Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,824 products)
- Apoptosis(6,303 products)
- Cell Cycle/Checkpoint(4,862 products)
- Chromatin/Epigenetics(2,607 products)
- Cytoskeletal Signaling(1,553 products)
- DNA Damage/DNA Repair(2,875 products)
- Endocrinology/Hormones(3,752 products)
- Enzyme(3,671 products)
- GPCR/G-Protein(8,998 products)
- Immunology and Inflammation(3,861 products)
- Influenza Virus(300 products)
- JAK/STAT signaling(416 products)
- MAPK Signaling(1,253 products)
- Membrane Transporter/Ion Channel(3,155 products)
- Metabolism(10,145 products)
- Microbiology/Virology(7,618 products)
- Neuroscience(10,355 products)
- Other Inhibitors(35,866 products)
- Oxidation-Reduction(40 products)
- PI3K/Akt/mTOR Signaling(1,426 products)
- Proteases/Proteasome(1,687 products)
- Stem Cell and Derivatives(737 products)
- Tyrosine Kinase/Adaptors(1,976 products)
- Ubiquitination(1,726 products)
Show 16 more subcategories
Found 66549 products of "Inhibitors"
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GSK864
CAS:GSK864 is an inhibitor of isocitrate dehydrogenase 1 (IDH1) mutant. GSK864 inhibits IDH1 mutants R132C, R132H, and R132G (IC50: 8.8, 15.2, and 16.6 nM).Formula:C30H31FN6O4Purity:97.07%Color and Shape:SolidMolecular weight:558.6NSC381467
CAS:NSC381467: Potent, oral EGFR-TK inhibitor with strong antiproliferative effects, promising for cancer research.Formula:C20H16O7Color and Shape:SolidMolecular weight:368.34PPO-IN-1
PPO-IN-1 is a potent inhibitor of protoporphyrinogen IX oxidase (PPO) (Ki: 2.5 nM).Formula:C18H10F3N3O4SColor and Shape:SolidMolecular weight:421.35Rpi 856 C
CAS:Rpi 856 C is a retrovirus protease inhibitor from Streptomyces that is effective against HIV-1 and HTLV-1 proteases.Formula:C39H56N6O10Purity:98%Color and Shape:SolidMolecular weight:768.90Clavicoronic acid
CAS:Clavicoronic acid, a β-lactamase inhibitor, boosts penicillin antibiotics against resistant bacteria.Formula:C15H18O4Color and Shape:SolidMolecular weight:262.3S-HP210
S-HP210: selective GR modulator, blocks NF-κB (IC50: 1.92 μM), non-toxic to mouse fibroblasts.Formula:C22H19N3O2S2Color and Shape:SolidMolecular weight:421.545-Iminodaunorubicin hydrochloride
CAS:5-Iminodaunorubicin HCl: quinone-modified anthracycline with antitumor properties, induces DNA breaks in cancer cells.Formula:C27H31ClN2O9Color and Shape:SolidMolecular weight:563.00Antibacterial agent 81
CAS:Antibacterial agent 81 blocks DNA transcription, targets S. aureus (MIC 12.5μM) & M. smegmatis (MIC 7.8μM). Used in infection research.Formula:C33H28N2O8Color and Shape:SolidMolecular weight:580.58O-GlcNAcase-IN-1
O-GlcNAcase-IN-1 is a potent and novel inhibitor of O-GlcNAcase(OGA) with an IC 50 value of 46 nM.Formula:C15H22N6Color and Shape:SolidMolecular weight:286.38GG-43
GG-43 is a potent inhibitor of LIN28. The IC50 value of GG-43 against human LIN28A is 4 μM [1].Formula:C21H21NO3Color and Shape:SolidMolecular weight:335.4Squalestatin 2
CAS:Squalestatin 2 is an inhibitor of squalene synthase.Formula:C33H44O13Purity:98%Color and Shape:SolidMolecular weight:648.698(S),15(S)-DiHETE
CAS:8(S),15(S)-DiHETE, from 15(S)-HETE's oxidation by 15-LO, triggers eosinophil movement at 1.5 μM; it counteracts pain and LTB4 effects.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47Murizatoclax
CAS:AMG 397 is an oral MCL1 inhibitor .Formula:C42H57ClN4O5SPurity:98%Color and Shape:SolidMolecular weight:765.44Antiproliferative agent-4
