Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,853 products)
- Apoptosis(6,368 products)
- Cell Cycle/Checkpoint(4,909 products)
- Chromatin/Epigenetics(2,633 products)
- Cytoskeletal Signaling(1,587 products)
- DNA Damage/DNA Repair(2,868 products)
- Endocrinology/Hormones(3,765 products)
- Enzyme(3,673 products)
- GPCR/G-Protein(9,054 products)
- Immunology and Inflammation(3,952 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(417 products)
- MAPK Signaling(1,259 products)
- Membrane Transporter/Ion Channel(3,163 products)
- Metabolism(10,156 products)
- Microbiology/Virology(7,674 products)
- Neuroscience(10,550 products)
- Other Inhibitors(35,855 products)
- Oxidation-Reduction(41 products)
- PI3K/Akt/mTOR Signaling(1,437 products)
- Proteases/Proteasome(1,692 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,992 products)
- Ubiquitination(1,744 products)
Show 16 more subcategories
Found 66513 products of "Inhibitors"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
FX-06
CAS:FX-06 (Fibrin-derived peptide Bβ15-42) is a peptide derived from the fibrin Bbeta chain.Formula:C133H216N44O38Color and Shape:SolidMolecular weight:3039.41CP-664511
CAS:CP-664511 is an alpha4beta1/ vascular cell adhesion molecule-1 (VCAM-1) inhibitor with therapeutic potential for allergic airway disease.Formula:C28H34N4O6Color and Shape:SolidMolecular weight:522.59NK3R-IN-1
CAS:NK3R-IN-1 (compound 16x), an orally active imidazolepiperazine derivative, acts as a Neurokinin Receptor NK3R inhibitor and has been shown to reduce bloodFormula:C17H16FN5OSPurity:98%Color and Shape:SolidMolecular weight:357.41PI5P4Kα-IN-1
CAS:PI5P4Kα-IN-1 (Compound 13) is a phosphatidylinositol 5-phosphate 4-kinase (PI5P4K) inhibitor, displaying IC50 values of 2 μM for PI5P4Kα and 9.4 μM for PI5P4KβFormula:C20H17N3O2SPurity:98%Color and Shape:SolidMolecular weight:363.43WRR139
CAS:WRR139, a peptide vinyl sulfone, plays a role in disease processes including inflammation and cancer, and acts as an inhibitor of cytosolic enzyme N-glycanase 1Formula:C25H32N2O4SColor and Shape:SolidMolecular weight:456.6VU0364739
CAS:VU0364739, a selective phospholipase D2 (PLD2) inhibitor with an IC50 of 22 nM, effectively reduces cancer cell proliferation [1].Formula:C26H27FN4O2Purity:98%Color and Shape:SolidMolecular weight:446.52CDD-1845
CAS:CDD-1845, a non-covalent, non-peptide inhibitor, exhibits potent inhibition of SARS-CoV-2 M^pro with a K_i value of 3 nM.Formula:C34H31N5O2Purity:98%Color and Shape:SolidMolecular weight:541.64CJ-42794
CAS:CJ-42794 (CJ-042794) is a selective antagonist of prostaglandin E receptor subtype 4 (EP4).Formula:C22H17ClFNO4Purity:99.92%Color and Shape:SolidMolecular weight:413.83L-ANAP hydrochloride (1313516-26-5 free base)
L-ANAP hydrochloride is a polarity-sensitive and genetically encodable fluorescent unnatural amino acid.Formula:C15H17ClN2O3Purity:98%Color and Shape:SolidMolecular weight:308.76Fulvestrant (R enantiomer)
