Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,833 products)
- Apoptosis(6,315 products)
- Cell Cycle/Checkpoint(4,875 products)
- Chromatin/Epigenetics(2,612 products)
- Cytoskeletal Signaling(1,566 products)
- DNA Damage/DNA Repair(2,872 products)
- Endocrinology/Hormones(3,754 products)
- Enzyme(3,672 products)
- GPCR/G-Protein(9,014 products)
- Immunology and Inflammation(3,901 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(415 products)
- MAPK Signaling(1,256 products)
- Membrane Transporter/Ion Channel(3,154 products)
- Metabolism(10,139 products)
- Microbiology/Virology(7,620 products)
- Neuroscience(10,377 products)
- Other Inhibitors(35,852 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,430 products)
- Proteases/Proteasome(1,691 products)
- Stem Cell and Derivatives(733 products)
- Tyrosine Kinase/Adaptors(1,983 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66522 products of "Inhibitors"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
KC-11404
CAS:KC-11404 is an LTB4 inhibitor for the treatment of b-cell leukemias and lymphomas, potently inhibiting histamine, platelet activating factor and 5-lipoxygenase.Formula:C28H38N4OColor and Shape:SolidMolecular weight:446.63Canosimibe
CAS:Canosimibe is a cholesterol absorption inhibitorFormula:C44H60FN3O10Color and Shape:SolidMolecular weight:809.96Fonsartan free acid
CAS:Fonsartan: Angiotensin receptor blocker, halts angiotensin II effects on rat vascular cells.Formula:C26H32N4O5S2Purity:98%Color and Shape:SolidMolecular weight:544.69Monoamine oxidase/Aromatase-IN-1
Compound 2q: Dual MAO/aromatase inhibitor; IC50: 39 nM (MAO-B), 31 nM (aromatase). Useful in neurological/breast cancer research.Formula:C19H19N3O3SColor and Shape:SolidMolecular weight:369.44γ-Secretase modulator 11 hydrochloride
CAS:γ-Secretase modulator 11 hydrochloride is a potent, orally active γ-secretase modulator (IC50: 0.029 μM).Formula:C28H23ClF2N4O2Color and Shape:SolidMolecular weight:520.96α-Glucosidase-IN-12
α-Glucosidase-IN-12 is a potent inhibitor of α-glucosidase (IC50: 10.20 μM).Formula:C25H30N4O4S2Color and Shape:SolidMolecular weight:514.66ERGi-USU-6 mesylate
ERGi-USU-6 (mesylate) is a new selective ERG positive prostate cancer inhibitor with an IC50 value of 0.089 μM that is an ERGi-USU-6 salt derivative.Formula:C14H18N4O4SColor and Shape:SolidMolecular weight:338.38Casein Kinase II Inhibitor IV Hydrochloride
CAS:Casein Kinase II Inhibitor IV HCl promotes keratinocyte differentiation, potential for skin disorder therapy.Formula:C24H24ClN5O3Purity:98%Color and Shape:SolidMolecular weight:465.93Antifungal agent 11
Antifungal agent 11 has a good antifungal effect.Formula:C21H19F2N7O3S2Color and Shape:SolidMolecular weight:519.55Mibefradil
CAS:Mibefradil is a calcium channel blocker with moderate selectivity for T-type Ca2+ channels (IC50s: 2.7 μM and 18.6 μM for T-type and L-type currents).Formula:C29H38FN3O3Purity:98%Color and Shape:SolidMolecular weight:495.63BW-10
CAS:BW-10 potently inhibits bombesin evoked release of gastrointestinal hormones in vitro and in vivo.Formula:C57H72N14O8Color and Shape:SolidMolecular weight:1081.27SID 26681509 quarterhydrate
SID 26681509 is a selective inhibitor of cathepsin L (IC50: 56 nM) and blocks Plasmodium falciparum (IC50: 15.4 μM) and Leishmania major (IC50: 12.5 μM).Formula:C27H35N5O6SColor and Shape:SolidMolecular weight:544.16Antitubercular agent-23
Antitubercular agent-23 combats Candida albicans (MIC: 1.1 μg/ml) and M. tuberculosis (MIC: 1 μg/ml).Formula:C20H22FN5O8SColor and Shape:SolidMolecular weight:511.48PDE4-IN-6