Antiproliferative agent-4 suppresses cancer cell growth with low toxicity, inhibits tumors in mice, and induces apoptosis in EC109 cells.Formula:C29H35ClO8Color and Shape:SolidMolecular weight:547.04Antitumor agent-50
Antitumor agent-50 (compound 1a) is a thiazolidinone.Formula:C17H14FNO3SColor and Shape:SolidMolecular weight:331.36MRS-2339
CAS:MRS-2339 is a P2X receptor activator.Formula:C12H15ClN5O6PColor and Shape:SolidMolecular weight:391.70Antifungal agent 28
Antifungal 28 disrupts Candida, hits fluconazole-resistant strains, and inhibits biofilms.Formula:C22H29N5OSColor and Shape:SolidMolecular weight:411.56Tubulin polymerization-IN-34
"Tubulin-IN-34 inhibits oxazolylisoindole microtubule assembly, selective for VL51 lymphoma."Formula:C31H35N3O6Color and Shape:SolidMolecular weight:545.63Enpp-1-IN-7
Enpp-1-IN-7: potent enpp-1 inhibitor, broad specificity, potential in cancer/infectious disease research. (WO2021203772A1)Formula:C18H19N7O4SColor and Shape:SolidMolecular weight:429.45FGFR4-IN-9
FGFR4-IN-9 is a selective inhibitor of FGFR4 (IC50: 75.3 nM) that effectively inhibits the growth and angiogenesis of hepatocellular carcinoma cells.Formula:C24H22ClF3N4O4Color and Shape:SolidMolecular weight:522.9TCMDC-125431
TCMDC-125431 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystals.Formula:C25H27N3O2SColor and Shape:SolidMolecular weight:433.57E7090 succinate
CAS:E7090 succinate inhibits FGFR1, FGFR2, and FGFR3 with IC50: 0.71, 0.50, 1.2 nM; less so FGFR4 at 120 nM.Formula:C76H92N10O24Color and Shape:SolidMolecular weight:1529.60Motuporin
CAS:Motuporin is an inhibitor of type-1 and type-2A protein phosphatase catalytic subunits (PP-1c and PP-2Ac).Formula:C40H57N5O10Color and Shape:SolidMolecular weight:767.91KDM1/CDK1-IN-1
KDM1/CDK1-IN-1 inhibits KDM1 (IC50: 0.096 μM) & CDK1 (IC50: 0.078 μM), blocks HOP-92 G2/M phase, induces apoptosis, toxic to cancer cells.Formula:C22H17N5O3SColor and Shape:SolidMolecular weight:431.47CD33 splicing modulator 1
Compound 1 modulates CD33, affects microglial cells, and may aid in neurodegenerative disease research.Formula:C25H25FN6OColor and Shape:SolidMolecular weight:444.5HPK1-IN-14
CAS:HPK1-IN-14 is a potent inhibitor of HPK1. HPK1-IN-14 has potential for the study of HPK1-related diseases.Formula:C24H23FN6O2Color and Shape:SolidMolecular weight:446.48IRAK4-IN-14
CAS:IRAK4-IN-14 is a selective, potent, orally active IRAK4 inhibitor (IC50: 0.003 μM) with favorable PK parameters in rats and mice. effect.Formula:C25H28FN9OColor and Shape:SolidMolecular weight:489.55α-Glucosidase-IN-14
α-Glucosidase-IN-14 is a potent inhibitor of α-glucosidase (IC50: 5.22 μM).Formula:C24H27N5O4S2Color and Shape:SolidMolecular weight:513.63Leukotriene F4
CAS:LTF4, made in vitro from LTE4 with enzymes, contracts vascular muscle weakly; potency is LTD4 > LTC4 > LTE4 >> LTF4.Formula:C28H44N2O8SColor and Shape:SolidMolecular weight:568.72L 689065
CAS:L 689065 is a 5-lipoxygenase inhibitor.Formula:C35H33ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:597.17RSV-IN-7
CAS:RSV-IN-7 (example 253) is a RSV inhibitor ( EC 50 : < 0.4 μΜ) .Formula:C27H22F3N7O3Color and Shape:SolidMolecular weight:549.50PI3K-IN-27
CAS:PI3K-IN-27 is a potent PI3K inhibitor, relevant for cancer and immune disease research. See patent WO2021233227A1.Formula:C30H26F2N6O2SColor and Shape:SolidMolecular weight:572.63PCSK9-IN-17