CAS:Fulvestrant R enantiomer is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.Formula:C32H47F5O3SPurity:98%Color and Shape:SolidMolecular weight:606.77PonatiLink-1-24
CAS:Ponatinib, also known as PonatiLink-1-24, is a selective inhibitor of the Abelson murine leukemia (ABL) enzyme [1].Formula:C101H144ClF5N12O29Color and Shape:SolidMolecular weight:2120.73Petesicatib
CAS:Petesicatib is an inhibitor of cathepsin S. Petesicatib used in the research of immune diseases.Formula:C25H23F6N5O4SPurity:99.76%Color and Shape:SolidMolecular weight:603.54Ref: TM-T16474
1mg100.00€5mg236.00€1mL*10mM (DMSO)314.00€10mg371.00€25mg735.00€50mg1,134.00€100mg1,468.00€200mg1,972.00€Proteasome β2c/i-IN-1
CAS:Proteasome β2c/i-IN-1 (compound 37) serves as a selective inhibitor targeting the β2c and β2i subunits of the human proteasome [1].Formula:C32H48N4O7Purity:98%Color and Shape:SolidMolecular weight:600.75JNJ4796
CAS:JNJ4796 is an oral fusion inhibitor that neutralizes influenza A group 1 by blocking HA-mediated fusion, mimicking bnAbs.Formula:C28H27N9O3Purity:98%Color and Shape:SolidMolecular weight:537.57Docosatrienoic Acid
CAS:Docosatrienoic acid is a rare omega-3 fatty acid; Ki value is 5×M, which inhibits the binding of LTB4 to porcine neutrophil membrane.Formula:C22H38O2Purity:98%Color and Shape:SolidMolecular weight:334.54Kif15-IN-2
CAS:Kif15-IN-2 is a kinesin Kif15 inhibitor with potential anticancer activity and can be used in prostate cancer research.Formula:C20H20N6O4SPurity:98.17%Color and Shape:SolidMolecular weight:440.48FC 11
CAS:FC 11 is a reversible FAK PROTAC Degrader with DC50 of 40-370 pM and degrades pFAKtyr397 in TM3 cells within 3 hours at 100 nM.Formula:C41H42F3N13O9SColor and Shape:SolidMolecular weight:949.91LTB4 antagonist 1
CAS:LTB4 Antagonist 1, a carboxamide-acid derivative, potently inhibits Leukotriene B4 (LTB4) activity with an IC50 value of 288 nM and exhibits notable anti-Formula:C26H23NO6Purity:98%Color and Shape:SolidMolecular weight:445.46KRAS G12C inhibitor 14
CAS:KRAS G12C inhibitor 14 is a potent KRAS G12C inhibitor with an IC 50 of 18 nM [1].Formula:C24H19ClF2N4O3Purity:98%Color and Shape:SolidMolecular weight:484.88PDE5-IN-2
CAS:PDE5-IN-2 is a potent, highly selective, and orally active inhibitor of PDE5(IC50 of 0.31 nM)Formula:C25H21N3O6SPurity:98%Color and Shape:SolidMolecular weight:491.52COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Formula:C16H16ClNO3SPurity:99.75%Color and Shape:SolidMolecular weight:337.82Ref: TM-T36520
1mg38.00€5mg86.00€1mL*10mM (DMSO)94.00€10mg123.00€25mg215.00€50mg299.00€100mg411.00€200mg560.00€HDAC-IN-63
CAS:HDAC-IN-63 (Compound 63) is a dual FLT3/HDAC inhibitor with IC50 values of 0.844 nM for FLT3 and 30.0 nM for HDAC1.Formula:C25H26Cl2N6O3Color and Shape:SolidMolecular weight:529.42JT002
CAS:JT002 is an orally active NLRP3 inflammasome inhibitor that decreases the production of NLRP3-dependent proinflammatory cytokines (such as IL-1β, IL-1α, IL-18)Formula:C20H24N4O5SPurity:98%Color and Shape:SolidMolecular weight:432.49Aurora kinase inhibitor-8
