight:555.71Curcumin-β-D-glucuronide
CAS:Curcumin-β-D-glucuronide, a principal metabolite detected in hepatic tissue and portal blood following oral consumption of Curcumin, is utilized in colon cancerFormula:C27H28O12Purity:98%Color and Shape:SolidMolecular weight:544.5IKK-IN-1
CAS:IKK-IN-1 is an inhibitor of IKK.Formula:C22H26ClN3O4Purity:98%Color and Shape:SolidMolecular weight:431.91S-Adenosyl-L-methionine (1,4-butanedisulfonate)
CAS:S-Adenosyl-L-methionine (SAMe) 1,4-butanedisulfonate functions as an orally active methyl group donor and serves as a dietary supplement known for itsFormula:C19H32N6O11S3Purity:98%Color and Shape:SolidMolecular weight:616.69SW IV-52
CAS:SW IV-52 is an XIAP-inhibitor that acts as a second mitochondria-derived activator of caspases (SMAC) mimetic.Formula:C25H39ClN4O3Purity:98%Color and Shape:SolidMolecular weight:479.05PF-02575799
CAS:PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).Formula:C42H37FN4O4Purity:98%Color and Shape:SolidMolecular weight:680.77CD235
CAS:CD235 is a structurally similar analog of CD161. CD161 is an orally bioavailable inhibitor of BET bromodomain.Formula:C26H20FN5O2Purity:98%Color and Shape:SolidMolecular weight:453.47(S)-(-)-MRJF22
CAS:(S)-(-)-MRJF22, a haloperidol metabolite II valproate ester, demonstrates potent antimigratory effects in both endothelial and tumor cells, and is considered aFormula:C29H39ClFNO3Color and Shape:SolidMolecular weight:504.08Xanthine amine congener
CAS:Xanthine amine congener is an Adenosine receptor antagonist.Formula:C21H28N6O4Purity:99.7%Color and Shape:SolidMolecular weight:428.48Orexin receptor modulator-1
CAS:Orexin Receptor Modulator-1 is a compound utilized in the study of various conditions including substance addiction, panic disorder, anxiety, post-traumaticFormula:C23H22ClF5N6OColor and Shape:SolidMolecular weight:528.91SLU-10482
CAS:SLU-10482, an antiparasitic agent, effectively reduces C.Formula:C18H16F4N6OColor and Shape:SolidMolecular weight:408.35h-NTPDase-IN-5
CAS:h-NTPDase-IN-5 (compound 3b) serves as a pan-inhibitor of NTPDase, exhibiting inhibitory concentration 50 (IC50) values of 1.10 μM (h-NTPDase1), 44.73 μM (h-Formula:C23H21N3O2SPurity:98%Color and Shape:SolidMolecular weight:403.5Sezolamide hydrochloride
CAS:Sezolamide hydrochloride is a potent topical carbonic anhydrase inhibitor.Formula:C11H19ClN2O4S3Color and Shape:SolidMolecular weight:374.93Formoterol HCl
CAS:Formoterol HCl is a long-acting beta-2 adrenergic agonist (LABA).Formula:C19H25ClN2O4Color and Shape:SolidMolecular weight:380.869HDAC6-IN-21
CAS:HDAC6-IN-21 (compound 13) is an irreversible inhibitor of histone deacetylase 6 (HDAC6) [1].Formula:C14H13F2N5O2Purity:98%Color and Shape:SolidMolecular weight:321.28