CAS:PCSK9-IN-17 is a PCSK9 inhibitor utilized in the research of cholesterol metabolism.Formula:C16H19N5OSColor and Shape:SolidMolecular weight:329.42RS 2135
CAS:RS 2135 is a novel class I antiarrhythmic agent to inhibit ischemia-induced ventricular arrhythmias.Formula:C18H21ClN2O2Purity:98%Color and Shape:SolidMolecular weight:332.83RMS5
CAS:RMS5: hambanine analogue, inhibits P-gp, anti-cancer with cytotoxic, anti-proliferative effects, reduces Bcl-2 proteins, cleaves PARP.Formula:C35H38N2O5SColor and Shape:SolidMolecular weight:598.75Antiproliferative agent-8
Compound 5a, an anticancer agent, enhances P53 and has antiproliferative effects.Formula:C22H16ClN3O3Color and Shape:SolidMolecular weight:405.83Galidesivir
CAS:Galidesivir (BCX4430) is an antiviral compound that inhibits viral RNA-dependent RNA polymerase (RdRp) activity and reduces lung infections in infected animals.Formula:C11H15N5O3Purity:96.73% - 99.13%Color and Shape:SolidMolecular weight:265.27Antibacterial agent 63
CAS:Aztreonam-siderophore conjugate 63 is an antibacterial agent that exhibits efficacy against Gram-negative bacteria through the linkage of aztreonam to aFormula:C35H43N9O14S2Color and Shape:SolidMolecular weight:877.9Azotomycin
CAS:Azotomycin is an antagonist of L-glutamine and may be used as an immunosuppressant.Formula:C17H23N7O8Purity:98%Color and Shape:SolidMolecular weight:453.41TRPA1 Antagonist 1
CAS:TRPA1 Antagonist 1 is an antagonist of TRPA1(IC50: 8 nM) and is a methylene phosphate prodrug which converts to its active parent drug.Formula:C24H20F6N5Na2O7PSPurity:98%Color and Shape:SolidMolecular weight:713.45ARG1-IN-1
CAS:ARG1-IN-1 is a human arginase 1 inhibitor with an IC 50 of 29 nM.Formula:C11H21BN2O4Color and Shape:SolidMolecular weight:256.11AA 497 (Free Base)
CAS:AA 497, a beta-2 agonist, causes relaxation and suppresses Ca spike frequency.Formula:C14H21NO3Purity:98%Color and Shape:SolidMolecular weight:251.32KMN-80
CAS:KMN-80 is a potent, selective EP4 agonist with IC50 3 nM, spurring osteoblast differentiation, and showing in vivo bone repair efficacy.Formula:C21H33NO4Color and Shape:SolidMolecular weight:363.49Numidargistat
CAS:CB-1158 is a potent and orally bioavailable inhibitor of arginase (IC50s: 86 and 296 nM for recombinant human arginase 1 and 2).Formula:C11H22BN3O5Purity:98%Color and Shape:SolidMolecular weight:287.12BMS-986104 HCl
CAS:BMS-986104 is a potent and selective S1P1 receptor modulator.Formula:C22H36ClNOPurity:98%Color and Shape:SolidMolecular weight:365.98Lunacalcipol
CAS:Lunacalcipol is used for the treatment of Secondary Hyperparathyroidism.Formula:C28H42O4SColor and Shape:SolidMolecular weight:474.7Hoe 892
CAS:Hoe 892 is a stable thia-thimo-analogue of prostacyclin and acts as a platelet aggregation inhibitor.Formula:C20H33NO4SColor and Shape:SolidMolecular weight:383.55ALOX15-IN-1
ALOX15-IN-1 (8b) inhibits rabbit/human ALOX15; IC50: 0.04 μM for LA, 2.06 μM for AA.Formula:C24H31N3O5SColor and Shape:SolidMolecular weight:473.59SARS-CoV-2 nsp14-IN-2
SARS-CoV-2 nsp14-IN-2: Strong Nsp14 methyltransferase inhibitor (IC50: 0.09 μM), potential for COVID-19 research.Formula:C21H21N5O5SColor and Shape:SolidMolecular weight:455.49Cleistanthin
CAS:Cleistanthin, a toxic Cleistanthus collinus compound, has antihypertensive, alpha-antagonist, and diuretic properties; a modified naphthofuran-xylose.Formula:C28H28O11Color and Shape:SolidMolecular weight:540.52