PDE4-IN-6: Potent PDE4 inhibitor, IC50 - 0.125μM (B), 0.43μM (D), anti-inflammatory, for arthritis research.Formula:C25H20FNO5SColor and Shape:SolidMolecular weight:465.49P-gp modulator 1
CAS:P-gp modulator 1 is a high affinity and orally available P-glycoprotein (Pgp) modulatorFormula:C41H72N2O6Purity:98%Color and Shape:SolidMolecular weight:689.02Resolvin E2
CAS:RvE2, a bioactive lipid from the SPM family, is made from EPA and reduces inflammatory neutrophil infiltration and helps treat NAFLD and other diseases.Formula:C20H30O4Color and Shape:SolidMolecular weight:334.45TRPA1 Antagonist 1
CAS:TRPA1 Antagonist 1 is an antagonist of TRPA1(IC50: 8 nM) and is a methylene phosphate prodrug which converts to its active parent drug.Formula:C24H20F6N5Na2O7PSPurity:98%Color and Shape:SolidMolecular weight:713.45Befiradol hydrochloride
CAS:Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 aggregation.Formula:C20H23Cl2F2N3OPurity:99.64%Color and Shape:SolidMolecular weight:430.32IRAK4-IN-9
CAS:IRAK4-IN-9 is a potent IRAK4 inhibitor with an IC50 of 1.5 nM, promising for inflammatory, autoimmune diseases, and cancer research.Formula:C22H25N7Color and Shape:SolidMolecular weight:387.48Antitubercular agent-11
Antitubercular agent-11 (Compound 1e) is an antitubercular agent with a bulkier electron-donating group (Bu-t) that shows the best MIC value of 0.060 μg/mL [1].Formula:C16H15N3O4Color and Shape:SolidMolecular weight:313.31Monoamine Oxidase B inhibitor 2
MAO-B inhibitor 2: potent, reversible, oral, selective (IC50=1.33 nM), BBB-penetrant, with anti-oxidant and anti-inflammatory effects for Parkinson's study.Formula:C19H19FO3Color and Shape:SolidMolecular weight:314.35CHNQD-01255
CAS:CHNQD-01255 is an orally active inhibitor of Arf-GEFs that is effective against hepatocellular carcinoma (HCC).Formula:C23H29NO6Color and Shape:SolidMolecular weight:415.48MLKL-IN-6
MLKL-IN-6 (compound P28) is a mixed lineage kinase inhibitor that specifically targets the Mixed Lineage Kinase domain-like (MLKL) protein.
Formula:C20H18N4O5Purity:98%Color and Shape:SolidMolecular weight:394.38Asukamycin
CAS:Asukamycin, from S. nodosus asukaensis, is a polyketide antibiotic inhibiting tumor cells by activating caspases 8 and 3.Formula:C31H34N2O7Color and Shape:SolidMolecular weight:546.61TS010
TS010 is a highly potent inhibitor of GLO-I, with an IC50 value of 0.57 μM. It holds significant promise for advancements in cancer research [1].Formula:C16H12N4O4SColor and Shape:SolidMolecular weight:356.365α-reductase-IN-1
CAS:5α-reductase-IN-1 is a potent inhibitor of the enzyme 5α-reductase.Formula:C31H37NO5Purity:98%Color and Shape:SolidMolecular weight:503.63GSK2945 hydrochloride
GSK2945 HCl is a specific Rev-erbα antagonist, EC50: 21.5 μM (mouse), 20.8 μM (human), increases cholesterol 7α-hydroxylase.Formula:C20H19Cl3N2O2SColor and Shape:SolidMolecular weight:457.8Spliceostatin A
CAS:Spliceostatin A is an anticancer agent and splicing inhibitor that induces apoptosis by inducing cell cycle arrest in the G1 and G2/M phases.Formula:C28H43NO8Purity:94.66%Color and Shape:SolidMolecular weight:521.643PX-316
CAS:PX-316: AKT inhibitor, reduces Akt activity by 78% in HT-29 xenografts, effective against MCF-7 and HT-29 cancers, well-tolerated intravenously.Formula:C28H57O10PColor and Shape:SolidMolecular weight:584.72TTA-P1
CAS:TTA-P1: potent T-type calcium channel inhibitor; impacts neuron firing, hormone secretion, cell growth; potential in absence epilepsy research.Formula:C19H27Cl2FN2OColor and Shape:SolidMolecular weight:389.33MDL-28050