CAS:Aurora kinase inhibitor-8 is a highly selective inhibitor of Aurora kinase.Formula:C30H29N7O3Color and Shape:SolidMolecular weight:535.6Glycosidase-IN-1
CAS:Glycosidase-IN-1, a D-mannose-derived inhibitor, has hypoglycemic effects and aids in creating immunosuppressants and β-glucosidase blockers.Formula:C13H23NO5Purity:98%Color and Shape:SolidMolecular weight:273.33WNY1613
CAS:WNY1613: Potent PI3Kδ inhibitor with anti-NHL properties, induces apoptosis in cells, affects phosphorylation in vitro/in vivo.Formula:C29H35N9O3Color and Shape:SolidMolecular weight:557.65Antiproliferative agent-40
CAS:Antiproliferative agent-40 (Compound 9) effectively inhibits the proliferation of HT1080 and MCF-7 cancer cells, displaying IC50 values of 52 μM and 8.2 μM,Formula:C20H18N4O3Color and Shape:SolidMolecular weight:362.38Antifungal agent 66
CAS:Antifungal agent 66 (compound 10) exhibits broad-spectrum antifungal activity against seven phytopathogenic fungal mycelia and significant inhibitory effects onFormula:C19H25ClO6Color and Shape:SolidMolecular weight:384.85PZ-1190
CAS:PZ-1190, a multitarget ligand for serotonin and dopamine receptors, exhibits potential antipsychotic activity in rodents [1].Formula:C27H30N4O2S2Purity:98%Color and Shape:SolidMolecular weight:506.68Collagen proline hydroxylase inhibitor
CAS:Collagen proline hydroxylase inhibitor is an inhibitor collagen proline hydroxylase and useful for antifibrotic proliferative agents.Formula:C18H18N4O4Purity:98%Color and Shape:SolidMolecular weight:354.36Oxilorphan
CAS:Oxilorphan is a μ-opioid blocker and a weak κ-opioid activator; similar to naloxone in strength; can cause hallucinations and dysphoria.Formula:C20H27NO2Purity:98%Color and Shape:SolidMolecular weight:313.43GPR120 Agonist 3
CAS:GPR120 Agonist 3 (GPR120-IN-1) is a selective agonist of Gpr120 ( logEC50: -7.62).Formula:C19H23ClF3NO3Purity:99.01%Color and Shape:SolidMolecular weight:405.84Ref: TM-T15413
1mg34.00€5mg84.00€1mL*10mM (DMSO)93.00€10mg137.00€25mg260.00€50mg371.00€100mg557.00€200mg790.00€Trk-IN-10
CAS:Trk-IN-10 inhibits TRK (IC50: 0.86 nM TrkA, 6.92 nM TrkA G595R, 350 nM ALK), promising for solid tumors with selective action and potential lower toxicity.Formula:C20H20FN5O3Color and Shape:SolidMolecular weight:397.4STAT3-IN-B9
CAS:STAT3-IN-B9 (B9) is an inhibitor of abnormal STAT3 activation and inhibits the proliferation of tumor cells including MDA-MB-468, MDA-MB-231, and DU145.Formula:C20H13NO5SPurity:98.19%Color and Shape:SolidMolecular weight:379.39Ref: TM-T28865
1mg109.00€2mg154.00€5mg235.00€1mL*10mM (DMSO)255.00€10mg349.00€25mg532.00€50mg745.00€100mg999.00€200mg1,333.00€TM-N1324
CAS:TM-N1324 is a GPR39 agonist; 280 nM potency without Zn2+, 9 nM with; similar effects on murine GPR39 (EC50s: 180 nM/5 nM).Formula:C18H13ClFN7OPurity:99.88%Color and Shape:SolidMolecular weight:397.79Ref: TM-T17103
1mg49.00€2mg64.00€5mg90.00€1mL*10mM (DMSO)92.00€10mg170.00€25mg371.00€50mg557.00€100mg792.00€SN38-COOH
CAS:SN38-COOH, the active metabolite of the topoisomerase I inhibitor irinotecan, is utilized in the synthesis of antibody-drug conjugates (ADCs).Formula:C26H24N2O8Color and Shape:SolidMolecular weight:492.48AMG-7549