CAS:MDL-28050 is a synthetic analog of hirudin 55-65 C-terminal fragment and a peptide inhibitor.Formula:C61H88N10O23Color and Shape:SolidMolecular weight:1329.4PDE4-IN-12
PDE4-IN-12 is a potent and safe PDE4 ubiquitous inhibitor that acts on PDE4 (IC50: 3.5 nM, SI: 2.71) and PDE7 (IC50: 15 nM, SI: 4.27).Formula:C34H35NO6Color and Shape:SolidMolecular weight:553.64LasR-IN-2
LasR-IN-2 blocks LasR via H-bond with TRY-56, useful in bacterial infection and CF research.Formula:C21H16ClN3O2Color and Shape:SolidMolecular weight:377.82WQ3810 TFA
WQ3810 TFA is an orally available fluoroquinolone with antimicrobial activity against Mycobacterium tuberculosis and inhibits the DNA rotamase activity ofFormula:C24H23F6N5O5Purity:99.52%Color and Shape:SoildMolecular weight:575.46Bleomycin Free Base
CAS:Bleomycin Free Base, a glycopeptide antibiotic, halts DNA function and treats solid tumors.Formula:C55H84N17O21S3Color and Shape:SolidMolecular weight:1415.55AM-9514
CAS:AM-9514: a potent Glucokinase activator with strong in vitro results, good pharmacokinetics, and efficacy in diabetes.Formula:C18H25N5O4Color and Shape:SolidMolecular weight:375.42sEH inhibitor-4
Compound B15: potent sEH inhibitor (0.03 nm), reduces inflammation & pain.Formula:C27H28Cl2N4O3Color and Shape:SolidMolecular weight:527.44SR121566A
CAS:SR121566A is a novel non-peptide antagonist of Glycoprotein IIb/IIIa (GP IIb-IIIa).Formula:C20H25N5O4SPurity:98%Color and Shape:SolidMolecular weight:431.51NCATS-SM4487
CAS:NCATS-SM4487 is a highly selective inhibitor of GALK1 (IC50: 0.05 μM).Formula:C25H24ClFN8O2Color and Shape:SolidMolecular weight:522.96HS-731
CAS:HS-731 is a μ-Opioid Receptor Agonist.Formula:C20H26N2O5Color and Shape:SolidMolecular weight:374.43J-104132
CAS:J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.Formula:C31H33NO7Purity:98%Color and Shape:SolidMolecular weight:531.60INCB-9471 dihydrochloride
CAS:INCB-9471 HCl: a potent CCR5 antagonist, blocks monocyte migration & HIV-1.Formula:C30H42Cl2F3N5O2Purity:98%Color and Shape:SolidMolecular weight:632.59FLT3-IN-13
FLT3-IN-13 inhibits topoisomerase II/FLT3 in leukemia with IC50 of 2.26 μM, causes G2/M arrest, and promotes apoptosis.Formula:C20H14N4O2Color and Shape:SolidMolecular weight:342.35WS-898
WS-898 boosts paclitaxel efficacy in resistant cells by inhibiting ABCB1; IC50: SW620/Ad300 - 5.0 nM, KB-C2 - 3.67 nM, HEK293/ABCB1 - 3.68 nM.Formula:C33H25N7OSColor and Shape:SolidMolecular weight:567.66PI3K-IN-23
PI3K-IN-23 is a (E)-9-oxooctadec-10-en-12-ynoic acid analogue that promotes glucose uptake (EC50: 7.00 μM).Formula:C24H33NO4SColor and Shape:SolidMolecular weight:431.59Epiderstatin
CAS:Epiderstatin is isolated from Streptomyces pulveraceus subsp. epiderstagenes; inhibits mitogenic activity of epidermal growth factor.Formula:C15H20N2O4Color and Shape:SolidMolecular weight:292.33Antiallergic agent-1
Antiallergic agent-1, an Src family kinase inhibitor, is a new and valuable lead compound with potential as an anti-allergic agent.Formula:C27H19F6N5OColor and Shape:SolidMolecular weight:543.46ATM-3507 trihydrochloride (1861449-70-8 free base)
ATM-3507 trihydrochloride is a potent tropomyosin inhibitor (IC50s: 3.83-6.84 μM in human melanoma cell lines).Formula:C37H49Cl3FN5O2Purity:98%Color and Shape:SolidMolecular weight:721.17HDAC6-IN-12
HDAC6-IN-12 is a potent inhibitor of HDAC6 that binds in the DNA chain, causing DNA damage and exhibiting anticancer effects that can be used in cancer researchFormula:C24H39F2N3O5Color and Shape:SolidMolecular weight:487.58