CAS:AMG-7549 is a disrupter of Glucokinase−Glucokinase Regulatory Protein (GK−GKRP) binding.Formula:C24H24ClN5O3S2Color and Shape:SolidMolecular weight:530.06PF-07059013
CAS:PF-07059013, an orally active and potent noncovalent modulator of sickled hemoglobin (HbS), specifically binds to Hb with nanomolar affinity and demonstratesFormula:C19H16FN5O2Color and Shape:SolidMolecular weight:365.36Nivocasan
CAS:Nivocasan (GS-9450/LB-84451), a caspase-inhibitor, reduces ALT in NASH, shows hepatoprotective effects in fibrosis models.Formula:C21H22FN3O5Color and Shape:SolidMolecular weight:415.41Raloxifene Bismethyl Ether hydrochloride
CAS:Raloxifene Bismethyl Ether hydrochloride is a Raloxifene metabolite and an estrogen receptor inactive compound on which both hydroxyl groups are absent.Formula:C30H32ClNO4SPurity:98%Color and Shape:SolidMolecular weight:538.1TMV-IN-2
CAS:TMV-IN-2, a chalcone, inhibits TMV with an EC50 of 89.9 μg/mL, used in infection and tumor studies.Formula:C27H23FO4Color and Shape:SolidMolecular weight:430.47KDM2B-IN-1
CAS:KDM2B-IN-1: Potent, specific KDM2B histone demethylase inhibitor for hyperproliferative disease research.Formula:C21H30N4O2SColor and Shape:SolidMolecular weight:402.56TM2 TEAD inhibitor
CAS:TM2 TEAD inhibitor, a robust and reversible inhibitor of the TEA domain transcription factor, presents dual inhibitory concentrations (IC50) of 38 nM for TEAD4Formula:C26H33N3O3Purity:99.91%Color and Shape:SolidMolecular weight:435.57TC-SP 14
CAS:TC-SP 14 (compound 14) is a potent, orally available S1P1 agonist with EC50 of 0.042 μM; minimal S1P3 binding (EC50 3.47 μM); reduces blood lymphocytes.Formula:C25H20F2N2O2SColor and Shape:SolidMolecular weight:450.5E-6123
CAS:E-6123 is an antagonist of platelet-activating factor (PAF) receptor.Formula:C23H22ClN5OSPurity:98%Color and Shape:SolidMolecular weight:451.97LMPTP INHIBITOR 1 hydrochloride
CAS:LMPTP INHIBITOR 1 hydrochloride is a selective inhibitor of low molecular weight protein tyrosine phosphatase ( LMPTP ), with an IC 50 of 0.8 μM for LMPTP-A.Formula:C28H37ClN4OPurity:99.89%Color and Shape:SolidMolecular weight:481.07Thioquinapiperifil
CAS:Thioquinapiperifil is a type of phosphodiesterase-5 (PDE-5) inhibitor found in dietary supplements.Formula:C24H28N6OSPurity:98%Color and Shape:SolidMolecular weight:448.58Pumaprazole
CAS:Pumaprazole (BY-841) is an antagonist of a reversible proton pump.Formula:C19H22N4O2Purity:99.91%Color and Shape:SolidMolecular weight:338.4Ref: TM-T16682
1mg87.00€5mg178.00€1mL*10mM (DMSO)203.00€10mg295.00€25mg602.00€50mg964.00€100mg1,558.00€200mg2,097.00€WAY-304671
CAS:WAY-304671 is an active compound with potential as a ubiquitin ligase inhibitor.Formula:C16H9ClN2OS2Color and Shape:SolidMolecular weight:344.84Ianthelliformisamine B TFA
CAS:Ianthelliformisamine B TFA, an antibiotic enhancer, is used to against resistant Gram-negative bacteria.Formula:C21H27Br2F6N3O6Purity:98%Color and Shape:SolidMolecular weight:691.25
